Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
10/2001
10/11/2001WO2001012154A3 Targeted lipid particles
10/11/2001CA2404628A1 7-and 9-carbamate, urea, thiourea, thiocarbamate, and heteroaryl-amino substituted tetracycline compounds
10/10/2001EP1142867A2 Cell adhesion inhibitors
10/10/2001EP1140854A2 Methods for the synthesis of alpha-hydroxy-beta-amino acid and amide derivatives
10/10/2001EP1140846A1 Aspartic protease inhibitors
10/10/2001EP1140829A1 Contrast media for angiography
10/10/2001EP1140787A1 Crosslinkers based on dibenzalacetone derivatives
10/10/2001EP1140745A1 Colchinol derivatives as vascular damaging agents
10/10/2001CN1316986A Novel compounds
10/04/2001WO2001072701A1 Ceramide derivatives and method of use
10/04/2001WO2001072699A1 Inhibition of angiogenesis and tumor growth
10/04/2001WO2001072687A1 Diphenyl ether compounds useful in therapy
10/04/2001WO2001072685A2 Polyamine analogues as cytotoxic agents
10/04/2001WO2001072297A1 Methods for inhibiting angiogenesis and tumor growth
10/04/2001WO2001021577A3 Melanin concentrating hormone antagonist
10/04/2001WO2001000663A3 Catalytically active recombinant memapsin and methods of use thereof
10/04/2001EP1137690A2 Peg-based macromonomers, chemically inert polymers prepared therefrom and the use of these polymers for organic synthesis and enzyme reactions
10/04/2001EP1137410A1 Novel 4-dedimethy laminotetra cycline derivatives
10/04/2001CA2659030A1 Methods for inhibiting angiogenesis and tumor growth
10/04/2001CA2404439A1 Diphenyl ether compounds useful in therapy
10/04/2001CA2403814A1 Polyamine analogues as cytotoxic agents
10/04/2001CA2402769A1 Ceramide derivatives and method of use
10/03/2001CN1315945A Nitrate salts of antihypertensive medicines
10/03/2001CN1315941A Process to continuously prepare aqueous mixture of epsi-caprolactam and epsi caprolactam precursors
10/02/2001US6297401 A 3-nitrosalicylamide derivative effective against plant pytopathogens
10/02/2001US6297283 Excellent inhibitory effect on the production of an ige antibody and are hence useful as antiallergic agents
09/2001
09/27/2001WO2001070675A2 Inhibitors of histone deacetylase
09/27/2001WO2001070672A2 Compounds and methods to treat alzheimer's disease
09/27/2001WO2001070671A2 Insecticidal anthranilamides
09/27/2001WO2001070670A1 Novel phenylalanine derivative
09/27/2001WO2001062705A8 Aminoalcohol derivatives
09/27/2001WO2001000665A3 Inhibitors of memapsin 2 and use thereof
09/27/2001WO2000061537A3 Pharmaceutical compounds
09/27/2001US20010025109 Process for the preparation of 3-amino-2-oxo-pyrrolidines, novel intermediates and their use
09/27/2001CA2404002A1 Inhibitors of histone deacetylase
09/27/2001CA2401749A1 Compounds and methods to treat alzheimer's disease
09/26/2001EP0842142B1 Process for producing alpha-(n,n dialkyl)-amino carboxylic acid amides
09/26/2001EP0800505B1 Novel immunotherapeutic aryl amides
09/26/2001CN1314880A Novel method for preparing optically active alpha-aminonitriles
09/26/2001CN1071751C Reversible protease inhibitors
09/25/2001US6294580 For therapy and prophylaxis of type ii or non-insulin dependent diabetes mellitus, hyperglycaemia, dyslipidemia, type ii diabetes, type i diabetes, hypertriglyceridemia, syndrome x, insulin resistance, heart failure
09/25/2001US6294569 Analgesic at central nervous system in the mammalian subject. also, these compounds are inflammatory pain caused, for example by burns (induced by a contact with heat, acid or the other rheumatism or the like, in the said subject.
09/25/2001US6294560 Synthesis of clasto-lactacystin β-lactone and analogs thereof
09/25/2001US6294557 Analgesic at central nervous system in the mammalian subject. also, these compounds are inflammatory pain caused, for example by burns (induced by a contact with heat, acid or the other rheumatism or the like, in the said subject.
