Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
06/2002
06/18/2002US6407102 Indole derivatives and their use for the treatment of malignant and other diseases based on pathological cell proliferation
06/18/2002CA1341370C Fused polycyclic compounds, methods of manufacture, and their use as paf antagonists, antihistamines and/or antiinflammatory agents
06/14/2002WO2001044187A1 Novel substituted tricyclic compounds
06/14/2002CA2394778A1 Novel substituted tricyclic compounds
06/13/2002WO2002046166A1 Phenylethenyl or phenylethinyl derivatives as glutamate receptor antagonists
06/13/2002WO2002046164A1 Therapeutic compounds
06/13/2002WO2002046155A1 Synthesis of fused pyrrolecarboxamides
06/13/2002WO2002046154A1 Peroxisome proliferator activated receptor d activators
06/13/2002WO2002046153A2 Process for the preparation of zafirlukast
06/13/2002WO2002046149A2 2-thio-5-amino substituted benzoquinones, their manufacture and their use in rubber
06/13/2002WO2002046129A2 Inhibitors of histone deacetylase
06/13/2002WO2002024648A3 Process for the preparation of cell proliferation inhibitors
06/13/2002WO2002015891A3 Pharmaceutical combination of angiotensin ii antagonists and ace inhibitors
06/13/2002WO2001037819A3 Use of indirubine derivatives for making medicines
06/13/2002US20020072636 Optically active diphosphines, preparation thereof according to a process for the resolution of the racemic mixture and use thereof
06/13/2002US20020072616 3-azabicyclo[3.1.0]hexane derivatives useful in therapy
06/13/2002US20020072531 Useful as anticoagulants in mammals; inhibitors of factor Xa
06/13/2002US20020072529 For therapy and prophylaxis of cerebral apoplexy and craniocerebral trauma
06/13/2002US20020072516 For therapy of diabetes, obesity, autoimmune disorders, acute and chronic inflammatory disorders, osteoporosis, cancer, malignant disorders
06/13/2002CA2430841A1 Synthesis of fused pyrrolecarboxamides
06/12/2002EP1212375A2 Ph sensitive cyanine dyes as reactive fluorescent reagents
06/12/2002EP1212320A2 Phenylpiperazines as serotonin reuptake inhibitors
06/12/2002EP1212318A1 Substituted indolinones as tyrosine kinase inhibitors
06/12/2002EP1212317A1 Indole derivatives and their use for the treatment of osteoporosis amongst other applications
06/12/2002EP1212303A2 Bicyclic androgen and progesterone receptor modulator compounds and methods
06/12/2002EP1212302A1 Compounds and pharmaceutical compositions as cathepsin s inhibitors
06/12/2002EP1212298A1 Isolation of natural l-beta-3-indolylalanine and enrichment of natural aliphatic amino acid mixtures with natural l-beta-3-indolylalanine
06/12/2002EP1212296A1 Phosphate mimics and methods of treatment using phosphatase inhibitors
06/12/2002EP1212268A1 Catalyst for pauson-khand reaction
06/12/2002EP1212081A2 Pharmaceutical formulations and use thereof in the prevention of stroke, diabetes and/or congestive heart failure
06/12/2002EP0885210B1 Tricylic compounds having binding affinity for melatonin receptors, their production and use
06/12/2002EP0782577B1 Asymmetric ligands useful for transition metal catalyzed bond forming reactions and epoxide reactions therewith
06/12/2002EP0688211B1 Thalidomide for inhibition of angiogenesis
06/12/2002CN1353691A Cell adhesion-inhibiting anti inflammatory and immune-suppresive compounds
06/11/2002US6403808 Treating mental disorders
06/11/2002US6403792 Sulfonyl isatin compounds and methods of blocking apoptosis therewith
06/11/2002US6403644 For prevention and/or treatment of diseases induced by overexpression and excess activity of matrix metalloproteinase; for example, rheumatoid, arthrosteitis, unusual bone resorption, osteoporosis, periodontitis
06/11/2002US6403632 Cyclic amide derivative
06/11/2002US6403587 Autoimmune diseases, acute and chronic inflammatory conditions, allergic conditions, infection associated with inflammation, viral, transplantation tissue rejection, atherosclerosis, restenosis, hiv infectivity, and
06/11/2002US6403577 Hexamethyleneiminyl tachykinin receptor antagonists
06/11/2002US6403561 Disorders associated with the inactivation or excessive degradation of cholecystokinin; inhibiting the enzymatic hydrolysis of cholecystokinin 1-(2(s)-aminobutyryl)-2(s)-indolinecarboxylic acid
06/11/2002US6403055 Carboxylated polyamine compound
06/11/2002CA2065192C Process for the production of 2-azabicyclo[2.2.1]hept-5-en-3-one
06/11/2002CA2031756C Isatine derivatives, their preparation and use
06/06/2002WO2002044416A2 Sulfonated diarylrhodamine dyes as fluorescent labels
06/06/2002WO2002044168A2 Indole-type inhibitors of p38 kinase
06/06/2002WO2002044152A1 Indoline derivatives and their use as 5-ht2 receptor ligands
06/06/2002WO2002044151A1 1,4-disubstituted piperazine derivatives useful as uro-selective $g(a)1-adrenoceptor blockers
06/06/2002WO2002044150A1 Chemical process and new intermediates
