Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
09/2003
09/04/2003US20030166517 Galenical formulations
09/04/2003US20030164482 Photochromatic pyrano-1,3-oxazinonaphthalene derivatives
09/03/2003EP1339721A2 Hydroxyesters of 7-desmethylrapamycin
09/03/2003EP1339709A1 Farnesyl transferase inhibiting benzoheterocyclic derivatives
09/03/2003EP1339687A1 4-6-diphenyl pyridine derivatives as antiinflammatory agents
09/03/2003EP0929533B1 4,4-disubstituted-1,4-dihydro-2h-3,1-benzoxazin-2-ones useful as hiv reverse transcriptase inhibitors and intermediates and processes for making the same
09/02/2003US6613913 Intermediate for antidepressant azaheterocyclylmethyl derivatives of 7,8-dihydro-1, 6,9-trioxa-3-aza-cyclopenta [a]naphthalene
09/02/2003US6613776 Protein serine/threonine kinase inhibitors used for treating diseases such as cancer, diabetes and Alzheimer's disease
08/2003
08/28/2003WO2003070236A2 Tricyclic pyrazole derivatives, process for their preparation and their use as antitumor agents
08/28/2003WO2003045315A3 Carbonylbenzoxazine compounds for enhancing glutamatergic synaptic responses
08/28/2003WO2003017990A3 Ophthalmic composition comprising an ascomycin
08/28/2003US20030163001 Method for oximating organic carbonyl compounds and/or ch-acid compounds
08/28/2003US20030162968 1,4-Disubstituted benzo-fused urea compounds
08/28/2003US20030162962 Streptogramin derivatives, their preparation and compositions containing them
08/28/2003US20030162805 Antidepressant azaheterocyclylmethyl derivatives of oxaheterocycle-fused-[1,4]-benzodioxans
08/28/2003US20030162802 Preferential enzyme inhibitors such as 2-((4-6-pyrimidinedion -2-yl)amino)-4-methyl-5-thiazolecarboxylic acid ethyl ester, used for prophylaxis of lymphocyte associated disorders
08/28/2003CA2476822A1 Tricyclic pyrazole derivatives, process for their preparation and their use as antitumor agents
08/27/2003EP1337247A1 Gaba enhancers in the treatment of diseases relating to reduced neurosteroid activity
08/27/2003EP1337150A2 Substituted 4,5-dihydro-1,2,4-triazin-6-ones, 1,2,4-triazin-6-ones, and their use as fungicides and insecticides
08/27/2003EP1124831B1 Sodium salt of 3-(4-cinnamyl-1-piperazinyl)imino-methyl rifamycin sv and process of preparation
08/27/2003EP0946567B1 Novel counterparts of camptothecin, their application as medicine and pharmaceutical compositions containing them
08/27/2003CN1439001A Tetrahydropyridino or piperidino hetlrocyclic derivatives
08/27/2003CN1438993A Ethylenediamine derivatives
08/27/2003CN1119346C Benzothiadiaxoles and derivatives
08/27/2003CN1119343C Substituted aminocycloalkylpyrrolidine derivatives
08/27/2003CN1119332C Intermediate of azepine
08/26/2003US6610722 Inhibitors of prenyl-protein transferase
08/26/2003US6610686 Use of pirenoxine for the protection of corneal tissues in photokeractomy
08/26/2003US6610677 Enhancing glycogen synthesis, lowering blood levels of glucose, treating colon, ovarian, or breast cancer, treating diabetes, treating schizophrenia
08/21/2003WO2003068980A2 Method for extracting a macrolide from biomatter
08/21/2003WO2003068779A1 Cyclic compounds and their use as complex ligands
08/21/2003WO2003068193A1 Pharmaceutical composition comprising n- ((1-n-butyl-4-piperidinyl) methyl)-3, 4-dihydro-2h- (1, 3) oxazino (3, 2-a) indole-10-carboxamide or salt and process therefor comprising dry granulation
08/21/2003WO2003022433A3 A derivatized macrocycle compound for covalent bonding to a substrate and method of forming and use
08/21/2003WO2002094844A3 Antiviral nucleosides
08/21/2003US20030158421 Method for the 1,3 dipolar cycloaddition of organic compounds in a microreactor
08/21/2003US20030158245 Fused heterocyclic derivatives, their production and use
08/21/2003US20030158243 Preparation and use of carbohydrate-based bicyclic ring structures with antimicrobial and cytostatic activity
08/21/2003US20030158219 N-substituted spiropiperidine compounds as ligands for ORL-1 receptor
08/21/2003US20030158173 NK 1 antagonists
08/21/2003CA2475659A1 Pharmaceutical composition comprising n- ((1-n-butyl-4-piperidinyl) methyl)-3, 4-dihydro-2h- (1, 3) oxazino (3, 2-a) indole-10-carboxamide or salt and process therefor comprising dry granulation
08/20/2003EP1336611A1 Dehalogeno compounds
08/20/2003EP1335924A2 Ethers of 7-desmethylrapamycin for use in immunosuppression
08/20/2003EP1335923A2 Condensed pyridoindole derivatives
08/20/2003EP1335725A2 Use of cci-779 as an antineoplastic agent
08/20/2003EP1189908B1 Indolocarbazole alkaloids from a marine actinomycete
08/20/2003EP1067935B1 Acylbenzoxazines for enhancing synaptic response(s)
08/20/2003CN1437602A Compounds for treating impaired fundic relaxation
