Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
08/2008
08/21/2008CA2672955A1 New 2, 4-dianilinopyrimidines, preparation thereof as drugs, pharmaceutical compositions and use thereof essentially as ikk inhibitors
08/20/2008EP1958948A1 Pyridazine compound and use thereof
08/20/2008EP1957485A2 Substituted 4-amino-pyrrolotriazine derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis
08/20/2008EP1957480A1 Substituted oxindol-derivatives, medicaments containing said derivatives and use thereof
08/20/2008EP1957461A1 Bisamide inhibitors of hedgehog signaling
08/20/2008EP1957076A2 Thiazole derivatives as cxcr3 receptor modulators
08/20/2008EP1957058A1 Compounds for the treatment of inflammatory disorders and microbial diseases
08/20/2008EP1670790B1 Benzimidazole derivatives, compositions containing them, preparation thereof and uses thereof
08/20/2008EP1660492B1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
08/20/2008EP1567523B1 Indolyl derivatives
08/20/2008EP1482935B1 Thiazole and oxazole derivatives which modulate ppar activity
08/20/2008EP1456203B1 Ethylene diamine derivatives and their use as orexin-receptor antagonists
08/20/2008EP1375489B1 Medicinal composition containing 1,3-thiazine derivative
08/20/2008CN101248068A 有丝分裂驱动蛋白抑制剂及其使用方法 Mitotic kinesin inhibitors and methods of use
08/20/2008CN101248067A Oxazolidinone derivatives and use thereof as antibiotics
08/20/2008CN101248064A Nitrocatechol derivatives as COMT inhibitors
08/20/2008CN101248059A Substituted amide derivatives as protein kinase inhibitors
08/20/2008CN101248054A Thiazole derivatives and use thereof
08/20/2008CN101248044A Novel indole compounds
08/20/2008CN101247807A Thiazole compounds and methods of use
08/20/2008CN101245097A Inhibitors of serine proteases, particular hcv NS3-NS4 protease
08/20/2008CN101244062A Sustained release pharmaceutical compositions and methods of treatment using the same
08/20/2008CN100412073C Novel thiophene amidines, compositions thereof, and methods of treating complement-mediated diseases and conditions
08/19/2008US7414071 Such as 5-(3-(2S-(3R-hydroxy-4-(3-trifluoromethyl-phenyl)-butyl)-5-oxo-pyrrolidin-1 -yl)-propyl)-thiophene-2-carboxylic acid; prostaglandin E2 agonists subtypes (EP4); for treatment of (ocular) hypertension, liver failure, and glaucoma
08/19/2008US7414067 Ophthalmic compositions for treating ocular hypertension
08/19/2008US7414066 Anticholesterol agents; antilipemic agents; antiischemic agents; cardiovascular disorders
08/19/2008US7414057 Piperazine urea derivatives as melanocortin-4 receptor agonists
08/19/2008US7414055 Inhibitors of Akt activity
08/19/2008US7414054 3-(arylamino)methylene-1, 3-dihydro-2H-indol-2-ones as kinase inhibitors
08/19/2008US7414050 e.g. 4-Cyano-1H-imidazole-2-carboxylic acid [2-cyclohex-1-enyl-4-(2,6-dioxo-piperidin-4-yl)-phenyl]-amide; tyrosine kinase inhibitor; autoimmune diseases, antiinflammatory, anticarcinogenic agent
08/19/2008US7414048 4,5-dihydro-isoxazole derivatives and their pharmaceutical use
08/19/2008US7414047 Piperazinyl and diazapanyl benzamides and benzthioamides
08/19/2008US7414040 e.g. 3'-(1-Cyclohexyl-5-hydroxy-3-methyl-1H-pyrazol-4-ylazo)-2'-hydroxy-biphenyl-3- carboxylic acid; agonists of TPO receptor; non-peptide; thrombocytopenia is due to bone marrow, stem cell, or liver transplant, idiopathic thrombocytopenia purpura, myelodysplastic syndromes, aplastic anemia or leukemia
