| Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773) |
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| 09/12/2008 | CA2679249A1 Compounds and compositions as modulators of gpr119 activity |
| 09/12/2008 | CA2679101A1 Heterocyclic compounds, compositions comprising them and methods of their use |
| 09/12/2008 | CA2678492A1 Bicyclic organic compounds suitable for the treatment of inflammatory or allergic conditions |
| 09/11/2008 | US20080221180 Thiazole Derivatives and Use Thereof |
| 09/11/2008 | US20080221178 Benzimidazole Derivatives,Compositions Containing Them, Preparation Thereof and Uses Thereof |
| 09/11/2008 | US20080221151 In which the amino is substituted by arylmethyl- or heteroarylmethyl- group, e.g., 2-Methoxybenzyl)-(2-phenylpyrrolidin-3-yl)-amine and 5-{[2-(3-Chloro-phenyl)-pyrrolidin-3-ylamino]-methyl}-6-methoxy-3-methyl-1,1a,3,7b-tetrahydro-3-aza-cyclopropa[a]naphalen-2-one; neurokinin 1 (Substance P) inhititors |
| 09/11/2008 | US20080221088 3,4-Substituted Thiazoles as Ampk Activators |
| 09/11/2008 | US20080221082 of the alpha V beta 3 integrin receptor; , thromboembolic events, cardiovascular disorders, lung diseases, disorders of the CNS, the kidney, the gastrointestinal tract or inflammation |
| 09/11/2008 | US20080219929 Introducing into the subject a ligand capable of labelling aggregated paired helical filament (PHF) tau protein, determining the presence and/or amount of ligand bound to extracellular aggregated PHF tau in the medial temporal lobe of the brain, correlating the result of the determination |
| 09/11/2008 | US20080216606 Grinding to uniform particle size; heating; pressurization;; extraction from ores, concentrates |
| 09/10/2008 | EP1967517A1 Probe for diagnosis of conformational disease |
| 09/10/2008 | EP1966187A1 Piperazine compounds useful as antagonists of c-c chemokines (ccr2b and ccr5) for the treatment of inflammatory diseases |
| 09/10/2008 | EP1966176A1 Heterocyclic gaba-b modulators |
| 09/10/2008 | EP1966170A2 Estrogen modulators |
| 09/10/2008 | EP1966161A1 Carboxamides for controlling undesired micro-organisms in plant protection |
| 09/10/2008 | EP1966152A2 Glucokinase activators |
| 09/10/2008 | EP1966151A1 Polycyclic indazole derivatives that are erk inhibitors |
| 09/10/2008 | EP1966144A1 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors |
| 09/10/2008 | EP1966139A1 Aspartic protease inhibitors |
| 09/10/2008 | EP1965807A2 S1p receptor modulating compounds and use thereof |
| 09/10/2008 | EP1965798A2 Useful combinations of monobactam antibiotics with beta-lactamase inhibitors |
| 09/10/2008 | EP1658071B1 Cyanoguanidine-based azole compounds useful as malonyl-coa decarboxylase inhibitors |
| 09/10/2008 | EP1438053B1 Pyrimidine derivatives, pharmaceutical agent containing said compounds, use and method for making same |
| 09/10/2008 | EP1437349B9 Substituted isoxazoles and the use thereof as antibiotics |
| 09/10/2008 | EP1362856B1 Water-soluble triazole fungicide |
| 09/10/2008 | EP1323710B1 Nitrogenous five-membered ring compounds |
| 09/10/2008 | CN101263130A 2-aniline-4-aryl substituted thiazole derivatives |
| 09/10/2008 | CN101263129A Pesticide thiazolyloxy substituted phenylamidine derivatives |
