Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
09/2002
09/10/2002US6448286 Imino pyrrolidine derivatives useful as nitric oxide synthase inhibitors
09/10/2002US6448285 Disorders associated with overactivity of 5 alpha reductase; androgen dependent disorders such as seborrhoea, acne, hirsutism and/or androgenic alopecia
09/10/2002US6448257 Tricyclic carboxamides contain a piperazine or piperidine moiety; antiinflammatory agents; heart and kidney conditions
09/10/2002US6447748 Benzamide compounds for cancer imaging and therapy
09/06/2002WO2002068424A1 Indole derivatives having an inhibitory effect on protein kinases
09/06/2002WO2002068414A2 Analogs of thalidomide as potential angiogenesis inhibitors
09/06/2002WO2002068399A1 Aryl carbamate derivatives, preparation and use thereof
09/06/2002WO2002068390A1 Diamides which inhibit tryptase and factor xa activity
09/06/2002WO2002068389A2 Indole derivatives with inhibitor effects on phenol oxidase
09/06/2002WO2002068380A1 Synthetic excitatory amino acids
09/06/2002WO2002067939A1 Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
09/06/2002WO2002067937A1 Indoline and tetrahydro-quinolines as prodrugs for tumour treatment
09/06/2002WO2002067930A1 Benz-indole and benzo-quinoline derivatives as prodrugs for tumor treatment
09/06/2002WO2002067918A1 Novel diallylmethylamine derivative
09/06/2002WO2002067865A2 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof
09/06/2002WO2002050029A3 Tetracyclic derivatives as spla2 inhibitors
09/06/2002WO2002046153A3 Process for the preparation of zafirlukast
09/06/2002WO2002032421A8 Indole compounds as minimally physiologial function monitioring agents
09/06/2002WO2002022577A3 Hydroxamate derivatives useful as deacetylase inhibitors
09/06/2002WO2002005796A3 Use of a spla2 inhibitor for the treatment of sepsis
09/06/2002CA2439265A1 Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
09/06/2002CA2438828A1 Aryl carbamate derivatives, preparation and use thereof
09/06/2002CA2437114A1 Diamides which inhibit tryptase and factor xa activity
09/05/2002US20020123513 Administering indole-2-carboxylic amide derivatives of given formula
09/05/2002US20020123485 For therapy of hypertension, cirrhosis and ascites
09/05/2002DE10109280A1 Indolderivate mit inhibitorischer Wirkung auf Proteinkinasen Indole derivatives having an inhibitory effect on protein kinases
09/04/2002EP1236728A2 S-type 2-substituted hydroxy-2-indolinylbutyric ester compounds and process for preparation thereof
09/04/2002EP1236723A1 Sulfamide derivatives useful as beta3 agonists and pharmaceutical uses thereof
09/04/2002EP1236711A2 Using allosteric hemoglobin modifiers to decrease oxygen affinity in blood
09/04/2002EP1235801A2 Solid pharmaceutical preparation
09/04/2002EP1235571A1 Use of melatonin for treating androgenetic and diffuse alopecia
09/04/2002EP1068184B1 N-aryloxyethylamine derivatives for the treatment of depression
09/04/2002CN1367168A Indoquinone compound and its preparation method
09/04/2002CN1090205C Condensed ring azo compound and its producing method and use
09/04/2002CN1090204C Multifunctional cyanate ester and epoxy blends
09/04/2002CN1090185C Pyridonecarboxylic acid derivative substituted by bicyclic amino group, ester thereof, salt thereof, and bicyclic amine as intermediate thereof
09/04/2002CN1090181C N-substituted 4-hydroxyindole derivatives and keratin fidre dyeing compsns. containing same
09/03/2002US6444849 Amide derivatives
09/03/2002US6444819 Benzylpiperazinyl and piperidinyl ethanone derivatives: dopamine receptor subtype specific ligands
09/03/2002US6444704 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
09/03/2002US6444697 Synthetic compounds for treatment of inflammation
09/03/2002CA2258960C A process for preparing naphthyridones and intermediates
09/01/2002CA2373578A1 .beta.3, agonists and uses thereof
08/2002
08/29/2002WO2002067053A2 High speed photothermographic materials containing tellurium compounds and methods of using same
08/29/2002WO2002066672A2 Treatment of cns disorders using d-amino acid oxidase and d-aspartate oxidase antagonists
08/29/2002WO2002066462A1 Pyrazole derivatives against tgf overexpression
08/29/2002WO2002066459A1 Indole derivatives and their use as gnrh antagonists
08/29/2002WO2002066446A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
08/29/2002WO2002066427A2 (+)-1-(3,4-dichlorophenyl)-3-azabicyclo[3.1.0]hexane, compositions and uses thereof
08/29/2002WO2002066426A2 Fluoro oxindole derivatives as modulators of kcnq potassium channels
08/29/2002WO2002066073A1 Method of examining effect of angionegesis inhibitor mediated by the inhibition of integrin expression
08/29/2002WO2002042304A3 Cyclopenta[b][1,4] diazepino[6,7,1-hi]indoles as 5ht2c antagonists
