Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
10/2002
10/10/2002CA2441077A1 Substituted carbazoles as inhibitors of spla2
10/10/2002CA2406832A1 Preventives/remedies for alzheimer's disease
10/09/2002EP1247803A2 Indolinone compounds suitable for modulation of protein kinases
10/09/2002EP1246819A1 A method for the preparation of substituted benzene derivatives
10/09/2002EP1246818A1 Novel indole derivatives
10/09/2002EP1246817A1 4-phenyl-1-piperazinyl, -piperidinyl and -tetrahydropyridyl derivatives
10/09/2002EP1246816A1 Substituted phenyl-piperazine derivatives, their preparation and use
10/09/2002EP1246815A1 Phenylpiperazinyl derivatives
10/09/2002EP1246803A1 Piperidine and piperazine derivatives which function as 5-ht 2a? receptor antagonists
10/09/2002EP1246795A2 Antibacterial agents
10/09/2002EP1246625A2 Methods and compositions for mitigating pain using nitrate esters
10/09/2002EP1246621A1 Nitrosated and nitrosylated cyclooxygenase-2 inhibitors, compositions and methods of use
10/09/2002EP1246620A1 Substituted acylhydroxamic acids and method of reducing tnf-g(a) levels
10/09/2002EP1000025A4 Substituted naphthopyrans
10/09/2002EP0946542B1 Indane or dihydroindole derivatives
10/09/2002CN1373754A Antibacterial agents
10/09/2002CN1092193C Prolylendopeptidase inhibitors
10/08/2002US6462234 Process to prepare (2S)-2-(dipropylamino)-6-ethoxy-2, 3-dihydro-1H-indene-5-carboxamide
10/08/2002US6462207 Which upon further chemical modification are useful in biomedical applications, permit the synthesis of new polymers, may be used as intermediates in the preparation of compositions possessing properties of interest
10/08/2002US6462092 Such as 3-((3-fluorophenyl)-((3-(trifluoromethyl)phenyl)-methyl)amino)-1,1,1 -trifluoro-2-propanol; cardiovascular disease, i.e. atherosclerosis and other coronary artery diseases
10/08/2002US6462073 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
10/08/2002US6462056 Oxazolidines as 5-HT2A-antagonists
10/08/2002US6462048 3-(2-(4-methylpiperazin-1-yl)-benzylidene)-1,3-dihydro-indol-2-one for example; useful as psychotherapeutic agents
10/08/2002US6462032 Cyclic regimens utilizing indoline derivatives
10/03/2002WO2002076988A2 Tert. alkylphenoxy substituted polycyclic compounds
10/03/2002WO2002076964A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
10/03/2002WO2002076963A1 Bicyclic guanidine derivatives and therapeutic uses thereof
10/03/2002WO2002076929A1 Aryl and biaryl compounds having mch modulatory activity
10/03/2002WO2002076402A2 Fatty amine drug conjugates
10/03/2002WO2000034265A3 Quinoline-indole antimicrobial agents
10/03/2002WO1998008787A3 Resolution of racemic mixtures using polymers containing chiral units
10/03/2002US20020143186 For prophylaxis and therapy of hyperglycemia, Type 1 diabetes, Type 2 diabetes, disorders of the lipid metabolism, such as dyslipidemia, and obesity
10/03/2002US20020143046 Used as calcium channel blockers
10/03/2002US20020143045 Reacting 4-(oxiran-2-ylmethoxy)-9H- carbazole with 2-(2-methoxyphenoxy)ethylamine to produce carvedilol
10/03/2002US20020143036 Pentafluorobenzenesulfonamides and analogs
10/03/2002US20020143027 As inhibitors of tumor necrosis factor; for therapy of cachexia, arthritis, rheumatoid arthritis, osteoarthritis, reperfusion injury, congestive heart failure, Crohn's disease, ulcerative colitis, systemic lupus erythrematosis
10/02/2002EP1245565A1 Indenoindolone derivatives, process for their preparation and pharmaceutical compositions containing them
10/02/2002EP1245229A2 Methods and compositions for inhibition of angiogenesis
10/02/2002EP1244626A2 Caspase inhibitors and uses thereof
10/02/2002EP1244621A1 Nitrile derivatives as cathepsin k inhibitors
10/02/2002EP1244616A1 (hetero)bicyclylmethanesulfonylamino-substituted hydroxamic acid derivatives
10/02/2002EP0917529A4 Catalyst compositions and processes for olefin oligomerization and polymerization
10/02/2002EP0843675B1 Aza-anthracyclinone derivatives
10/02/2002EP0706521B1 Imides as tnf alpha inhibitors
10/02/2002EP0679641B1 Sulfonamide and sulfonic ester derivatives each having tricyclic hetero ring
10/02/2002DE10114138A1 Cdk-inhibitorische Indirubinderivate mit erhöhter Löslichkeit Cdk-inhibitory indirubin derivatives with increased solubility
10/02/2002CN1372547A Aminoalkoxy carbazoles for the treatment of CNS diseases
10/02/2002CN1372546A Fused pyrrolecarboxamides GABA brain receptor ligands
10/02/2002CN1372545A 吲哚衍生物 Indole derivatives
