Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
05/2001
05/09/2001CN1294576A VLA-4 antagonists
05/09/2001CN1294121A N-acyl amino-acid amide prodn. process
05/08/2001US6229026 Reacting an isobenzofuran derivative with grignard reagents 4-halogen-fluorophenyl and 3-halogen-n,n-dimethylpropylamine; causing ring-closure of the product and conversion to 5-cyano derivative
05/08/2001US6229011 N-aroylphenylalanine derivative VCAM-1 inhibitors
05/08/2001US6228985 Derivatives of aminobenzoic and aminobiphenylcarboxylic acids useful as anti-cancer agents
05/08/2001US6228982 Stable compounds that form double-stranded, helical structures mimicking double-stranded dna; diagnosis; prophylaxis; therapy; antisense agents
05/03/2001WO2001030747A1 Hydroxamic acid derivative as inhibitor of the formation of soluble human cd23
05/03/2001WO2001030745A1 Anthranilic acid derivatives as inhibitors of the cgmp-phosphodiesterase
05/03/2001CA2389319A1 Hydroxamic acid derivative as inhibitor of the formation of soluble human cd23
05/02/2001EP1095930A1 Novel compounds
05/02/2001EP1095011A1 Novel fluorescent lanthanide chelates
05/02/2001EP1094826A1 Novel therapeutic agents that modulate alpha-1a adrenergic receptors
05/02/2001EP0966427B1 Preparation of acid amides and metallisation of compounds
05/02/2001EP0743853B1 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
05/02/2001CN1065237C Cyclopentane-and-cyclo pentene-beta-amino acids
05/01/2001USRE37160 Synthesis of tyrosine derived diphenol monomers
05/01/2001US6225625 Signal detection methods and apparatus
05/01/2001US6225352 Low molecular weight dendritic compounds as pharmaceutical agents
04/2001
04/26/2001WO2001028982A1 Diethylenetriaminepenta acetic acid derivatives
04/26/2001WO2001028979A2 Inhibitors of neuraminidases
04/25/2001EP1094059A1 Process for production of N-acyl amino acid amide
04/25/2001EP1093819A2 Compounds and compositions for delivering active agents
04/25/2001EP0701568B1 New peptide derivatives
04/25/2001CN1064954C Orthosubstituted benzoylguanidine, preparation of same, pharmaceutical containing same and application of same
04/24/2001US6222052 Process for preparing optically active 2-amino-ω-oxoalkanoic acid derivatives
04/24/2001US6221865 Inhibitors of protein farnesyltransferase and protein geranylgeranyltransferase.
04/24/2001US6221367 Exposing a biologically active agent to a complexing perturbant to reversibly transform the biologically active agent to the intermediate state and to form a transportable supramolecular complex
04/22/2001WO2002102250A1 $g(in vivo) imaging
04/22/2001CA2422767A1 In vivo imaging
04/19/2001WO2000073274A3 Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors
04/19/2001WO2000050623A3 Method for preparing optically active 3,3,3-trifluoromethyl-2-alkyl propionic acid derivatives
04/18/2001EP1091930A1 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES
04/18/2001EP1091929A2 Secondary aspartic acid amide esters
04/18/2001EP1091928A1 Novel acyl pseudodipeptides, preparation method and pharmaceutical compositions containing same
04/18/2001CN1291973A N-sulphonyl and N-sulphinyl phenylglycinamide
04/17/2001US6218393 Anthranilic acid derivatives as multi drug resistance modulators
04/17/2001US6218370 Useful for cell transfection
04/17/2001CA2103044C Novel bi-aromatic compounds derived from a salicylic pattern, method of preparation and use in human and veterinary medicine and in cosmetics
04/12/2001WO2001025190A1 Novel diarylamide derivatives and use thereof as medicines
04/12/2001WO2001025189A1 2'-substituted 1,1'-biphenyl-2-carbonamides, method for the production thereof, use thereof as a medicament and pharmaceutical preparations containing said compounds
04/12/2001WO2001025172A1 A method for preparing and screening one or more compounds
04/12/2001WO2001025170A1 N-SUBSTITUTED DIALKYL α-AMINO ACIDS FOR USE AS AMINO PROTECTING GROUPS
04/12/2001WO2001024925A1 Method for activating passivated iron
04/12/2001WO1999063939A9 Multibinding inhibitors of cyclooxygenase-2
04/12/2001CA2385972A1 Novel diarylamide derivatives and use thereof as medicines
04/12/2001CA2385715A1 A method for preparing and screening one or more compounds
04/12/2001CA2385597A1 Method for activating passivated iron
04/11/2001EP1090914A2 Processes and intermediates for manufacturing retroviral protease inhibiting compounds
04/11/2001EP1090909A1 Novel inhibitors of prenylated pyrophosphate consuming enzymes
04/11/2001EP1090625A2 Topical composition for the skin and use thereof
04/11/2001EP1090106A2 Alkylamines and their precursors as specific modulators of human gamma-delta t cell function
04/11/2001EP1089963A1 Hydroxamic acid derivatives as inhibitors of the production of human cd23 and of the tnf release
04/11/2001EP0809625B1 Anionic amphiphilic compounds with at least two hydrophilic and at least two hydrophobic groups based on dicarboxylic acid diamides
04/10/2001US6214877 Antidiabetic agents; modulator of glucose concentration
04/10/2001US6214799 Unsaturated amide compounds
04/05/2001WO2001023347A1 Novel aromatic compounds
04/05/2001WO2001023067A1 Polyamide-containing ligands covalently bonded to supports, polyamide-containing resins, and methods for removing metals from solutions
04/05/2001DE19947508A1 Activation of passivated iron to form a catalyst component, useful for hydrogenation, comprises treatment with hydrogen at elevated temperature and pressure in the presence of a nitrile compound.