08/19/2008CA2432799C Pyrazole compounds useful as protein kinase inhibitors
08/19/2008CA2257448C Pyridyl alkene- and pyridyl alkine-acid amides as cytostatics and immunosuppressives
08/19/2008CA2200871C Aniline derivatives
08/14/2008WO2008098143A2 Antimicrobial compounds and methods of use
08/14/2008WO2008097976A1 Heterocyclic modulators of tgr5 for treatment of disease
08/14/2008WO2008096746A1 Spiro compound and use thereof
08/14/2008WO2008096129A1 Nitrogen containing hetrocyclic compounds useful as bifunctional modulators of m3 receptors and beta- 2 receptors
08/14/2008WO2008096127A2 Bicyclo[2.2.1]hept-7-ylamine derivatives and their use as m3 muscarinic receptor modulators
08/14/2008WO2008096001A1 Hcv inhibiting macrocyclic phenylcarbamates
08/14/2008WO2008095852A1 Bronchorelaxing arylamides
08/14/2008WO2008095293A1 [1,2,3] triazolyl substituted coumarins as inhibitors of leukotriene biosynthesis
08/14/2008WO2008095292A1 [1,2,3] triazolyl substituted quinolines and coumarins as inhibitors of leukotriene biosynthesis
08/14/2008WO2008038136A3 Substituted heterocyclylcarbonylamino-acetic-acid-derivatives as inhibitors of bacterial heptose synthesis, methods for their preparation and biological applications of said inhibitors
08/14/2008WO2007065288A8 Useful combinations of monobactam antibiotics with beta-lactamase inhibitors
08/14/2008US20080194656 Benzotriazole Derivatives as Cannabinoid Receptor Antagonists
08/14/2008US20080194629 3-Mono-and 3,5-Disubstituted Piperidine Derivatives as Renin Inhibitors
08/14/2008US20080194625 Tetrahydroquinoline derivatives as cannabinoid receptor modulators
08/14/2008US20080194597 Platelet adp receptor inhibitors
08/14/2008US20080194558 Quinazoline analogs as receptor Tyrosine Kinase inhibitors
08/14/2008US20080194555 Tyrosine kinase inhibitors; antiproliferation agents; metabolism diseases; antiallergens; central nervous system disorders; vision and skin disorders; antiarthritic agents
08/14/2008US20080194545 Antimicrobial compositions and methods of use
08/14/2008US20080194466 (5Z)-5-(6-Quinoxalinylmethylidene)-2-[(2,4,6-Trichlorophenyl)Amino]-1,3-Thiazol-4(5H)-One
08/14/2008US20080191201 Composition containing thiazole rings, organic semiconductor polymer containing the composition, organic active layer containing the organic semiconductor polymer, organic thin film transistor containing the organic active layer, electronic device containing the organic thin film transistor and method of preparing the same
08/14/2008CA2677481A1 Triazole compounds that modulate hsp90 activity
08/14/2008CA2677263A1 Compounds and compositions as modulators of gpr119 activity
08/14/2008CA2677015A1 Hcv inhibiting macrocyclic phenylcarbamates
08/14/2008CA2676498A1 [1,2,3] triazolyl substituted quinolines and coumarins as inhibitors of leukotriene biosynthesis
08/13/2008EP1956020A2 1-[2-(heterocyclyl-aminomethyl)-piperidin-1-YL]-1-(2-methyl-5-phenyl-heterocyclyl)-methanone derivatives and related compounds as orexin-1 antagonists for the treatment of obesity
08/13/2008EP1956013A1 Diagnostic and remedy for disease caused by amyloid aggregation and/or deposition
08/13/2008EP1955697A1 2-aminobenzamide derivative
08/13/2008EP1954696A2 2-phenoxy-n-(1,3,4-thiadizol-2-yl)pyridin-3-amine derivatives and related compounds as p2y1 receptor inhibitors for the treatment of thromboembolic disorders
08/13/2008EP1954695A1 Novel method of preparation of 5-chloro-3-imidazol-1-yl-[1,2,4]thiadiazole and (3-imidazol-1-yl-[1,2,4]thiadiazol-5-yl)-dialkyl-amines
