| Patents for C07C 257 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines (2,984) |
|---|
| 11/12/2002 | US6479485 Benzamidine derivatives and their use as anti-coagulants |
| 11/06/2002 | EP1254159A2 Process for the preparation of acetyl-amidiniophenylalanyl-cyclohexylglycyl-pyridinioalaninamides |
| 11/06/2002 | EP1254136A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF |
| 11/06/2002 | EP0923528B1 Oligosaccharide synthesis |
| 11/05/2002 | US6476264 N-(4-carbamimidoyl-phenyl)-glycine derivatives |
| 10/30/2002 | CN1093533C Process for preparing N-(2- or 3-M, 5- or 6-M', 4-amino-phenyl)-N', N'-dimethyl acetamidine |
| 10/29/2002 | US6472405 Glycoprotein IIB/IIIA antagonists |
| 10/29/2002 | US6472393 Serine protease inhibitors |
| 10/24/2002 | WO2002083630A1 Oxalic acid derivatives |
| 10/24/2002 | WO2002083030A2 Bifunctional energy-reversible acyl-compositions |
| 10/24/2002 | WO2002002516A3 Inhibitors of hiv integrase |
| 10/24/2002 | US20020156212 Catalyst systems of alpha -diimine, urethane or urea ligands complexed to nickel, palladium or other transition metals |
| 10/24/2002 | CA2445538A1 Oxalic acid derivatives |
| 10/24/2002 | CA2444262A1 Bifunctional energy-reversible acyl-compositions |
| 10/23/2002 | EP1250317A2 Bis-basic compounds for use as tryptase inhibitors, method for producing the same and their use as medicaments |
| 10/23/2002 | EP1250315A1 Functional monomers for molecular recognition and catalysis |
| 10/17/2002 | US20020151545 Anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and metastasis inhibitors in treating cancer |
| 10/17/2002 | US20020151534 Antithrombotic compounds |
| 10/17/2002 | US20020151524 Aromatic fungicide compound containing N=C-G group wherein G= O, S, S=O, S(O)2 or N(NRR') |
| 10/17/2002 | DE10117823A1 New N-phenyl-oxalamide derivatives, are factor Xa and factor VIIa inhibitors useful e.g. for treating thrombosis, myocardial infarction, inflammation, angina pectoris or tumor diseases |
| 10/16/2002 | CN1374951A Process for the preparation of 4(5)-amino-5(4) carboxamidoimidazoles and intermediates thereof |
| 10/15/2002 | US6465686 Halogenated 2-amino-5,6 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| 10/15/2002 | US6465518 2-amino-5-fluoro-6-(1-iminoethylamino)-hept-4-enoic acid, for example; treating or preventing various causes of inflammation |
| 10/15/2002 | US6465459 Inhibit the enzyme, factor xa |
| 10/10/2002 | WO2002079145A1 BENZAMIDE INHIBITORS OF FACTOR Xa |
| 10/09/2002 | EP1037874B1 1-(adamantyl)amidines and their use in the treatment of conditions generally associated with abnormalities in glutamatergic transmission |
| 10/03/2002 | WO2002076395A2 Agents and methods for treatment of cancer |
| 10/03/2002 | WO2002062766A3 Melanocortin-4 receptor binding compounds and methods of use thereof |
| 10/03/2002 | US20020143061 2-amino-5, 6 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| 10/03/2002 | CA2441394A1 Agents and methods for treatment of cancer |
| 10/02/2002 | EP1244613A2 Methods for producing cyanobenzoic acid derivatives |
| 10/01/2002 | CA2203850C Novel n-phenyl-n-phenyliminonethylbenzamidines and their analogues as muscarinic receptor agonists |
| 09/26/2002 | WO1997019953A8 New lh-rh antagonists with improved effectiveness |
| 09/26/2002 | US20020137730 Positively charged non-natural amino acids, methods of making and using thereof in peptides |
| 09/26/2002 | US20020137687 Novel compounds that inhibit tryptase activity |
