| Patents for C07C 257 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines (2,984) |
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| 04/15/2003 | US6548675 1-Cyclopropylcarbonyl-2-hydroxy(optional),4-isopropylbenzene used as starting materials for 1-((2-hydroxy(optional),4-alkylphenyl)carbonylalkyl-),4-(diphenylmethyl -)piperidine derivatives; antihistamines; antiallergens; bronchodilators |
| 04/10/2003 | WO2003029224A1 6-membered unsaturated heterocyclic compounds useful for selective inhibition of the coagulation cascade |
| 04/10/2003 | WO2003029216A1 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade |
| 04/10/2003 | WO2003029200A2 Compounds useful as reversible inhibitors of cysteine proteases |
| 04/10/2003 | WO2003028729A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade |
| 04/10/2003 | US20030069250 Anticoagulants |
| 04/10/2003 | US20030066988 Electroconductivity coloring |
| 04/10/2003 | CA2462647A1 6-membered unsaturated heterocyclic compounds useful for selective inhibition of the coagulation cascade |
| 04/10/2003 | CA2462601A1 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade |
| 04/10/2003 | CA2462305A1 6-membered heterocyclic compounds useful for selective inhibition of the coagulation cascade |
| 04/10/2003 | CA2459825A1 Compounds useful as reversible inhibitors of cysteine proteases |
| 04/09/2003 | CN1105101C Beta-sultonamido hydroxamic acids as matrix metalloproteinase and TACE inhibitors |
| 04/08/2003 | US6545170 For therapy of rheumatoid arthritis and in osteoarthritis, inflammatory bowel disease, cardivascular ischemia, diabetes, congestive heart failure, myocarditis, atherosclerosis, migraine, glaucoma, aortic aneurysm, reflux esophagitis |
| 04/08/2003 | US6545108 Catalysts containing N-pyrrolyl substituted nitrogen donors |
| 04/08/2003 | US6545054 Alkenyl and alkynyl compounds as inhibitors of factor Xa |
| 04/03/2003 | WO2003027076A2 1h-imidazole derivatives having cb1 agonistic, cb1 partial agonistic or cb1- antagonistic activity |
| 04/03/2003 | WO2003027061A2 Muscarinic agonists |
| 04/03/2003 | US20030065176 Anticoagulant; cardiovascular disorders |
| 04/02/2003 | EP1296940A1 Amidine derivatives as selective antagonists of nmda receptors |
| 04/02/2003 | CN1104412C Benzamidine derivatives and use thereof as medicaments with LTB4-antagonistic effect |
| 03/27/2003 | WO2003024407A2 Inhibitors of rnase p proteins as antibacterial compounds |
| 03/27/2003 | US20030060653 N-unsubstituted amidinium salts |
| 03/26/2003 | EP1294741A2 Dipeptide inhibitors for the blood-clotting factor xa |
| 03/26/2003 | EP0885186B1 Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them |
| 03/26/2003 | CN1406226A Novel malonic acid derivatives, process for their preparation, their use as inhibitor of factor XA activity and pharmaceutical compositions containing them |
| 03/20/2003 | US20030052310 Perfluorinated amide salts and their uses as ionic conducting materials |
| 03/19/2003 | CN1103333C Selective thrombin inhibitors |
| 03/13/2003 | WO2003020685A1 Fluorine compound and fluorinating agent comprising the compound |
| 03/12/2003 | EP1289939A1 Phenylglycine derivatives |
| 03/12/2003 | EP0670835B1 Process for preparing benzopyran compounds |
| 03/06/2003 | WO2003017994A1 Amidine derivatives for treating amyloidosis |
| 03/06/2003 | US20030045712 Substituted aryl and heteroaryl derivatives, the preparation thereof and the use therof as pharmaceutical compositions |
| 03/06/2003 | CA2455497A1 Amidine derivatives for treating amyloidosis |
| 03/05/2003 | EP1288197A2 N-Unsubstituted amidinium salts |
