Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
02/2003
02/06/2003WO2002085914A3 ENZYMATIC PROCESS FOR PREPARING CEPHALOSPORANIC ACID DERIVATIVES USING α-KETOACID DERIVATIVES
02/06/2003WO2002079146A3 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
02/06/2003WO2002066418A3 Process for the preparation of arylethanoldiamines useful as agonists of the beta-3-adrenoceptor
02/06/2003WO2002061110A3 Nucleic acid derivatives
02/06/2003WO2002059112A3 Pyrazole compounds useful as protein kinase inhibitors
02/06/2003US20030027821 Administering 2-oxy substituted benzoxazin-5-one derivative to a human or animal for the prevention or treatment of obesity or an obesity related disorder
02/05/2003EP1280807A1 Photochromatic pyrano-1,3-oxazinonaphthalene derivatives
02/05/2003EP1280798A1 Bicyclic heterocylces, medicaments containing said compounds, the use thereof and method for producing them
02/05/2003EP1280572A1 Delivery devices for treatment of vascular disease
02/05/2003EP1280570A2 Delivery devices for treatment of vascular disease
02/05/2003EP1280569A1 Delivery systems for treatment of vascular disease
02/05/2003EP1280568A1 Delivery devices for treatment of vascular disease
02/05/2003EP1280512A2 Delivery systems for treatment of vascular disease
02/05/2003EP1086078B1 Neuropeptide y5 receptor antagonists
02/05/2003CN1100538C Lotion
02/04/2003US6515123 Triphendioxazine pigments, intermediates, their method of making and uses thereof
02/04/2003US6514983 Inhibitors of the nucleic enzyme poly(adenosine 5'-diphospho-ribose)polymerase
02/04/2003US6514972 Heteropolycyclic inhibitors of protein kinases
01/2003
01/30/2003WO2003008399A1 Synthesis of udp-glucose: n-acylsphingosine glucosyltransferase inhibitors
01/30/2003WO2002088079A3 Dual inhibitors of pde 7 and pde 4
01/30/2003WO2002059129A3 Substituted tetracyclic pyridoindoles as serotonin agonists and antagonists
01/30/2003WO2002018376A1 Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
01/30/2003WO2002014536A3 Odulating multiple lineage kinase proteins
01/30/2003US20030023082 Epothilone derivatives and methods for making and using the same
01/30/2003US20030022885 Pyrazole compounds useful as protein kinase inhibitors
01/30/2003CA2417907A1 Bicyclic heterocycles, pharmaceutical compositions containing these compounds, their use and processes for preparing them
01/29/2003EP1279674A2 Acetylenic ortho-sulfonamido and phosphinic acid amido bicyclic heteroaryl hydroxamic acids as TACE inhibitors
01/29/2003EP1278744A1 Heterobicyclic sulfonamides and their use as platelet adp receptor inhibitors
01/29/2003EP1129097B1 Novel type condensed pyridazinone compounds
01/29/2003EP0946553B1 8-azabicyclo 3.2.1]octane derivatives, their preparation and their use as insecticides
01/29/2003CN1393448A Process for synthesizing oxazole [4,5-6] pyridine-2 (3H) one
01/28/2003WO2002018372A1 Bicyclic heterocycles, medicaments containing these compounds, their use, and methods for the production thereof
01/28/2003US6512115 Preparation of pigments
01/28/2003US6512113 A process for preparing 4,10-dinitro-2,6,8,12-tetraoxa-4,10-diazatetracyclo(5.5.0.05,903,11) -dodecane involves reacting at least one hexa-substituted piperazine derivative with at least one nitrate source and optionally at least one strong
01/28/2003CA2124375C Compounds containing a fused bicyclic ring and processes therefor
01/23/2003WO2003006469A1 New picolinamine derivatives and their use a fungicides
01/23/2003WO2002050066A3 Pyrazole compounds useful as protein kinase inhibitors
01/23/2003WO2002017893A3 Sgk2 and sgk3 used as diagnostic and therapeutic targets
01/23/2003US20030017975 Immunosuppressants; activation of lipopeptide fungicides
01/22/2003EP1276740A2 Novel epothilone derivatives, method for the preparation thereof and their pharmaceutical use
01/22/2003EP0646115B1 Heterocyclic-cyclic amine derivatives
01/22/2003CN1392875A Condensed azepines as vasopressino agonists
01/22/2003CN1099419C Azebicyclic compound
01/16/2003WO2003004098A1 Composition for topical administration comprising an interleukin-2 inhibitor and an antimicrobial agent
01/16/2003WO2001051049A9 O-methylated rapamycin derivatives for alleviation and inhibition of lymphoproliferative disorders
01/16/2003US20030013737 Antimicrobial quinolone derivatives and use of the same to treat bacterial infections