10/01/2002US6458985 Use of compressed CO2 in chemical reactions
10/01/2002US6458965 Herbicides, antigrowth agents and surfactants for wood preservatives
10/01/2002US6458852 Use of substituted N, N-bis-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
10/01/2002US6458849 Method of treating or preventing a ceip-mediated disorder in a subject by administering a therapeutically effective amount of a compound for strokes
10/01/2002US6458824 Solid preparation
10/01/2002US6458806 Aryl alkenamides derivatives as MCP-1 antagonists
10/01/2002US6458803 Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
10/01/2002US6458781 Blockers calcium channel antagonists for strokes, brain disorders
10/01/2002US6458337 Diagnostic imaging contrast agent with improved in serum relaxivity
10/01/2002CA2209018C Sulfonamides and their use
10/01/2002CA2059708C Indole derivatives
09/2002
09/26/2002WO2002074764A2 Piperazine derivatives and their use as 5-ht1b ligands
09/26/2002WO2002074742A2 Cdk-inhibitory indirubin derivatives having an increased solubility
09/26/2002WO2002074740A1 Biguanide derivatives
09/26/2002WO2002074342A1 Remedies for arteriosclerosis
09/26/2002WO2002074309A2 Use of tryptophan derivatives for the specific cytostatic treatment of serotonin-producing tumors
09/26/2002WO2002074306A1 Remedies for fatty liver
09/26/2002WO2002074296A1 Remedies for solid cancer containing hydroxamic acid derivatives as the active ingredient
09/26/2002WO2002055517A3 4-(hetero)aryl substituted indolinones
09/26/2002WO2002038544A3 3-substituted oxindole beta 3 agonists
09/26/2002WO2002024636A3 N-acylsulfonamide apoptosis promoters
09/26/2002WO2002003975A3 Combinations of ssri and estrogenic agents
09/26/2002WO2001091756A3 S-methyl-dihydro-ziprasidone for treatment of psychiatric and ocular disorders
09/26/2002WO2000043375A3 Substituted aryl heterocyclic compounds
09/26/2002WO1997019953A8 New lh-rh antagonists with improved effectiveness
09/26/2002US20020137968 Treating with amides, ureas, amidines, carbamates, carboximidamides and other derivatives of given formula, e.g. (+)-N-((2,2-dimethylcyclopentyl)methyl)-4-hexyloxybenzamide
09/26/2002US20020137961 Use as skin lightening agents; 4-(1,4-Dioxaspiro(4.5)dec-8-yl)-1,3-benzenediol for example
09/26/2002US20020137939 Novel guanidinobenzamides
09/26/2002US20020137929 1 - (3-heterocyclylphenyl) isothiourea, -isourea, -guanidine and -amidine herbicidal agents
09/26/2002US20020137774 Carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
09/26/2002US20020137745 N-(3,5-dichloropyridin-4-yl)-2-(1-(4-fluorobenzyl)-5 -hydroxyindol-3-yl)-2-oxoacetamide, for example; treating eosinophil-related conditions, including chronic obstructive pulmonary disease
09/26/2002US20020137687 Novel compounds that inhibit tryptase activity
09/26/2002US20020137686 Inhibitors of the ICE/ced-3 family of cysteine proteases
09/26/2002US20020137201 Detection of transmembrane potentials by optical methods
09/25/2002EP1242471A1 Substituted group 4 metal complexes, catalysts and olefin polymerization process
09/25/2002EP1242399A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS
09/25/2002EP1242379A1 Curcumin analogues for treating cancer
09/25/2002EP1242376A1 Method for producing oxindoles
09/25/2002EP1242375A2 Method for purifying lactames
09/25/2002EP1242366A1 Salicylamides as serine protease and factor xa inhibitors
09/25/2002EP1242360A2 Exciplexes
09/25/2002EP1242327A1 Pigmented vitreous material its precursor glass items coated therewith and method of its preparation
09/25/2002EP1242082A1 Methods and compositions for the prevention and treatment of atherosclerosis, restenosis and related disorders
09/25/2002EP1242081A1 Caspases and apoptosis
09/25/2002EP1242074A1 5-benzyl-octahydroindole and 6-benzyl-decahydroquinoline nmda/nr2b antagonists
09/25/2002EP1242069A2 Albumin-binding compounds that prevent nonenzymatic glycation and that may be used for treatment of glycation-related pathologies
09/25/2002EP0976731B1 Process for producing 5-methylindolines
09/25/2002EP0968179B1 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
09/25/2002EP0923550B1 Acylaminoalkenylene-amide derivatives as nk1 and nk2 antagonists
09/25/2002EP0835258B1 Novel camptothecin analogues, preparation methods therefor, use thereof as drugs, and pharmaceutical compositions containing said analogues
09/24/2002US6455709 Such as 1,3-dimethyl-fulleropyrrolidine-1,3-dicarboxylic n-amide oligomer