Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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12/09/2004 | US20040248890 Voltage gated sodium and calcium channel inhibitors |
12/09/2004 | US20040248222 Monoclonal antibodies specific for buprenorphine and metabolites thereof |
12/09/2004 | CA2525282A1 Indole derivatives with an improved antipsychotic activity |
12/08/2004 | EP1484327A1 Nitrogenous heterocyclic compound and medicine thereof |
12/08/2004 | EP1483267A2 Microtubule stabilizing compounds |
12/08/2004 | EP1483265A1 Purine derivatives as kinase inhibitors |
12/08/2004 | EP1482936A1 Ophthalmic composition comprising ascomycin |
12/08/2004 | EP1482933A2 Potent, simplified derivatives of immunosuppressive agents |
12/08/2004 | EP1385850B1 New process for the preparation of oxabispidines |
12/08/2004 | EP1363898A4 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same |
12/08/2004 | EP0831094B1 Fused polycyclic heterocycle derivatives |
12/08/2004 | CN1179046C Erythromycins and its preparation method, use and compositions |
12/08/2004 | CN1178656C Pharmaceutical composition |
12/07/2004 | US6828327 Macroheterocylic compounds useful as kinase inhibitors |
12/07/2004 | US6828326 Pyrimidinone fused bicyclic metalloproteinase inhibitors |
12/07/2004 | CA2316921C Aryl fused azapolycyclic compounds |
12/07/2004 | CA2154668C Condensed heterocyclic glutamic acid derivatives as antiproliferative agents |
12/02/2004 | WO2004103272A2 Improved cytotoxic agents comprising new maytansinoids |
12/02/2004 | WO2004034961A3 Antimicrobial agents and uses thereof |
12/02/2004 | US20040243097 Antiproliferative drug and delivery device |
12/02/2004 | US20040242866 Tricyclic benzodiazepines as vasopressin receptor antagonists |
12/02/2004 | US20040242660 Combinations of oxazolidinones with other active ingredients for the prophylaxis and/or treatment of thromboembolic disorders |
12/02/2004 | US20040242627 2-Iminoimidazole derivatives (1) |
12/02/2004 | US20040242596 such as N-(3-Amino-propyl)-N-[1-(5-benzyl-3-methyl-4-oxo-4,5-dihydro-isothiazolo[5,4-d]pyrimidin-6-yl)-propyl]-4-chloro-benzamide; for interrupting mitosis; antiproliferatives and anticancer agents |
12/02/2004 | US20040242580 can be applied as sprays by methods commonly employed in crops such as vegetables, fruits, ornamentals, seeds, turf, cereal and vines among other plants |
12/02/2004 | US20040242573 Novel compounds |
12/02/2004 | US20040242533 such as 5-iodo-O6-5'-cyclo-5,6-dihydro-3'-azido-3'-deoxythymidine for prophylaxis or diagnosis of viral diseases caused by hepatitis virus, herpes viruses such as Epstein-Barr virus |
12/02/2004 | CA2525507A1 Process for synthesizing .beta.-lactamase inhibitor intermediates |
12/02/2004 | CA2525130A1 Improved cytotoxic agents comprising new maytansinoids |
12/01/2004 | EP1481077A2 Mitotic kinesin inhibitors |
12/01/2004 | EP1480985A1 Salt of benzosulfonic acid containing clopidogrel and use thereof for the production of pharmaceutical formulations |
12/01/2004 | EP1480644A2 Novel heterocyclic compounds which are active as inhibitors of beta+lactamases |
12/01/2004 | CN1551885A Cyclic indole and heteroindole derivatives, the production and use thereof as medicaments |
12/01/2004 | CN1551767A Cancer treatment |
11/30/2004 | US6825184 For use as anti-inflammatory agents |
11/30/2004 | US6825170 Erythromycin type macrolide with a fused oxazolone ring |
11/25/2004 | WO2004101803A2 Process for producing anticancer agent ll-d45042 |
11/25/2004 | WO2004101583A1 Rapamycin carbohydrate derivatives |
11/25/2004 | WO2004101573A1 Synthesis of substituted heterocyclic compounds |
11/25/2004 | WO2004101564A1 Pyrimidine derivatives possessing cell-cycle inhibitory activity |
11/25/2004 | WO2004101536A1 Novel phenoxazinone derivatives as enzyme substrates and use thereof as indictor in the detection of microorganisms with peptidase activity |
11/25/2004 | WO2004047755A3 Fused bicyclic nitrogen-containing heterocycles |
11/25/2004 | WO2004021984A3 Heterocyclic aromatic compounds useful as growth hormone secretagogues |
11/25/2004 | US20040235939 Macrolactone having very dense functionalization; antiproliferative activity |
11/25/2004 | US20040235880 2-(9-Chloro-3-methyl-4oxo-5H-isoxazolo[4,3-c]quinolin-5-yl)-pyridine, optionally substituted in the 6 positionof the pyridine ring; coadministering with vincristine, epirubicin, daunorubucin, doxorubicin, or etoposide to reduce the severity of MRP1 derived drug resistance |
11/25/2004 | US20040235869 For therapy of subject infected with a retrovirus |
11/25/2004 | US20040235841 For therapy and prophylaxis of diseases and disorders associated with cyclin-dependent kinases (CDKs) activity |
11/25/2004 | US20040235840 For therapy of tumors |
11/25/2004 | US20040235762 Host vs. graft disease, leukemia, lymphoma; autoimmune disorders; fungicides; antitumor and antiproliferative agents |
11/25/2004 | US20040235753 Oxytocin agonists |
11/25/2004 | US20040234573 Medical devices containing rapamycin analogs |
