Patents for C07B 53 - Asymmetric syntheses (6,231)
01/1995
01/10/1995US5380927 Process for preparing optically active 2-aryl-alkanoic acids, in particular 2-aryl-propionic acids
01/10/1995US5380755 Alkyl and alkylbenzyl ethers of substituted hydroquinones
01/04/1995EP0423300B1 Chiral reaction medium for organic reactions
12/1994
12/28/1994CN1096782A Process for preparation benzothiazepine derivatives
12/22/1994WO1994029253A1 Method for preparing difunctional compounds having high enantiomeric purity
12/22/1994CA2164724A1 Process for preparing difunctional compounds having high enantiomeric purity
12/20/1994US5374727 Asymmetric hydrogenation of dihydro-pyrido [1,2-a]indoles
12/14/1994EP0628534A1 Process for the stereospecific synthesis of leucotriene B4 having configuration 6Z, 8E, 10E and intermediate products
12/07/1994EP0626967A1 Process for preparing enantiomerically pure fluorinated epoxychromans
12/06/1994US5371256 With rhodium and iridium
11/1994
11/30/1994CN1026785C Process for the preparation of clausenamide and neoclausenamide, and of their derivatives
11/24/1994WO1994026751A1 Enantioselective oxazaborolidine catalysts
11/24/1994WO1994026708A1 Optically active 3-(1-(alkylamino))alkyl pyrrolidines
11/24/1994CA2160124A1 Optically active 3-(1-(alkylamino)) alkyl pyrrolidines
11/23/1994EP0625523A1 Cis-oxalato(trans-L-1,2-cyclohexanediamine) Pt(II) complex having high optical purity and process of preparing same
11/17/1994EP0624587A2 Assymetric hydrogenation of furolimidazol derivatives
11/17/1994EP0624152A1 Process for preparing ketone enantiomer.
11/15/1994CA2122511A1 Asymmetric hydrogenation of furoimidazole derivatives
11/08/1994US5362886 Asymmetric synthesis
11/08/1994US5362757 Administering for treatment of cardiovascular disorders while reducing side effects
11/01/1994US5360938 Asymmetric syntheses
10/1994
10/27/1994WO1994024104A1 Improvements in or relating to chiral auxiliaries
10/18/1994US5357001 Optically active amino acid sulphoxide and amino acid sulphone derivatives, their preparation, their polymerisation and use as adsorbents for chromatographic resolution of racemates
10/05/1994EP0618197A1 Synthesis of CIS-decahydroisoquinoline-3-carboxylic acids
10/05/1994EP0618196A1 Stereocontrolled synthesis of cis-bicyclic compounds
10/04/1994US5352832 Asymmetric process for preparing florfenicol, thiamphenicol chloramphenicol and oxazoline intermediates
10/01/1994CA2119732A1 Stereocontrolled synthesis of cis-bicyclic compounds
10/01/1994CA2119730A1 Synthesis of cis-decahydroisoquinoline-3-carboxylic acids
09/1994
09/28/1994EP0617028A1 Enantiomers of 1-(4-chlorophenyl)phenylmethyl)-4-(4-methylphenyl)sulfonyl piperazine
09/20/1994US5348870 Using hydrolase to effect ester interchange and resolution, then alcoholysis or hydrolysis and dehydration with cyclization and crystallization
09/15/1994WO1994020483A1 Process to derivatives of piperizinylcamphorsulfonyl oxytocin antagonists
09/14/1994EP0614902A1 Phosphine compounds and transition metal-phosphine complexes containing them as ligands
09/14/1994EP0614901A1 Phosphine compound and transition metal-phosphine complex containing the same as ligand
09/14/1994EP0614895A1 Bis-dihydropyran derivatives and their use in chiral transformations
09/14/1994EP0614894A1 Process for the synthesis of substituted amide derivatives of piperazinylcamphorsulfonyl oxytocin antagonists
09/14/1994EP0614871A1 Process for producing optically active beta-hydroxyketone
09/14/1994EP0614870A2 Process for producing optically active aldehydes
09/13/1994CA2118756A1 Process for the synthesis of substituted amide derivatives of piperizinylcamphorsulfonyl oxytocin antagonists
08/1994
08/31/1994EP0612716A1 Process for the preparation of an optically pure aminoalcohol
08/16/1994US5338851 Synthesis of cis-decahydroisoquinoline-3-carboxylic acids
08/04/1994WO1994017079A1 OPTICALLY ACTIVE β-AMINOALKOXYBORANE COMPLEX
08/04/1994CA2153695A1 Optically active .beta.-aminoalkoxyborane complex
08/03/1994EP0609031A1 Process for preparing benzothiazepine derivatives
08/03/1994EP0609025A1 Process for producing optically active epoxy alcohol derivatives
08/03/1994EP0608307A1 New ligands for asymmetric dihydroxylation: multiple cinchona alkaloid units attached to a central heterocyclic core
08/02/1994CA1331197C Enantiomeric glutaramide diuretic agents
07/1994
07/28/1994CA2114036A1 Process for preparing benzothiazepine derivatives
07/20/1994CN1089614A Alpha-phosphonosulfonate squalene synthetase inhibitors and method
07/12/1994US5329015 Chiral phospholanes via chiral 1,4-diol cyclic sulfates
07/07/1994WO1994014835A1 Use of molecularly imprinted polymers for stereo- and/or regioselective synthesis
07/07/1994WO1994014802A1 Process for preparing substituted 1,3-oxathiolanes with antiviral properties
07/07/1994WO1994014764A1 Asymmetric process for preparing florfenicol, thiamphenicol, chloramphenicol and oxazoline intermediates
07/07/1994CA2152627A1 Use of molecularly imprinted polymers for stereo- and/or regioselective synthesis
07/06/1994EP0604857A1 Process for preparing optically active 4-mercapto-2-pyrrolidone derivative and intermediate therefor
06/1994
06/29/1994EP0603414A1 (-)-ritodrine
06/08/1994EP0600020A1 Asymmetric syntheses.
