Patents
Patents for C07D 501 - Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula: , e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (7,574)
07/2005
07/27/2005EP1556389A1 Cephem compounds
07/27/2005EP1556388A2 A method for manufacture of ceftiofur
07/27/2005CN1644583A Cephe alkene onium salt compound and its preparation and use in preparation of cefepime
07/27/2005CN1212327C Preparation of N-protected-3-pyrrolidine-lactam substituted phosphonium salts
07/27/2005CN1212324C Method for preparing crystalline cefathiamidine and its usage
07/20/2005EP1554289A1 A cefdinir intermediate
07/20/2005EP1554288A1 Process for the preparation of (z)-isomer enriched 7-amino-3-propen-1-yl-3-cephem-4- carboxylic acid
07/20/2005CN1640879A One-step method for preparing high-purity cefpoxime proxetil
07/20/2005CN1640878A Method for preparing cefathiamidide
07/19/2005US6919449 Process for the preparation of cephalosporin intermediate and its use for the manufacture of cephalosporin compounds
07/14/2005WO2005063772A1 Process for production of intermediates for use in cefalosporin synthesis
07/14/2005WO2005044824A3 Processes for the preparation of highly pure 3-(2-substituted vinyl) cephalosporin
07/14/2005US20050153950 Broad -spectrum cephem compounds
07/13/2005CN1639169A An improved synthesis of ceftiofur intermediate
07/13/2005CN1637002A Cephalosporin ester compound resisting beta-lactamase and its salt
07/13/2005CN1637001A Process of preparing amorphous cefuroxin axetil
07/12/2005US6916801 Bactericides, antibiotic
07/06/2005CN1634933A Process for preparing ceftriaxone sodium
07/06/2005CN1634932A Process for preparing cefotaxime sodium
07/06/2005CN1634931A Cefuroxime axetil diastereoisomer separating method
07/06/2005CN1634930A Cephalosporins medicine intermediate crystal and method for preparing same
07/06/2005CN1209364C Amine salt of cefathiamiding, its preparing method and application
06/2005
06/29/2005EP1546155A2 Intermediate cefdinir salts
06/29/2005EP1546154A1 Process for the preparation of cefdinir
06/29/2005EP1546096A1 Process for the preparation of amino-pyrrolidine derivatives
06/23/2005US20050137182 Novel crystalline form of cefdinir
06/22/2005EP1544197A1 Intermediates for cephem compounds
06/21/2005US6908996 Compounds and method for preparing 3-methylcephams
06/15/2005EP1228074B1 Method of preparing highly pure cefpodoxime proxetil
06/15/2005EP1222194B1 7-acylamino-3-heteroarylthio-3-cephem carboxylic acid antibiotics and prodrugs thereof
06/15/2005CN1628118A Process for prepn. of cefdinir
06/15/2005CN1628108A Process for the preparation of 4-methyl-thiazole-5-carbaldehyde intermediate
06/15/2005CN1626566A Process for the removal of porogens from temperature sensitive macroreticular polymers using steam at reduced pressure
06/15/2005CN1206231C 7-acylamino-3-heteroarylthio-3-cephem carboxylic and prodrugs thereof
06/14/2005US6906187 Manufacture of cefalosporins and intermediates
06/14/2005US6906055 Bactericides; antibiotiucs; dissolving in water, crystallization; Ceftaroline fosamil acetate
06/14/2005US6906054 Alkylidene or dialkylidene cephalosporin-type derivatives
06/09/2005WO2005051959A1 Β-lactamase-resistant cephalosporin ester compounds and salts of thereof
06/09/2005WO2004062558A3 Process for enzymatic synthesis of βετα-lactam antibiotics
06/07/2005US6903211 Reacting a 3-cephem-4-protected carboxy derivative with acetaldehyde to produce an intermediate, deesterifying the carboxy protecting group using an acid, forming salt with a base, neutralizing, silylating, condensing with an anhydride
06/02/2005WO2004098500A3 CARBACEPHEM ss-LACTAM ANTIBIOTICS
06/02/2005US20050119478 Reacting a benzathenium salt with thiourea
06/02/2005US20050119244 Process for preparing cephalosporins with salified intermediate
06/02/2005US20050118669 Reporter genes; fluorescence activated cell sorting
05/2005
05/26/2005WO2005003367A3 Process for the preparation of cephradine
05/26/2005US20050113570 Process for preparation of 7-[alpha-amino (4-hydroxyphenyl) acetamido]-3-substituted-3-cephem-4-carboxylic acid
05/26/2005US20050113355 Suspending cefdinir in pyridine; salt formation
05/26/2005CA2534342A1 Amino acid prodrugs
05/25/2005CN1620460A Crystalline hydrochloride of 7-(((5-amino-1, 2, 4-thiadiazol-3-yl)(fluoromethoxyimino) acetyl) amino) -3- ((imino-1-piperazinylmethyl)methylhydrazono)-methyl-3-cephem-4-carboxylic acid
05/25/2005CN1203075C Prepn of cefotaxime
05/24/2005US6897304 Cephem compounds and ESBL-detecting reagents containing the same
05/19/2005WO2005044824A2 Processes for the preparation of highly pure 3-(2-substituted vinyl) cephalosporin
