Patents
Patents for C07C 257 - Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines (2,984)
04/2005
04/14/2005WO2005033065A1 Novel amidine compounds for treating microbial infections
04/14/2005CA2537791A1 Novel amidine compounds for treating microbial infections
04/12/2005US6878828 Coupling cysteine with benzonitrile, then esterifying, alkylating, hydrolyzing and reacting with acids to form 2-methylcysteine
04/12/2005CA2081836C Aromatic amidine derivatives and salts thereof
04/07/2005US20050075513 Method for preparing nitrogen-containing compounds
04/07/2005US20050074668 Perfluorinated amide salts and their uses as ionic conducting materials
04/06/2005CN1603291A Novel intermediates useful for the preparation of antihistaminic piperidine derivatives
04/06/2005CN1195783C Polymerization of olefins
04/05/2005US6875883 Forming a phenyl-thiazoles chemical intermediates for making antioxidants, ferrielectric liquid crystal dopant, picornaviral viricides, antiinflammatory agents, anti-asthma agents, and fibringoen antagonists
04/05/2005US6875882 Ferroelectric liquid crystals, antihistamines, antiinflammatory agents, viricides
03/2005
03/31/2005WO2005028425A2 Amidines and derivatives thereof and pharmaceutical compositions containing them
03/31/2005CA2539842A1 Amidines and derivatives thereof and pharmaceutical compositions containing them
03/24/2005US20050065346 anticoagulants; thrombosis; factor x inhibitor
03/22/2005US6870021 Mixtures of condensation polymers comprising organonitrogen or organosulfur polymers and curing agents, having preferential binding, used for analysis, separation and resolution of racemic mixtures
03/16/2005EP1115758B1 Polymerization of olefins
03/16/2005EP0874625B1 Indane derivatives for antipsychotic compositions
03/10/2005US20050054679 For therapy of psychiatric and neurological disorders
03/09/2005EP1512679A1 Novel adamantane derivatives with neuroprotective, antidepressant and anti-ischaemic activities, and process for preparing them
03/03/2005US20050049421 amidation; reacting an amine and an ester in the presence of a silylating agent as catalyst under mild conditions
03/03/2005US20050049312 N-(1-adamantyl)alkyl]alkano-amidines, guanidines or N'-nitroguanidines; non-competitive receptor antagonists for the NMDA receptor
03/02/2005EP1509525A1 Process for preparing xanthine phosphodiesterase v inhibitors and precursors thereof
03/02/2005CA2479613A1 Novel adamantane derivatives with neuroprotective, antidepressant and anti-ischaemic activities, and process for preparing them
03/01/2005US6861532 Synthesis of 2-alkylcysteine
02/2005
02/24/2005US20050043569 preparing an amidine by reacting a NH group-containing compound with a nitrile in the presence of a silylating agent (trimethylsilyl trifluoromethanesulfonate); direct and efficient synthesis ; large-scale synthesis.
02/24/2005US20050043403 Reacting carboxamide compound with sulphuric diester to form imidic ester alkyl sulfate; then reacting with ammonia to form amidinium alkyl sulfate
02/24/2005US20050042372 Class of volatile compounds for the deposition of thin films of metals and metal compounds
02/23/2005EP1317421B1 2-amino-2-alkyl-5 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors
02/23/2005EP0876337B1 New lh-rh antagonists with improved effectiveness
02/23/2005CN1190416C Substituted phenyl alkyl nitrogen monoxide synthase inhibitor and its prepn. and use
02/22/2005US6858396 Amino acids where primary amine group is replaced by azide; use in peptides screening for bioactivity, crossing blood-brain barrier, increasing selectivity; treating brain disorders
02/16/2005EP1506162A2 Synthesis of benzonitriles and benzimidates
02/16/2005EP1294741B1 Dipeptide inhibitors for the blood-clotting factor xa
02/08/2005US6852761 Inhibitors of serine proteases of the coagulation cascade and compounds, compositions and methods for anticoagulant therapy for the treatment and prevention of a variety of thrombotic conditions including coronary artery and cerebrovascular
02/02/2005EP1501789A1 Amidinylphenyl compounds and their use as fungicides
02/02/2005CN1187056C Cyclo-oxygenase inhibitor and amidine derivative salts, preparation method thereof, use thereof as drugs, and pharmaceutical compositions containing said salts
01/2005
01/25/2005US6846958 Synthesis of benzimidate from benzoic acid
01/18/2005US6844446 Catalysts containing per-ortho aryl substituted aryl or heteroaryl substituted nitrogen donors
01/18/2005US6844404 Catalyst compositions for the polymerization of olefins
01/11/2005US6841701 Inhibitors for the blood-clotting factor Xa
01/11/2005US6841696 N-unsubstituted amidinium salts
01/05/2005EP1492774A2 Pyrimidone derivatives useful for the treatment of inflammation and immunological diseases
12/2004
12/28/2004US6835495 Pentacyclic anion salts or tetrazapentalene derivatives and their uses as ionic conducting materials
12/23/2004US20040259891 Novel pyrimidon derivatives
12/22/2004CN1556788A Muscarinic agonists
12/22/2004CN1556703A 1H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1 antagonistic activity
12/21/2004CA2241904C Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides
12/16/2004WO2004069900A3 Bisaminophenyl-based curatives and amidine-based curatives and cure accelerators for perfluoroelastomeric compositions
12/15/2004CN1555356A Bisphenol derivative as NHE-3 inhibitor
12/09/2004US20040248897 Substituted N-acylaniline derivatives, the preparation thereof, and their use as pharmaceutical compositions
12/08/2004EP1482940A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
12/08/2004CN1178905C Novel peptide derivative
12/07/2004US6828456 2-amino-2-alkyl-3 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors
12/07/2004US6828454 Metal complexes of iminohydroxamic acids
12/02/2004US20040242584 Muscarinic agonists
12/01/2004EP1481966A1 Novel arylamidine derivative or salt thereof
11/2004
11/30/2004US6825231 Substituted norbornylamino derivatives, processes for their preparation, their use as medicaments or diagnostics, and a medicament comprising them
11/25/2004US20040235962 Conformationally restricted polyamine analogs as disease therapies
11/25/2004US20040235854 1H-imidazole derivatives having cb1 agonistic, cb1 partial agonistic or cb1 antagonistic activity
11/24/2004CN1176918C Intermediate of alpha-substituted benzene acetic acid derivate with farm pesticide activity
11/23/2004US6822062 Supported group 8-10 transition metal olefin polymerization catalysts
11/17/2004EP1476421A2 Novel amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative
11/17/2004CN1176104C Process for preparation of acetyl-guanylphenylalanyl-cyclohexylglycyl-pyridinioalaninamides
11/11/2004US20040225109 Process for the preparation of acetyl-amidiniophenylalanyl-cyclohexylglycyl-pyridinioalaninamides
11/10/2004CN1174962C Amidine compound and its preparing process
11/04/2004WO2004094363A1 Muscarinic agonists
11/04/2004US20040220411 Oxalic acid derivatives
11/04/2004US20040220241 Substituted biphenyl derivatives
11/04/2004CA2518700A1 Muscarinic agonists
11/02/2004US6812231 Inhibiting activated blood-coagulation factor x
10/2004
10/28/2004US20040214956 Synthesis with amidines and curing promoters with high molecular weight
10/27/2004EP1470752A1 Insecticides containing hydrazone derivatives as the active ingredient and novel hydrazone derivatives
10/27/2004EP1470104A2 Novel compounds that inhibit factor xa activity
10/27/2004CN1541215A HIV inhibiting pyrimidines derivatives
10/20/2004CN1171861C Halogenated amidino amino acid dervatives useful as nitric oxide synthase inhibitors
10/19/2004US6806380 Modified safe and efficient process for the environmentally friendly synthesis of imidoesters
10/14/2004WO2004087124A1 Compounds having serotonin 5-ht17 receptor antagonist activity and muscarinic m4 receptor agonist activity and their use in the treatment of psychotic disorders
10/14/2004US20040204582 Substituted sulfonamides and ureas useful for inhibiting kinase activity
10/13/2004CN1170813C N2 phenylamidine derivatives and fungicidal composition and use
10/12/2004US6803472 Method for preparing nitrogen containing compounds
10/12/2004US6803464 Reacting acid salt of aminoacetamidine with a source-of cyanide and reacting with 2,3,5-trichlorobenzaldehyde to produce 2-((cyano-(2,3,5-trichlorophenyl)-methyl)-amino)-acetamidine or a salt thereof
10/07/2004US20040198739 Prevention reproduction of virus
10/06/2004EP1463495A2 Agents and methods for treatment of cancer
09/2004
09/30/2004US20040192779 2-amino-2-alkyl-4 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors
09/29/2004EP1062201B1 Halogenated amidino amino acid derivatives useful as nitric oxide synthase inhibitors
09/29/2004CN1168717C Novel intermediates for prepn. of antihisatminic piperidine derivatives
09/28/2004US6797828 Processes for the preparation of 4(5)-amino-5(4)-carboxamidoimidazoles and intermediates thereof
09/28/2004US6797699 Exemplified by n'-l-arginylspermidine
09/21/2004US6794545 Conformationally restricted polyamine analogs as disease therapies
09/21/2004US6794515 Synthesis of 2-alkylcysteine via substituted thiazoline amide
09/21/2004US6794365 Inhibitors of the blood clotting enzyme factor xa; treating thromboembolic diseases; trifluoroacetic acid salt of 2-(4-carbamimidoyl-benzyl)-n-((1-carbamoyl-4-guanidino-butylcarbamoyl) -cyclohexyl-methyl)-n',n'-dimethyl-malonamide
09/16/2004WO2003028729A3 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
09/08/2004EP1311492B1 Method for producing lamotrigine from alpha-oxo-2,3-dichlorophenyl acetamidino-aminoguanidino hydrazone by ring closure reaction
09/07/2004US6787668 2-amino-4,5 heptenoic acid derivatives useful as nitric oxide synthase inhibitors
09/02/2004WO2004073709A1 Antimicrobial agents
09/02/2004US20040171839 Serine protease inhibitor; therapy for thrombosis , cardiovascular disorders
09/02/2004US20040171670 Neurological diseases and disorders; such as 3-fluoro-10,11-dihydro-5-(2-aminoethyl)-5H-dibenzo[a,d]cycloheptene
09/02/2004US20040171616 preventing and treating thrombotic conditions, such as coronary artery disease, cerebrovascular disease, and other coagulation related disorders
08/2004
08/31/2004US6783946 Positively charged non-natural amino acids, methods of making thereof, and use thereof in peptides
08/25/2004EP1448534A1 6-membered unsaturated heterocyclic compounds useful for selective inhibition ofthe coagulation cascade
08/25/2004EP1149069B1 Phenylglycine derivatives
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