| 09/25/2002 | EP1242366A1 Salicylamides as serine protease and factor xa inhibitors |
| 09/24/2002 | US6455529 Adhesion receptor antagonists |
| 09/19/2002 | US20020132849 2-Amino-2-alkyl-5 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors |
| 09/18/2002 | WO2001070678A2 Substituted biphenyl derivatives |
| 09/18/2002 | EP1240149A2 Process to prepare aryltriazolinones and novel intermediates thereto |
| 09/18/2002 | EP0934259B1 Beta-sulfonamido hydroxamic acids as matrix metalloproteinase and tace inhibitors |
| 09/18/2002 | EP0929516B1 Benzamidine derivatives and the use thereof as medicaments with ltb4-antagonistic effect |
| 09/18/2002 | CA2403500A1 Substituted biphenyl derivatives |
| 09/17/2002 | US6451792 Matrix metalloprotease inhibitors |
| 09/17/2002 | CA2041832C Hydrazones |
| 09/12/2002 | WO2002070471A1 Phenyl derivatives and their use in the treatment of thromboembolic disorders or tumours |
| 09/12/2002 | WO2002070468A2 Novel benzamidine derivatives having anti-inflammatory and immunosuppressive activity |
| 09/12/2002 | US20020128510 Antiarthritic agents; rheumatic diseases; osteoarthritis; inhibition of the inducible nitric oxide synthase - induced after activation of vascular smooth muscle, macrophages, endothelial cells by enotoxin and cytokines |
| 09/12/2002 | US20020128315 Amidinophenol derivatives as leukotriene B4 (LTB4)antagonists, phospholipase A2 inhibitors, and trypsin inhibitors. |
| 09/12/2002 | CA2439644A1 Phenyl derivatives and their use in the treatment of thromboembolic disorders or tumours |
| 09/11/2002 | EP0912504B1 Oxazolidine ester |
| 09/10/2002 | USRE37839 Fungicides, insecticides, miticides, nematocides, and pesticides |
| 09/10/2002 | US6448269 Such as 6-(n-(4-(aminoiminomethyl)benzoyl)amino)-3,4-dihydro-4,4-dimethyl-2h-1 -benzopyran-2-yl)acetic acid; inhibiting platelet aggregation or fibrinogen binding or preventing thrombosis |
| 09/05/2002 | DE10110325A1 Phenylderivate 2 Phenyl derivatives 2 |
| 09/04/2002 | EP1236712A1 Amidinophenylpyruvic acid derivative |
| 08/29/2002 | WO2002066418A2 Process for the preparation of arylethanoldiamines useful as agonists of the beta-3-adrenoceptor |
| 08/29/2002 | WO2002042273A3 Acid derivatives useful as serine protease inhibitors |
| 08/29/2002 | WO2002037937A3 Acid derivatives useful as serine protease inhibitors |
| 08/29/2002 | US20020120007 Benzamide inhibitors of factor Xa |
| 08/27/2002 | US6441179 Intermediates useful for the preparation of antihistaminic piperidine derivatives |
| 08/22/2002 | WO2002064136A2 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators |
| 08/21/2002 | EP0802179B1 Substituted amidinonaphthyl ester derivatives |
| 08/15/2002 | WO2002062778A2 Anti-thrombotic compounds, production and use thereof as medicaments |
| 08/15/2002 | WO2002062766A2 Melanocortin-4 receptor binding compounds and methods of use thereof |
| 08/15/2002 | CA2435492A1 Antithrombotic compounds, the preparation thereof and their use as pharmaceutical compositions |
| 08/14/2002 | EP0724435B1 Amidino derivatives useful as nitric oxide synthase inhibitors |
| 08/08/2002 | WO2002060861A1 Benzamidine derivatives and process for production thereof |
| 08/08/2002 | US20020107290 Inhibiting activated blood-coagulation factor X |
| 08/08/2002 | DE10104597A1 Antithrombotische Verbindungen, deren Herstellung und deren Verwendung als Arzneimittel Antithrombotic compounds, their preparation and their use as medicaments |
| 08/07/2002 | EP1227721A1 Novel substituted succinic acid metallo-beta-lactamase inhibitors and their use in treating bacterial infections |