05/19/2005US20050107581 Steam stripping beads under vacuum; divinyl benzene/ethyl vinyl benzene copolymers; dilution; for production of cephalosporin C and insulin
05/18/2005EP1531168A1 Process for the removal of porogens from temperature sensitive macroreticular polymers using steam at reduced pressure
05/18/2005CN1617875A Crystalline cefdinir potassium dihydrate
05/17/2005US6894162 Intermediates in cephalosporin production
05/17/2005CA2486752A1 Process for the removal of porogens from temperature sensitive macroreticular polymers using steam at reduced pressure
05/12/2005WO2005042544A1 Processes for the preparation of cephalosporin derivatives
05/12/2005WO2005042543A1 Processes for the preparation of cephem derivatives
05/11/2005EP1529050A1 Cephalosporins
05/11/2005CN1613860A Cephaene onium salt compound and its preparation, and synthesis of cephapyrazde sulfate therefrom
05/11/2005CN1200941C Intermediates in cephalosporing production, intermediate and its use therein
05/06/2005WO2005040175A2 Process for the preparation of cephem carboxylic acids
05/06/2005WO2005020904A3 Oral neurotherapeutic cefazolin compositions
05/05/2005US20050096306 Such as 7-[-2-(5-amino-1,2,4-thiadiazol-3-yl)-2-(1-carboxy-1-methylethoxyimino)acetamido]-3-[3-amino-4-(3-aminopropyl)-2-methyl-1-pyrazolio]methyl-3-cephem-4-carboxylate; antimicrobial agents; synthesis
05/03/2005US6887992 Clathrate compound comprising p-methoxybenzyl ester of 7-phenylacetamide-3-formyl-3-cephem-4-carboxylic acid and dimethylformamide; intermediate or final product of pharmaceuticals such as cefixime, ceftibuten and cefdinir
05/03/2005CA2158999C Crystalline benzathine salt of cefonicid and its preparation
04/2005
04/27/2005EP1463734B1 An improved synthesis of ceftiofur intermediate
04/27/2005CN1198833C Vinyl pyrrolidone cephlosporins with basic substitutent group
04/21/2005WO2005034957A1 Noncrystalline antibacterial composition containing cefditoren pivoxil
04/21/2005WO2005003141B1 An improved process for the preparation of cefditoren
04/20/2005CN1608070A Process for the stabilization of an acidic aqueous phase comprising cephradine
04/19/2005CA2096709C Process for the cleavage of cephalosporin prodrug esters to 7-amino-3-methoxymethylceph-3-em-4-carboxylic acid
04/14/2005US20050080255 Reacting cefdinir with potassium compound; salt formation; crystallization from solvent
04/14/2005US20050080070 Process for the preparation of cephalosporin antibiotic
04/13/2005EP1134222B1 IMIDAZO[4,5-b]PYRIDINIUMMETHYL-CONTAINING CEPHEM COMPOUNDS HAVING BROAD ANTIBACTERIAL SPECTRUM
04/13/2005CN1606558A Novel cephalosporin compounds and process for preparing the same
04/13/2005CN1606463A Methods of treating bacterial infections in dogs and cats
04/13/2005CN1196686C Method for storing quaternary ammonium salt
04/06/2005CN1603327A New process for the preparation of vinyl pyrrolidinone cephalosporine derivatives
04/06/2005CN1603326A Cefathiamidine mixed salt and process for preparing same
04/06/2005CN1195761C Cephalosporin Intermediates
03/2005
03/31/2005WO2005027909A1 Cephem compounds
03/31/2005US20050070722 Chemical intermediate for cephalosporin bactericides
03/31/2005US20050070705 Cyclization of the corresponding tertiary amide azetidine compound
03/31/2005CA2536636A1 Cephem compounds
03/30/2005EP1289998B1 New process for the preparation of vinyl-pyrrolidinone cephalosporine derivatives
03/30/2005CN1600785A Method for preparing unformed cefuroxime axetil
03/30/2005CN1194980C Phosphonocephem derivatives, process for preparation of same, and use thereof
03/29/2005US6872836 Converting a protected 1,4- dihydroxy-2-amino or protected amino butane in presence of hydroxylamine or an acid additon salt into N-hydroxy-pyrrolidone derivative, reducting N-hydroxy group to secondary amine by hydrogenation
03/24/2005WO2005026176A1 Process for producing 3-chloromethyl-3-cephem derivative
03/23/2005CN1597684A Sodium ceftriaxone and its preparation method
03/17/2005US20050059821 Method for manufacture of ceftriaxone sodium
03/17/2005US20050059820 Method for manufacture of ceftriaxone sodium
03/17/2005US20050059819 Cefdinir pyridine salt
03/17/2005US20050059818 Crystal structure; suspension in ethanol, acetonitrile, formamide, triethylamine, toluene, ethyl acetate, tetrahydrofuran, methylene chloride, hexane, acetone, methyl ethyl ketone, dimethyl sulfoxide, pyridine, and/or nitromethane solvent
03/16/2005CN1594324A Process for preparing cefpiramide sodium
03/16/2005CN1594323A Amorphous cephalosporin
03/16/2005CN1594322A Cefixime sodium pharmaceutical composition and its preparation and application
03/16/2005CN1594321A Process for preparing cephazoline three-position intermediate
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