09/24/2001WO2003006652A2 Inhibition of specific histone deacetylase isoforms
09/24/2001CA2408385A1 Inhibition of specific histone deacetylase isoforms
09/20/2001WO2001068619A1 5-amide substituted diarylamines as mex inhibitors
09/20/2001WO2001068587A1 Novel crystal of stilbene derivative and process for producing the same
09/20/2001US20010023257 Hypotensive agents; anticholesterol agents
09/20/2001US20010023249 Calcium channel blockers
09/20/2001US20010023240 Compounds and compositions for delivering active agents
09/20/2001CA2403017A1 5-amide substituted diarylamines as mex inhibitors
09/19/2001EP1133485A1 A process for the synthesis of ritonavir
09/19/2001EP1133466A1 A process for the preparation of n,n'-bis 2, 3-dihydroxypropyl] -5-[(hydroxyacetyl) methylamino]-2, 4,6-triiodo-1, 3-benzenedi carboxamide
09/19/2001EP1133465A1 Amphiphilic polyamine compounds
09/19/2001EP1015416B1 Method for the preparation of citalopram
09/19/2001CN1313846A C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cystenine proteases
09/18/2001US6291701 Used as chemical intermeidate
09/18/2001US6291687 Used aspartyl protease inhibitors of human immunodeficiency virus (hiv)
09/18/2001US6291478 Compounds of the benzylaminodiacetamide family, compositions comprising them, preparation process and uses
09/18/2001US6291423 Lipid complexes for transferring at least a therapeutically active substance, in particular a polynucleotide into a target cell and use in gene therapy
09/18/2001US6291183 A plurality of oligonucleotide linker molecules are attached on a planar solid support, photoremovable groups react with terminal ends of oligonucleotides, substrates exposed to light activate binding at selected areas; peptide synthesis
09/12/2001EP1132376A1 Beta-amyloid protein production/secretion inhibitors
09/12/2001EP1131280A1 Preparation of 5-amino-isophthalamides
09/12/2001EP0888317B1 Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma
09/12/2001CN1070843C Process for crystallization frame water of (S)-N, N'-bis[2-hydroxyl-1-(hydroxymethyl)ethyl]-5-[(2-hydroxy-1-oxopropyl)amino]-2,4,6-triiodo-benzendicarboxamide
09/11/2001US6288234 Fluorinated heterocyclic amido amine compounds as drugs
09/11/2001US6288055 Analgesic agents
09/11/2001US6287538 DTPA monoamides, pharmaceutical agents containing these compounds, their use and process for their production
09/11/2001CA2125175C New peptide derivatives
09/07/2001WO2001064638A1 METHOD FOR PRODUCING β-ALANINAMIDES
09/07/2001WO2001064637A1 2-oxo-1-pyrrolidine derivatives, process for preparing them and their uses
09/07/2001WO2001019780A3 Novel derivatives of dicarboxylic acid having pharmaceutical properties
09/07/2001WO2001010383A3 Caspase inhibitors and uses thereof
09/06/2001US20010020097 Treatment of Alzheimer's disease
09/06/2001US20010020024 Opioid analgesics
09/06/2001DE10008522A1 Verwendung von 2-PHenylendiaminderivaten zur Behandlung von Infektionen Use of 2-phenylenediamine for the treatment of infections
09/05/2001EP1129075A1 N-aryl(thio)anthranilic acid amide derivatives, their preparation and their use as vegf receptor tyrosine kinase inhibitors
09/05/2001EP1129074A2 Antrhranilic acid amides and the use thereof as medicaments
09/05/2001EP1129069A1 Method for the crystallization of iopamidol
09/05/2001EP1129068A1 Bicyclic signal transduction inhibitors, composition containing them and uses thereof
09/05/2001EP1129064A1 Transfection reagents
09/05/2001EP0873304B1 Metalloproteinase inhibitors
09/05/2001EP0832061B1 Benzamide derivatives and their use as vasopressin antagonists
09/05/2001EP0777646B1 Metalloproteinase inhibitors
09/05/2001CN1311776A Quanternary ammonium compounds as anti-tussive agents
09/04/2001US6284924 Bis/oxynaphthalene derivatives of carboxylic acids
09/04/2001US6284780 Prevent tumor necrosis factor retrovirus reproduction
09/04/2001CA1341289C Amide complexes
08/2001
08/30/2001WO2001062726A2 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
08/30/2001WO2001062712A1 (2s)-aminoindan derivatives, a process for their preparation and their use as selective dopamine d3 ligands
08/30/2001WO2001062711A2 Substituted alkylene diamine compounds
08/30/2001WO2001062709A2 Use of 2-phenylene diamine derivatives for the treatment of infections
08/30/2001WO2001062705A2 Aminoalcohol derivatives
08/30/2001US20010018441 Antiinflammatory agent, immunosuppressant, anticancer agents, antiarthritic agents
08/30/2001CA2401030A1 Use of 2-phenylene diamine derivatives for the treatment of infections
08/29/2001EP1127055A2 Stereoselective process for producing cryptophycins
08/29/2001EP1127052A1 Substituted 2-phenylbenzimidazoles, the production thereof and their use
08/29/2001EP0968185B1 Process to continuously prepare an aqueous mixture of (e)-caprolactam and (e)-caprolactam precursors
08/29/2001CN1310621A Substituted anilide compounds and methods