Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
01/2001
01/25/2001WO2001005746A1 AMINOBENZOPHENONES AS INHIBITORS OF IL-1β AND TNF-$g(a)
01/25/2001CA2379273A1 Aminobenzophenones as inhibitors of il-1.beta. and tnf-.alpha.
01/24/2001EP1070047A2 Lipids
01/24/2001EP1070046A1 Propanolamine derivatives
01/24/2001EP0712389B1 Therapeutic compound - fatty acid conjugates
01/24/2001CN1281430A N-alkanoylphenylalanine derivatives
01/23/2001US6177573 Process to prepare taxol
01/23/2001US6177561 Preparation of acid amides and metallization of compounds
01/23/2001US6177414 Polymaminoamide dendrimer star polymer carrying salicylic acid moieties; drug delivery
01/23/2001US6177060 Nmr or x-ray lymphography images
01/18/2001WO1999064049A9 Novel antibacterial agents
01/17/2001EP1069109A1 Process for production of optically active N-protected-N-methyl-phenylalanine derivative
01/17/2001EP1068176A1 Cysteine amides as farnesyl transferase inhibitors
01/17/2001CN1280571A New heterocyclic compounds and their use in medicine, process for their preparation and pharmaceutical compositions containing them
01/17/2001CN1280561A Amidocarboxylic acid derivatives
01/17/2001CN1280560A Adamantane derivatives
01/16/2001US6174923 Administering ethynyl alanine amino diol compound for treating hypertension
01/16/2001US6174905 As carcinostatic agent to a hematologic malignancy and a solid carcinoma
01/16/2001US6174887 Amide compounds and use of the same
01/16/2001US6174711 Method for producing L-allysine acetal
01/11/2001WO2001002466A1 Diaminobenzene derivative, polyimide obtained therefrom, and liquid-crystal alignment film
01/11/2001WO2000052019A3 Crystallization products of neotame and methods for producing same
01/10/2001EP1067136A1 New peptide derivatives
01/10/2001EP1066247A1 Inhibitors of serine proteases, particularly hepatitis c virus ns3 protease
01/10/2001EP1066245A1 Novel local anesthetic compounds and uses
01/09/2001US6172261 Biosynthesis using chain extension
01/09/2001US6172113 Bicyclic amino derivatives and PGD2 antagonist containing the same
01/09/2001US6171866 N-substituted iminodiacetic acid derivatives
01/09/2001US6171612 Gene therapy
01/04/2001WO2001000665A2 Inhibitors of memapsin 2 and use thereof
01/04/2001WO2001000663A2 Catalytically active recombinant memapsin and methods of use thereof
01/04/2001WO2001000621A1 Novel quaternary ammonium derivatives, method for preparing same and pharmaceutical use
01/04/2001WO2001000566A2 Substituted phenoxyacetic acids
01/04/2001WO2000035868A3 Methods for the synthesis of alpha-hydroxy-beta-amino acid and amide derivatives
01/04/2001CA2385798A1 Substituted phenoxyacetic acids
01/04/2001CA2377154A1 Novel quaternary ammonium derivatives, method for preparing same and pharmaceutical use
01/04/2001CA2374610A1 Catalytically active recombinant memapsin and methods of use thereof
01/03/2001CN1278530A Novel peptide derivative
01/02/2001US6169192 Ligands for transition metal complexes suitable for enantioselective hydrogenation of organic double or triple bonds
01/02/2001US6169116 Amino-tetralines, pharmaceutical compositions containing them and their pharmaceutical uses
01/02/2001CA2068064C Fibrinogen receptor antagonists
01/02/2001CA1341162C Sbustituted aminomethyltetralins and their heterocyclic analogues
12/2000
12/28/2000WO2000078708A1 Substituted benzamide inhibitors of rhinovirus 3c protease
12/28/2000CA2375356A1 Substituted benzamide inhibitors of rhinovirus 3c protease
12/27/2000EP1062218A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
12/27/2000EP1061934A1 Fibrinogen receptor antagonists
12/27/2000EP1021099A4 Anti-bacterial amine derivatives
12/27/2000EP0821666B1 Derivatives of succinamide and their use as metalloproteinase inhibitors
12/27/2000EP0751768B1 Anti-viral and anti-cancer agent
12/27/2000EP0530358B2 Polyaspartic acid compostion, method of its production and its use
12/27/2000CN1278167A Amide derivatives
12/26/2000US6166200 Cascade polymer complexes, process for their production and pharmaceutical agents containing said complexes
12/26/2000US6166057 Fungicides for the control of take-all disease of plants
