Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
04/2004
04/07/2004EP1210351B1 Method for separating lactone-containing high-molecular weight compounds
04/07/2004EP0741731B1 Process for epoxidising prochiral olefins
04/07/2004CN1487940A Lactam compounds and medicinal use thereof
04/07/2004CN1487933A Pyrazole compounds useful as protein kinase inhibitors
04/07/2004CN1487916A Process for the preparation of arylethanoldiamines useful as agonists the beta-3-adrenoceptor
04/07/2004CN1144793C Polar-substituted hydrocarbons
04/07/2004CN1144789C Pyrrolidine and piperidine derivatives, producing process and application thereof
04/01/2004WO2004026881A1 Macrocyclic pyrimidines, the production thereof and the use of the same as medicaments
04/01/2004WO2004026819A2 OPIATE ANALOGS SELECTIVE FOR THE delta-OPIOID RECEPTOR
04/01/2004WO2004018482A3 C6- and c9-substituted chromeno[4, 3-c]isoxazoline derivatives and their use as anti-depressants
04/01/2004WO2003084965A8 N-(3-rifamycinyl)-carbamates, method of preparing them and their use for treating and preventing tuberculosis
04/01/2004WO2002102314A3 Purine inhibitors of phosphodiesterase (pde) 7
04/01/2004US20040063955 Antichoelsterol agents; cardiovascular disorders; antihistamines; multiple sclerosis; antihistamines
04/01/2004US20040063926 L-nucleic acid derivative and processes for the synthesis thereof
04/01/2004US20040063754 Dehalogeno compounds
04/01/2004US20040063735 Calcitonin gene related peptide receptor antagonists
04/01/2004US20040063718 Targeted therapeutics and uses thereof
04/01/2004US20040063716 Cholesterol biosynthesis inhibitors containing as the active ingredient tricyclic spiro compounds
04/01/2004US20040063713 Such as 2-((4-(2-fluorophenyl)-1-piperazinyl)methyl)-1H-thieno(3,4-d)imidazole
04/01/2004US20040060478 Formed by chlorosulfonating an organic pigment and reacting with an amino carboxylic acid to form carboxy substituted sulfonamide derivatives
04/01/2004CA2498046A1 Opiate analogs selective for the delta-opioid receptor
04/01/2004CA2492319A1 Macrocyclic pyrimidines, the production thereof and the use of the same as medicaments
03/2004
03/31/2004EP1401841A1 Substituted 1-oxa-2,8-diaza-spiro 4,5]dec-2-ene derivatives as medicaments for the treatment of pain
03/31/2004EP1401834A1 New derivatives of oxazolidinones as antibacterial agents
03/31/2004EP1401830A2 Quinazolinediones as antibacterial agents
03/31/2004EP1401829A1 Novel heterocyclic antibacterial compounds
03/31/2004EP0874852B1 Oxazolidinone antibacterial agent with tricyclic substituents
03/31/2004CN1486315A Dehalogeno compounds
03/31/2004CN1486312A Pyrazole compounds useful as protein kinase inhibitors
03/31/2004CN1486311A Pyrazole compounds useful as protein kinase inhibitors
03/31/2004CN1486310A Pyrazole compounds useful as protein kinase inhibitors
03/31/2004CN1143853C Preparing method for anti-viral compounds
03/30/2004US6713487 Heterocyclic amine derivatives; for treating an inflammatory or immune disease, a cardiovascular disease, or a neurodegenerative condition
03/30/2004US6713484 Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
03/30/2004US6713475 Tricyclic benzodiazepines (cyclic oligopeptides), useful for treatment of hypertension, congestive heart failure, cardiac insufficiency, coronary vasospasm, cardiac ischemia, liver cirrhosis, renal failure, stroke or thrombosis
03/25/2004WO2004024939A2 Ligands for the peroxisome proliferator-activated receptor, and methods of use thereof
03/25/2004WO2004024736A1 Antidepressant azaheterocyclylmethyl derivatives of 4,5-dihydroimidazo[1,4,5-de]benzoxazine
03/25/2004WO2004024734A1 Antidepressant indolealkyl derivatives of heterocycle-fused benzodioxan methylamines
03/25/2004WO2004024733A1 Antidepressant piperidine derivatives of heterocycle-fused benzodioxans
03/25/2004WO2004024732A1 Antidepressant cycloalkylamine derivatives of heterocycle-fused benzodioxans
03/25/2004WO2004024731A1 Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans
03/25/2004WO2004024149A1 Medicament containing disorazoles and derivatives thereof for the treatment of benign and malignant tumoral diseases
03/25/2004WO2004024065A2 Substituted bicyclic thiophene derivatives, compostions containing such compounds and methods of use
03/25/2004WO2004000849A3 Tetracyclic arylsulfonyl indoles having serotonin receptor affinity
03/25/2004WO2003077862A3 Potent, simplified derivatives of immunosuppressive agents
03/25/2004WO2003022214A3 Piperazine and homopiperazine compounds
03/25/2004WO2003014121A9 Compounds, derivatives, compositions, preparation and uses
03/25/2004US20040058969 React with tubulin; forming microtubes; stabilization; antitumor, anticancer agents; antiinflammatory agnets; psoriasis; antiarthritic agents
03/25/2004CA2498532A1 Antidepressant piperidine derivatives of heterocycle-fused benzodioxans
03/25/2004CA2498131A1 Antidepressant cycloalkylamine derivatives of heterocycle-fused benzodioxans
