Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
03/2001
03/21/2001EP1083920A1 Novel antibacterial compounds
03/21/2001EP1083919A1 Novel antiviral compounds
03/21/2001EP1083917A1 Novel analgesic agents
03/21/2001EP1083894A1 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE
03/21/2001EP1083893A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the d 1? receptors
03/21/2001EP1083888A1 MULTIBINDING AGENTS THAT MODULATE PPARgamma AND RXR RECEPTORS
03/21/2001CN1288457A Inhibitors of & alpha; 4 mediated cell adhesion
03/20/2001US6204293 Inhibitors of protein isoprenyl transferases
03/20/2001US6204238 Fatty acid derivatives and their use as surfactants in detergents and cleaners
03/20/2001US6204222 Substituted cyclohexene-1,2-dicarboxylic acid derivatives and intermediates for their preparation
03/15/2001WO2001018171A2 Novel class of cytodifferentiating agents and histone deacetylase inhibitors, and methods of use thereof
03/15/2001WO2001017982A1 Benzophenones as inhibitors of reverse transcriptase
03/15/2001WO2001017953A1 Non-peptidic cyclophilin binding compounds and their use
03/15/2001WO2000053583A8 Inhibitors of protein tyrosine phosphatase
03/15/2001WO2000051972A8 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy
03/15/2001DE19943635A1 Neuartige Aminodicarbonsäurederivate mit pharmazeutischen Eigenschaften Novel Aminodicarbonsäurederivate with pharmaceutical properties
03/15/2001CA2383999A1 Novel class of cytodifferentiating agents and histone deacetylase inhibitors, and methods of use thereof
03/15/2001CA2383782A1 Compounds for the treatment of viral infections
03/15/2001CA2383086A1 Non-peptidic cyclophilin binding compounds and their use
03/15/2001CA2318004A1 Novel polyamine analogues as therapeutic and diagnostic agents
03/14/2001EP1082289A1 Methods for identifying novel multimeric agents that modulate receptors
03/13/2001US6201153 Synthesis of midodrine HCI from a novel intermediate 1-(2′,5′-dimethoxyphenyl)-2-azidoethanone
03/13/2001US6201024 Effective p2x7 receptor antagonists for use in the treatment of inflammatory, immune or cardiovascular disorders
03/13/2001US6201007 Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists
03/13/2001CA2167651C Biologically highly active bicyclic aromatic compositions; pharmaceutical and cosmetic compositions containing the same and their use
03/08/2001WO2001016211A1 Amphipathic compound having dendritic structure
03/08/2001WO2001016090A1 Enantiomerically-enriched compounds having photocleavable bond(s) and methods related thereto
03/08/2001WO1999064047A8 Novel antiviral compounds
03/08/2001WO1999063930A8 Novel angiotensin receptor modulators and their uses
03/08/2001WO1999019296A8 Aminobutanoic acid derivatives
03/08/2001CA2384191A1 Enantiomerically-enriched compounds having photocleavable bond(s) and methods related thereto
03/07/2001EP1080083A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
03/07/2001EP1080080A1 Novel therapeutic agents that modulate neurokinin receptors
03/07/2001EP1080070A2 Antiangiogenic drug to treat cancer, arthritis and retinopathy
03/07/2001EP1080069A1 Anthranilic acid derivatives as inhibitors of the cgmp-phosphodiesterase
03/07/2001EP1080068A1 Modulators of protein tyrosine phosphatases
03/07/2001EP1080067A1 Biodegradable corrosion inhibitors
03/07/2001CN1286254A Aromatic amino ether as analgesics
03/06/2001US6197798 Inhibitors of microsomal triglyceride transfer protein
03/06/2001US6197750 C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases
03/06/2001US6197332 Lipid-conjugated polyamide compounds and related compositions and methods thereof
03/01/2001WO2000058270A3 Hsv primase inhibitors
02/2001
02/28/2001EP1077931A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
02/28/2001EP1077930A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
02/28/2001EP1077929A1 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
02/28/2001EP1077928A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
02/28/2001EP1077927A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
02/28/2001CN1285346A Process for preparation of 4.4' diaminophenylacyl substituted aniline
02/27/2001US6194615 Useful as crosslinkers in coatings applications
02/27/2001US6194612 Template for solution phase synthesis of combination libraries
