Patents
Patents for C07D 501 - Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula: , e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (7,574)
02/2006
02/23/2006WO2006018807A1 Crystalline forms of cefdinir
02/23/2006US20060040915 Process for the preparation of cefdinir
02/22/2006EP1392704B1 Cephem compounds
02/15/2006EP0537255B1 Process for preparation of beta-lactams
02/15/2006CN1241928C Crystal of 7-phenylacetyl amido-3-picolyl-3-cephalosporin-4-carboxylic p-methoxy benzyl ester crystal and preparation method
02/09/2006US20060029674 Stable amorphous Cefdinir
02/08/2006EP0831869B1 Diphosphonate derivatives of therapeutic agents
02/02/2006US20060025586 Crystalline salt of phosphate, mesylate, tosylate, sulfate, hydrogen sulfate; chemical intermediate for producing pure cephalosporin with antibacterial properties; chemical synthesis, salt formation, crystallization, isolation
02/02/2006US20060025399 Crystalline anhydrous cefdinir and crystalline cefdinir hydrates
02/02/2006US20060025327 Hybrid molecules QA, wherein Q is an aminoquinoline and a is an antibiotic or a resistance enzyme inhibitor, their synthesis and their uses as antibacterial agent
02/01/2006CN1727347A Methylene containing aminobeterocycle substitutional cephalosporin of amidinothioacetamide, preparation method and application
02/01/2006CN1727346A Derivant of gamma carbon alkenyl cephalosporin, preparing method and application
02/01/2006CN1727345A Derivant of Deacetoxy cephalosporanicacid, preparation and application
02/01/2006CN1727344A Derivant of cephalosporin of amidinothioacetamide, preparation method and application
01/2006
01/26/2006WO2006008161A1 Alkanoyl amide solvates of 2-(2-aminothiazole-4-yl)-2-(acyloxyimino)acetic acid
01/26/2006US20060020130 Spraying a cefuroxime axetil solution via an atomizer into a stirred reactor containing an antisolvent to precipitate and crystallize the cefuroxime axetil into a slurry via antisolvent recrystallization; filtering and drying to obtain amorphous cefuroxime axetil powder; particle size of 20nm-30mu m.
01/25/2006EP1619198A1 Amorphous cefuroxime axetil and preparation process therefore
01/25/2006EP1618114A2 Processes for the preparations of cefepime
01/25/2006EP1618106A2 Carbacephem -lactam antibiotics
01/19/2006US20060014230 Beta-lactamase detecting reagent composition, detection kit and detection method
01/12/2006US20060009639 Process for the preparation of cefpodoxime proxetil
01/11/2006CN1235902C Crystalline acid salts of cefdinir and process for preparing cefdinir using same
12/2005
12/28/2005EP1609793A1 Novel crystal of 7- 2-(2-aminothiazole-4-yl)-2-hydroxyiminoa cetamido-3-vinyl-3-cephem-4-carboxylic acid (syn isomer) and method for preparation thereof
12/28/2005EP1608661A2 Process for the preparaton of 7-(p-hydroxyphenylglycylamido)cephem compounds
12/28/2005EP1434779B1 Cross-linked glycopeptide-cephalosporin antibiotics
12/28/2005EP1178043B1 Method for storing quaternary ammonium salt
12/22/2005WO2005121154A1 Process for the preparation of cefdinir
12/21/2005EP1606293A1 Cephalosporin in crystalline form
12/21/2005CN1711271A Process for the preparation of (Z)-isomer enriched 7-amino-3-propen-1-yl-3-cephem-4-carboxylic acid
12/15/2005WO2005118596A1 3-alkenylcephem compounds and process for production thereof
12/15/2005WO2005118595A1 Process for production of 3-alkenylcephem compounds
12/15/2005WO2005071096A3 Derivatives of cephalosporin and clavulanic acid for detecting beta-lacamase in a sample
12/14/2005CN1708502A Cephem compounds
12/14/2005CN1708501A An improved process for the preparation of chloro methyl cephem derivatives
12/13/2005US6974797 Bactericides for drug resistant bacteria
12/01/2005WO2005112648A1 Sulphur-containing oils for controlling plant pathogens and stimulating nutrient uptake
12/01/2005WO2005076694A3 Improved process for the production of cefotaxime sodium
12/01/2005US20050267092 Novel cephalosporin compounds and process for preparing the same
12/01/2005CA2562915A1 Sulphur-containing oils for controlling plant pathogens and stimulating nutrient uptake
11/2005
11/24/2005WO2005094800A3 A co-precipitated cefepime composition and process for preparation thereof
11/16/2005CN1697837A Method for crystallization of 7-aminocephalosporanic acid
11/16/2005CN1696134A Method for preparing cefixime
11/10/2005WO2005105813A1 Improved process for the manufacture of ceftriaxone sodium
11/09/2005CN1694888A Process for the preparation of 3-propenyl cephalosporin DMF solvate
11/03/2005US20050245738 Stable bioavailable crystalline form or cefdinir and a process for the preparation thereof
11/03/2005US20050245498 Sterically-awkward beta-lactamase inhibitors
11/02/2005EP1590354A2 Carboxylic acid esters of pharmaceutical compounds
