Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
07/2008
07/30/2008CN101233104A Cyanopyrrole-sulfonamide progesterone receptor modulators and uses thereof
07/30/2008CN101233103A Cyanopyrrole-phenyl amide progesterone receptor modulators and uses thereof
07/30/2008CN101230067A Broadspectrum 2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors
07/30/2008CN101230038A Pyridine carboxamide derivatives and their use as pesticides
07/30/2008CN101230034A Nitrogen hetero-cycle compounds for use in the treatment of 5-hydroxide tryptamines related diseases
07/30/2008CN101230008A Substituted heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them
07/30/2008CN101229166A Therapeutic agent for keratoconjunctival disorder
07/30/2008CN100406454C Pyrazole compounds useful as protein kinase inhibitors.
07/30/2008CN100406453C 4-anilino-quinazoline derivatives as antiproliferative agents
07/30/2008CN100406439C Pyrrolidine derivatives as metalloprotease inhibitors
07/29/2008US7405310 Non-nucleoside reverse transcriptase inhibitors
07/29/2008US7405295 Certain imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of Bruton's tyrosine kinase by such compounds
07/29/2008US7405231 Oxidized thioether derivatives
07/29/2008US7405228 Antibacterial cyano-(substituted)-methylenepiperidinophenyl oxazolidinones targeting multiple ribonucleoprotein sites
07/29/2008US7405218 Isothiazole derivatives useful as anticancer agents
07/29/2008US7405217 N-aroyl piperazine derivatives as orexin receptor antagonists
07/29/2008US7405215 e.g. [3-(3-benzyl-4-oxo-3,4-dihydro-phthalazin-1-yl)-indol-1-yl]-acetic acid; inhibit binding of endogenous ligands, including prostaglandin PGD2 and its metabolites and certain thromboxane metabolites (such as 11-dehydro-TXB2), to CRTH2; antiallergent; asthma, bronchitis, rhinitis, cough, psoriasis
07/29/2008US7405209 Protease inhibitors
07/29/2008CA2432222C Pyrazole compounds useful as protein kinase inhibitors
07/29/2008CA2432132C Pyrazole compounds useful as protein kinase inhibitors
07/29/2008CA2401033C 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
07/29/2008CA2359592C Pharmaceutical compositions for alleviating discomfort
07/29/2008CA2256022C 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling chemical synaptic transmission
07/24/2008WO2008089005A2 Renin inhibitors
07/24/2008WO2008087514A2 Hdac inhibitors
07/24/2008WO2008086854A1 5-([1,3,4] oxadiazol-2-yl)-1h-indazol and 5-([1,3,4] thiadiazol-2-yl)-1h-indazol derivatives as sgk inhibitors for the treatment of diabetes
07/24/2008WO2008073956A3 Cyclic sulfonamide derivatives and methods of their use
07/24/2008WO2008068272A3 Antibacterial quinoline derivatives
07/24/2008WO2008065626A3 3-heteroaryl (amino or amido)-1- (biphenyl or phenylthiazolyl) carbonylpiperidine derivativesas orexin receptor inhibitors
07/24/2008WO2008051406A3 Substituted imidazoles as bombesin receptor subtype-3 modulators
07/24/2008WO2008032858A3 Thiadiazole compound and use thereof
07/24/2008WO2008011392A8 Proline urea ccr1 antagonists for the treatment of autoimmune diseases or inflammation
07/24/2008WO2007134169A9 Indole, benzimidazole, and benzolactam boronic acid compounds, analogs thereof and methods of use thereof
07/24/2008WO2007120638A3 Methods and compositions for modulating glycosylation
07/24/2008WO2007077574A8 SULFOXIMINE DERIVATIVES AS p38 MAP KINASE INHIBITORS
07/24/2008US20080177082 N3 alkylated benzimidazole derivatives as mek inhibitors
07/24/2008US20080177080 Oxazole derivatives of tetracyclines
07/24/2008US20080177029 Halogenation and sulfonation of a 4-hydroxy-quinolone, ring closing metathesis with 2nd generation Hoveyda's catalyst of 2-(2-(cyclopropyl-2-propenyl)aminocarbonyl)-4-hydroxy-5-alkenoyl) pyrrolidine, etherification with the quinolone; one pot process; Hepatitis C viricides
