Patents
Patents for C07C 257 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines (2,984)
10/2003
10/07/2003US6630510 Substituted succinic acid metallo-β-lactamase inhibitors and their use in treating bacterial infections
10/02/2003US20030187037 Cardiovascular disorders; antiinflammatory agents; antitumor agents
10/01/2003EP0813525B1 Benzamidine derivatives their preparation and their use as anti-coagulants
09/2003
09/25/2003US20030181766 Amidino derivatives, and anticoagulants and thrombosis therapeutic agents containing them
09/25/2003US20030180804 (Serine) protease modulators; membrane proteins
09/24/2003CN1444561A Acetamide derivatives and use thereof as inhibitors of coagulation factors XA and VIIA
09/17/2003CN1121375C Oligosaccharide synthesis
09/12/2003WO2003074476A1 Novel arylamidine derivative or salt thereof
09/11/2003US20030171349 Novel muscarinic receptor agonists
09/10/2003EP1163230B1 Formamidine sulfate and phosphate salts, their production and their use in the synthesis of 1,3,5-triazine
09/09/2003US6617330 For controlling and preventing pests
09/04/2003WO2002070468A3 Novel benzamidine derivatives having anti-inflammatory and immunosuppressive activity
09/04/2003US20030166798 Mixtures of condensation polymers comprising organonitrogen or organosulfur polymers and curing agents, having preferential binding, used for analysis, separation and resolution of racemic mixtures
09/04/2003US20030166685 Acid derivatives of benzene useful as anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and as metastasis inhibitors in treating cancer
09/04/2003US20030166577 Inhibitors for the blood-clotting factor xa
09/03/2003EP1339673A1 Malonamide and malonamic ester derivatives with antithrombotic activity, their preparation and their use
09/03/2003EP1339663A2 Naphthalene derivatives
09/03/2003EP0744435B1 Water-absorbent resin, process for production thereof, and water-absorbent resin composition
09/02/2003US6613351 Vector including a complex between at least one compound having an amidine polar head of formula where m is 14 and at least one of nucleic acids molecules, polypeptides, glycosylated polypeptides and membrane
08/2003
08/28/2003WO2003070690A2 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative
08/28/2003US20030162776 Substituted 5-membered polycyclic compounds useful for selective inhibition of the coagulation cascade
08/28/2003CA2474785A1 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative
08/27/2003EP1337504A2 Novel polyamine analog-amino acid conjugates useful as anticancer agents
08/21/2003US20030158442 Process for the production of nitrogen compounds
08/20/2003EP1336615A2 Metal complexes with iminohyrdoxamic acid as a ligand
08/20/2003EP1335908A2 Peroxisome proliferator activated receptor alpha agonists
08/20/2003EP1150944B1 N2-phenylamidine derivatives
08/20/2003CN1437468A Halogentated 2-amino-5.6-heptenoic aicd derivatives useful as nitric oxide synthase inhibitors
08/14/2003US20030153728 Such as 1-methoxy-2-(3-methylphenyl)ethanimine by treating nitrile with anhydrous hydrogen chloride solution and anhydrous alcohol
08/12/2003US6605677 Olefin polymerization processes using supported catalysts
08/12/2003US6605626 Antithrombotic agents
08/07/2003WO2003064378A2 Novel compounds that inhibit factor xa activity
08/07/2003US20030149053 Reacting acid salt of aminoacetamidine with a source-of cyanide and reacting with 2,3,5- trichlorobenzaldehyde to produce 2-((Cyano-(2,3,5-trichlorophenyl)-methyl)-amino)-acetamidine or a salt thereof
08/07/2003CA2473164A1 Novel compounds that inhibit factor xa activity
08/06/2003EP1332131A2 Acid derivatives useful as serine protease inhibitors
08/06/2003EP1332129A2 Acid derivatives useful as serine protease inhibitors
08/06/2003EP0711762B1 Process for producing tetrazole compounds
07/2003
07/31/2003WO2003027061A3 Muscarinic agonists
07/31/2003US20030144528 Production of commercial herbicides: carbonylating an amidrazone of formula (A) with one or more carbonylating agent, or by (ii) condensing a hydrazonoyl derivative of formula (A) with one or more ring-forming agent, wherein
07/29/2003US6600049 Carbonylating an amidrazone compound with at least one carbonylating agent for preparing 1-aryltriazolinones compound
07/29/2003CA2188690C Selective thrombin inhibitors
07/24/2003WO2003059064A1 Insecticides containing hydrazone derivatives as the active ingredient and novel hydrazone derivatives
07/24/2003US20030139405 6-Membered heterocyclic compounds useful for selective inhibition of the coagulation cascade
07/23/2003CN1115330C N-(4-carbamimido-phenyl)-phenylglycinamid derivatives
07/22/2003US6596863 Matrix metalloproteinase inhibitor is useful as an anticancer agent, angiogenesis inhibitor, a tumor cell infiltration inhibitor or a tumor metastasis inhibitor; inflammatory diseases, osteoarthritis, rheumatoid arthritis
07/17/2003US20030135045 Glycoprotein IIb/IIIa antagonists
07/17/2003US20030134904 Inhibitors of RNase P proteins as antibacterial compounds
07/16/2003CN1430599A Phenylglycine derivatives
