Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
09/2000
09/21/2000WO2000055120A1 Amide derivatives
09/21/2000CA2367348A1 Novel compounds and compositions as protease inhibitors
09/21/2000CA2361819A1 Amide derivatives
09/20/2000EP1036059A1 Adamantane derivatives
09/20/2000EP1036058A1 Adamantane derivatives
09/20/2000EP1035772A1 Fungicidal compositions and methods, and compounds and methods for the preparation thereof
09/20/2000EP0932658B1 Asymmetrical imide bleach activators and compositions employing the same
09/20/2000CN1056602C Esters and amides as PLAZ inhibitors
09/19/2000US6121487 Method of producing amino acids and amino-acid derivatives
09/19/2000US6121482 Amphiphilic compounds with at least two hydrophilic and at least two hydrophobic groups based on dicarboxamides
09/19/2000US6121418 PNA synthesis using a base-labile amino protecting group
09/14/2000WO2000053583A1 Inhibitors of protein tyrosine phosphatase
09/14/2000WO2000053172A1 Ccr-3 receptor antagonists
09/14/2000WO1999063999A8 H1-histamine receptor antagonists
09/14/2000CA2366308A1 Inhibitors of protein tyrosine phosphatase
09/13/2000EP1035110A1 Benzylaminodiacetamide derivatives, compositions containing the same, process for their preparation and uses
09/13/2000EP1034783A1 Amide derivatives
09/13/2000EP1033910A1 Dipeptide apoptosis inhibitors and the use thereof
09/13/2000EP0871611B1 New derivatives of glycylanilides, preparation and therapeutical application
09/13/2000EP0839056A4 Process for producing ioversol
09/13/2000CN1266426A Microbicidal N-sulfonylglycin alkynyloxyphenemethyl amide derivatives
09/12/2000US6118010 Catalytic reduction of the 1-alkoxycarbonyl-3-oxo-3-phenylpropyl derivative
09/12/2000US6117841 Used to treat stroke, cerebral ischemia, pain, head trauma or epilepsy
09/08/2000WO2000052019A2 Crystallization products of neotame and methods for producing same
09/08/2000WO2000051973A1 Cyclobutene-3,4-dione derivatives, preparation method and therapeutic use
09/08/2000WO2000051972A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy
09/08/2000CA2365032A1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy
09/07/2000DE19910396A1 New anthranilic acid amide and isatoic acid derivatives useful in treatment of angiogenic disorders, e.g. tumors, psoriasis, arthritis and arteriosclerosis, and for prevention of vascular reocclusion
09/06/2000EP1033366A2 Amide derivatives useful as Neuropeptide Y (NPY) antagonists
09/06/2000EP1032377A1 Substituted 2-aminoacetamides and the use thereof
09/06/2000CN1265642A Aryloxyaniline derivatives
09/05/2000US6114391 α-amino acid amides, preparation thereof and the therapeutical use thereof
09/05/2000US6114381 To control brain damage associated with anoxia or ischemia which typically follows stroke, cardiac arrest or perinatal asphyxia; compound is an antagonist to inhibit excitotoxic actions at excitatory amino acid receptor sites
09/05/2000US6114325 1,2-di-substituted benzene-carboxamide derivative, hair growth promoter and external composition for skin using the same
09/05/2000CA2020340C Enantioselective synthesis of antifolates
08/2000
08/31/2000WO2000050623A2 Method for preparing optically active 3,3,3-trifluoromethyl-2-alkyl propionic acid derivatives
08/31/2000WO2000050385A1 Process for the preparation of iopamidol
08/31/2000WO2000040558A8 Aspartic protease inhibitors
08/30/2000EP1030853A1 Novel signal transduction inhibitors, compositions containing them
08/29/2000US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor
08/24/2000WO2000048993A1 Arylaminoalkylamides
08/24/2000WO2000048989A1 Mevinolin derivatives
08/24/2000WO2000048623A1 Novel amide derivatives as growth hormone secretagogues
08/24/2000CA2362290A1 Novel amide derivatives as growth hormone secretagogues
08/23/2000EP0861228B1 Lipopolyamines as transfection agents and pharmaceutical uses thereof
08/23/2000EP0828705B1 Iodination process
08/23/2000EP0821668B1 Derivatives of succinamide and their use as metalloproteinase inhibitor