07/24/2008US20080176911 2-{2-[2-hydroxy(3-methyl)butyrylamino]pentanoyl}amino-5-(1-methylethyl-4-(3-phenyl-1,2,4-oxadiazol-5-yl)thiazole; neurodegenerative diseases: senile dementia, Alzheimer's and Parkinson's diseases, Down's syndrome, amyloid angiopathy, cerebrovascular disorders, Pick's disease, post-traumatic dementias
07/24/2008US20080176899 Such as 1-Benzo[1,3]dioxol-5-yl-cyclopropanecarboxylic acid [5-(2-methoxy-pyridin-3-ylmethyl)-thiazol-2-yl]-amide 5-(2-Methoxy-pyridin-3-ylmethyl)-thiazol-2-ylamine; cystic fibrosis transmembrane conductance regulator disorders
07/24/2008US20080176865 Substituted arylpyrazoles
07/24/2008US20080176849 e.g. N-hydroxy-3-[4-[[(2-hydroxyethyl)[2-(1H-indol-3-yl)ethyl]-amino]methyl]phenyl]-2E-2-propenamide; histone deacetylase inhibitor; anticarcinogenic, antitumor, antiproliferative agents; improved stability
07/24/2008US20080176842 N1-[1-[N-(2-methylpropyl)-N-(phenylsulfonyl)amino]-2R-hydroxy-3S-(phenylmethyl)prop-3-yl]-3-(1-morpholinosulfonyl)-2R-methylpropionamide; viricide; human T-cell leukemia/limphoma virus
07/24/2008DE102007002717A1 Heterocyclische Indazolderivate Heterocyclic indazole derivatives
07/24/2008CA2712109A1 Thiazolidine derivatives and methods for the preparation thereof
07/24/2008CA2675735A1 5-(1,3,4-oxadiazol-2-yl)-1h-indazole and 5-(1,3,4-thiadiazol-2-yl)-1h-indazole derivatives as sgk inhibitors for the treatment of diabetes
07/23/2008EP1947098A1 Cyclic amine compounds and pest control agent
07/23/2008EP1947093A1 Substituted morpholine and thiomorpholine derivatives
07/23/2008EP1947086A1 Benzene derivative or salt thereof
07/23/2008EP1945635A2 Thiazolyl piperidine derivatives useful as h3 receptor modulators
07/23/2008EP1945620A2 Compounds and compositions as ppar modulators
07/23/2008EP1945617A2 Histone deacetylase inhibitors with aryl-pyrazolyl motifs
07/23/2008EP1945612A2 Heterocyclic compounds as pstat3/il-6 inhibitors
07/23/2008EP1945609A2 Amino acid derivatives as histone deacetylase (hdac) inhibitors
07/23/2008EP1945029A2 Inhibitors of ion channels
07/23/2008EP1615909B1 Piperazine derivatives and their use for the treatment of neurological and psychiatric diseases
07/23/2008EP1567489B1 Pyrrolidin-2-one derivatives as inhibitors of thrombin and factor xa
07/23/2008EP1382603B1 Nitrogenous fused-ring compound having pyrazolyl group as substituent and medicinal composition thereof
07/23/2008EP1071680B1 N,n-disubstituted amides that inhibit the binding of integrins to their receptors
07/23/2008CN101228157A Amino acid salts of rosiglitazone
07/23/2008CN101228156A Fungicidal carboxamides
07/23/2008CN101228155A Substituted oxadiazole derivatives as positive allosteric modulators of metabotropic glutamate receptors
07/23/2008CN101228154A Novel tetracyclic tetrahydrofuran derivatives containing a cyclic amine side chain
07/23/2008CN101228152A N-(heteroaryl)-1-heteroarylalkyl-1h-indole-2-carboxamide derivatives, preparation and therapeutic use thereof
07/23/2008CN101228143A Thiazole derivative
07/23/2008CN101228134A Substituted arylpyrazoles as antiparasitic agent
07/23/2008CN101228128A A process for the preparation of substituted phenyl ether compounds and rosiglitazone
07/23/2008CN100404544C 9-ketospinosyn derivatives
07/23/2008CN100404511C 4,4-difluoro-1,2,3,4-tetrahydro-5h-1-benzoazepine derivative or salt of the same
07/23/2008CN100404505C Novel substituted indoles
07/22/2008US7402704 Arylsulfones and uses related thereto
07/22/2008US7402696 exert an ACC activity-inhibiting effect that is effective in the treatment of obesity, hyperlipemia, fatty liver, hyperglycemia, impaired glucose tolerance, diabetes, diabetic complications (diabetic peripheral neuropathy, diabetic nephropathy, diabetic retinopathy, and diabetic macroangiopathy, hyperten