| 03/05/2003 | EP1286982A2 Process for the preparation of benzoyl substituted bicylic compounds and chiral bnezopyran derivatives |
| 02/27/2003 | WO2003016306A1 Hiv inhibiting pyrimidines derivatives |
| 02/27/2003 | WO2002038105A3 Novel polyamine analog-amino acid conjugates useful as anticancer agents |
| 02/27/2003 | US20030040521 For controlling and preventing pests |
| 02/26/2003 | EP1285909A1 Process for the production of nitrogen compounds |
| 02/20/2003 | US20030036657 Carbonylating an amidrazone compound with at least one carbonylating agent for preparing 1-aryltriazolinones compound |
| 02/19/2003 | CN1398247A Colchinol derivatives as vascular damaging agents |
| 02/13/2003 | WO2003011210A2 Arylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase |
| 02/12/2003 | EP1282420A2 Halogenated 2-amino-3, 4 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| 02/12/2003 | EP1282413A1 Halogenated 2-amino-5,6 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| 02/12/2003 | CN1396928A Process for preparation of acetyl-amidiniophenylalanyl-cyclohexylglycyl-pyridinioalaninamides |
| 02/06/2003 | WO2002066418A3 Process for the preparation of arylethanoldiamines useful as agonists of the beta-3-adrenoceptor |
| 02/06/2003 | US20030027925 Use of a 2-substituted-1,3-dioxocycloalkyl linker group to couple saccharide groups of both the O-glycoside and N-glycoside type to a polymer support in a solid phase systhesis process |
| 02/06/2003 | US20030027828 Malonamid and malonamic ester derivatives with antithrombotic activity, their preparation, and their use |
| 02/06/2003 | US20030026521 Optical interleaver |
| 02/05/2003 | CN1395467A Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents |
| 02/05/2003 | CN1394846A Alpha-substituted benzene acetic acid its preparation and farm pesticide containing said compound |
| 02/04/2003 | US6514486 Inhibits tyrosinase or the synthesis of melanin; N'-(4-hydroxyphenyl)-N,N-dimethylformamidine |
| 01/30/2003 | WO2003008393A1 Method for producing lamotrigine from alpha-oxo-2,3-dichlorophenyl acetamidino-aminoguanidino hydrazone by ring closure reaction |
| 01/29/2003 | EP1279662A1 Process for preparing phenylcyclohexan-1-ylcarboxylic acids |
| 01/29/2003 | EP1278784A2 Catalysts containing n-pyrrolyl substituted nitrogen donors |
| 01/29/2003 | EP1278721A1 Process for the preparation of pyrazine compounds |
| 01/29/2003 | EP0973735B1 Polyaromatic antiviral compositions |
| 01/29/2003 | CN1100036C Prourokinase and urokinase affinity ligand and its usage |
| 01/27/2003 | WO2002010127A1 Acetamide derivatives and the use thereof as inhibitors of coagulation factors xa and viia |
| 01/27/2003 | CA2417427A1 Acetamide derivatives and the use thereof as inhibitors of coagulation factors xa and viia |
| 01/23/2003 | WO2003006444A2 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity |
| 01/23/2003 | WO2002022559A3 2-amino-2-alkyl-4 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors |
| 01/23/2003 | CA2453169A1 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity |
| 01/22/2003 | CN1099425C 新的肽衍生物 New peptide derivatives |
| 01/16/2003 | US20030013702 Agents and methods for treatment of cancer |
| 01/15/2003 | EP1274676A2 Polycyclic aryl and heteroaryl substituted 1,4-quinones useful for selective inhibition of the coagulation cascade |
| 01/15/2003 | EP0713483B1 Amidine derivatives with nitric oxide synthetase activities |
| 01/14/2003 | US6506517 Surface modified carbonaceous materials |
| 01/08/2003 | EP1272455A1 Halogenated 2-amino-4, 5 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| 01/07/2003 | US6504031 Enzyme inhibitor such as 6-(2-(1-isopropyl-1,2,3,4-tetrahydro -7-isoquinolinyl)ethenyl)-2-naphthalenecarboximidamide, used as angiogenesis inhibitors; antiarthritic, antiinflammatory and antitumor agents |
