Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
12/1999
12/16/1999CA2319120A1 Phosphodiesterase-v modulator drugs and their uses
12/16/1999CA2319068A1 Novel angiotensin receptor modulators and their uses
12/16/1999CA2318894A1 .beta.2-adrenergic receptor agonists
12/16/1999CA2318547A1 Combinatorial synthesis of multibinding libraries
12/16/1999CA2318286A1 Multibinding agents that modulate ppar.gamma. and rxr receptors
12/16/1999CA2318055A1 .beta.2-adrenergic receptor agonists
12/16/1999CA2316999A1 Inhibitors of hiv reverse transcriptase
12/15/1999EP0767780B1 Amino acid derivatives and their use as pesticides
12/15/1999EP0685457B1 Glycerol derivative, device and pharmaceutical composition
12/15/1999CN1238779A Method and compounds for inhibiting 'beta'-amyloid peptide release and/or synthesis
12/15/1999CN1238761A Benzamidoaldehydes and their use as cryteine protease inhibitors
12/15/1999CN1238760A N-(aryl/heteroaryl/alkyl acetyl) amino acid esters, pharmaceutical composition comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
12/14/1999US6001880 Disubstituted n-(2-dialkylaminoethyl)benzamide derivatives of given formula; antibacterial activity against helicobacter pyroli, administering for the prevention or cure of peptic ulcers
12/14/1999US6001879 Suitable for controlling pests, preferably fungi, insects and bacteria, in plants and industrial materials; methods of their sybnthesis including reacting aminosalicylamides with acylating agents
12/14/1999US6001824 Butyryl-tyrosinyl spermine, analogs thereof and methods of preparing and using same
12/14/1999US6001347 Organic acid compound of given structure having an aromatic amide group, a methoxy group in the ortho position on the aromatic ring, and a lipophilic chain terminated with a carboxylic acid is useful as a nontoxic carrier
12/14/1999CA2136007C Novel compound with platelet aggregation inhibitor activity
12/09/1999WO1999062867A1 Indan derivatives
12/09/1999CA2334412A1 Indan derivatives
12/08/1999EP0962552A1 A process for the preparation of 4-(des-dimethylamino)-tetracyclines
12/08/1999EP0850320B1 Methods for detecting binding of ligand pair with enhanced sensitivity
12/08/1999EP0790979B1 Process for the crystallization from water of (s)-n,n'-bis[2-hydroxy-1-(hydroxymethyl)ethyl]-5-[(2-hydroxy-1-oxopropyl)amino]-2,4,6-triiodo-1,3-benzendicarboxamide
12/08/1999EP0712387B1 2-aminoindans as selective dopamine d3 ligands
12/08/1999EP0577675B1 Contrast media
12/08/1999CN1237962A Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists
12/08/1999CN1237959A Process for preparation of an inorganic salt of an optically active
12/08/1999CN1237637A 四环素发酵工艺 Tetracycline fermentation process
12/08/1999CN1047162C Acetylglutaminylzinc compound and its preparation and usage
12/07/1999USRE36433 Dissolving in secondary butanol; crystallization
12/07/1999US5998666 Phenoxyethylamine derivatives, method of preparation, application as medicine and pharmaceutical compositions containing same
12/07/1999US5998466 Preplanting
12/07/1999CA2017126C Reaction products of aminoalkylene polycarboxylic acids with secondary amines and middle distillate compositions containing the aforesaid
12/02/1999WO1999061410A1 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
12/02/1999WO1999061406A2 Antiangiogenic drug to treat cancer, arthritis and retinopathy
12/02/1999WO1999051565A9 Novel local anesthetic compounds and uses
12/02/1999CA2331056A1 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
12/01/1999EP0960084A1 Novel solid-phase synthesis techniques for preparing multiple analogous compounds
12/01/1999CN1236775A Process for preparation of 4-(des-dimethylamino)-tetracyclines
11/1999
11/30/1999US5994408 Compositions containing and methods of using 1-aminoindan and derivatives thereof and process for preparing optically active 1-aminoindan derivatives
11/30/1999US5994270 Fungicides for the control of take-all disease of plants
11/30/1999US5993780 Contrast media
11/25/1999WO1999059960A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
11/25/1999WO1999059959A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
11/25/1999WO1999059958A1 Biodegradable corrosion inhibitors
11/25/1999WO1999059527A2 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives
11/25/1999DE19822912A1 Verfahren zur Herstellung von 3-Amino-2-oxo-pyrrolidinen, neue Zwischenprodukte und deren Verwendung A process for the preparation of 3-amino-2-oxo-pyrrolidines, to novel intermediates and their use
11/25/1999DE19822791A1 Verwendung von Amiden polymerisierter Fettsäuren als Verdickungsmittel Use of polymerized fatty acid amides as thickening agents
11/25/1999CA2332836A1 Biodegradable corrosion inhibitors