08/13/2008EP1954694A1 Imidazole derivatives as nitric oxide synthase dimerisation inhibitor
08/13/2008EP1954288A1 Amidine derivatives and their uses as medicine
08/13/2008EP1954277A2 Aminopyrimidines useful as kinase inhibitors
08/13/2008EP1954138A2 Insecticidal methods using 3-amino-1,2-benzisothiazole derivatives
08/13/2008EP1954128A2 Diphenylmethane derivatives as inhibitors of leukotriene biosynthesis
08/13/2008EP1828177B1 Novel mch receptor antagonists
08/13/2008EP1781649B1 Substituted hydantoins
08/13/2008EP1590337B1 Acylaminothiazole derivatives, preparation method thereof and use of same as beta-amyloid peptide production inhibitors
08/13/2008EP1541558B1 Heterocyclic compounds having hiv integrase inhibitory activity
08/13/2008EP1322309B1 High affinity small molecule c5a receptor modulators
08/13/2008EP1020445B1 Fused pyridine derivatives
08/13/2008CN101243096A 抗病毒化合物 Antiviral compounds
08/13/2008CN101243078A Thiazolyl piperidine derivatives useful as h3 receptor modulators
08/13/2008CN101243063A Sulfonamide derivatives having carbonic anhydrase inhibiting activity and their use as therapeutic and diagnostic agents
08/13/2008CN101243048A 1-acyldihydropyrazol derivatives
08/13/2008CN101240166A Bromobenzothiazoles luminous agent and preparation method thereof
08/13/2008CN101239972A Heterocyclic n-aryl carboxamides as cytokine inhibitors
08/13/2008CN101239955A Method for producing fungicide composition
08/13/2008CN100410250C Spiroheterocyclic compoundsus reversible inhibitors of cysteine proteases
08/13/2008CN100410245C Arylmethyl-carbonylamino-thiazole derivatives and their use as antitumor agents
08/12/2008US7411065 Peptide nucleic acid monomers: diphenylmethyl, benzyl, alkylthioalkyl, or phenylthioalkyl esters of N-(1-[4-(2-benzothiazolyl-, 2-benzoxazolyl-, 2-benzofuranyl- or 2-benzothiophenyl-sulfonyl)-3-piperazinon-1-ylcarbonylmethyl]pyrimidon-4-yl)carbamic acids
08/12/2008US7410995 N-linked sulfonamide of heterocyclic thioesters for vision and memory disorders
08/12/2008US7410987 Treating pruritus or pain, particularly that caused by a rheumatic disease, by administering a 2-[o-(aminoalkoxy)phenyl])-3-acylbenzothiazoline, e.g., 3-Acetyl-6-chloro-2-[2-(3-(N-(2-hydroxyethyl)-N-isopropylamino)-propoxy)-5-methoxyphenyl]benzothiazoline
08/12/2008US7410972 Compounds
08/12/2008US7410970 Substituted 1,4,-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
08/12/2008US7410961 2,6-disubstituted piperiddines as modulators
08/07/2008WO2008094992A2 2-aminopyridine derivatives useful as kinase inhibitors
08/07/2008WO2008093677A1 Novel oxadiazole derivatives and thiadiazole derivatives having neovascularization inhibiting activity
08/07/2008WO2008093674A1 Novel thiadiazole derivative having kinase inhibitory activity
08/07/2008WO2008093065A1 L-ALANINE DERIVATIVES AS α5βL ANTAGONISTS
08/07/2008WO2008092955A1 Processes and intermediates for preparing a macrocyclic protease inhibitor of hcv
08/07/2008WO2008092954A2 Polymorphic forms of a macrocyclic inhibitor of hcv
08/07/2008WO2008092891A1 1-oxa-3-azaspiro(4.5)decan-2-one derivatives for the treatment of eating disorders
08/07/2008WO2008092888A1 1-oxa-3-azaspiro[4,5]decan--2-one derivatives for the treatment of eating disorders
08/07/2008WO2008092887A1 I-oxa-3-azaspiro (4.5) decan-2-one and 1-oxa-3, 8-diazaspiro (4.5) decan-2-one derivatives for the treatment of eating disorders