07/10/2003US20030130354 Such as 3,5-dimethyl-1-adamantanecarboximidamide hydrochloride; glutamate receptors; methyl-D-aspartate receptors; neurodegenerative diseases; side effect reduction
07/10/2003US20030130342 Such as anticoagulant 3-(6-(4-(aminoiminomethyl)phenyl methoxy)-2-methyl-2H-1-benzopyran-2-yl)propanoic acid hydrochloride
07/10/2003US20030130232 Amidine derivatives, the preparation and use thereof as medicaments with LTB4 antagonistic effect
07/09/2003EP1040096B1 Neuroprotective agents
07/09/2003EP0966490B1 Catalyst compositions for the polymerization of olefins
07/01/2003US6586471 Halogenated 2-amino-3, 4 heptenoic acid derivatives useful as nitric oxide synthase inhibitors
06/2003
06/26/2003US20030119871 Amidine derivatives as selective antagonists of ndma receptors
06/25/2003EP0906094B1 Substituted n- (aminoiminomethyl or aminomethyl)phenyl]propyl amides
06/25/2003CN1112353C Amino benzene amidine derivative and its use
06/24/2003US6583177 Leukotriene B4 antagonist compounds and method for treatment
06/18/2003EP1319642A2 Method of Preparing a Halogenated Compound
06/17/2003US6579823 Group 8-10 metal complex comprising a bidentate or variable denticity ligand; polymerization of olefins
06/12/2003US20030109547 Amidinophenylpyruvic acid derivatives
06/11/2003EP1317490A1 Catalysts containing per-ortho aryl substituted aryl or heteroaryl substituted nitrogen donors
06/11/2003EP1317456A2 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
06/11/2003EP1317421A1 2-amino-2-alkyl-5 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors
06/11/2003EP1317420A1 2-amino-2-alkyl-3 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors
06/11/2003EP1317418A2 2-amino-2-alkyl-4 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors
06/11/2003EP1317417A2 2-amino-2-alkyl-3 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors
06/11/2003EP1317416A2 2-amino-2-alkyl-4 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors
06/10/2003US6576780 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors
06/10/2003US6576596 Substituted 2-benzoyl-cyclohexan-1,3-diones with herbicidal effect
06/10/2003US6576159 Colorants, electroconductive materials; solubility, dissociation
06/04/2003CN1110305C Naphthyl-substituted benzimidazole derivatives as anticoagulants
06/03/2003US6573337 Dioxocyclohexane compound linker for solid-phase synthesis of oligosaccharides
06/03/2003CA2115432C Substituted .beta.-amino acid derivatives useful as platelet aggregation inhibitors
05/2003
05/28/2003CN1420874A Process for preparing aryltriazolinones and novel intermediates thereto
05/21/2003EP1312602A1 Amidino derivatives, and anticoagulants and thrombosis therapeutic agents containing them
05/21/2003EP1311492A1 Method for producing lamotrigine from alpha-oxo-2,3-dichlorophenyl acetamidino-aminoguanidino hydrazone by ring closure reaction
05/20/2003US6566526 Intermediates useful for the preparation of antihistaminic piperidine derivatives
05/20/2003US6566330 Positively charged non-natural amino acids, methods of making and using thereof in peptides
05/20/2003CA2099994C Phenyl amidines derivatives useful as platelet aggregation inhibitors
05/15/2003US20030092915 Using phase transfer catalyst and quaternary ammonium compound
05/14/2003EP1309549A1 Acetamide derivatives and the use thereof as inhibitors of coagulation factors xa and viia
05/08/2003WO2003037326A1 Solid phase synthesis of chemical libraries
05/08/2003US20030087832 Anticancer agents; antidiabetic agents, anticholesterol agents, cardiovascular disorders, osteoporosis
05/07/2003EP1042268B1 1,7-dibromodibenzosuberone and procedures for its preparation
05/07/2003EP0889863B1 Surface modified carbonate materials
05/07/2003EP0749417B1 Cyano compounds and preparations thereof
05/06/2003US6559312 Intermediates useful for the preparation of antihistaminic piperidine derivatives
05/02/2003EP1306366A2 New dibenzosuberone derivatives
05/01/2003WO2002038553A3 Triazole derivatives and their use as peroxisome proliferator activated receptor alpha agonists
05/01/2003US20030083504 N- (4-carbamimidoyl-phenyl) -glycine derivatives
04/2003
04/29/2003US6555711 Reacting an N-allylimino nitrobenzene compound with a diamino-dinucleophile to form an alpha-amino-N- allylamidino-nitrobenzene compound; chemical intermediate for a pyrazolo(1,5-b)(1,2,4)triazole color photographic coupler
04/29/2003US6555689 Intermediates useful for the preparation of antihistaminic piperidine derivatives
04/24/2003WO2002058690A3 Methods for the treatment of diseases using malonyl-coa decarbox ylase inhibitors
04/24/2003WO2002022553A3 Non-natural basic amino acids, their preparation and use
04/24/2003US20030078418 Useful potentiators of beta -lactam antibiotics; therapy
04/22/2003US6552200 Intermediates useful for the preparation of antihistaminic piperidine derivatives
04/16/2003EP0998451B1 Substituted 3,3-diamino-2-propenenitriles, their preparation and use
04/16/2003CN1105703C Alpha-substituted phenylacetic acid derivative, process for producing same, and agricultural bactericide containing same
04/15/2003US6548694 N-(4-carbamimidoyl-phenyl)-glycine derivatives
1 ... 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 ... 30