Patents
Patents for C07C 257 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines (2,984)
09/1999
09/08/1999CN1228089A Pesticidal 3-(substituted phenyl)-5-(thienyl or furyl)-1,2,4-triazoles
09/07/1999US5948819 α-substituted phenylacetic acid derivative, its production and agricultural fungicide containing it
09/01/1999EP0939075A1 A novel azoamidine compound
08/1999
08/31/1999US5945455 Amine and amidine containing compounds as weight reducing agents
08/31/1999US5945408 Hydroxyanidino derivatives useful as nitric oxide synthase inhibitors
08/26/1999CA2263391A1 Azoamidine compound and its use as polymerization initiator
08/24/1999US5942614 Process to produce midazolam
08/24/1999US5942547 2-Deoxystreptamine derivatives, pharmaceutical compositions thereof and therapeutic methods using same
08/24/1999US5942544 Anticoagulants and treatment of thromboembolic disoeders
08/19/1999WO1999041231A1 Amidino derivatives and drugs containing the same as the active ingredient
08/19/1999WO1999041214A1 Halogenating agent and process for halogenating hydroxyl group
08/18/1999CN1226230A Pesticidal composition
08/17/1999US5939392 Thrombin inhibitors, anticoagulants and antiinflammatory agents
08/11/1999EP0934259A1 Beta-sulfonamido hydroxamic acids as matrix metalloproteinase and tace inhibitors
08/11/1999CN1044600C N-arylhydrazine derivatives as insecticidal and acaricidal agents
08/05/1999WO1999038841A1 Adamantanecarboximidamide derivatives and their use as nmda antagonists
08/04/1999CN1224714A N-(4-carbamimido-phenyl)-phenylglycinamid derivatives
07/1999
07/29/1999WO1999030695A8 Substituted amidino compounds in the treatment of chronic obstructive pulmonary disease
07/28/1999EP0931069A1 Process for preparing amidines
07/28/1999EP0931060A1 Substituted n- (aminoiminomethyl or aminomethyl)phenyl]propyl amides
07/27/1999US5929120 Guainidino, formamidino, amino and related compounds for inhibiting osteoclast-mediated bone resorption
07/21/1999EP0929516A1 Benzamidine derivatives and the use thereof as medicaments with ltb4-antagonistic effect
07/13/1999US5922892 Process to produce midazolam
07/13/1999US5922763 Biphenyl derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
07/07/1999EP0927035A1 Thrombin inhibitors
07/06/1999US5919787 Aminotetrazole derivatives useful as nitric oxide synthase inhibitors
07/01/1999WO1999032105A1 Esters of conjugated linoleic acid or conjugated linolenic acid and uses thereof
06/1999
06/24/1999WO1999031092A1 Benzamine derivatives
06/24/1999WO1999031051A1 1-(adamantyl)amidines and their use in the treatment of conditions generally associated with abnormalities in glutamatergic transmission
06/24/1999WO1999031049A1 Neuroprotective agents
06/24/1999WO1999030695A1 Substituted amidino compounds in the treatment of chronic obstructive pulmonary disease
06/24/1999CA2314395A1 Use of substituted amidino compounds in the treatment of chronic obstructive pulmonary disease
06/24/1999CA2313651A1 Benzamine derivatives
06/23/1999EP0923528A1 Oligosaccharide synthesis
06/17/1999WO1999029670A2 Aminocarbonyltetralin and dihydronaphtalene derivates as thrombin inhibitors
06/17/1999DE19755268A1 Benzamidinderivate Benzamidine derivatives
06/16/1999EP0922043A1 Pesticidal 3-(substituted phenyl)-5-(thienyl or furyl)-1,2,4-triazoles
06/10/1999WO1999028284A1 Dibenzosuberone derivatives and procedures for their preparation
06/10/1999DE19754490A1 Durch einen Aminocarbonylrest substituierte Bicyclen, ihre Herstellung und ihre Verwendung als Arzneimittel By an aminocarbonyl radical substituted bicyclic compounds, their preparation and their use as medicaments
06/09/1999EP0921116A1 N-(4-carbamimido-phenyl)-glycine amide derivatives
06/08/1999US5910602 Method for preparing 3-amino substituted crotonates
06/04/1999CA2255180A1 N-(4-carbamimido-phenyl)-phenylglycinamid derivatives
06/03/1999WO1999026919A1 Biphenylamidine derivatives
06/03/1999WO1999026918A1 Biphenylamidine derivatives
06/03/1999WO1999005096A3 Urokinase inhibitors
06/03/1999CA2310331A1 Biphenylamidine derivatives
06/03/1999CA2310330A1 Biphenylamidine derivatives
06/02/1999EP0918773A1 Process for the production of 8-chloro-6-(2-fluorophenyl)-1-methyl-4h-imidazo 1,5-a]benzodiazepine
06/02/1999EP0625138B1 Novel amidine derivatives, their preparation and their use as medicaments with ltb4 antagonistic effect