06/06/2002WO2002044149A1 Indole and dihydroindole derivatives
06/06/2002WO2002044148A2 Aryl-substituted indirubin derivatives, the production thereof and use of the same
06/06/2002WO2002044120A1 Compounds active at the glucocorticoid receptor iii
06/06/2002WO2002043667A2 HYDROLYSIS OF [R(R*,R*)]-2-(4-FLUOROPHENYL)-β,δ -DIHYDROXY-5-(1-METHYLETHYL)-3-PHENYL-4-[(PHENYLAMINO)CARBONYL]-1H-PYRROLE-1-HEPTANOIC ACID ESTERS WITH CALCIUM HYDROXIDE
06/06/2002WO2002014294A3 Heterocyclic sulfonamide derivatives and their use for potentiating glutamate receptor function
06/06/2002WO2001003684A3 Albumin-binding compounds that prevent nonenzymatic glycation and that may be used for treatment of glycation-related pathologies
06/06/2002US20020068831 Intermediate for the synthesis of amlodipine, a process for the preparation there and corresponding use
06/06/2002US20020068756 Inhibition of phosphodiesterase; 3-carbocyclic(alkyl)oxy-2-aryl(alkyl)aminocarbonyl-1-aryl(alkyl)indole or azaindole derivatives
06/06/2002US20020068692 Administration a melatonin blocker to patients with disorders associated with altered dopamine function; preclinical diagnosis by administering melatonin to induce a mild transient form of the disorder
06/06/2002CA2430343A1 1,4-disubstituted piperazine derivatives useful as uro-selective .alpha.1-adrenoceptor blockers
06/06/2002CA2430064A1 Chemical process and new intermediates
06/06/2002CA2429816A1 Sulfonated diarylrhodamine dyes as fluorescent labels
06/06/2002CA2429382A1 Indole-type inhibitors of p38 kinase
06/06/2002CA2427255A1 Hydrolysis of [r(r*,r*)]-2-(4-fluorophenyl)-.beta.,.delta. -dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid esters with calcium hydroxide
06/05/2002EP1211301A1 Organic electroluminescent device
06/05/2002EP1210343A2 Benzoic acid derivatives and their use as ppar receptor agonists
06/05/2002EP1210333A2 Novel herbicides
06/05/2002EP1210329A2 Aminoalkoxy carbazoles and their use as 5-ht ligands
06/05/2002EP1210328A1 Fused pyrrolecarboxamides: a new class of gaba brain receptor ligands
06/05/2002EP1210321A1 Aminosalicylclic acid amides and their use for combating organisms that are harmful to plants
06/05/2002EP0966430B1 Anti-inflammatory compounds
06/05/2002EP0934319B1 1H-PYRIDO[3,4-b]INDOLE-4-CARBOXAMIDE DERIVATIVES, PREPARATION AND APPLICATION THEREOF IN THERAPEUTICS
06/05/2002EP0923551B1 4-aminoethoxy indolone derivatives
06/05/2002EP0851855B1 Acylated derivatives of melatonin and its analogues, useful as medicaments
06/05/2002CN1352545A 吲哚衍生物 Indole derivatives
06/05/2002CN1085980C Meta-guanidine, urea, thiourea or azacyclic amino benzoic and derivatives as integrin antagaonists
06/04/2002US6399808 Reacting amine with carbon dioxide in anhydrous solvent
06/04/2002US6399785 Multiply-substituted fullerenes
06/04/2002US6399780 Kinase inhibitors; anticancer agents
06/04/2002US6399656 Using a benzopyran-3-carboxamide compound
06/04/2002US6399631 Carbazole neuropeptide Y5 antagonists
06/04/2002US6399614 1-(N-phenylaminoalkyl)piperazine derivatives substituted at position 2 of the phenyl ring
06/04/2002US6399601 Antidiabetic agents; nervous system disorders; anticholesterol agents
05/2002
05/30/2002WO2002043449A1 Luminescent element material and luminescent element comprising the same
05/30/2002WO2002042412A2 Protease inhibitors and their pharmaceutical uses
05/30/2002WO2002042304A2 Cyclopenta[b][1,4] diazepino[6,7,1-hi]indoles as 5ht2c antagonists
05/30/2002WO2002042294A1 1-sulfonyl substituted tryptophane derivatives and its use as integrin inhibitors
05/30/2002WO2002042292A2 Indol derivative and their use as inhibitors of p38 kinase
05/30/2002WO2002042273A2 Acid derivatives useful as serine protease inhibitors
05/30/2002WO2002042269A1 3-arylindole derivatives and their use as cb2 receptor agonists
05/30/2002WO2002042250A1 DERIVATIVES OF 4-HYDROXYBUTANOIC ACID AND OF ITS HIGHER HOMOLOGUE AS LIGANDS OF η-HYDROXYBUTYRATE (GHB) RECEPTORS, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND PHARMACEUTICAL USES
05/30/2002WO2002041889A2 Indolsulfonyl compounds useful in the treatment of cns disorders
05/30/2002WO2002041835A2 Estrogen receptor modulators
05/30/2002WO2002020526A3 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
05/30/2002WO2002014275A3 Heterocyclic sulfonamide derivatives and their use for potentiating glutamate receptor function
05/30/2002WO2001064646A3 Hydrazones and analogs as cholesterol lowering agents
05/30/2002WO2001047882A3 Substance library which can be obtained by reacting aldehydes with secondary amines, acid chlorides and naphthol, pyrrole and/or indole compounds
05/30/2002WO2000076489A3 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
05/30/2002US20020065192 Productivity catalysts and microstructure control
05/30/2002US20020064794 Modified carbocyanine dyes and their conjugates
05/30/2002US20020064782 Fluorescent nucleotides