02/27/2001US6194418 Bactericides, pesticides
02/22/2001WO2001012591A1 Novel naphthylsulfonic acids and related compounds as glucose uptake agonists
02/22/2001WO2001012588A1 Salicylamide derivatives
02/22/2001WO2001012587A1 Aminosalicylclic acid amides and their use for combating organisms that are harmful to plants
02/22/2001WO2001012154A2 Targeted lipid particles
02/22/2001WO1999063996A8 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
02/22/2001DE19938737A1 Aminosalicylsäureamide Aminosalicylamides
02/22/2001CA2379431A1 Targeted lipid particles
02/21/2001EP1077070A2 Oral drug delivery compositions
02/21/2001EP1076641A1 Inhibitors of impdh enzyme
02/21/2001EP0835238B1 New cationic and polycationic amphiphiles, reactives containing the same and their use
02/21/2001CN1284942A Matrix metalloprotease inhibitors
02/20/2001US6191165 Pharmaceutical for treatment of neurological and neuropsychiatric disorders
02/20/2001US6191157 Anticholesterol agents; cardiovascular disorders
02/15/2001WO2001010821A1 Multivalent exocyclic diketo compounds
02/15/2001WO2001010799A1 Methods for preparing n-[(aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds
02/15/2001WO2001010429A2 Long chain n-alkyl compounds and oxa-derivatives thereof and use as antiviral compositions
02/15/2001WO2001010383A2 Caspase inhibitors and uses thereof
02/15/2001DE19741356C2 Verwendung von Glucoprotaminen Use of Glucoprotaminen
02/14/2001EP1075462A2 Process for the preparation of s- n,n'- bis 2- hydroxy-1- (hydroxymethyl) ethyl]-5- (2- hydroxy-1- oxopropyl)- amino]- 2,4,6- triiodo- 1,3- benzenedicarboxamide
02/14/2001EP0877729B1 Azlactone-based surfactants
02/14/2001CN1284060A Novel metalloproteinase inhibitors
02/14/2001CN1284058A Neuroprotective agents
02/14/2001CN1284057A Adamantane derivatives
02/14/2001CN1284056A Anticonvulsant and sentral nervous system-active bis (fluorophenyl) alkylamides
02/13/2001US6187905 Peptide compound which inhibits viral proteinases; viricides for hepatitis c, hepatitis g, and human gb viruses
02/08/2001WO2001009083A1 Production of n-substituted 2,7-dialkyl-4-hydroxy-5-amino-8-aryl-octanoylamides
02/08/2001WO2001009079A1 2-alkyl-5-halogen-pent-4-ene carboxylic acids and their production
02/08/2001WO2000066528A3 Quinones for treatment of diseases
02/07/2001EP1073643A2 New heterocyclic compounds and their use in medicine, process for their preparation and pharmaceutical compositions containing them
02/07/2001EP1073641A2 New substituted amides, their production and their use
02/07/2001EP1073633A2 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
02/07/2001EP1073632A1 Substituted benzamides, their production and their use as cysteine protease inhibitors
02/07/2001EP1073631A1 New substituted amides, their production and their use
02/07/2001EP1073623A1 Substituted amino acids as erythropoietin mimetics
02/07/2001CN1283181A Substituted beta-alanines
02/06/2001US6184389 Feature a plurality of functional groups attached to backbone and phosphoramidate sites
02/06/2001US6184345 Stable under solid phase synthesis conditions
02/06/2001US6184249 Androgen receptor suppressors in the therapy and diagnosis of prostate cancer, alopecia and other hyper-androgenic syndromes
02/06/2001US6184210 Dipeptide-based caspase (proteolytic family of cysteine proteases whose active site cysteine residue is essential for ice-mediated apoptosis) inhibitors of given formula are potent inhibitors of apoptosis
02/01/2001WO2001007400A1 Carboxylic acid derivatives and adhesion molecule inhibitors containing the same as the active ingredient
02/01/2001WO2001007020A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof
02/01/2001DE19935219A1 Carbonsäureamide, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Herstellung Carboxamides, medicaments containing these compounds, their use and production
02/01/2001CA2382757A1 Carboxylic acid derivatives and adhesion molecule inhibitors which contain the same as effective ingredients
01/2001
01/31/2001EP1072255A2 Desferrioxamine oral delivery system
01/31/2001EP1071660A1 N-sulphonyl and n-sulphinyl phenylglycinamide
01/31/2001CN1282319A Aminobutanoic acid derivatives
01/30/2001US6180140 Modified amino acids for drug delivery
01/30/2001CA2010929C Process for preparing nitriloamides
01/30/2001CA1341173C Fungicides