08/29/2002WO2002042273A3 Acid derivatives useful as serine protease inhibitors
08/29/2002WO2000066104A9 Ace-2 inhibiting compounds and methods of use thereof
08/29/2002WO1999064055A9 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht4 receptors
08/29/2002US20020120583 Dynamic number authentication for credit/debit cards
08/29/2002US20020120148 Benzocycloheptenylamino derivatives; treatment of pollakiuria or urinary incontinence
08/29/2002US20020120137 FXR modulators
08/29/2002US20020120011 Substituted N, N-disubstituted diamino compounds useful for inhibiting cholesteryl ester transfer protein activity
08/29/2002US20020120007 Benzamide inhibitors of factor Xa
08/29/2002US20020119976 Tetracyclic derivatives, process of preparation and use
08/29/2002US20020119972 Cannabinoid receptor modulators, their processes of preparation, and use of cannabinoid receptor modulators for treating respiratory and non-respiratory diseases
08/29/2002US20020119971 Antiinflammatory agents; skin disorders; central nervous system disorders
08/29/2002US20020119966 Central nervous system disorders
08/29/2002US20020119961 Bridged piperazine derivatives
08/29/2002US20020119956 Using thalidomine
08/29/2002US20020119910 Drug delivery
08/29/2002US20020119191 Pharmaceutical or food composition for treatment or prevention of brain edema
08/29/2002CA2438805A1 Fluoro oxindole derivatives as modulators of kcnq potassium channels
08/29/2002CA2438264A1 Heterocyclic substituted carbonyl derivatives and their use as dopamine d3 receptor ligands
08/29/2002CA2433866A1 Treatment of cns disorders using d-amino acid oxidase and d-aspartate oxidase antagonists
08/28/2002EP1233768A1 Carvedilol methanesulfonate
08/28/2002EP1140898B1 Amide and urea derivatives as 5-ht reuptake inhibitors and as 5-ht1b/1d ligands
08/28/2002EP0846110B1 Thf-containing sulfonamide inhibitors of aspartyl protease
08/28/2002CN1365972A Indole derivatives and its anticancer usage
08/28/2002CN1365971A Antibacterial activity, induction, separation and synthesis of N-acyltryptamine derivative as plant protecting chemical
08/28/2002CN1089765C 1H-pyrido [3,4-b] indole-4-carboxamide derivatives, preparation and application thereof in therapeutics
08/28/2002CN1089764C Substituted heterocyclic compounds, preparation method thereof and pharmaceutical compositions containing same
08/27/2002US6441192 Adding acid chloride and alkyl or aryl magnesium halide separately and simultaneously to a stirred solution of an indole such that the two reagents do not come into immediate contact; synchronised rates of molar addition
08/27/2002US6441175 Useful in treating various neuropsychological disorders including, schizophrenia, dementia, depression, anxiety, parkinson-like motor disorders and motion disorders
08/27/2002US6441023 For therapy of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone disease, diabetes (insulin resistance) and hiv infection
08/27/2002US6441021 Type-iv collagenase inhibitors
08/27/2002US6441004 Monocyte chemoattractant protein-1 inhibitor compounds
08/27/2002US6440889 Amine elimination process for making single-site catalysts
08/27/2002CA2167039C Alkylated (hetero)cyclic compounds; process for preparing the same and pharmaceutical compositions containing them
08/27/2002CA2045955C Indole derivatives
08/22/2002WO2002064576A1 Heteroaryl alkyl piperazine derivatives as fatty acid oxidation inhibitors
08/22/2002WO2002064565A1 Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical
08/22/2002WO2002064564A1 Benzo'f!isoindole derivatives with affinity to the ep4 receptor
08/22/2002WO2002064551A1 Hiv protease inhibitors based on amino acid derivatives
08/22/2002WO2002064546A2 Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical
08/22/2002WO2002064545A1 Acylated indanyl amines and their use as pharmaceuticals
08/22/2002WO2002064533A1 Obtaining anthracene and carbazole by melt-crystallization
08/22/2002WO2002064133A1 Preparations for controlling concentration in blood
08/22/2002WO2002040008A3 Treatment of sexual dysfunction with non peptide bombesin receptor antagonists
08/22/2002WO2002038557A3 Benzoylbenzofurane derivatives for treatment of cardiac arrhythmia
08/22/2002WO2002004412A3 Tyrosine derivatives as phosphatase inhibitors
08/22/2002US20020115869 Lambda-shaped carbazole and main-chain NLO polyurethane containing the same
08/22/2002US20020115857 Useful as an intermediate of a carbocyclic nucleoside anti-viral agent; reacting 2-azabicyclo(2.2.1)hept-5-en-3-one with a sulfonyl halide or phosphoryl halide and then with a nucleic acid base
08/22/2002US20020115826 Enzyme inhibitor for use for use in the treatment of cell proliferative defects