Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
01/2004
01/14/2004CN1468247A Ethers of 7-desmethylrapamycin
01/14/2004CN1468246A Hydroxyesters of 7-desmethylrapamycin
01/14/2004CN1468245A New process for the production of oxabispidines
01/14/2004CN1468244A New oxabispidine compound useful in the treatment of cardiac arrhythmias
01/14/2004CN1468242A Azabicyclic compounds, preparation thereof and use as medicines, in particular as antibacterial agents
01/14/2004CN1468241A Heterocyclic compounds as ligands of the gabaa receptor
01/14/2004CN1468112A The use of 5ht4 receptor antagonists in the prophylaxis or treatment of certain cardiovascular conditions
01/13/2004US6677334 Oxazolo, thiazolo and selenazolo [4,5-c]-quinolin-4-amines and analogs thereof
01/13/2004US6677309 Anthracycline derivatives
01/08/2004WO2004002992A1 Compounds
01/08/2004WO2004002491A1 Morpholine and tetrahydropyran drivatives and their use as cathepsin inhibitors
01/08/2004WO2004002490A2 Piperidine compounds as antibacterials
01/08/2004WO2003076445A3 Microtubule stabilizing compounds
01/08/2004WO2003055856A3 BICYCLIC LACTAM DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-α CONVERTING ENZYME (TACE)
01/08/2004WO2002059124A3 Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists
01/08/2004US20040006063 Dipeptide derivatives
01/08/2004DE10226943A1 Phenylaminopyrimidine und ihre Verwendung Phenylaminopyrimidine and their use
01/08/2004CA2488525A1 Morpholine and tetrahydropyran derivatives and their use as cathepsin inhibitors
01/07/2004EP1378570A1 Flk-1 is a receptor for vascular endothelial growth factor
01/07/2004EP1377589A1 Oxazolyl-pyrazole derivatives as kinase inhibitors
01/07/2004EP1377556A1 Pyrazole derivatives for treating hiv
01/07/2004EP1289997B1 Macrolides
01/07/2004CN1466456A Sgk2 and Sgk3 used as diagnostic and therapeutic targets
01/07/2004CN1465578A Indolinospirobenzoxazine compound, and synthesis method and use thereof
01/07/2004CN1133429C Use of macrolide compounds for treatment of ARDS
01/06/2004US6673809 Tricyclic compounds as MRP1-inhibitors
01/06/2004US6673808 Pharmaceutical consisting of tacrolimus tricyclic compound, diethyl sebacate dissolution/absorption promoter, hydrophilic glycol pharmaceutical base, diethylene glycol monoethyl ether compatibilizer and cellulose or carboxyvinyl polymer thickener
01/06/2004US6673793 Oxazinoquinolones useful for the treatment of viral infections
01/06/2004US6673781 Inhibit secretory phospholipase a2-mediated fatty acid release; treating adult respiratory syndrome, pancreatitis, bronchial asthma, allergic rhinitis, chronic rheumatism, arteriosclerosis, cerebral infarction and psoriasis
01/02/2004EP1373273A1 Process for preparing maytansinol
01/02/2004EP1373224A1 New spirotricyclic derivatives and their use as phosphodiesterase-7 inhibitors
01/01/2004US20040002528 CBI analogs of CC-1065 and the duocarmycins
01/01/2004US20040002495 Lactam glycogen phosphorylase inhibitors and method of use
01/01/2004US20040002488 Fused bicyclic aromatic compounds that are useful in treating sexual dysfunction
12/2003
12/31/2003WO2004000849A2 Tetracyclic arylsulfonyl indoles having serotonin receptor affinity
12/31/2003WO2004000324A1 Pharmaceutical compositions for the treatment of diseases related to neurotrophines
12/31/2003WO2004000307A1 Novel use of ansamycin antibiotics and method of screening novel angiogenesis inhibitor
12/31/2003WO2003068980A3 Method for extracting a macrolide from biomatter
12/31/2003WO2003059269A3 Acridone inhibitors of impdh enzyme
12/31/2003CN1463975A Novel harringtonlne derivative, method for making same and its pharmaceutical composition and use thereof
12/31/2003CA2445515A1 Transcription factor modulating compounds and methods of use thereof
12/30/2003US6670507 Process for the preparation of aryloctanoyl amides
12/30/2003US6670389 Laulimalide derivatives
12/30/2003US6670373 Compounds and method for inhibiting MRP1
12/30/2003US6670364 Antagonists of MCP-1 function and methods of use thereof
12/30/2003US6670358 Substituted thioacetamides
12/30/2003US6670168 Recombinant Streptomyces hygroscopicus host cells that produce 17-desmethylrapamycin
12/30/2003CA2102241C Use of macrolide compounds for eye diseases
12/30/2003CA2099970C Composition for curing sjoegren syndrome disease