12/26/2000US6165999 Tetracycline derivatives
12/26/2000US6165971 Polyamides or polylactams or amides of dimerized fatty acid as thickner and a surfactant
12/21/2000WO2000077032A2 Spermine:peptide-based surfactant compounds
12/21/2000WO2000077027A2 Serine protease inhibitors
12/21/2000WO2000076971A2 Serine protease inhibitors
12/21/2000WO2000076970A2 Serine protease inhibitors
12/21/2000WO2000076489A2 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
12/21/2000CA2383008A1 Compounds
12/21/2000CA2375920A1 Compounds
12/21/2000CA2375551A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
12/20/2000EP1060175A2 Tryptase inhibitors
12/20/2000EP1060171A2 Tryptase inhibitors
12/20/2000EP1060160A2 Disubstituted lavendustin a analogs and pharmaceutical compositions comprising the analogs
12/20/2000EP0915835B1 A process for the preparation of 5- acetyl (2,3-dihydroxypropyl)amino]-n,n'-bis (2,3-dihydroxypropyl)-2,4,6- triiodo-1,3-benzenedicarboxamide
12/19/2000US6162812 Pharmaceutical compositions containing HIV protease inhibitors and methods of their use
12/14/2000WO2000075104A1 Novel method for preparing optically active alpha-aminonitriles
12/14/2000WO2000046187A3 Antizyme modulators and their use
12/13/2000CN1276785A N-aroylphenylalanine derivs.
12/12/2000US6160009 Excitatory amino acid receptor modulators
12/12/2000CA2131186C Isosteric antiherpes peptide derivatives
12/12/2000CA2058560C Trifluoromethylketone derivatives, processes for preparation thereof and use thereof
12/12/2000CA2036413C Hiv protease inhibitors
12/12/2000CA2036397C Hiv protease inhibitors containing derived amino acid units
12/07/2000WO2000073274A2 Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors
12/07/2000WO2000073263A1 Cytofectin dimers and methods of use thereof
12/07/2000WO2000073260A1 Squaric acid derivatives as cell adhesion molecules
12/07/2000WO2000072920A1 Substituted biaryl ether compounds
12/07/2000CA2375822A1 Substituted biaryl ether compounds
12/07/2000CA2375218A1 Squaric acid derivatives as cell adhesion molecules
12/07/2000CA2375188A1 Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors
12/06/2000EP1056714A1 Phenylalanine derivatives as inhibitors of alpha4 integrins
12/06/2000EP1056475A1 Dendrimeric fullerene derivatives, method for producing same and their use as neuroprotectors
12/05/2000US6156924 Inhibit an envelope virus such as influenza virus by inhibiting the fusion of the virus with the host cell
12/05/2000US6156896 Fluorous reaction and separation systems
12/05/2000US6156884 Bifunctional boronic compound complexing reagents and complexes
12/05/2000US6156750 Bioactive bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof
11/2000
11/30/2000WO2000071529A1 Substituted phenyl compounds with immunosuppressing activity and pharmaceutical compositions
11/30/2000DE19924819A1 Substituierte Phenylcyclohexancarbonsäurebenzylamid (Adenosinaufnahmeinhibitoren) Substituted Phenylcyclohexancarbonsäurebenzylamid (adenosine uptake inhibitors)
11/30/2000CA2372580A1 Substituted phenyl compounds with immunosuppressing activity and pharmaceutical compositions
11/29/2000EP1055665A1 3-(3-Hydroxyphenyl)-3-amino-propionamide derivatives
11/28/2000US6153796 Reaction of acetamido-n,n'-bis(2,3-hydroxypropyl)-2,4,6-triiodoisophthalamide with 2,3-dihydroxypropylating agent in the presence of alcohol solvent
11/28/2000US6153771 Intermediates for the preparation of iodinated contrast agents
11/28/2000US6153659 3-{N-[2-(N',N'-dimethylamino ethoxy)ethyl]-N-methylamino}propionamide for the production of polyurethanes
11/28/2000US6153171 Methods for identifying compounds effective for treating neurodegenerative disorders and for monitoring the therapeutic intervention therefor
11/23/2000WO2000069810A1 Glucagon antagonists/inverse agonists
11/23/2000WO2000043354A3 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4
11/23/2000DE19923274A1 Homo-conjugated triene preparation in high yield, by sequential Wittig reactions of bis-ylid with two aldehyde components, useful in synthesis of highly unsaturated fatty acids, leukotrienes or pheromones