Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
10/2003
10/02/2003WO2003080064A1 Kinase inhibitors
10/02/2003WO2003079980A2 Caboxylic acid glycuronides, glycosamides and glycosides of quinolones, penicillins, analogs, and uses thereof
10/02/2003WO2003064385A3 Delta1-pyrrolines and their use as pest control agents
10/02/2003WO2003016316A8 Diazacycloalkanes as oxytocin agonists
10/02/2003US20030187291 Iodohydroxylation of olefins
10/02/2003US20030186995 Substituted bicyclic derivatives useful as anticancer agents
10/02/2003US20030186987 Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
10/02/2003US20030186970 Androgen receptor modulator compounds and methods
10/02/2003CA2479338A1 Substituted phenylacetic acids
10/02/2003CA2479279A1 Fused bicyclic pyridine derivative as tachykinin receptor antagonist
10/02/2003CA2477651A1 Kinase inhibitors
10/01/2003EP1348712A1 L-nucleic acid derivatives and processes for the synthesis thereof
10/01/2003EP1200447B1 Oxazinocarbazoles for the treatment of cns diseases
10/01/2003EP0970079B1 Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with n- or c-linked imidazoles
09/2003
09/30/2003US6627753 Agricultural insecticides
09/30/2003US6627640 Oxazolo, thiazolo and selenazolo [4,5-c]-quinolin-4-amines and analogs thereof
09/30/2003US6627638 Viricides, anticarcinogneic agents
09/30/2003US6627637 I kappa B kinase inhibitors for treating various disorders including arthritis
09/30/2003US6627634 Antitumor agents, treatment of the lungs and respiratory tract
09/25/2003WO2003078439A1 10-(3-cyclopropylaminomethyl-1-pyrrolidinyl)pyridobenzoxazinecarboxylic acid derivative effective against resistant bacterium
09/25/2003WO2003078398A1 NON-PEPTIDE GnRH ANTAGONISTS
09/25/2003WO2003077915A1 Use of rapamycin for inhibiting of cell death
09/25/2003WO2003077862A2 Potent, simplified derivatives of immunosuppressive agents
09/25/2003US20030181497 Heterocyclic acridone inhibitors of IMPDH enzyme
09/25/2003US20030181468 Thiopyrimidine and isothiazolopyrimidine kinase inhibitors
09/25/2003US20030181438 Bicyclic lactam derivatives as inhibitors of matrix metalloproteinases and/or TNF-alpha converting enzyme (TACE)
09/25/2003US20030181437 By reaction of pyrrolobenzothiazepin-9-one with amine to give the corresponding enamine, which is subsequently transformed into the final compound
09/25/2003CA2478795A1 Use of rapamycin for inhibiting cell death
09/25/2003CA2478763A1 10-(3-cyclopropylaminomethyl-1-pyrrolidinyl)pyridobenzoxazine carboxylic acid derivatives effective against drug-resistant bacteria
09/25/2003CA2478713A1 Non-peptide gnrh antagonists
09/24/2003EP1346994A1 Cholesterol biosynthesis inhibitors containing as the active ingredient tricyclic spiro compounds
09/24/2003EP1346993A1 Lactam compounds and medicinal use thereof
09/24/2003EP1345946A1 Macroheterocylic compounds useful as kinase inhibitors
09/24/2003EP1345945A1 Streptogramin derivatives, preparation thereof and compositions containing same
09/24/2003EP1345929A2 Pyrazole compounds useful as protein kinase inhibitors
09/24/2003EP1345928A2 Pyrazole compounds useful as protein kinase inhibitors
09/24/2003EP1345927A1 Pyrazole compounds useful as protein kinase inhibitors
09/24/2003EP1345926A2 Pyrazole compounds useful as protein kinase inhibitors
09/24/2003EP1345925A2 Pyrazole compounds useful as protein kinase inhibitors
09/24/2003EP1345922A1 Pyrazole compounds useful as protein kinase inhibitors
09/24/2003EP1252163B1 4-pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy
09/24/2003EP1100802B1 OXAZOLO, THIAZOLO AND SELENAZOLO [4,5-c]-QUINOLINE-4-AMINES AND ANALOGS THEREOF
09/24/2003EP1051415B1 Benzamide derivatives as vasopressin antagonists
09/24/2003EP0994879B1 Photochromatic compounds, process for their preparation and their use in polymeric materials
09/23/2003US6624302 Polyketide derivatives
09/23/2003US6624202 Inhibitors of copper-containing amine oxidases
09/23/2003US6624161 Administering 2-oxy substituted benzoxazin-5-one derivative to a human or animal for the prevention or treatment of obesity or an obesity related disorder
09/23/2003US6624159 Herpes virus
09/18/2003WO2003076938A1 Novel fluorescent label compounds
09/18/2003WO2003076639A1 Osteoclast differentiation inhibitors
09/18/2003WO2003076447A1 An optically acitve pyridine derivative and a medicament containing the same
09/18/2003WO2003076445A2 Microtubule stabilizing compounds
09/18/2003WO2003076442A1 Purine derivatives as kinase inhibitors