| 09/10/2008 | CN101263125A Quinazoline derivatives useful in cancer treatment |
| 09/10/2008 | CN101260107A Diheterocycle compound containing 4-thiazolidinone and pyrimidine, synthetic method and application thereof |
| 09/10/2008 | CN101260106A Raf kinase inhibitor, preparing method and use thereof |
| 09/10/2008 | CN101260086A Protein-tyrosine-phosphatase 1B inhibitor and its preparation method and use |
| 09/10/2008 | CN101259128A Polymorph medicine |
| 09/09/2008 | US7423159 Agent for preventing or treating neuropathy |
| 09/09/2008 | US7423156 Optionally fused oxazolyl- or thiazolyl-aminophenylbenzoyl(cyclo)alkanoic acid derivatives, e.g., trans-(1R,2R)-2-({3'-fluoro-4'-,[(6-fluoro-1,3-benzothiazol-2-yl)amino]-1,1'-biphenyl-4-yl}carbonyl)cyclopentanecarboxylic acid; diacylglycerol O-acyltransferase type 1 inhibitors |
| 09/09/2008 | US7423150 Substituted benzazoles and methods of their use as inhibitors of Raf kinase |
| 09/09/2008 | US7423148 Small molecule PI 3-kinase inhibitors and methods of their use |
| 09/09/2008 | US7423058 Inhibitors of hepatitis C virus NS3 protease |
| 09/09/2008 | US7423055 e.g., 2-(2-methyl-5-amino)phenyl-4-(3-pyridyl)-thiazole; c-kit inhibitors; treating cell proliferative, metabolic, allergic, and degenerative disorders. |
| 09/09/2008 | US7423053 e.g. 4-[4-Amino-5-(3-fluorobenzoyl)thiazol-2-ylamino]piperidine-1-carboxylic acid tert-butyl ester; inhibit cyclin-dependent kinases; antiproliferative, anticarcinogenic agent; solid tumor such as breast, lung, colon and prostate |
| 09/09/2008 | US7423052 Piperidine compounds for use as orexin receptor antagoinst |
| 09/09/2008 | US7423050 2,4,6-trifluoro-N-[6-[(1-methyl-4-piperidinyl)carbonyl]-2-pyridinyl]-benzamide (hemisuccinate/hydrochloride salt); migraine; inhibit peptide extravasation, while avoiding significant vasoconstrictive activity; improved solubility |
| 09/09/2008 | US7423048 eating disorders of disturbed fundus such as dyspepsia, early satiety, bloating, anorexia; fundic relaxation; 1-(1-((2,3-dihydro(1,4)dioxino(2,3-b)pyridin-3-yl)methyl) -4- piperidinyl)-2-imidazolidinone; improved pharmacokinetics, less vasoconstriction, side effect reduction, sustain release |
| 09/09/2008 | US7423030 1-amino-phthalazine derivatives, the preparation and the therapeutic use thereof |
| 09/09/2008 | CA2252163C D-proline derivatives |
| 09/09/2008 | CA2225756C Substituted cyanophenyl uracils |
| 09/04/2008 | WO2008105607A1 Heteroaryl-imidazole derivatives as cannabinoid cb1 receptor antagonists |
| 09/04/2008 | WO2008105408A1 Novel pyrrole derivative having ureide group and aminocarbonyl group as substituents |
| 09/04/2008 | WO2008105326A1 Process for production of 2-imino-4-thiazolidinone derivative and 2,4-thiazolidinedione derivative |
| 09/04/2008 | WO2008104869A1 Nicotinamide derivatives as inhibitors of h-pgds and their use for treating prostaglandin d2 mediated diseases |
| 09/04/2008 | WO2008104580A1 New use of glutaminyl cyclase inhibitors |
| 09/04/2008 | WO2008104524A1 Thiadiazole derivatives, inhibitors of stearoyl-coa desaturase |
| 09/04/2008 | WO2008104077A1 Small molecule inhibitors of protein arginine methyltransferases (prmts) |