07/22/2008US7402606 Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin K inhibitors for the treatment of bone loss
07/22/2008US7402605 E.g., 17,17-propano-16-hydroxy-5-(4-ethoxycarbonylthiazol-2-yl)-9-oxo-1,2,3,4,20-pentanor-5-thia-8-azaprost-13-ene; EP2 and/or EP4 receptor agonist; immune disease; antiallergens; alopecia; dysmenorrhea; erectile dysfuncction; antiarthritic agents; liver, respiratory, vascular, urogenital disorder
07/22/2008US7402600 Nitroderivatives of cardiovascular agents
07/22/2008US7402597 e.g. [[7-Allyl-3-[2-[2-(2,4-dichlorophenyl)-5-isopropyl-4-oxazolyl]ethyl]-1,2-benzisoxazol-6-yl]oxy]acetic acid; with vehicles (lactose, D-mannitol, glucose), disintegrators (starch or carboxymethylcellulose calcium ), binders (hydroxypropylcellulose) and lubricants (magnesium stearate or talc)
07/22/2008US7402583 Substituted quinolines as antitumor agents
07/22/2008US7402581 3,5-Dibromo-N-[(2S)-2-(4-fluorophenyl)-4-(3-morpholin-4-ylazetidin-1-yl)butyl]-N-methylbenzamide; neurokinin 1 and 2 (NK1,2) receptors, antagonist; improved pharmacokinetics: not inhibit liver enzyme cytochrome P450, prevent drug-drug interactions, oral bioavailability, antiinflammatory and analgesic
07/22/2008US7402580 Polymerase inhibitors; antiischemic agents; brain disorders; cardiovascular disorders; antiinflammatory agents; antiarthritic agents; neurodegenerative agents; Alzheimer's disease; muscular disorders; antidiabetic agents; kidney disorders; viricides; anticancer agents; immunosuppressants
07/22/2008US7402579 Quinobenzoxazine analogs and compositions
07/22/2008US7402548 Benzoxazole compounds, process for producing the same and herbicides
07/22/2008US7402421 Recombinant methods and materials for producing epothilone and epothilone derivatives
07/22/2008CA2474511C Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders
07/22/2008CA2238171C Quinoline derivatives as nk3 antagonists
07/17/2008WO2008085316A1 Bipiperidinyl compounds, compositions containing such compounds and methods of treatment
07/17/2008WO2008084873A1 Oxime derivative
07/17/2008WO2008084872A1 Hydrazone derivative
07/17/2008WO2008084671A1 Process for producing 1-substituted-2-pyridone-3-carboxylic acid derivative
07/17/2008WO2008084218A1 Benzazole derivatives for the treatment of inflammations
07/17/2008WO2008084043A1 Urea glucokinase activators
07/17/2008WO2008063625A3 Pyridine compounds and methods of their use
07/17/2008WO2008056257A3 Novel triazinedione derivatives as gaba-b receptor modulators
07/17/2008WO2008050101A3 Benzoyl amino heterocyclyl compounds useful in the treatment of a disease mediated through glk
07/17/2008WO2008045564A8 Carboxamide compounds and their use as antagonists of the chemokine ccr2 receptor
07/17/2008WO2008020405A3 Azetidine compounds as orexin receptor antagonists
07/17/2008WO2007146039A3 Crystalline forms of n-[5-[[[5-(1,1-dimethylethyl)-2-oxazolyl]methyl] thio]-2-thiazolyl]-4-piperidinecarboxamide
07/17/2008US20080171882 [(4S)-4-Methyl-2,5-dioxoimidazolidin-4-yl]methanesulfonyl chloride and [(4R)-4-methyl-2,5-dioxoimidazolidin-4-yl]methanesulfonyl chloride; chemical intermediates for enzyme inhibitors
07/17/2008US20080171871 2,2-Dichloro-N-[2-[3-(2-chloro-6-fluorophenyl)-5-isoxazolyl]-(4-pyridyl)]Acetamide; Hepatitis C virus
07/17/2008US20080171778 N3 alkylated benzimidazole derivatives as mek inhibitors
07/17/2008US20080171733 Antiinflammatory agents, antidepressants, analgesics, purinergic receptor antagonists; neurodegenerative diseases, spinal cord injuries; 1-(2,3-dichlorophenyl)-N-[(2-methylphenyl)methyl]-1H-tetraazol-5-amine