| 01/03/2003 | WO2003000653A1 Substituted n-acyl aniline derivatives, production and use thereof as medicaments |
| 01/03/2003 | CA2451625A1 Substituted n-acyl-aniline derivatives, the preparation thereof and the use thereof as pharmaceutical compositions |
| 01/02/2003 | EP1268413A2 Substituted biphenyl derivatives |
| 01/02/2003 | EP0804431B9 GLYCOPROTEIN IIb/IIIa ANTAGONISTS |
| 01/02/2003 | EP0705245B1 Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives |
| 01/01/2003 | CN1388118A Substituted phenyl alkyl nitrogen monoxide synthase inhibitor and its prepn and use |
| 12/31/2002 | US6500866 1-(adamantyl)amidines and their use in the treatment of conditions generally associated with abnormalities in glutamatergic transmission |
| 12/26/2002 | US20020198407 Antiallergy agents and bronchodilators |
| 12/26/2002 | US20020198184 Matrix metalloproteinase inhibitor is useful as an anticancer agent, angiogenesis inhibitor, a tumor cell infiltration inhibitor or a tumor metastasis inhibitor; inflammatory diseases, osteoarthritis, rheumatoid arthritis |
| 12/25/2002 | CN1097052C Process for production of amidinoindole derivs, and salts thereof |
| 12/19/2002 | WO2002042248A3 Naphthalene derivatives |
| 12/18/2002 | EP1265867A1 Novel malonic acid derivates, processes for their preparation, their use as inhibitor of factor xa activity and pharmaceutical compositions containing them |
| 12/18/2002 | EP0736002B9 Compound capable of introducing at least one molecule into a cell |
| 12/12/2002 | US20020187993 Bifunctional energy-reversible acyl-compositions |
| 12/11/2002 | EP1264820A1 Novel amide compounds |
| 12/10/2002 | US6492527 Process to prepare aryltriazolinones and novel intermediates thereto |
| 12/09/2002 | WO2001096366A2 Dipeptide inhibitors for the blood-clotting factor xa |
| 12/09/2002 | CA2412181A1 Dipeptide inhibitors for the blood-clotting factor xa |
| 12/03/2002 | US6489365 Ltb4-antagonistic compounds for treatment of inflammation, allergy or gastropathy induced by non-steroidal antiinflammatory agents in a warm-blooded animals |
| 11/28/2002 | DE10124867A1 New substituted (hetero)aryl-alkenes or -alkynes, used as thrombin inhibitors, serine protease inhibitors, antithrombotic agents and intermediates |
| 11/27/2002 | EP1260504A1 Process for the preparation of antihistaminic 4-diphenylmethyl piperidine derivatives |
| 11/22/2002 | WO2003101942A1 Amidine substituted aryl and heteroaryl derivatives with an antithrombotic and factor xa inhibiting action |
| 11/22/2002 | CA2445571A1 Substituted aryl and heteroaryl derivatives, the preparation thereof and the use thereof as pharmaceutical compositions |
| 11/21/2002 | WO2002091989A2 Antiviral therapies using polyamine or polyamine analog-amino acid conjugates |
| 11/20/2002 | EP0892780B1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS |
| 11/13/2002 | EP1255724A1 Substituted norbornylamino derivatives, method for the production thereof, use thereof as a medicament or a diagnostic reagent and medicaments containing said compounds |
| 11/13/2002 | EP0760658B1 Compounds for inhibiting osteoclast-mediated bone resorption |
| 11/13/2002 | CN1379756A Substituted nor bornylamino derivatives, method for production thereof, use thereof as medicament or diagnostic reagent medicaments containing said compounds |
| 11/12/2002 | US6479663 Intermediates useful for the preparation of antihistaminic piperidine derivatives |
| 11/12/2002 | US6479524 To prolong the thrombin time |