| 09/04/2008 | WO2008080965A3 Hiv inhibiting 5,6-substituted pyrimidines |
| 09/04/2008 | US20080214816 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)ethyl)-6-chloro-1,3-dihydro-2H-indol-2-one; high yield, reduced formation of by-products, avoids special purification procedures like column chromatography |
| 09/04/2008 | US20080214640 3'-{[1-(3,4-Dimethylphenyl)-3-methyl-5-oxo-1,5-dihydropyrazol-4-ylidene]hydrazino}-2'-hydroxybiphenyl-3-carboxylic acid or a salt; treatment of thrombocytopenia; may be coadministered with a colony stimulating factor, cytokine, chemokine, or an interleukin or cytokine receptor agonist or antagonist |
| 09/04/2008 | US20080214610 Thiazolylimidazole Derivatives and Their Use as Inhibitors of Microsmal Triglyceride Transfer Protein |
| 09/04/2008 | US20080214540 3-[(phenyl or benzothiazol-2-yl)methyl]indole-N-acetic acids and esters; analgesics; aldose reductase inhibitors; diabetes complications including cataracts, retinopathy, nephropathy, and neuropathy; side effect reduction |
| 09/04/2008 | US20080214533 Anticoagulants, thrombolytic agents; amidating a p-(hydroxy-protected alkylamino)aniline with a (hetero)arylaminocarbonyl-(hetero)aryl carboxylic acid; deblocking, reacting with cyanogen bromide and cyclizing |
| 09/04/2008 | US20080214529 Such as n-{3-[1-(3,3-dimethyl-butyl)-4-hydroxy-2-oxo-1,2,4a,5,6,7-hexahydro-pyrrolo[1,2-b]pyridazin-3-yl]-1,1-dioxo-1,4-dihydro-1 lambda-6-benzo[1,2,4]thiadiazin-7-yl}-methane sulfonamide; hepatitis C viral infections; inhibiting replication |
| 09/04/2008 | US20080214524 e.g. N-[2-(3-fluorophenyl)ethyl]-N'-isoquinolin-5-ylurea; opioid receptor inhibitor; analgesic, antiinflammatory agent; inflammatory thermal hyperalgesia, urinary incontinence and bladder overactivity |
| 09/04/2008 | US20080214455 5Z)-2-[(2,6-Dichlorophenyl)amino]-5-{[3-(4-morpholinyl)-6-quinoxalinyl]methylidene}-1,3-thiazol-4(5H)-one; inhibiting hYAK3 proteins; autoimmunity, HIV, cancer, drug-induced anemias, myelodysplastic syndrome, aplastic anemia myelosuppression, cytopenia |
| 09/04/2008 | CA2679446A1 New use of glutaminyl cyclase inhibitors |
| 09/04/2008 | CA2679185A1 2,2,2-tri-substituted acetamide derivatives as glucokinase activators, their process and pharmaceutical application |
| 09/04/2008 | CA2678735A1 Novel pyrrole derivative having ureido group and aminocarbonyl group as substituents |
| 09/03/2008 | EP1964561A1 Inhibitors of IMPDH enzyme |
| 09/03/2008 | EP1963313A2 Inhibitors of diacylglycerol acyltransferase (dgat) |
| 09/03/2008 | EP1963295A1 3, 6-dihydro-2-oxo-6h-(1,3,4)thiadiazine derivatives |
| 09/03/2008 | EP1963293A1 1-orthofluorophenyl substituted 1, 2 , 5-thiazolidinedione derivatives as ptp-as inhibitors |
| 09/03/2008 | EP1963292A2 Organic compounds |
| 09/03/2008 | EP1963282A1 Sulfoximine-substituted pyrimidines , their preparation and use as drugs |
| 09/03/2008 | EP1963281A2 Heterocyclic derivatives as modulators of ion channels |
| 09/03/2008 | EP1963273A2 Substituted isoquinoline-1,3(2h,4h)-diones, 1-thioxo-1,4-dihydro-2h-isoquinoline-3-ones and 1,4-dihydro-3(2h)-isoquinolones and use thereof as kinase inhibitors |