04/05/2001DE19947457A1 New 2'-aminomethyl-biphenyl-2-carboxamide derivatives, are potassium channel blockers especially useful for treating re-entry or supraventricular arrhythmia or atrial fibrillation or flutter
04/05/2001CA2384631A1 Polyamide-containing ligands covalently bonded to supports, polyamide-containing resins, and methods for removing metals from solutions
04/04/2001EP1088481A2 Fungicides for the control of take-all disease of plants
04/04/2001EP1087953A1 Nitrate salts of antihypertensive medicines
04/04/2001EP1087940A1 Novel compounds useful in pain management
04/04/2001EP1087938A1 Inhibitors of neuraminidases
04/03/2001US6211245 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
04/03/2001US6211242 Benzamide derivatives as vasopressin antagonists
03/2001
03/29/2001WO2001021603A1 A process for the synthesis of ritonavir
03/29/2001WO2001021584A1 Tyrosine derivatives
03/29/2001WO2001021577A2 Melanin concentrating hormone antagonist
03/29/2001WO2001021576A1 Aromatic diamide derivatives or salts thereof, agricultural/horticultural chemicals and method of using the same
03/29/2001WO2000059875A3 Novel inhibitors of formation of advanced glycation endproducts (age's)
03/29/2001CA2386474A1 Melanin concentrating hormone antagonist
03/28/2001EP1086081A1 Quarternary ammonium compounds as anti-tussive agents
03/28/2001EP1086065A4 Combinatorial synthesis of multibinding libraries
03/28/2001EP1086065A1 Combinatorial synthesis of multibinding libraries
03/28/2001EP1085894A1 Beta 3-adrenergic receptor agonists
03/28/2001EP1085893A1 Phosphodiesterase-v modulator drugs and their uses
03/28/2001EP1085891A1 Multibinding inhibitors of topoisomerase
03/28/2001EP1085889A2 Novel therapeutic agents that modulate endothelin receptors
03/28/2001EP1085887A2 Novel angiotensin receptor modulators and their uses
03/28/2001EP1085870A2 Multivalent agonists, partial agonists and antagonists of the gaba receptors
03/28/2001EP1085868A1 H1-histamine receptor antagonists
03/28/2001EP1085861A1 Inhibitors of nitric oxide synthase
03/28/2001EP1085847A2 Novel therapeutic agents that modulate estrogen receptors
03/28/2001EP1085846A2 Multibinding inhibitors of microsomal triglyceride transferase protein
03/28/2001EP1085845A2 Multibinding inhibitors of cyclooxygenase-2
03/28/2001EP1035772A4 Fungicidal compositions and methods, and compounds and methods for the preparation thereof
03/28/2001CN1289324A Method for preparing an N-[(aliphatic or aromatic) carbonyl]-2-aminoacetamide compound and a cyclyzed compound
03/27/2001US6207712 Isolating or synthesizing fatty acid amino acid conjugate selected from n(17-hydroxylinolenoyl)-l-glutamine, n(linolenoyl)-l-glutamine; applying to plant such that plant produces and/or releases volatile compounds
03/27/2001US6207693 Benzamide derivatives having a vasopressin antagonistic activity
03/22/2001WO2001019809A1 Tryptase inhibitors
03/22/2001WO2001019784A1 Methods of preparing substituted tetracyclines with transition metal-based chemistries
03/22/2001WO2001019780A2 Novel derivatives of dicarboxylic acid having pharmaceutical properties
03/22/2001WO1999063936A8 Novel therapeutic agents that modulate endothelin receptors
03/22/2001CA2672722A1 Methods of preparing substituted tetracyclines with transition metal-based chemistries
03/22/2001CA2384763A1 Tryptase inhibitors
03/21/2001EP1085011A1 Novel polyamine analogues as therapeutic and diagnostic agents
03/21/2001EP1085009A1 Indan derivatives
03/21/2001EP1084137A1 Peptide inhibitors of hepatitis c virus ns3 protease
03/21/2001EP1083921A1 Novel leukotriene receptor antagonists and their uses