Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
10/1999
10/28/1999WO1999054294A1 New substituted amides, their production and their use
10/28/1999WO1999054293A1 Substituted benzamides, their production and their use as cysteine protease inhibitors
10/28/1999WO1999054290A1 Inhibitors of neuraminidases
10/28/1999WO1999054284A1 Anthranilic acid derivatives as inhibitors of the cgmp-phosphodiesterase
10/28/1999WO1999054283A1 Polyamine transport inhibitors
10/28/1999WO1999054279A1 Substituted amino acids as erythropoietin mimetics
10/28/1999CA2329660A1 Inhibitors of neuraminidases
10/28/1999CA2328720A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
10/28/1999CA2328435A1 New substituted amides, their production and their use
10/28/1999CA2328430A1 Substituted benzamides, their production and their use as cysteine protease inhibitors
10/28/1999CA2328413A1 Anthranilic acid derivatives as inhibitors of the cgmp-phosphodiesterase
10/27/1999EP0951466A2 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
10/27/1999EP0951465A1 Alpha-amino acid amides, preparation thereof and the therapeutical use thereof
10/27/1999CN1233238A Acylaminoalkenylene-amide derivatives as NK1 and NK2 antagonists
10/26/1999US5973188 Anticoagulant; prevention cell, protein binding
10/26/1999US5973006 Nervous system disorders; alzheimer's disease; huntington disease; parkinson's disease
10/26/1999US5972307 Administering to human or animal body an effective amount of a diagnostic agent comprises a metal chelate of a compound having two macrocyclic chelant groups linked by a bridge containing ester or amide bond
10/21/1999WO1999052858A2 Lipids
10/21/1999WO1999032428A8 Synthesis of diamines
10/21/1999DE19818614A1 New benzamide derivatives useful as cysteine protease inhibitors for treating neurodegenerative diseases, neuronal damage, stroke, cranial trauma, Alzheimer's disease, etc.
10/21/1999DE19817461A1 New benzamide derivatives useful as cysteine protease inhibitors for treating neurodegenerative diseases, neuronal damage, stroke, cranial trauma, Alzheimer's disease, etc.
10/20/1999EP0783318A4 Inhibitors of farnesyl-protein transferase
10/20/1999EP0740655B1 Metalloproteinase inhibitors
10/20/1999CN1232447A Hydroxamic acid derivs.
10/19/1999US5969100 Peptide, peptide analog and amino acid analog protease inhibitors
10/14/1999WO1999051565A1 Novel local anesthetic compounds and uses
10/14/1999WO1999051564A1 Propanolamine derivatives
10/14/1999CA2315946A1 Novel local anesthetic compounds and uses
10/13/1999EP0948481A1 Aminobutyric acid fungicides
10/13/1999EP0948360A1 Novel lipid compounds and compositions containing same used for the transfer of at least an active substance, in particular a polynucleotide, in a target cell and therapeutic use
10/13/1999EP0782562B1 Process for the manufacturing of iodinated contrast agents
10/13/1999EP0763523B1 Naphthalene derivative
10/13/1999CN1045589C N-acylaminoglutaricamide derivative
10/12/1999US5965772 Process for the preparation of 5-(acetyl(2,3-dihydroxypropyl)amino-N,N-bis(2,3-dihydroxypropyl)-2,4,6-t riiodo
10/12/1999US5965763 Biphenyl compounds
10/12/1999US5965744 Ortho-substituted benzoylguanidines, including composition and methods of using them
10/12/1999US5965188 Anti-bacterial amine derivatives
10/12/1999US5965121 Compounds and compositions for delivering active agents
10/12/1999US5965119 Trialkyl-lock-facilitated polymeric prodrugs of amino-containing bioactive agents
10/07/1999WO1999050230A1 Inhibitors of serine proteases, particularly hepatitis c virus ns3 protease
10/07/1999WO1999050229A1 Fatty acid analogs and prodrugs
10/06/1999EP0946519A1 Benzamide derivatives having a vasopressin antagonistic activity
10/06/1999EP0946499A1 N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
10/06/1999EP0946497A1 Process for the preparation of nmda antagonists
10/06/1999CN1230876A Anti-bacterial amine derivatives
10/05/1999US5962507 O-acyl-4-phenyl-cyclohexanols, their salts, medicaments containing such compounds, and their use, as well as a method of preparing them
10/05/1999US5962506 Glycol and hydroxyphosphonate peptidomimetics as inhibitors of aspartyl proteases
10/05/1999US5962492 Antiasthma agents; antiinflammatory agents
