Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
03/2000
03/16/2000CA2342364A1 Process to continuously prepare an aqueous mixture of .epsilon.-caprolactam and .epsilon.caprolactam precursors
03/15/2000EP0984922A1 Preparation of tri-iodo benzene compounds
03/14/2000US6037496 3-{N-[2-(N',N'-dimethylamino ethoxy)ethyl]-N-methylamino}propionamide for the production of polyurethanes
03/14/2000US6037494 Crystallizing pure iopamidol from the alcohol solvents which give azeotropes with water forming two separate layers; lower has minimal removable solvent content, and upper layer can be recycled to reduce amount of solvent used
03/14/2000US6037472 For treating disease-states characterized by excessive activity of matrix metalloproteases such as rheumatoid arthritis, osteoarthritis, periodontal disease, aberrant angiogenesis, tumor invasion and metastasis
03/14/2000CA2045543C Iodinated esters
03/09/2000WO2000012462A1 Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
03/09/2000WO2000012454A1 Novel polycationic lipids
03/09/2000CA2341458A1 Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
03/08/2000EP0984002A1 Process to continuously prepare an aqueous mixture of epsilon-caprolactam and epsilon-caprolactam precursors
03/08/2000EP0983290A1 Method for producing polymers having nucleo-bases as side-groups
03/08/2000EP0983230A1 Yellow polymorph of 5-amino-2,4,6-triiodo-n,n'-bis(2,3-dihydroxypropyl)-isophthalamide
03/08/2000EP0983227A1 Preparation of tri-iodo benzene compounds
03/08/2000EP0983226A1 New nitromethyl ketones, process for preparing them and compositions containing them
03/08/2000EP0854857B1 Method of preparing optically active alpha-amino acids and alpha-amino acid derivatives
03/08/2000CN1246844A Process for preparation of iodinated contrast agents and intermediates
03/07/2000US6034275 Tertiary amines
03/07/2000US6034266 Gem-difluoro derivative of phenylacetamide and phenylacetic acid and their pharmaceutical uses
03/07/2000US6034137 Cationic lipids for gene therapy
03/07/2000US6034095 Rheumatic diseases; osteoporosis
03/07/2000CA2109646C Para-nitroanilide peptides
03/02/2000WO1999064054A9 Multibinding inhibitors of topoisomerase
03/02/2000WO1999063937A3 Multivalent macrolide antibiotics
03/01/2000EP0618926B1 New peptide derivatives
03/01/2000CN1245812A Cinnamic acid derivative
02/2000
02/29/2000US6031126 Rearranging a hydrazobenzene compound to form a diaminodiphenyl compound, diazotising, catalytic reacting with a styryl compound to form a distyryl-biphenyl fluorescent whitening agent
02/23/2000EP0861226B1 Synthesis of carboxylic acid derivatives
02/23/2000CN1245486A Ketobenzamides as calpain inhibitors
02/23/2000CN1049651C Metalloproteinase inhibitors
02/22/2000US6028111 Compositions and use of benzamides and nicotinamides as anti-inflammatory agents
02/22/2000US6028110 Succinyl hydroxamic acid, N-formyl-N-hydroxy amino carboxylic acid and succinic acid amide derivatives as metalloprotease inhibitors
02/22/2000US6028101 Fungicides for the control of take-all disease of plants
02/22/2000CA2170607C Difluoro statone antiviral analogs
02/22/2000CA1340904C Amino acid derivative anticonvulsant
02/22/2000CA1340902C Amino acid derivative anticonvulsant
02/17/2000WO2000007981A1 Open chain alkoxyamine compounds and their use as polymerization regulators
02/17/2000WO2000007980A1 Amide derivatives which are useful as cytokine inhibitors
02/17/2000WO1999054310A3 New substituted amides, their production and their use
02/17/2000CA2337482A1 Open chain alkoxyamine compounds and their use as polymerization regulators
02/16/2000EP0979225A1 Compounds and compositions for delivering active agents
02/16/2000EP0979107A1 Light imaging contrast agents
02/16/2000CN1244858A Preparation of alpha-amino carboxylic acid amides
02/16/2000CN1244857A Preparation of acylated alpha-amino carboxylic acid amides
02/16/2000CN1244523A Extraction and purification of tetracyclic antibiotics with alcohol solvents
02/15/2000US6025516 Synthesis of chemical intermediates for forming anti-cancer drug paclitaxel (taxol) and its analogs
02/15/2000US6025444 Cinnamic acid derivative
02/15/2000US6025295 Supported catalysts
02/10/2000WO2000006658A2 Adhesives and sealants
02/10/2000WO2000006610A2 Polymer production
02/10/2000WO2000006559A1 Reduced dipeptide analogues as calcium channel antagonists
02/10/2000WO2000006535A1 Tyrosine-derived compounds as calcium channel antagonists
02/10/2000WO2000006525A2 Synthesis of combinatorial libraries of compounds reminiscent of natural products