05/1999
05/25/1999CA2124522C A method of preparing ortho esters
05/20/1999WO1999024407A1 Compounds which inhibit tryptase activity
05/20/1999WO1999024395A1 Compounds which inhibit tryptase activity
05/14/1999WO1999022707A1 Composition for topical application on the skin and/or its appendages comprising at least a compound containing an iminophenol fragment
05/06/1999EP0912504A1 Process to prepare taxol
05/06/1999EP0912494A1 Coumpounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
05/05/1999CN1216039A Process to prepare taxol
04/1999
04/07/1999EP0906094A1 Substituted n- (aminoiminomethyl or aminomethyl)phenyl]propyl amides
04/07/1999EP0770059B1 Substituted benzamidines, their production and their use as medicaments
04/06/1999US5892061 Reacting a mono- or polycarboxylic acid with a mono- or polyamide in the presence of a haloiminium salt and base; catalyst selectivity
03/1999
03/30/1999US5889056 Of nitric oxide synthase; hypotensive agent, antiinflammatory agents, antiarthritic agents
03/30/1999US5889005 Benzamidine derivatives and their use for treating thrombotic diseases
03/24/1999EP0673432B1 Process for preparing clavulanic acid
03/23/1999US5886208 Substituted B-amino acid derivatives useful as platelet aggregation inhibitors
03/23/1999US5885990 Fibrinolysis promoting action; thrombolysis action
03/17/1999EP0902090A1 Compound capable of introducing at least one molecule into a cell.
03/17/1999EP0902013A1 Novel amidine derivatives, their preparation and their use as medicaments with LTB-4 antagonistic effect
03/17/1999EP0902000A1 A method of preparing 1, 1-Dialkoxycycloalkanes
03/17/1999CN1211232A Benzamidine derivatives substituted by amino acid and hydroxy acid derivatives and their use as anti-coagulants
03/16/1999US5883100 Benzamidine derivatives and their use as anti-coagulants
03/04/1999WO1999010316A1 3-amidinoaniline derivatives, activated blood coagulation factor x inhibitors, and intermediates for producing both
03/04/1999CA2301559A1 3-amidinoaniline derivatives, activated blood coagulation factor x inhibitors, and intermediates for producing both
03/02/1999US5877190 Substituted biphenyl compounds
03/02/1999US5877181 Benzamidine derivatives and their use as anti-coagulants
02/1999
02/25/1999WO1998045259A3 Polyaromatic antiviral compositions
02/24/1999CN1209062A Naphthyl-substituted benzimidazole derivatives as anticoagulants
02/23/1999US5874593 Production process and intermediate of tetrazole compound
02/23/1999US5874472 Aminoacid derivatives as no synthase inhibitors
02/17/1999CN1208347A Substituted N-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides
02/16/1999US5872138 Thrombin inhibitors
02/11/1999WO1998040420A3 Catalyst compositions for the polymerization of olefins
02/09/1999US5869299 Using an enzyme system from streptomyces, particularly s. clavuligerus.
02/09/1999US5869067 Bi-aromatic compounds and pharmaceutical and cosmetic compositions
02/04/1999WO1999005096A2 Urokinase inhibitors
02/04/1999WO1999004778A1 Pharmaceutical compounds
02/04/1999CA2297906A1 Pharmaceutical compounds
02/04/1999CA2294300A1 Urokinase inhibitors
02/02/1999US5866612 Acetamidine derivatives and their use as inhibitors for the nitric oxide synthase
02/02/1999US5866577 Aromatic amidine derivatives and salts thereof
01/1999
01/27/1999EP0893437A1 Tryptase inhibitor and novel guanidino derivatives
01/27/1999EP0892780A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS
01/26/1999US5863931 Amidino derivatives and their use as nitric oxide synthase inhibitors
01/20/1999EP0891325A1 Para-substituted phenylpropanoic acid derivatives as integrin antagonists
01/20/1999CN1205687A Tyrosin-derivate as alpha-V-integrin inhibitors
01/13/1999EP0890176A1 Proton conductor in liquid form
01/13/1999EP0889877A1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS
01/13/1999EP0889863A2 Surface modified carbonate materials
01/07/1999WO1999000356A1 Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides
01/07/1999WO1999000127A1 Antithrombotic agents
01/07/1999WO1999000121A1 Antithrombotic agents
01/07/1999EP0888271A1 Benzamidine derivatives substituted by amino acid and hydroxy acid derivatives and their use as anti-coagulants
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