08/22/2000US6107410 A photosensitive crosslinked cinnamic acid-spacer-poly-saccharide forming a cyclobutane ring when dimerized; medical material having biocompatibility, bioresorptivity and solubility; films, gels and powders
08/17/2000WO2000047549A1 Preparation of iodixanol
08/17/2000WO2000047548A1 Improved compounds for protein binding
08/17/2000WO2000027819A3 Antrhranilic acid amides and the use thereof as medicaments
08/17/2000WO2000018823A3 Peg-based macromonomers, chemically inert polymers prepared therefrom and the use of these polymers for organic synthesis and enzyme reactions
08/17/2000CA2341348A1 Improved compounds for protein binding
08/16/2000EP1028112A1 Phenylglycinolamides linked by a hetero-atom with antiatherosclerotic agents
08/16/2000EP0703790B1 Iodinated paramagnetic chelates, and their use as contrast agents
08/15/2000US6103767 Physiologically active substances TKR1785's, process for the preparation thereof, and microbe
08/15/2000US6103720 Ketobenzamides as calpain inhibitors
08/10/2000WO2000046187A2 Antizyme modulators and their use
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/10/2000DE19904812A1 Verfahren zur Herstellung von Folsäure A process for preparing folic acid
08/10/2000CA2362259A1 Antizyme modulators and their use
08/09/2000EP1026166A1 Process for the preparation of folic acid
08/09/2000EP1026149A1 Amidocarboxylic acid derivatives
08/09/2000EP1025840A2 Oral drug compositions and methods
08/09/2000EP1025067A1 Process for the crystallisation of sterically hindered compounds
08/09/2000EP0820434B1 Phenoxyethylamine derivatives having high affinity for the 5-ht 1a receptor, preparation thereof, use thereof as drugs, and pharmaceutical compositions containing said derivatives
08/09/2000CN1262272A HIV proteinase inhibitor
08/08/2000US6100298 Mixture of drug and n-(4-(carboxypropyl)phenyl-4-phenyl-butyramide for improved oral drug delivery
08/08/2000US6099856 Increased bioavailable
08/03/2000WO2000044770A1 Substituted phenethylamine derivatives
08/03/2000WO2000006610A3 Polymer production
08/03/2000WO2000006146A9 Substituted anilide compounds and methods
08/03/2000CA2359030A1 Substituted phenethylamine derivatives
08/02/2000EP1024134A1 Aminobutanoic acid derivatives
08/02/2000EP0886634A4 Process for producing ioversol
08/02/2000CN1261894A Polyol-amino-acid compounds having anti-helicobactor pylori activity
08/01/2000US6096874 High affinity tamoxifen derivatives
08/01/2000US6096782 Administering an alanine containing peptide to the alzhiemer's patient
07/2000
07/27/2000WO2000043354A2 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4
07/27/2000WO2000043352A1 A method for the synthesis of compounds of formula 1 and derivatives thereof
07/27/2000WO2000043000A1 Proteasome inhibitors
07/27/2000WO2000023429A3 Stereoselective process for producing cryptophycins
07/27/2000WO1999066944A9 Methods for identifying novel multimeric agents that modulate receptors
07/27/2000WO1999064033A9 Phosphodiesterase-v modulator drugs and their uses
07/27/2000WO1999063994A9 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE
07/27/2000WO1999057098A3 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
07/27/2000CA2359561A1 Proteasome inhibitors
07/27/2000CA2359076A1 A method for the synthesis of compounds of formula 1 and derivatives thereof
07/27/2000CA2357781A1 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4
07/26/2000EP1021407A1 Synthesis of clasto-lactacystin beta-lactone and analogs thereof
07/26/2000EP1021169A1 Active agent transport systems
07/26/2000EP1021099A1 Anti-bacterial amine derivatives
07/25/2000CA2205285C Benzoic acid derivative and pharmaceutical composition
07/20/2000WO2000042010A1 Contrast media for angiography
07/20/2000WO1999064048A9 Inhibitors of hiv reverse transcriptase
07/20/2000CA2360560A1 Contrast media for angiography
07/19/2000EP1020431A1 Method of purifying and recovering sweetener
07/19/2000EP1020429A1 Sphingosine derivatives and medicinal composition
07/19/2000EP1019365A1 Novel compositions for the delivery of negatively charged molecules
07/19/2000EP1019364A2 Inhibitors of protein tyrosine phosphatase