05/1994
05/25/1994CN1087079A (-)-Ritodrine
05/17/1994US5312957 Enantioselective hydrocyanation of aromatic vinyl compounds
05/17/1994US5312939 2,2'-bis (dicyclopentylphosphino)-1,1'-binaphthyl and transition metal complex using the same as ligand
05/11/1994EP0595868A1 Process for the preparation of intermediates in the synthesis of chiral thiazolidine-2,4-dione derivatives
05/10/1994US5310956 Optically active epoxides and a process for the production thereof
05/04/1994EP0595635A1 Alpha-phosphorous substituted sulfonate derivatives as squalene synthetase inhibitors
05/04/1994EP0594608A1 Chiral catalysts for enantioselective synthesis.
05/03/1994US5308820 Of an amino acid amide derivative and a titanium alkoxide
05/03/1994US5308819 Diphosphines containing silane groups, immobilised diphosphines and the use thereof as hydrogenation catalysts
05/03/1994CA1329214C 2-hydroxy-3-(4-methoxyphenyl)-3-(2- aminophenylthio)propionic acid, 8'-phenylmenthyl ester, especially for diltiazem
04/1994
04/29/1994CA2107644A1 .alpha.-phosphonosulfonae squalene synthetase inhibitors and methd
04/28/1994WO1994008983A1 Amide derivatives
04/27/1994EP0593917A1 Process for the preparation of optically active esters and thioesters
04/26/1994US5306834 Process for preparing optically active 4-methyl-2-oxetanone
04/26/1994US5306820 Process for the preparation of enantiomerically pure substituted (quinolin-2-yl-methoxy)phenylacetic acids
04/20/1994EP0592552A1 Chiral phospholanes via chiral 1,4-diol cyclic sulfates.
04/14/1994WO1994007850A1 Process for the stereoselective synthesis of 3-substituted 2-sulphonyl methyl propionic acids and intermediate products
04/14/1994WO1994007849A1 Process for the stereoselective synthesis of 3-substituted 2-thiomethyl propionic acids
04/14/1994CA2146144A1 Process for the stereoselective synthesis of 3-substituted 2-thiomethylpropionic acids
04/14/1994CA2146142A1 Process for the stereoselective synthesis of 3-substituted 2-sulfonylmethylpropionic acids, and intermediate products
04/07/1994DE4233100A1 Verfahren zur stereoselektiven Synthese von 3-substituierten 2-Sulfonylmethylpropionsäuren sowie Zwischenprodukte Method for the stereoselective synthesis of 3-substituted 2-Sulfonylmethylpropionsäuren and intermediates
04/07/1994DE4233099A1 Verfahren zur stereoselektiven Synthese von 3-substituierten 2-Thiomethylpropionsäuren Method for the stereoselective synthesis of 3-substituted 2-Thiomethylpropionsäuren
04/05/1994US5300638 Reacting imine derivative of threonine with an acetyl halide in the presence of a base; preferential
03/1994
03/31/1994WO1994006792A1 Optically active hydroquinine (amino-3 phenyl)-1 ethanesulfonate, preparation and use thereof
03/31/1994CA2144158A1 Optically active hydroquinine 1-(3-aminophenyl)ethanesulfonate; preparation thereof and its use
03/29/1994US5298660 Compound containing an assymetrical carbon atom
03/22/1994US5296595 Metal complexes with bridging ligands
03/16/1994EP0587471A1 Use of carbohydrates in the solid state as chiral supports for chemical reactions
03/15/1994CA1327804C Process for the minimization of racemization in the preparation of optically active ((aryloxy)phenoxy)proprionates herbicides
03/08/1994US5292946 In-situ preparation of diisopinocamphenyl chloroborane
03/08/1994US5292893 Catalytic asymmetric and non-asymmetric reduction of times and oximes using metal catalysts
03/08/1994CA1327593C Enantioselective process and intermediates for preparing trans or cis hemicaronic aldehyde derivatives
03/03/1994WO1994004486A1 Chemical process for preparing an optically active aminodiol
02/1994
02/23/1994EP0583433A1 Diphosphine ligands
02/17/1994WO1994003271A1 Chiral catalysts and epoxidation reactions catalyzed thereby
02/17/1994CA2141790A1 Chiral catalysts and epoxidation reactions catalyzed thereby
02/16/1994EP0583171A2 (3R,5S)-3,5,6-trihydroxyhexanoic acid derivatives and methods for their production
02/16/1994EP0582692A1 Diphosphine ligands
02/15/1994US5286883 (3R,5S)-3,5,6-trihydroxyhexanoic acid derivative and production method thereof
02/09/1994EP0581777A1 Stereoselective preparation of substituted piperidines
01/1994
01/26/1994EP0580336A1 Process for preparing optically active 4-methyl-2-oxetanone
01/26/1994EP0580210A1 Process for the preparation of optically active methionine amide
01/26/1994EP0579797A1 Diphosphine ligands
01/25/1994US5281750 Chiral polymers for the production of excess enantiomers
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