10/05/1999US5962483 Antiasthma agents; antiinflammatory agents
10/05/1999US5962419 Nervous system disorders; brain disorders
10/02/1999CA2267815A1 Amino acid derivatives and anti-inflammatory agents
09/1999
09/29/1999EP0945517A2 Process for the preparation of the disodium salt of z-l-aspartic acid from fumaric acid
09/29/1999EP0944587A1 Metalloproteinase inhibitors
09/29/1999EP0944584A1 Benzamidoaldehydes and their use as cysteine protease inhibitors
09/29/1999EP0944582A1 Ketobenzamides as calpain inhibitors
09/29/1999CN1229794A Synthetic process of benzobenzyl ammonium amide
09/28/1999US5958971 Chemical compounds
09/28/1999US5958960 Excitatory amino acid receptor modulators
09/28/1999US5958457 Compositions for the delivery of antigens
09/28/1999US5958376 Iodinated X-ray contrast media
09/28/1999US5958375 Urea-linked, iodinated bis phenyl compounds for X-ray contrast media
09/23/1999WO1999047494A1 Novel bis-benzamide derivatives, method for making same pharmaceutical compositions containing them and use thereof as medicine
09/22/1999EP0942924A2 METHODS AND COMPOUNDS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS
09/21/1999US5955506 Acetamidobenzamide compounds for treatment of parkinson's disease
09/21/1999US5955503 Modified amino acid compounds useful as carriers in the delivery of biologically active agents such as, for example, bioactive peptides and the like
09/21/1999US5955491 Method for treating osteoporosis
09/21/1999US5955433 Method of thrombin inhibition
09/16/1999WO1999046268A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
09/16/1999WO1999046267A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999046244A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999046237A1 Modulators of protein tyrosine phosphatases
09/16/1999WO1999046236A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999045939A1 Fibrinogen receptor antagonists
09/16/1999CA2322743A1 Fibrinogen receptor antagonists
09/15/1999EP0941084A1 Raf kinase inhibitors
09/15/1999EP0741697B1 Amino acid derivatives and their use as phospholipase a2 inhibitors
09/15/1999CN1228763A Process for iohexol manufacture
09/15/1999CN1228762A Process for preparation of contrast agent
09/15/1999CN1045084C Novel compound with platelet aggregation inhibitor activity and its use, and drug composition containing the same
09/14/1999US5952499 Therapeutic compound-fatty acid conjugates
09/14/1999US5952462 Transition state analogs
09/14/1999US5952377 Fatty acid analogs and prodrugs
09/14/1999US5952343 HIV protease inhibitors
09/14/1999US5952316 2-amino-1,3-propanediol compound and immunosuppressant
09/10/1999WO1999032428A3 Synthesis of diamines
09/09/1999DE19807475A1 New myxocheline derivatives useful e.g. for treating disorders associated with deficient metal ion metabolism, especially iron or aluminium metabolism, e.g. hemosiderosis, thalassemia or Alzheimer's disease
09/08/1999EP0731797B1 Paramagnetic chelates for nuclear magnetic resonance diagnosis
09/08/1999EP0617009B1 Novel amino acid derivative
09/08/1999CN1228079A Process for preparation of 5-[acetyl (2,3-dihydroxypropyl) amino]-N,N'-bis (2,3-dihydroxypropyl)-2,4,6-triiodo-1,3-benzenedicarboxamide
09/07/1999US5948940 Process for iohexol manufacture
09/07/1999US5948935 Process and intermediates for (s)-α-amino-1-carboxycyclopentaneacetic acid
09/07/1999US5948819 α-substituted phenylacetic acid derivative, its production and agricultural fungicide containing it
09/07/1999US5948778 Difluoro statone antiviral analogs
09/07/1999CA2050334C Iodinated non-ionic compounds, process for their preparation and contrast materials containing them
09/02/1999WO1999043644A1 N-sulphonyl and n-sulphinyl phenylglycinamide___________________
09/02/1999WO1999043642A1 Phenylalanine derivatives as inhibitors of alpha4 integrins
09/02/1999WO1999043636A2 Disubstituted lavendustin a analogs and pharmaceutical compositions comprising the analogs
09/02/1999WO1999043358A1 Dendrimeric fullerene derivatives, method for producing same and their use as neuroprotectors
09/02/1999WO1998034632A9 Compounds and compositions for delivering active agents
09/02/1999CA2321307A1 Disubstituted lavendustin a analogs and pharmaceutical compositions comprising the analogs