| 08/06/2002 | US6429317 Indane derivatives for antipsychotic compositions |
| 08/01/2002 | WO2002058690A2 Methods for the treatment of diseases using malonyl-coa decarbox ylase inhibitors |
| 08/01/2002 | WO2001078654A3 Halogentated 2-amino-3, 4 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| 08/01/2002 | US20020103398 Double bond acts as a rigidifying element, for unexpected potency and selectivity for inhibition of inducible nitric oxide synthase over the constitutive isoforms |
| 08/01/2002 | US20020103194 Secondary amine, imine, amidine, guanidine, or other nitrogen functional group compounds; for treatment or prevention of diseases in which treatment is mediated by muscarinic receptor agonism such as cognitive decline and Alzheimer's disease |
| 08/01/2002 | US20020102380 Ionic compounds in which the anionic load has been delocalized; ionic conducting materials, electronic conducting materials, colorant, and the catalysis of various chemical reactions including polymerization |
| 07/25/2002 | WO2002057236A1 Phenyl derivatives |
| 07/25/2002 | DE10102322A1 New disubstituted and trisubstituted benzene derivatives useful as coagulation inhibitors for the treatment of thromboembolic diseases |
| 07/24/2002 | EP0804431B1 GLYCOPROTEIN IIb/IIIa ANTAGONISTS |
| 07/23/2002 | US6423737 Benzamidoxime prodrugs as antipneumocystic agents |
| 07/18/2002 | WO2002022558A3 2-amino-2-alkyl-3 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors |
| 07/18/2002 | WO2002022557A3 2-amino-2-alkyl-4 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors |
| 07/17/2002 | EP1222162A1 Novel ltb 4? antagonist, method for the production thereof and its use as a medicament |
| 07/17/2002 | CN1359373A 6[(aryl and heteroaryl)oxy] methyl] naphthalene-2-carboximidamide derivatives, preparation and therapeutic application thereof |
| 07/11/2002 | US20020091210 Group 8-10 transition metal based supported catalyst where the support is treated with a pore-filling agent; improved the catalyst productivity in the presence of hydrogen |
| 07/10/2002 | CN1087283C New LH-RH antigonists with improved effectiveness |
| 07/09/2002 | US6417386 Hydrazone derivatives; acarina; miticides |
| 07/09/2002 | US6417200 Antithrombotic agents |
| 07/09/2002 | CA2217455C New substituted derivatives, of biphenyl or phenylpiridine, their preparation process and the pharmaceutical compositions that contain them |
| 07/03/2002 | CN1356998A Method of producing nitroguanidine-and nitroenamine derivatives |
| 06/27/2002 | US20020082267 Fungicidal phenylamidine derivatives |
| 06/25/2002 | US6410542 Aminotetrazole derivatives useful as nitric oxide synthase inhibitors |
| 06/25/2002 | US6410538 Benzamidine derivatives |
| 06/20/2002 | US20020077482 Novel intermediates useful for the preparation of antihistaminic piperidine derivatives |
| 06/20/2002 | US20020077363 2-amino-4,5 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| 06/19/2002 | EP1215206A1 Processes for the preparation of 4(5)-amino-5(4)-carboxamidoimidazoles and intermediates thereof |
| 06/19/2002 | EP1214291A1 Biphenyl derivatives used as nhe-3 inhibitors |
| 06/19/2002 | EP0837856B1 Pesticidal tris-oximino heterocyclic compounds |
| 06/18/2002 | US6407219 Process for preparing azoiminoethers and azocarboxylic acid esters and novel azocboxylic acid mixed esters |
| 06/13/2002 | US20020072631 2-amino-2-alkyl-3 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors |