| Patents for C07C 257 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines (2,984) |
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| 10/24/2006 | US7125879 Prevention reproduction of virus |
| 10/24/2006 | CA2237650C Benzamidoxime prodrugs as antipneumocystic agents |
| 10/17/2006 | US7122676 Reacting oxalimidic acid dihydrazide with sodium nitrite |
| 10/17/2006 | US7122580 management, treatment and/or control of diseases caused in intrinsic clotting pathway utilizing factor IX such as stroke, myocardial infarction, aneurysm surgery, and deep vein thrombosis associated with surgical procedures etc |
| 10/04/2006 | EP1706375A2 Substituted n-aryl amidines as selective d1 dopamine receptor antagonists for the treatment of obesity and cns disorders |
| 10/04/2006 | EP1377290B1 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators |
| 10/03/2006 | US7115769 Catalyzing the alkylation, forming a 2-alkylcysteine derivatives, a chemical intermediates for iron chelating agents |
| 09/28/2006 | US20060217561 Synthesis of substituted thiazoline carboxylic acids |
| 09/20/2006 | CN1275916C Novel intermediates useful for the preparation of antihistaminic piperidine derivatives |
| 09/19/2006 | US7109216 For therapy of psychiatric and neurological disorders |
| 09/14/2006 | US20060205943 Process for preparing xanthine phosphodiesterase V inhibitors and precursers thereof |
| 09/13/2006 | CN1830955A Method for synthesizing O-ethoxy phenyl formamidine acetate |
| 09/12/2006 | US7105559 Substituted 5-membered polycyclic compounds useful for selective inhibition of the coagulation cascade |
| 09/12/2006 | US7105502 Releasing nitric oxide; controlling blood pressure; cytotoxic compound |
| 09/07/2006 | US20060199978 Compounds having serotonin 5-ht17 receptor antagonist activity and muscarinic m4 receptor agonist activity and their use in the treatment of psychotic disorders |
| 09/06/2006 | EP1698629A2 Polyamines and their use in therapy |
| 09/06/2006 | CN1273128C Substituted N-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides |
| 08/31/2006 | WO2006091669A1 Anti-cancer and anti-microbial oxazolidinones and analogues |
| 08/31/2006 | CA2597667A1 Anti-cancer and anti-microbial oxazolidinones and analogues |
| 08/30/2006 | EP1255724B1 Substituted norbornylamino derivatives, method for the production thereof, use thereof as a medicament or a diagnostic reagent and medicaments containing said compounds |
| 08/17/2006 | WO2005107762A3 Certain chemical entities, compositions, and methods |
| 08/17/2006 | CA2596646A1 Inhibitors of transthyretin amyloid fibril formation |
| 08/16/2006 | EP1509525B1 Process for preparing xanthine phosphodiesterase v inhibitors and precursors thereof |
| 08/10/2006 | WO2006084031A1 Imines as ion channel modulators |
| 08/10/2006 | WO2006083003A1 Novel benzamidine compound |
| 08/10/2006 | US20060178438 Muscarinic agonists |
| 08/10/2006 | CA2594505A1 Imines as ion channel modulators |
| 08/09/2006 | EP1177197B1 Polyamines and their use in therapy |
| 08/08/2006 | US7087783 Method for preparing nitrogen-containing compounds |
| 08/08/2006 | US7087765 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases |
| 08/03/2006 | WO2005113011A3 Prodrugs of ion channel modulating compounds and uses thereof |
| 08/03/2006 | US20060173211 Binaphthol derivatives and their use in optical resolution or optical transformation |
| 08/02/2006 | EP1215206B1 Processes for the preparation of 4(5)-amino-5(4)-carboxamidoimidazoles and intermediates thereof |
| 08/01/2006 | US7084250 asymmetric hydrogenation of 2-[2-acetylamino-3-(4-cyanophenyl)acryloylamino]-2-cyclohexylacetic acid and conversion of the cyano group into the amidine, or a salt thereof, with a 3-(2-amino-2-carbamoylethyl)-1-methylpyridinium salt; claimed intermediates |
| 08/01/2006 | CA2234611C New phenylamidine derivatives, processes for preparing them and their use as pharmaceutical compositions |
| 07/27/2006 | WO2006077854A1 Method for producing imide ether compound |
| 07/27/2006 | WO2004033397A3 Activity-based probes, and methods of their preparation and use |
| 07/27/2006 | US20060167267 Michael-type addition of a nucleophile to a dialkyl 2-methylidenylpropan-1,3-dioate and the conversion of a ester moiety into an amino moiety; S)-2-methylcysteine; desferrithiocin |
| 07/13/2006 | WO2006021833A3 Bisbenzamidines for the treatment of pneumonia |
| 07/11/2006 | US7074923 Process for preparing xanthine phosphodiesterase V inhibitors and precursors thereof |
| 07/11/2006 | CA2262566C Benzamidine derivatives and the use thereof as medicaments with ltb4-antagonistic effect |
| 07/06/2006 | WO2006070878A1 Carboxylic acid derivative or salt thereof |
| 07/05/2006 | EP1240149B1 Process to prepare aryltriazolinones |
| 07/04/2006 | US7071212 N-(4-carbamimidoyl-phenyl)-glycine derivatives |
| 06/29/2006 | US20060142594 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases |
| 06/29/2006 | US20060142586 Synthesis of 2-alkyl amino acids |
| 06/29/2006 | DE102004060248A1 New substituted 3-amino-acrylic acid-imino ester compounds useful as ligands in metal catalysts, which are useful as catalysts in polymerization-, copolymerization- and oligomerization-reactions |
| 06/28/2006 | EP1254159B9 Process for the preparation of acetyl-amidiniophenylalanyl-cyclohexylglycyl-pyridylalaninamides |
| 06/22/2006 | WO2006064757A1 Aminocarboxylic acid derivative and medicinal use thereof |
| 06/22/2006 | WO2005094897A3 Pegylated ion channel modulating compounds |
| 06/22/2006 | CA2591399A1 Aminocarboxylic acid derivative and medicinal use thereof |
| 06/21/2006 | EP1671945A1 Process for production of 1-aryl-5-(trifluoromethyl)-1h- tetrazoles |
| 06/15/2006 | US20060128776 Opioid receptor active compounds |
| 06/15/2006 | US20060128633 Colchinol derivatives as vascular damaging agents |
| 06/08/2006 | US20060122280 Muscarinic agonists |
| 06/07/2006 | EP1663960A2 Amidines and derivatives thereof and pharmaceutical compositions containing them |
| 06/07/2006 | EP1663959A1 Novel amidine compounds for treating microbial infections |
| 06/06/2006 | CA2136903C Acetic acid derivatives |
| 05/31/2006 | CN1257889C Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative |
| 05/18/2006 | US20060106204 Bifunctional energy-reversible acyl-compositions |
| 05/16/2006 | US7045533 Such as naphthalen-1-yl-(4-pentyloxy-naphthalen-1-yl)-mehtane for treatment/prevention of diseases/conditions associated with cannobinoid receptor activation such as chronic pain, osteo- and rheumatoid arthritis, teno-synovitis and gout |
| 05/10/2006 | EP1254159B1 Process for the preparation of acetyl-amidiniophenylalanyl-cyclohexylglycyl-pyridylalaninamides |
| 05/04/2006 | US20060094708 to treat cellular proliferative diseases, hyperplasias, solid tumor, cardiac hypertrophy, immune disorders and inflammation; modulators of one or more mitotic kinesins; N-(2-(2-dimethylamino-acetylamino)-1-{4-[8-(1-hydroxy-ethyl)-imidazo[1,2-a]pyridin-2-yl]-benzyl}-ethyl)-3-chloro-4-isopropoxy-benzamide |
| 05/03/2006 | CN1765893A Process for the preparation of arylethanoldiamines useful as agonists of the beta-3-adrenoceptor |
| 05/03/2006 | CN1765886A Process for the preparation of arylethanoldiamines useful as agonists of the beta-3-adrenoceptor |
| 05/02/2006 | US7038073 Synthesis of 2-alkyl amino acids |
| 04/27/2006 | US20060089513 Fluorine compound and fluorinating agent comprising the compound |
| 04/25/2006 | CA2194885C Substituted benzamidines, their preparation and their use as pharmaceutical compounds |
| 04/20/2006 | WO2006041119A1 Hydrazide derivatives |
| 04/18/2006 | CA2360943C N2-phenylamidine derivatives |
| 04/13/2006 | WO2006031556A3 Amidine substituted aryl aniline compounds |
| 04/12/2006 | EP1644337A1 Melanocortin-4 receptor binding compounds and methods of use thereof |
| 04/11/2006 | US7026297 Neuroprotective agents |
| 03/30/2006 | US20060069265 Reacting cysteine (or a salt or an ester) and an aryl carboxylic acid to form a thiazoline ring; stereospecifically alkylating the thiazoline ring, and hydrolyzing the thiazoline ring to obtain a 2-alkylcysteine; chelation |
| 03/29/2006 | CN1247572C Method of producing nitroguanidine-and nitroenamine derivatives |
| 03/28/2006 | US7019173 Fluorine compound and fluorinating agent comprising the compound |
| 03/23/2006 | WO2006031556A2 Amidine substituted aryl aniline compounds |
| 03/22/2006 | EP1637141A1 Stabilized protease composition comprising a serine protease, morpholino derivatives and reversible inhibitors of said serine protease |
| 03/16/2006 | WO2006027135A1 4-aminomethyl benzamidine derivatives and their use as factor viiia inhibitors |
| 03/16/2006 | US20060058389 Novel compounds that inhibit factor xa activity |
| 03/16/2006 | CA2577608A1 4-aminomethyl benzamidine derivatives and their use as factor viia inhibitors |
| 03/15/2006 | CN1245381C Phenylglycine derivatives |
| 03/14/2006 | US7012098 Inhibitors of inducible nitric oxide synthase for chemoprevention and treatment of cancers |
| 03/09/2006 | WO2003103598A3 Amidine derivatives for treating amyloidosis |
| 02/28/2006 | US7005450 2-amino-2-alkyl-4 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors |
| 02/28/2006 | US7005437 Substituted aryl and heteroaryl derivatives, the preparation thereof and the use therof as pharmaceutical compositions |
| 02/21/2006 | US7002036 For production of (poly)peptides; comprises Michael-type addition of nucleophile to a dialkyl 2-methylidenylpropan-1,3-dioate and conversion of ester to amino moiety |
| 02/21/2006 | US7001924 Inhibitors of RNase P proteins as antibacterial compounds |
| 02/21/2006 | CA2186224C Amidino derivatives useful as nitric oxide synthase inhibitors |
| 02/21/2006 | CA2184691C L-n6-(1-iminoethyl)lysine derivatives useful as nitric oxide synthase inhibitors |
| 02/14/2006 | US6998503 crystallized as an anhydrous, stoichiometric 1.5 HCl salt; inhibiting or modulating nitric oxide synthesis |
| 02/14/2006 | CA2248598C Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors |
| 01/31/2006 | US6992221 Production of commercial herbicides: carbonylating an amidrazone of formula (A) with one or more carbonylating agent, or by (ii) condensing a hydrazonoyl derivative of formula (A) with one or more ring-forming agent, wherein |
| 01/26/2006 | WO2006009590A1 Copper (i) compounds useful as deposition precursors of copper thin films |
| 01/25/2006 | CN1238338C Process for the preparation of 4(5)-amino-5(4) carboxamidoimidoimidazoles intermediates |
| 01/03/2006 | US6982335 Synthesis of substituted thiazoline carboxylic acids |
| 12/28/2005 | EP1608617A1 Muscarinic agonists |
| 12/28/2005 | EP1608354A1 Compounds having serotonin 5-ht7 receptor antagonist activity and muscarinic m4 receptor agonist activity and their use in the treatment of psychotic disorders |
| 12/28/2005 | EP1265867B1 Malonic acid derivates, processes for their preparation, their use as inhibitor of factor xa activity and pharmaceutical compositions containing them |
| 12/28/2005 | CN1714079A Mandelic acid derivatives |