12/30/2003CA2051399C Therapeutically useful 2-aminotetralin derivatives
12/25/2003US20030236296 Novel interleukin-1beta converting enzyme inhibitors
12/25/2003US20030236291 Antitumor agents
12/25/2003US20030236265 Bactericides; autoimmune disease; antiinflammatory agents; administering a synergistic mixture of rifamycin and another antibiotic
12/25/2003US20030236245 Helix mimetics and composition and methods related thereto
12/25/2003US20030236240 Macrocycles useful in the treatment of alzheimer's disease
12/25/2003US20030236229 For stimulating the immune system, treating proliferative disorders, or microbial infections
12/25/2003US20030235614 Time release agents comprising drugs such as tacrolimus in solid solutions
12/24/2003WO2003106460A1 Novel interleukin-1 beta converting enzyme inhibitors
12/24/2003WO2003106450A1 Phenylaminopyrimidines and their use as rho-kinase inhibitors
12/24/2003WO2003106438A1 Synthesis of diazonamide "a" core
12/24/2003WO2003105868A1 Novel maxi-k channel blockers, methods of use and process for making the same
12/24/2003WO2003051299A3 Sulfhydryl rifamycins and uses thereof
12/24/2003WO2003019697A3 Organic electroluminescent device based on 2,5-diaminoterephthalic acid derivatives
12/24/2003CN1131869C 新的含三(噁唑)的细胞毒性大环内酯化合物 New cytotoxic macrolide compounds containing tris (oxazole) of
12/24/2003CA2488884A1 Novel maxi-k channel blockers, methods of use and process for making the same
12/23/2003US6667304 Affinity for melatonin receptors; sleep disorders; N-(2-(2-methoxy-6H-pyrido(2',3':4,5)pyrrolo(2,1-a)isoindol-11 -yl)ethyl)acetamide; N-(2-(3-methoxy-6,7,8,9-tetrahydropyrido (3,2-b)indolizin-5-yl) ethyl)acetamide
12/23/2003CA2233178C (methylsulfonyl)phenyl-2-(5h)-furanones as cox-2 inhibitors
12/23/2003CA2116387C Oxazolidinedione derivatives, their production and use
12/18/2003WO2003104236A1 Calcitonin gene related peptide receptor antagonists
12/18/2003WO2003104231A1 NOVEL INTERLEUKIN-1beta CONVERTING ENZYME INHIBITORS
12/18/2003WO2003082192A3 Certain pharmaceutically useful substituted aminoalkyl heterocycles
12/18/2003WO2003050064B1 Mitotic kinesin inhibitors
12/18/2003WO2002014536A9 Odulating multiple lineage kinase proteins
12/18/2003US20030232821 Oxadiazine derivatives
12/18/2003US20030232215 Organic Red Electro-Luminescent Device and Dopant
12/17/2003EP0937075B1 New Imidazo- and Oxazolopyridines as Phosphodiesterase Inhibitors.
12/17/2003CN1462269A Fused azepine drivatives and their use as antidiuretic agents
12/16/2003US6664247 Pyrazole compounds useful as protein kinase inhibitors
12/11/2003WO2003101994A1 Fused bicyclic aromatic compounds that are useful in treating sexual dysfunction
12/11/2003WO2003101956A1 Pharmaceutical combination
12/11/2003WO2003101490A1 Drug composition containing calcium channel antagonist
12/11/2003WO2003101445A1 Intravenous rifalazil formulation and methods of use thereof
12/11/2003WO2003079980A3 Caboxylic acid glycuronides, glycosamides and glycosides of quinolones, penicillins, analogs, and uses thereof
12/11/2003WO2003051300A3 Metal complexes and formulations of rifamycin analogues and uses therof
12/11/2003WO2003022807A8 Medical devices containing rapamycin analogs
12/11/2003US20030229115 Organ rejection disease; autoimmune disease; immunosuppressants
12/11/2003US20030229095 Sexual disorders
12/11/2003US20030229079 1-(Aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
12/11/2003US20030229066 Central nervous system diosrders; psychological disorders
12/11/2003US20030229065 Measuring drug resistance, calibration; reducing antibiotic resistance
12/11/2003CA2486110A1 Pharmaceutical combination
12/10/2003EP1368358A1 Isoxazoline derivatives as anti-depressants
12/10/2003EP1368357A1 Tricyclic quinolinone and tricyclic quinoline as androgen receptor modulator compounds
12/10/2003EP1368029A2 Method and composition for rejuvinating cells, tissues, organs, hair and nails
12/09/2003US6660862 Genetic engineering
12/09/2003US6660740 Sorbitol dehydrogenase inhibitors
12/09/2003US6660731 Pyrazole compounds useful as protein kinase inhibitors
12/09/2003US6660526 Potassium fluoroionophore
12/09/2003CA2078758C 2-substituted indane-2-mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
12/04/2003WO2003099823A2 1,3-diaza-dibenzoazulenes as inhibitors of tumour necrosis factor production and intermediates for the preparation thereof