11/02/2005EP1590353A1 A process for the preparation of cefpodoxime proxetil
11/02/2005EP1311518B1 Preparation of n-protected-3-pyrrolidine-lactam substituted phosphonium salts
11/02/2005CN1225468C Cephem compounds and ESBL detecting reagents containing same
10/2005
10/27/2005WO2005100369A1 Depletion of e-isomers in preparation of z-enriched 3-(2-substituted vinyl) cephalosporins
10/27/2005WO2005100368A2 Stable amorphous cefdinir
10/27/2005WO2005100367A1 Intermediates useful in the synthesis of 3-(2-substituted vinyl) cephalosporins
10/27/2005WO2005100330A1 Preparation of intermediate for 3-[2-(4-methylthiazole-5-yl)vinyl] cephalosporins
10/27/2005US20050239691 Cross-linked glycopeptide - cephalosporin antibiotics
10/27/2005CA2562083A1 Stable amorphous cefdinir
10/26/2005EP1045852B1 Process for the preparation of cefpodoxim proxetil diastereoisomers
10/26/2005CN1687076A Compound of dual functional esterified prodrug of Cefetamet, and oral preparation
10/20/2005US20050234233 Cephalosporins
10/13/2005WO2005094800A2 A co-precipitated cefepime composition and process for preparation thereof
10/13/2005US20050227309 Optically-detectable enzyme substrates and their method of use
10/12/2005EP1583764A1 A process for the manufacture of cefpodoxime proxetil
10/12/2005CN1679595A Phosphonocephem derivatives, their production and use
10/12/2005CN1222508C Process for preparation of condensed sulfamide
10/06/2005WO2005092900A1 PROCESS FOR PREPARING CEPHALOSPORIN INTERMEDIATES USING α-IODO-1-AZETIDINEACETIC ACID ESTERS AND TRIALKYLPHOSPHITES
10/06/2005CA2557798A1 Process for preparing cephalosporin intermediates using alpha-iodo-1-azetidineacetic acid esters and trialkylphosphites
10/05/2005CN1678616A Cephalosporins
09/2005
09/29/2005WO2005090361A1 Trihemihydrate, anhydrate and hydrate forms of cefdinir
09/29/2005WO2005090360A1 Novel polymorph of cefdinir
09/29/2005US20050215782 Process for preparing crystalline 3-chloromethyl-3-cephem derivatives
09/29/2005US20050215781 Novel polymorph of cefdinir
09/29/2005CA2558629A1 Trihemihydrate, anhydrate and hydrate forms of cefdinir
09/28/2005CN1220693C Process for preparation of 3-sulfonyloxy-3-cephem compounds
09/27/2005US6949641 Crystalline β-lactam intermediate
09/27/2005US6949521 Therapeutic azide compounds
09/22/2005US20050209451 Crystalline form of cefdinir
09/22/2005US20050209450 High yield for industrial production; beta -lactam antibacterial agents; allyl (5R,6S)-6((R)-1-t-butyldimethyl-silyloxyethyl)-7-oxo-3-((R)-2-tetrahydrofuryl)-4-thia-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylate (3-2)
09/22/2005US20050209211 Trihemihydrate, anhydrate and novel hydrate forms of Cefdinir
09/21/2005EP1575913A1 Novel intermediates for synthesis of cephalosporins and process for preparation of such intermediates
09/21/2005CN1671658A Process for the manufacture of amino-pyrrolidine derivatives
09/15/2005WO2005085258A1 3-pyridinium methylcephem compound
09/15/2005CA2557988A1 3-pyridinium methylcephem compound
09/14/2005EP1572699A1 Crystalline cefdinir salts
08/2005
08/31/2005EP1458727B1 Process for the stabilization of an acidic aqueous phase comprising cephradine
08/31/2005EP1382608B1 Sulfate of cephem compound
08/31/2005EP1365764B1 Oral pharmaceutical composition of cefpodoxime proxetil
08/25/2005WO2005076694A2 Improved process for the production of cefotaxime sodium
08/24/2005EP1565192A2 Method and compositions for temporarily incapaciting subjets
08/24/2005EP1565178A2 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
08/18/2005US20050181469 Beta-lactamase substrates having phenolic ethers
08/17/2005EP1562957A1 Process for the preparation of 3-propenyl cephalosporin dmf solvate
08/17/2005CN1656046A Process for producing cyclic compound
08/11/2005WO2005016936A3 Process for selective preparation of z-isomer of cefditoren and pharmaceutically acceptable salts and esters thereof
08/11/2005US20050176697 crystal of 3-[4-(1-methyl-4-pyridinio)-2-thiazolylthio]-7 beta -[2-(5-phosphonoamino-1,2,4-thiadiazol-3-yl)-2(Z)-ethoxyiminoacetamido]-3-cephem-4-carboxylate with acetic acid and water, crystals; anti-Methicillin Resistant Staphylococcus aureus agent; storage stability, high purity
08/10/2005CN1653072A Broad -spectrum cephem compounds
08/04/2005WO2005071096A2 Derivatives of cephalosporin and clavulanic acid for detecting beta-lacamase in a sample
08/03/2005CN1213144C Recombination nucleic acid molecule and application thereof
07/2005
07/28/2005WO2005040175A3 Process for the preparation of cephem carboxylic acids
07/28/2005US20050165229 Cyclization cepham derivative; 1,4-dihydroxylbut-1-yl side chain is cyclized to form cyclic ether, such as tetrahydrofuranyl system; acid catalyst
07/27/2005EP1556500A1 Simple enzymatic process for preparing cefazolin
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