11/25/2004 | CA2525907A1 Rapamycin carbohydrate derivatives |
11/25/2004 | CA2524706A1 Synthesis of substituted heterocyclic compounds |
11/24/2004 | EP1478648A2 Phosphorus-containing compounds uses thereof |
11/24/2004 | EP1478357A2 Tricyclic pyrazole derivatives, process for their preparation and their use as antitumor agents |
11/24/2004 | CN1549812A Pyrazole compounds useful as protein kinase inhibitors. |
11/24/2004 | CN1176925C Regioselective synthesis of rapamycin derivs. |
11/23/2004 | US6822098 Carbocyclic carbo, oxo amines such as n-heptyl-3-methyl-4-oxo -1,4-dihydroquinoline-2-carboxamide, used for prophylaxis of gastrointerstinal disorders |
11/23/2004 | US6821970 Useful for treating diseases wherein modulation of 5-ht activity is desired; nervous system disorders |
11/23/2004 | US6821969 Thioxazinoquinolones as antiviral agents |
11/23/2004 | US6821651 Red fluorescent material and organic electroluminescent device containing same |
11/23/2004 | CA2295061C Storage-stable ophthalmic compositions comprising diclofenac and ofloxacin |
11/18/2004 | US20040229910 Therapeutic compounds |
11/18/2004 | US20040229895 Tetracyclic benzamide derivatives and methods of use thereof |
11/18/2004 | US20040229893 Substituted benzothiazole amide derivatives |
11/18/2004 | US20040229882 dipeptide or tripeptide MC-1R and MC-4R agonists |
11/18/2004 | US20040229323 aerobic fermentation of a biologically pure strain of Streptomyces hygroscopicus LL-D45042 until macrocyclic lactone LL-D45042 is formed, recovery, purification |
11/18/2004 | US20040226501 Crystallization and purification of macrolides |
11/18/2004 | CA2524624A1 Imidazo and thiazolopyridines as jak3 kinase inhibitors |
11/17/2004 | EP1476447A1 Cyclic compounds and their use as complex ligands |
11/17/2004 | EP1476136A1 Pharmaceutical composition comprising n-((1-n-butyl-4-piperidinyl)menthyl)-3,4-dihydro-2h-(1,3)oxazino(3,2-a)indole-10-carboxamide or salt and process therefor comprising dry granulation |
11/17/2004 | EP1250340B1 Methods and compounds for inhibiting mrp1 |
11/17/2004 | CN1547584A Substituted 1-oxa-2,8-diaza-spiro[4,5]dec-2-ene derivatives and related treatment methods |
11/17/2004 | CN1546470A 6-phenylpyridyl-2-amine derivatives |
11/16/2004 | US6818764 Process for preparing substance GM-95 |
11/16/2004 | US6818641 Arthropodicidal carboxanilides |
11/16/2004 | CA2145383C O-alkylated rapamycin derivatives and their use, particularly as immunosuppressants |
11/11/2004 | WO2004096366A1 9-azabicyclo’3.3.1!non-6-ee derivatives with a heteroatom at the 3-position as renin inhibitors |
11/11/2004 | WO2004071345A8 A device and method for the determination of lithium ion concentration in a biological fluid |
11/11/2004 | US20040225111 Therapy for osteoporosis |
11/11/2004 | US20040224944 Pyrazole compounds useful as protein kinase inhibitors |
11/11/2004 | US20040224904 Carbohydrate scaffold, carrying two side chains, which form a macrocyclic ring that may be unsaturated and contains ether, amide, ester and/or carbamate groups; for therapy of bacterial, fungal, viral or protozoal infections or tumors |
11/11/2004 | US20040224394 Transgenic cells, rapamycin biosynthetic cluster for use in production of compounds used as antifungals, neurophins, immunosuppressant and antitumor agents; bioreactors |
11/11/2004 | CA2521938A1 9-azabicyclo[3.3.1]non-6-ene derivatives with a heteroatom at the 3-position as renin inhibitors |
11/10/2004 | EP1474404A2 Method for extracting a macrolide from biomatter |
11/10/2004 | EP1474389A2 Delta1-pyrrolines |
11/10/2004 | CN1545741A Organic electroluminescent device based on 2,5-diaminoterephthalic acid derivatives |
11/10/2004 | CN1545414A Organic compounds |
11/10/2004 | CN1174986C Tricyclic benzodiazepines as vasopressin receptor antagonists |
11/09/2004 | US6815546 Analogues of camptothecin, their use as medicaments and the pharmaceutical compositions containing them |
11/09/2004 | US6815544 Coupling, acylation, treating with an allyl bromide, reduction, desilylation, cyclization and reduction |
11/09/2004 | US6815463 For therapy of disease of cellular hyperproliferation in a subject |
11/09/2004 | US6815448 For therapy of ognitive deficits due to aging, stroke, head trauma, alzheimer's disease or other neurodegenerative diseases, or schizophrenia; anxiety, aggression and stress, and for the control of various physiological phenomena |
11/04/2004 | WO2004094645A1 Process for the recovery of staurosporine from a fermentation broth |
11/04/2004 | WO2004093805A2 Selective spirocyclic glucocorticoid receptor modulators |
11/04/2004 | WO2004087145A3 Antibacterial agents |
11/04/2004 | WO2004083215A3 Nitrogeneous polycyclic derivatives useful as chelators of metal ions and their applications |
11/04/2004 | US20040220204 mixture of fatty ester, alkylene carbonate, butylene glycol, diethylene glycol, monoalkyl ether and thickeners |
11/04/2004 | US20040220176 Particle-forming compositions containing fused pyrrolocarbazoles |
11/04/2004 | US20040220175 (Pyrido/thieno) - [f] - oxazepine-5-one derivatives |