03/25/2004CA2498106A1 Substituted bicyclic thiophene derivatives, compositions containing such compounds and methods of use
03/25/2004CA2497783A1 Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans
03/25/2004CA2497214A1 Antidepressant indolealkyl derivatives of heterocycle-fused benzodioxan methylamines
03/24/2004EP1399450A1 Benzoxazepine derivatives and their use as ampa receptor stimulators
03/24/2004EP1399445A2 Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists
03/24/2004EP1399444A2 Novel heterocyclic compounds, method for preparing same and use thereof as medicines, in particular as anti-bacterial agents
03/24/2004EP1399443A1 Nitrogen-containing bicyclic heterocycles for use as antibacterials
03/24/2004EP1399436A2 Oxytocin agonists
03/24/2004CN1484679A Acid pigment dispersamts and pigment preparations
03/23/2004US6710053 Deuterated rapamycin compounds, method and uses thereof
03/18/2004WO2004022767A1 Solid state fermentation and fed batch for the production of an immunosuppressant
03/18/2004WO2004021984A2 Heterocyclic aromatic compounds useful as growth hormone secretagogues
03/18/2004WO2003011298A8 Antibacterial oxazinones and methods for their use and synthesis
03/18/2004WO2003011222A3 Thrombin inhibitors
03/18/2004US20040053955 An immunosuppressants for treating allograft rejection, transplant rejection, psoriasis, and rheumatoid arthritis, a 9,10-dihydro-9-oxo-acridine-3-yl- derivatives
03/18/2004US20040053952 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
03/18/2004US20040053923 Novel isoindole derivatives
03/17/2004EP1397364A1 Novel pyrrole derivatives as pharmaceutical agents
03/17/2004EP1397361A1 Carboline derivatives as pdev inhibitors
03/17/2004EP1397340A2 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
03/17/2004EP1397142A2 Pyrimidine inhibitors of phosphodiesterase (pde) 7
03/17/2004EP1354020A4 Novel red fluorescent material and organic electroluminescent device containing same
03/17/2004EP1305318B1 Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b] [1,3]benzothiazepines
03/17/2004EP0891332B1 6-phenylpyridyl-2-amine derivatives
03/16/2004US6706736 Antidepressant azaheterocyclylmethyl derivatives of oxaheterocycle-fused-[1,4]-benzodioxans
03/16/2004US6706727 ethyl-4-chloro- or 4-hydroxy- Ascomycin derivatives; pimecrolimus homologues; cultivating Streptomyces hygroscopius to produce the 4-hydroxy derivative; replacement of the hydroxy with chloro under epimerization; antiinflammatory; immunosupression
03/16/2004US6706707 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles
03/16/2004CA2096460C Dual action inhibitors
03/16/2004CA2079143C Novel 2-substituted indane-2-carboxyalkyl derivatives useful as inhibitors of enkephalinase and ace
03/11/2004WO2004019907A1 Methods and reagents for treating infections of clostridium difficile and diseases associated therewith
03/11/2004WO2004009578A3 Pentacyclic oxepines and derivatives thereof, process for their preparation and pharmaceutical compositions containing them
03/11/2004WO2003096782A3 Process for preparing maytansinol
03/11/2004WO2003063864A3 Heterocyclic compounds which are active as inhibitors of beta lactamases
03/11/2004US20040049029 Process for preparing substance GM-95
03/11/2004US20040048884 3-aminoalkyluracil derivatives, e.g., 1-(2,6-Difluorobenzyl)-5-(3-methoxyphenyl)-6-methyl-3-(N-methyl-N-(2 -pyridylethyl)-aminoethyl)uracil; contraceptives; treating lupus, sex hormone related cancer, benign prostatic hypertrophy, etc.
03/11/2004US20040048883 Novel fused quinazoline derivatives useful as tyrosine kinase inhibitors
03/11/2004US20040048847 Increasing the sugar-transporting capacity; preventing and/or treating diabetes, diabetic peripheral neuropathy, diabetic nephropathy, diabetic retinopathy, diabetic macroangiopathy, impaired glucose tolerance or adiposis
03/11/2004US20040048845 Containing indolecarbazole compounds, such as staurosporine.
03/11/2004CA2495144A1 Methods and reagents for treating infections of clostridium difficile and diseases associated therewith
03/10/2004EP1395606A1 Pyrrolidin-2-one derivatives as inhibitors of factor xa
03/10/2004EP1395570A1 Oxazin(thi)one compounds used as fungicides
03/10/2004EP1395290A2 Cytotoxic cd44 antibody immunoconjugates
03/10/2004EP1395257A1 Macrocycles useful in the treatment of alzheimer's disease
03/10/2004EP1054673B1 Benzoxazine compounds for enhancing synaptic response
03/10/2004CN1481368A Gyrase imhibitors and uses thereof
03/10/2004CN1481365A Cyclization process step in making of quinolones and naphthyridines
03/09/2004US6703402 Oxazolo, thiazolo and selenazolo [4,5-c]-quinolin-4-amines and analogs thereof
03/09/2004US6703401 Compounds, their preparation and use
03/09/2004US6703348 Heterocyclyl-substituted benzoylcyclohexandiones, their preparation, and their use as herbicides
03/04/2004WO2004018483A1 Fused heterocyclic isoxazoline derivatives and their use as anti-depressants