Patents
Patents for C07C 257 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines (2,984)
08/2004
08/25/2004CN1524072A Phenyl derivatives and their use in the treatment of thromboembolic disorders or tumours
08/24/2004US6780863 Treat inflammatory and/or allergic conditions
08/19/2004WO2004069900A2 Bisaminophenyl-based curatives and amidine-based curatives and cure accelerators for perfluoroelastomeric compositions
08/19/2004WO2004048335A3 Mandelic acid derivatives
08/19/2004US20040162281 Pyridine ring containing biaryl compound useful to treat and/or prevent clotting disorders, and as antiinflammatory and anticoagulant agents
08/17/2004US6777577 Anticancer agents; antidiabetic agents, anticholesterol agents, cardiovascular disorders, osteoporosis
08/17/2004US6777555 3-(optionally hydroxyl)-4-(cyclopropylcarbonyl)-cumene intermediate
08/12/2004WO2002076395A3 Agents and methods for treatment of cancer
08/11/2004EP0977552B1 Composition for topical application on the skin and/or its appendages comprising at least a compound containing an iminophenol fragment
08/04/2004CN1518541A Phenyl derivatives
08/03/2004US6770771 Catalyst systems of alpha -diimine, urethane or urea ligands complexed to nickel, palladium or other transition metals
07/2004
07/29/2004US20040147531 Neurodegradation diseases; alzheimer's disease; down's syndrome; antidiabetic agents
07/28/2004EP1440968A1 Process to prepare aryltriazolinones and novel intermediates thereto
07/28/2004EP0976700B1 Process for halogenating hydroxyl group
07/28/2004CN1515550A Thrombosis resisting preparation
07/28/2004CN1159277C New intermediate for preparation of anti-histamine piperdine derivatives
07/21/2004EP1438296A2 1h-imidazole derivatives having cb1 agonistic, cb1 partial agonistic or cb1- antagonistic activity
07/21/2004EP1438292A1 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade
07/21/2004CN1514823A 草酸衍生物 Oxalic acid derivatives
07/20/2004CA2085555C Dual inhibitors of no synthase and cyclooxygenase, process for their preparation and therapeutical compositions containing them
07/15/2004US20040138275 Serine protease inhibitor; cardiovascular disorders
07/14/2004EP1436249A2 Muscarinic agonists
07/14/2004EP1435932A2 Inhibitors of rnase p proteins as antibacterial compounds
07/08/2004US20040133013 Novel polyamine analog-amino acid conjugates useful as anticancer agents
07/08/2004US20040132822 Crystalline solid form of (2S,5Z)-2-amino-7-(ethanimidoylamino)-2-methylhept-5-enoic acid
07/07/2004EP1434769A2 Compounds useful as reversible inhibitors of cysteine proteases
07/06/2004US6759420 Low molecular weight, factor xa specific blood clotting inhibitors without side effects
07/01/2004US20040127658 Productivity catalysts and microstructure control
06/2004
06/30/2004EP1432687A2 Substituted 5-membered polycyclic compounds useful for selective inhibition of the coagulation cascade
06/29/2004US6756406 Antiarthritic agents; rheumatic diseases; osteoarthritis; inhibition of the inducible nitric oxide synthase - induced after activation of vascular smooth muscle, macrophages, endothelial cells by enotoxin and cytokines
06/24/2004US20040122057 Novel mandelic acid derivatives
06/15/2004US6750244 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
06/10/2004WO2004048335A2 Mandelic acid derivatives
06/10/2004US20040110832 management, treatment and/or control of diseases caused in intrinsic clotting pathway utilizing factor IX such as stroke, myocardial infarction, aneurysm surgery, and deep vein thrombosis associated with surgical procedures etc
06/10/2004US20040110801 Prevention of degenerative joint diseases, rheumatoid arthritis, osteoarthritis, ulcerative colitis, irritable colon and Crohn's diseas, antitumor agents; drug mixture for transdermal drug delivery, sustained release; chemical synthesis
06/10/2004CA2505542A1 Mandelic acid derivatives
06/09/2004EP1043310B1 Biphenylamidine derivatives
06/09/2004CN1502604A Process for the preparation of 4(5)-amino-5(4)carboxamidoimidoimidazoles and intermediates thereof
06/08/2004US6747146 Method of producing nitroguanidine- and nitroenamine derivatives
06/03/2004WO2003084937A3 Pyrimidinedione derivatives useful for the treatment of inflammation and immunological diseases
06/03/2004US20040106626 amidine containing compounds which inhibit serine proteases
06/03/2004US20040106560 such as N1-L-Arginylspermidine for protecting from damage from extended ischemic/hypoxic events
06/02/2004EP1423373A2 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
05/2004
05/27/2004US20040102500 Peroxisome proliferator activated receptor alpha agonists
05/26/2004EP1422216A1 Fluorine compound and fluorinating agent comprising the compound
05/26/2004EP1420773A1 Amidine derivatives for treating amyloidosis
05/26/2004EP1206446B1 Carboxylic acid amides, their production and their use as drugs
05/21/2004WO2003084935A3 Diaryl pyrimidinone derivatives useful for the treatment of inflammation and immunogolical diseases
05/19/2004EP1419152A1 Hiv inhibiting pyrimidines derivatives