| 09/03/2008 | EP1761497B1 Azadecalin glucocorticoid receptor modulators |
| 09/03/2008 | EP1636217B1 2-imidazo-benzothiazoles as adenosine receptor ligands |
| 09/03/2008 | EP1465626B1 Pharmaceutical compositions (kit) comprising dihydropyridinone compounds and an immunoregulatory (or an antiinflammatory) agent and their uses |
| 09/03/2008 | EP1311480B1 New amidino derivatives and their use as thrombin inhibitors |
| 09/03/2008 | CN101258150A Heteroaryl benzamide derivatives for use as glk activators in the treatment of diabetes |
| 09/03/2008 | CN101258149A Thiazole derivatives and use thereof |
| 09/03/2008 | CN101258147A Derivatives of 4-piperazin-1-yl-4-benz0[B]thiophene suitable for the treatment of CNS disorders |
| 09/03/2008 | CN101258142A 2-aminoaryl pyridines as protein kinases inhibitors |
| 09/03/2008 | CN101258137A Dicycloalkyl urea glucokinase activators |
| 09/03/2008 | CN101258131A 6-arylalkylamino- 2,3,4,5-tetrahydro-1h-benzo[d]azepines as 5-ht2c receptor agonists |
| 09/03/2008 | CN101255156A Composition containing thiazole rings, polymer, active layer, transistor, electronic device and method of preparing the same |
| 09/03/2008 | CN101255130A Benzofluoranthene alkynes compounds and uses thereof |
| 09/03/2008 | CN100415741C Thiazolidinedione derivative and its use as antidiabetic |
| 09/03/2008 | CN100415740C Pyrimidine compounds |
| 09/03/2008 | CN100415724C Pyrimidine derivatives |
| 09/03/2008 | CN100415717C Diarylmethylidene piperidine derivatives and their use as delta opioid receptor agonists |
| 09/03/2008 | CN100415716C 1-(1,2-disubstituted piperidyl)-4-substituted diethylenediamine derivative |
| 09/02/2008 | US7420089 for hepatitis C; histone deacetylase inhibitors; N-hydroxy-4-{[(naphthyl-carbonylamino]alkoxy}benzamides; anticarcinogenic agent; acute promyelocytic leukemia; cell-cycle arrest in late G1 phase or at the G2/M transition |
| 09/02/2008 | US7420062 Hetaryl-substituted pyrazolidindione derivatives with pesticidal characteristics |
| 09/02/2008 | US7420061 Process for preparing prodrugs of benzenesulfonamide-containing COX-2 inhibitors |
| 09/02/2008 | US7420053 2-imino-1,3-thiazine derivatives |
| 09/02/2008 | US7420001 N-({4'-[(1-benzofuran-2-ylcarbonyl)amino]-1,1'-biphenyl-4-yl}sulfonyl)glycine; metalloproteinase inhibitors; arthritis, macular degeneration, graft versus host disease, cancer, osteoarthritis |
| 09/02/2008 | US7419990 e.g. benzyl {1-[2-(1-{[1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidin-3-yl]carbonyl}piperidin-4-yl)-4,5-dimethylphenyl]propyl}carbamate; antidiabetic agent, obesity, sexual disfunctions |
| 09/02/2008 | US7419980 Treating conditions improved by monoamine reuptake; 1-[1-(2-naphthyl)-2-piperazin-1-ylethyl]cyclobutanol; sexual disorders, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders, hot flashes |
| 09/02/2008 | US7419975 Organic compounds |
| 09/02/2008 | US7419967 e.g. hexahydrofuro[2,3-b]furan-3-yl N-((1S,2R)-1-benzyl-3-(cyclopentyloxy)[(3-[2-(dimethylamino)ethyl]aminophenyl)sulfonyl]amino-2-hydroxypropyl)carbamate; against human immunodeficiency virus, chronic and acute viral infections |
| 09/02/2008 | CA2466728C Azetidinyl diamines useful as ligands of the nociceptin receptor orl-1 |