08/20/2003CN1118457C Cyclic diamine compound and medicine containing the same
08/19/2003US6608197 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
08/19/2003US6608098 Isoindole derivatives
08/19/2003US6608081 Treating pneumonia
08/19/2003US6608077 Il-8 receptor antagonists
08/19/2003US6608048 Tricyclic protein kinase inhibitors
08/19/2003CA2085347C Novel cyclic aminophenylacetic acid derivative, production therof, and immune response modulator containing the same as active ingredient
08/14/2003US20030153801 Compositions of cyclooxygenase-2 selective inhibitors and radiation for inhibition or prevention of cardiovascular disease
08/14/2003US20030153610 Substituted oxazolidinones and their in the field of blood coagulation
08/14/2003US20030153593 Use of CCI-779 as an antineoplastic agent
08/14/2003US20030153564 New oxabispidine compounds useful in the treatment of cardiac arrhythmias
08/14/2003US20030153563 CRF receptor antagonists and methods relating thereto
08/14/2003US20030153558 Immunomodulators and/or inhibiting cytokine release
08/14/2003US20030153556 Anticoagulants and antiagglomerants
08/13/2003EP1216244B1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists
08/13/2003EP0808313B1 Antipsychotic 4-(1h-indolyl-1-yl)-1-substituted piperidine derivatives
08/13/2003CN1436076A Method of treating cardiovascular disease
08/13/2003CN1117750C 3-heterocyclyl-substd. benzoyl derivs.
08/12/2003US6605707 Process for the preparation of 6-O-propargyl erythromycin derivatives
08/12/2003US6605630 Active against drug resistant gram positive pathogens
08/12/2003US6605613 Polyene macrolide antibiotic, especially a rapamycin, and an antioxidant, especially 2,6-di-t-butyl-4-methylphenol; 40-O-(2-hydroxy)ethyl-rapamycin in crystalline form.
08/12/2003US6605610 Aryl fused azapolycyclic compounds
08/12/2003US6605599 Epothilone derivatives
08/12/2003US6605295 Storage-stable ophthalmic compositions comprising diclofenac and ofloxacin
08/07/2003WO2003064432A1 Process for total synthesis of ecteinascidins and intermediates therefor
08/07/2003WO2003064425A1 N-substituted spiropiperidine compounds as ligands for orl-1 receptor
08/07/2003WO2003064421A1 Aminopiperidine derivatives
08/07/2003WO2003064415A1 Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterial, related compositions and methods
08/07/2003WO2003064385A2 Delta1-pyrrolines and their use as pest control agents
08/07/2003WO2003064383A2 Phosphorus-containing compounds & uses thereof
08/07/2003WO2003063874A1 Condensed heterocyclic compounds
08/07/2003WO2003063864A2 Heterocyclic compounds which are active as inhibitors of beta lactamases
08/07/2003WO2002048150A3 Agents useful for reducing amyloid precursor protein and treating demantia and methods of use thereof
08/07/2003US20030149266 Administering to a patient (a warm blooded animal, such as man) an effective amount of a pyrimidine derivative for treating cancer, cell proliferation, and inhibition of focal adhesion kinase effect
08/07/2003US20030149074 Modulators of phosphoinositide 3-kinase
08/07/2003US20030149036 Substituted benzothiazole amide derivatives
08/07/2003US20030149033 For prophylaxis and therapy of cerebrovascular diseases such as cerebral ischemia, stroke, reperfusion damage, brain trauma, edemas, cerebral thrombosis, dementia and Alzheimer's diseass
08/07/2003CA2474718A1 Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterial, related compositions and methods
08/07/2003CA2474594A1 Delta1-pyrrolines
08/07/2003CA2474434A1 Condensed heterocyclic compounds
08/07/2003CA2466915A1 N-substituted spiropiperidine compounds as ligands for orl-1 receptor
08/06/2003EP1332134A2 Inhibitors of prenyl-protein transferase
08/06/2003CN1434822A Substituted oxazolidinones and their use in the field of blood coagulation
08/05/2003US6602875 Sorbitol dehydrogenase inhibitors
08/05/2003US6602871 Thrombin or factor Xa inhibitors
08/05/2003US6602865 Pyridazino(4,5-b)(1,5)oxazepinone, -thiazepinone and -diazepinone compounds
08/05/2003US6602826 Heterocyclically substituted aromatic amino compounds with a herbicidal effect
07/2003
07/31/2003WO2003062245A1 Fused bicyclic pyrimidine derivatives
07/31/2003WO2003062244A1 Phenyl substituted heterocyclic compounds useful as herbicides
07/31/2003WO2003057698A3 Spiroazacyclic compounds as monoamine receptor modulators
07/31/2003WO2002092065A3 Novel methods for the treatment and prevention of pain using stress-activated protein kinase inhibitors
07/31/2003US20030144562 Hetero diels-alder adducts of pentacene as soluble precursors of pentacene
07/31/2003US20030144512 Process for preparing piperazinepentaneamide HIV protease inhibitors