09/18/2003WO2003076440A1 Condensed heterocyclic compounds as calcitonin agonists
09/18/2003WO2003057163A3 Methods for preparing immunoconjugates
09/18/2003WO2003048122A3 Inhibitors of cytosolic phospholipase a2
09/18/2003US20030176717 Process for the preparation of aryloctanoyl amides
09/18/2003US20030176702 N-(azabicyclo moieties)-substituted hetero-bicyclic aromatic compounds for the treatment of disease
09/18/2003US20030176701 Di-or triaza-spiro [4,5] decane derivatives
09/18/2003US20030176670 Multivalent macrolide antibiotics
09/18/2003US20030176455 Inhibiting cell death following cellular regeneration in a mammal in need thereof, which comprises providing with an effective amount of a rapamycin
09/18/2003US20030176454 N-coating heterocyclic compounds
09/18/2003US20030176433 For therapy and prophylaxis of hepatitis C virus (HCV) infection
09/18/2003US20030176422 Pyridoarylphenyl oxazolidinone antibacterials, and related compositions and methods
09/18/2003US20030176414 3-aza-6,8-dioxabicyclo [3.2.1] octanes and analogues and combinatorial libraries
09/18/2003US20030176400 For therapy of allergic diseases such as allergic rhinitis, allergic conjunctivitis, atopic dermatitis, bronchial rhinitis, allergic conjunctivitis, atopic dermatitis, bronchial asthma, food allergy, etc., systemic mastocytosis
09/18/2003US20030175901 Genetic engineering; polyketides
09/18/2003CA2478942A1 An optically active pyridine derivative and a medicament containing the same
09/18/2003CA2478110A1 Novel fluorescent label compounds
09/18/2003CA2478087A1 Microtubule stabilizing compounds
09/17/2003EP1343791A2 Substituted tetracyclic pyridoindoles as serotonin agonists and antagonists
09/17/2003EP1343766A1 Cyclization process step in the making of quinolones and naphthyridines
09/17/2003EP1343499A2 Heterocyclic substituted 2-methyl-benzimidazole antiviral agents
09/17/2003EP1282622B1 Crf receptor antagonists and methods relating thereto
09/17/2003EP1183317B1 Process for the preparation of herbicidal derivatives
09/17/2003CN1443188A Process for preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b] [1,3] benzotiazepines
09/17/2003CN1121376C Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives and matrix metalloprotease inhibitors
09/16/2003US6620931 Process for preparing new crystal polymorphs of a methyl-substituted benzimidazolone-dioxazine pigment
09/16/2003US6620807 Pyridobenzodiazepine and pyridobenzoxazepine carboxyamide vasopressin agonists
09/16/2003CA2078759C Novel carboxyalkyl derivatives useful as inhibitors of enkephalinase and ace
09/11/2003WO2003074054A1 Ophthalmic composition comprising ascomycin
09/11/2003US20030171599 An alpha-diazoacetamide is reacted under conditions promoting intramolecular C-H insertion, for example in the presence of a rhodium salt such as Rh2(OAc)4
09/11/2003US20030171394 Tricyclic dihydropyrazolone and tricyclic dihydroisoxazolone potassium channel openers
09/11/2003US20030171373 Spiro compounds as inhibitors of fibrinogen-dependent platelet aggregation
09/11/2003US20030171366 Having antibacterial activity against Gram-positive and Gram-negative bacteria
09/11/2003US20030170831 Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
09/11/2003US20030170765 Biological Conjugation with an enzyme donor, enzyme acceptor, and a substrate, competetive binding, detecting kinases or phosphatases
09/11/2003US20030168409 Method for separating lactone-containing high-molecular weight compounds
09/10/2003EP1341781A1 Antimicrobial quinolones
09/10/2003EP1341769A2 Bacterial gyrase inhibitors and uses thereof
09/10/2003EP1147115B1 Tricyclic benzodiazepines as vasopressin receptor antagonists
09/10/2003CN1441779A Proline derivatives and use thereof as drugs
09/09/2003US6617453 Triphendioxazine compounds
09/09/2003US6617437 Modified oligonucleotide of given formula; useful in diagnostics and therapeutics
09/09/2003US6617334 Antidepressant azaheterocyclylmethyl derivatives of 7,8-dihydro-1,6,9-trioxa-3-aza-cyclopenta[a]naphthalene
09/09/2003US6617333 Antineoplastic combinations comprising
09/09/2003US6617329 Aminoquinazolines and their use as medicaments
09/04/2003US20030166928 Central nervous system disorders, sleep disorders, eating disorders. sexual disorders, hypotensive agents
09/04/2003US20030166924 Method for extracting a macrolide from biomatter
09/04/2003US20030166640 Heterocyclic amides and/or isosteres used as antiinflammatory agents or for prophylaxis of nervous system disorders; combinatorial chemistry; substance P antagonists