01/16/2003US20030013707 Enzyme inhibitor
01/16/2003CA2452372A1 Composition for topical administration comprising an interleukin-2 inhibitor and an antimicrobial agent
01/15/2003EP1275653A1 Oxazolopyridines and their use as fungicides
01/15/2003EP1095045B1 Method for producing anellated triazoles and new anellated triazoles and their use
01/15/2003EP0790988B1 Use of dioxomorpholines to combat endoparasites, novel dioxomorpholines and process for their production
01/15/2003CN1391576A Androgen receptor modulator compounds and methods
01/15/2003CN1098843C Isoxazoles
01/14/2003CA2231540C Color-safe bleach boosters, compositions and laundry methods employing same
01/09/2003WO2003002569A1 Method of inhibiting ptp 1b and/or t-cell ptp and/or other ptpases with an asp residue at position 48
01/09/2003WO2003002560A1 New derivatives of oxazolidinones as antibacterial agents
01/09/2003WO2002086143A3 Enzymatic process for preparing cephalosporin derivatives
01/09/2003WO2002059111A3 Pyrazole compounds useful as protein kinase inhibitors
01/09/2003WO2002020558A3 Method for binding, in solution, a peptide and a lipophilic vector and uses thereof
01/09/2003WO2002020436A3 Methods for forming combinatorial libraries combining amide bond formation with epoxide opening
01/09/2003US20030009030 Novel selective deacetylating agents
01/09/2003US20030008894 Antimicrobial quinolones, their compositions and uses
01/09/2003US20030008861 N-arylsulfonyl aza-bicyclic derivatives as potent cell adhesion inhibitors
01/09/2003US20030008848 Small molecules useful in the treatment of inflammatory disease
01/09/2003CA2450982A1 New derivatives of oxazolidinones as antibacterial agents
01/08/2003EP1272494A2 Photochromic spiro(indoline)naphthoxazines
01/08/2003CN1390222A Imidazole compounds used as phosphodiesterase VII inhibitors
01/07/2003US6503926 Nitrogen heterocycle compounds
01/07/2003US6503921 Deuterated rapamycin compounds, methods and uses thereof
01/07/2003US6503737 Isolated nucleic acids relating to the fkbA gene within the FK-520 polyketide synthase gene cluster
01/07/2003CA2229892C Liposome preparations of indolocarbazole derivatives
01/03/2003WO2003000699A1 Substituted 1-oxa-2,8-diaza-spiro[4,5]dec-2-ene derivatives as medicaments for the treatment of pain
01/03/2003WO2003000694A1 6-phenyldihydropyrrolopyrimidinedione derivatives
01/03/2003WO2003000692A2 Oxytocin agonists
01/03/2003WO2003000691A1 Carboline derivatives as pdev inhibitors
01/03/2003WO2003000680A1 Diamine derivatives
01/03/2003WO2003000657A1 Diamine derivatives
01/03/2003WO2003000256A1 Substituted oxazolidinones for combinational therapy
01/03/2003WO2002060868A3 Inhibitors of prenyl-protein transferase
01/03/2003WO2002020531A3 Method for producing anellated tetrahydro-[1h]-triazoles
01/03/2003CA2450480A1 Oxytocin agonists
01/02/2003US20030004351 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
01/02/2003US20030004344 Thrombin or factor Xa inhibitors
01/02/2003US20030004337 Efficient lactam synthesis
01/02/2003US20030004164 Anticancer agents; autoimmune diseases
01/02/2003US20030004163 Antiinflammatory agents; headaches; antiarthritic agents
01/02/2003US20030004161 Anticancer agents; autoimmune diseases
01/02/2003US20030004150 New analogues of camptothecin, their use as medicaments and the pharmaceutical compositions containing them
01/02/2003EP1270557A1 Ethylenediamine derivatives
01/02/2003EP1268487A1 Tricyclic protein kinase inhibitors
01/02/2003EP1268486A2 Fused heterocyclic derivatives, their production and use
01/02/2003EP1268485A1 Method for the 1,3 dipolar cycloaddition of organic compounds in a microreactor
01/02/2003EP1268466A1 Decahydro-isoquinolines
01/02/2003EP1268444A1 2,4-di(hetero-)arylamino(-oxy)-5-substituted pyrmidines as antineoplastic agents
01/02/2003EP1268408A1 Arthropodicidal carboxanilides
01/02/2003EP1268406A1 Method for oximating organic carbonyl compounds and/or ch-acid compounds
01/02/2003EP1267876A1 Thrombin inhibitors
01/02/2003EP1139755A4 Method for treatment of bacterial infections with once or twice-weekly administered rifalazil
01/02/2003EP1053246B1 Beta-sheet mimetics and methods relating to the use thereof
12/2002
12/31/2002US6500855 Nitrogen containing aromatic heterocycles with ortho-substituted p1 groups; anticoagulants