11/25/1999CA2328699A1 Benzamide derivatives for the treatment of diseases mediated by cytokines
11/24/1999EP0959070A1 Process for the production of 3-amino-2-oxopyrrolidines, novel intermediates and their use
11/24/1999EP0959066A2 Use of amides of polymerised fatty acids as thickening agent
11/24/1999EP0958404A1 Polymethylenepolyamine dipropionamides as environmentally safe inhibitors of the carbon corrosion of iron
11/24/1999CN1235962A Use of amides of polymerized fatty acids as thickeners
11/24/1999CN1046704C Iodinated derivatives, preparation and use thereof as contrast agents in X-ray radiology
11/23/1999US5990341 Diastereoselective synthesis hydroxyethylene dipeptide isosteres
11/23/1999US5990278 Reacting an organic carboxylic acid with an amine derivative containing a protective group to form protected carbamide, reacting protected carbamide at a first ph to split off protective group, reacting in second ph to form carbamide
11/23/1999US5990166 Compounds and compositions for delivering active agents
11/23/1999US5990158 Carboxylic acid derivatives, method of manufacturing the same and therapeutic agents containing these compounds
11/23/1999US5990116 Trisubstituted phenyl derivatives
11/23/1999US5989539 Compounds and compositions for delivering active agents
11/22/1999CA2272664A1 Process for the preparation of 3-amino-2-oxo-pyrrolidines, novel intermediates and their use
11/18/1999WO1999058496A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
11/18/1999WO1999058495A1 Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
11/18/1999WO1999058494A2 Process for the preparation of s- n,n'- bis[2- hydroxy-1- (hydroxymethyl) ethyl]-5- [(2- hydroxy-1- oxopropyl)- amino]- 2,4,6- triiodo- 1,3- benzenedicarboxamide
11/17/1999EP0956050A1 Novel lipid complexes for transferring at least a therapeutically active substance, in particular a polynucleotide into a target cell and use in gene therapy
11/17/1999EP0656026B1 Polyarylates containing derivatives of the natural amino acid l-tyrosine
11/16/1999US5986132 Synthesis of carboxylic acid derivatives
11/16/1999US5986129 Multistage process of diazotization, acidification, hydrolysis and acylation
11/16/1999US5986053 Peptide nucleic acids complexes of two peptide nucleic acid strands and one nucleic acid strand
11/16/1999US5985928 Bioactive bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof
11/16/1999US5985922 Amino acid derivatives and active oxygen-resisting agent
11/16/1999US5985838 Peptide analogs as irreversible interleukin-1β protease inhibitors
11/16/1999US5985632 Peptide amidase from xanthomonas
11/11/1999WO1999057098A2 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
11/11/1999WO1999040083A3 Bifunctional tryptase inhibitors
11/11/1999WO1999040073A3 Tryptase inhibitors
11/11/1999DE19820400A1 Kationische Azofarbstoffe auf der Bais von Aminobenzoesäure Cationic azo dyes on the bais of aminobenzoic acid
11/11/1999CA2329704A1 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
11/10/1999EP0955342A1 Cationic azo dyes derived from aminobenzoic acid
11/10/1999EP0955066A2 Metal complexes of hydroxyaryl containing aminocarboxylic acid chelating agents
11/10/1999EP0955046A2 Amino acid derivatives and anti-inflammatory agents
11/10/1999EP0954375A1 Novel supported catalysts
11/10/1999CN1046269C HIV protease inhibitors
11/09/1999US5981600 Antineoplastic activity; for chemotherapeutic treatment of cancerous diseases
11/09/1999US5981580 Fatty acid analogs and prodrugs
11/09/1999US5981115 Recording layer comprises a resin an isocyanate compound crosslinked with resin, electron donating coloring agent and an electron accepting coloring developer
11/09/1999CA2140858C Method for denaturing road salt and denatured road salt
11/06/1999CA2270847A1 Alpha-ketoamide derivatives
11/04/1999WO1999055688A1 Substituted diarylalkyl amides as calcium channel antagonists
11/04/1999WO1999055663A1 Inhibitors of impdh enzyme
11/03/1999EP0953835A1 Apparatus for detection of a fluorescence pattern corresponding to ligand binding on a substrate
11/03/1999EP0655069B1 Amphiphilic compounds derived from amino acids or peptides, their methods of synthesis and their application as drug delivery systems
11/02/1999US5977406 Process for preparing α-amino acid amides, α-amino acids and derivatives thereof
11/02/1999US5977387 Process for preparing pharmaceutical compounds
11/02/1999US5977371 Tandem asymmetric transformation process
11/02/1999US5977178 Compounds with growth hormone releasing properties
11/02/1999US5977074 Inhibitors of β-amyloid protein production
11/02/1999US5976569 Diketopiperazine-based delivery systems
10/1999
10/28/1999WO1999054320A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
10/28/1999WO1999054310A2 New substituted amides, their production and their use