02/10/2000WO2000006146A1 Substituted anilide compounds and methods
02/10/2000WO1999063944A3 Novel therapeutic agents that modulate estrogen receptors
02/10/2000WO1999063939A3 Multibinding inhibitors of cyclooxygenase-2
02/10/2000CA2338764A1 Substituted anilide compounds and methods
02/08/2000USRE36562 Fungicides for the control of take-all disease of plants
02/08/2000US6022892 Bis-platinum complexes with polyamine ligands as antitumor agents
02/03/2000WO2000005201A1 N-benzocycloalkyl-amide derivatives and their use as medicaments
02/03/2000WO1999063936A3 Novel therapeutic agents that modulate endothelin receptors
02/03/2000WO1999063933A3 Multivalent agonists, partial agonists and antagonists of the gaba receptors
02/03/2000WO1999063929A3 Multibinding inhibitors of microsomal triglyceride transferase protein
02/03/2000DE19833853A1 Verfahren zur Herstellung von Aminosäuren und Aminosäurederivaten A process for the production of amino acids and amino acid derivatives
02/03/2000CA2338198A1 N-benzocycloalkyl-amide derivatives and their use as medicaments
02/02/2000EP0976760A2 Oligopeptides with fungicidal activity
02/02/2000EP0976721A2 Process for the preparation of amino acids and amino acid derivatives
02/01/2000US6020526 Amide-based cationic lipids
02/01/2000US6020373 Chelate derivatives as protectors against tissue injury
02/01/2000US6020317 Glycerol derivative, device and pharmaceutical composition
01/2000
01/27/2000WO1999063930A3 Novel angiotensin receptor modulators and their uses
01/27/2000WO1999061406A3 Antiangiogenic drug to treat cancer, arthritis and retinopathy
01/26/2000EP0973513A1 Compositions and methods for treating bone deficit conditions
01/26/2000EP0927030A4 Use of aryl n-substituted carboxamides to kill tumors
01/26/2000EP0763016B1 Compositions and methods for treating mast-cell mediated conditions
01/26/2000EP0670677B1 Potentiator of Bacillus pesticidal activity
01/26/2000CN1048719C Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxytetracyclines, prepn. method, their compositions and use thereof
01/26/2000CN1048718C Phenylethyl and phenylpropylamines compounds, prepn. method, pharmaceutical agent and use thereof
01/25/2000US6018050 Enantiomerically pure compounds obtained in high yields; preparing sterically demanding amino acids and their derivatives, such as the preparation of cis-4-hydroxyproline precursors; asymmetric synthesis
01/25/2000US6017965 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
01/25/2000US6017928 Retroviral protease inhibiting compounds
01/25/2000US6017919 Compounds and pharmaceutical use thereof
01/25/2000US6017889 Metalloproteinase inhibitors
01/25/2000US6017887 Peptide, peptide analog and amino acid analog protease inhibitors
01/25/2000US6017768 For screening agonists or antagonists of alpha adrenergic receptors, dopamine receptors, sigma opiate receptors, potassium ion channels, carbonic anhydrase inhibitors; for treatment of glaucoma
01/20/2000WO1999059527A3 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives
01/20/2000WO1999058494A3 Process for the preparation of s- n,n'- bis[2- hydroxy-1- (hydroxymethyl) ethyl]-5- [(2- hydroxy-1- oxopropyl)- amino]- 2,4,6- triiodo- 1,3- benzenedicarboxamide
01/19/2000EP0972845A1 Method for producing L-Allysine acetal
01/19/2000EP0971881A1 Process for the preparation of n-(3-hydroxy-succinyl)-amino acid derivatives
01/19/2000CN1242007A Cycloalkyl, lactam lactone and related compounds as 'beta'-amyloid peptide release inhibitors
01/18/2000US6015879 Compounds for treatment of nervous system disorders including alzheimer's disease, cognition defects, down's syndrome, parkinson's disease, cerebral hemorrhage with amyloidosis, dementia pugilistica, and head trauma
01/13/2000WO2000001666A1 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES
01/13/2000WO2000001665A2 Secondary aspartic acid amide esters
01/13/2000WO2000001663A1 Novel fluorescent lanthanide chelates
01/13/2000DE19920966A1 alpha-Ketoamidderivate alpha-Ketoamidderivate
01/13/2000CA2336904A1 Novel fluorescent lanthanide chelates
01/12/2000EP0970057A2 Substituted aminosalicyclic acid amides with fungicidal effect and intermediate products for production thereof
01/12/2000CN1048240C Process for preparing 7-substed-9-substed. amino-6-demethyl-6-deoxytetracyclines
01/12/2000CN1048239C Naphthalene deriv.
01/11/2000US6013658 Animal growth regulators
01/11/2000US6013626 To inhibit the proliferation of mammalian cells; antitumor agents