05/19/2004EP0975682B1 Group 8-10 transition metal olefin polymerization catalysts
05/19/2004CN1150169C Process for preparation of 4(5)-amino-5(4) carboxamidoimidazoles and intermediates thereof
05/19/2004CN1150162C Biphenylamidine derivatives
05/13/2004US20040092517 Phenyl derivatives and their use in the treatment of thromboembolic disorders or tumours
05/13/2004US20040092484 Novel nitric oxide-releasing imidate and thioimidate diazeniumdiolates, compositions, uses thereof and method of making same
05/12/2004CN1495173A Alpha-amino-N-allylamidinonitrobenzene compound and its synthesis
05/06/2004US20040087798 Novel amide compounds
05/06/2004US20040087627 Decarboxylase inhibitors; cardiovascular diosrders; antidiabetic agents; anticancer agents; dietetics
05/06/2004US20040087582 Anticaogulants; cardiovascular disorders; Factor x inhibitors; antiinflammatory agents
05/06/2004EP1415982A1 Halogenated amidino amino acid derivatives useful as nitric oxide synthase inhibitors
05/06/2004EP1414790A1 Substituted n-acyl aniline derivatives, production and use thereof as medicaments
05/06/2004EP1222162B1 Novel ltb4-antagonist, method for the production thereof and its use as a medicament
04/2004
04/29/2004WO2004035529A1 Process for producing n-(2-amino-1,2-dicyanovinyl)formamidine
04/29/2004WO2003093242A3 Substituted 5-membered polycyclic compounds useful for selective inhibition of the coagulation cascade
04/29/2004WO1992004317A3 Novel imidate insecticides
04/29/2004US20040082796 Reacting a substituted benzonitrile with a cysteine compound
04/29/2004US20040082779 Melanocortin-4 receptor binding compounds and methods of use thereof
04/29/2004US20040082585 Anticoagulants; controlling thrombosis; cardiovascular disorders
04/28/2004EP0888271B1 Benzamidine derivatives substituted by amino acid and hydroxy acid derivatives and their use as anti-coagulants
04/22/2004WO2004033397A2 Activity-based probes, and methods of their preparation and use
04/22/2004US20040077868 Process
04/22/2004US20040077865 Making 1-amino-6-nitroisoquinoline by reacting beta-(dimethylamino)-2-cyano-5-nitro-styrene with lithium hexamethyldisilazane or reacting said styrene compound with 2,4-dimethoxybenzylamine and then with anisole
04/22/2004CA2501831A1 Activity-based probes, and methods of their preparation and use
04/20/2004US6723843 Oligosaccharide synthesis
04/15/2004US20040073065 Fluorine compound and fluorinating agent comprising the compound
04/14/2004EP1408026A1 Alpha-amino-N-allylamidino nitrobenzene compound and synthesis
04/14/2004EP0839041B1 Cyclo-oxygenase inhibitor and amidine derivative salts, preparation method therefor, use thereof as drugs, and pharmaceutical compositions containing said salts
04/14/2004CN1489575A Benzamidine derivatives and process for producing same
04/08/2004WO2004005244B1 Method for carrying out the catalyst-free production of o-alkyl-n-cyanoformimidates
04/08/2004WO2003097622A3 Synthesis of 2-alkylcysteines, 2-(hydroxylated phenyl)-4-alkylthiazoline-4-carboxylic acids and derivatives thereof
04/08/2004WO2003070690A3 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative
04/07/2004EP1404648A1 Amidine substituted aryl and heteroaryl derivatives with an antithrombotic and factor xa inhibiting action
04/07/2004CN1487916A Process for the preparation of arylethanoldiamines useful as agonists the beta-3-adrenoceptor
04/06/2004CA2067381C Treatment of hiv infections and compounds useful therein
04/01/2004US20040063679 Amidino and guanidino peptidyl compounds; autoimmune diseases
04/01/2004US20040063671 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
03/2004
03/31/2004EP1015421B1 New phenylamidine derivatives, a process for preparing the same and their use as medicaments
03/30/2004US6713467 Anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and metastasis inhibitors in treating cancer
03/23/2004US6710056 Pharmaceutically acceptable salts thereof have an excellent antagonistic effect against activated blood coagulation factor vii.
03/18/2004WO2003084936A3 Amino substituted pyrimidinone derivatives useful in the treatment of inflammation and immunological
03/18/2004US20040053890 Naphthalene derivatives
03/17/2004EP1140802B1 Substituted aryl and heteroaryl derivatives, their production and their use as medicines
03/16/2004US6706745 Biphenylamidine derivatives
03/11/2004WO2003006444A3 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
03/04/2004WO2004018412A1 Crystalline solid form of (2s-5z)-2-amino-7-(ethanimidoylamino)-2-methylhept-5-enoic acid
03/04/2004WO2004018411A1 Muscarinic agonists
03/03/2004EP1392204A2 Bifunctional energy-reversible acyl-compositions
03/03/2004CN1479728A Pexoxisome proliferator activated receptor alpha agonists
03/02/2004US6699994 Biaryl compounds as serine protease inhibitors
02/2004
02/25/2004EP1391952A2 Salts of pentacyclic or tetrapentaline derived anions, and their uses as ionic conductive materials
02/25/2004EP1390357A2 Anti-thrombotic compounds, production and use thereof as medicaments
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