Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
11/2008
11/20/2008CA2684563A1 2-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-3-phenyl pyrazines and pyridines and 3-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-2-phenyl pyridines as 5-ht7 receptor antagonists
11/19/2008EP1992623A1 Heteroaryl benzamide derivative for use as GLK activator in the treatment of diabetes
11/19/2008EP1992621A1 Heteroarylamide-substituted pyrimidone derivatives for the treatment of neurodegenerative diseases
11/19/2008EP1991544A2 Substituted imidazole derivatives and their use as ptpase inhibitors
11/19/2008EP1991543A1 4-phenyl-thiazole-5-carboxylic acids and 4-phenyl-thiazole-5-carboxylic acid amides as plk1 inhibitors
11/19/2008EP1991536A2 Novel acetyl-coa carboxylase (acc) inhibitors and their use in diabetes, obesity and metabolic syndrome
11/19/2008EP1991532A2 Compositions and methods for inhibition of the jak pathway
11/19/2008EP1991531A1 Cinnoline and quinoxaline derivates as phosphodiesterase 10 inhibitors
11/19/2008EP1991530A1 Cinnoline derivatives as phosphodiesterase 10 inhibitors
11/19/2008EP1751131B1 Mtp inhibiting aryl piperidines or piperazines substituted with 5-membered heterocycles
11/19/2008EP1542675A4 Compounds useful for the inhibition of aldh
11/19/2008EP1532138B1 Inhibitors of tyrosine kinases
11/19/2008EP1372650B1 Combinations comprising an antidiarrheal agent and an epothilone or an epothilone derivative
11/19/2008CN101309908A Substituted 1h-benzimidazole-4-carboxamides are potent parp inhibitors
11/19/2008CN101309586A Thiazoles used as fungicides
11/19/2008CN101307046A Tripeptidyl peptidase inhibitors
11/19/2008CN100434428C Furazanobenzimidazoles
11/19/2008CN100434420C Compound inhibiting dipeptidyl peptidase iv
11/18/2008US7453002 Five-membered heterocycles useful as serine protease inhibitors
11/18/2008US7453000 Substituted oxazolobenzoisothiazole dioxide derivatives method for production and use thereof
11/18/2008US7452999 Chemical process for the preparation of intermediates to obtain N-formyl hydroxy-lamine compounds
11/18/2008US7452992 Heterocyclic compounds as CCR5 antagonists
11/18/2008US7452991 Aztreonam β polymorph with very low residual solvent content
11/18/2008US7452903 ligands for Calcitonin gene related peptide; azepinone ligands; migranes; N-[5-(2,3-Difluorophenyl)-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]-4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxamide
11/18/2008US7452899 Alzheimer's disease; bridged bicycloalkyl sulphonamide and sulphamide derivatives; [9-endo]2',3', 4',5'-Tetrahydro-5'-(2.2.2-trifluoroethyl)spiro[3-{(E)-2-[5-(4-fluorophenyl)-1-methyl-1H-pyrazol-3-yl]ethenyl}-4-methyl bicyclo[4.2.1]non-3-ene]-9,3'-[1,2,5]thiadiazol-1',1'-dioxide
11/18/2008US7452895 Such as N6-(4,5-dihydrooxazol-2-yl)-N4-[3-methyl-4-(6-methylpyridin-3-yloxy)-phenyl]-quinazoline-4,6-diamine; for treatment of hyperproliferative disorders such as cancer
11/18/2008US7452889 e.g. 3-(2-methylbenzothiazol-5-yloxy)-1-[4-(3-phenoxypropyl)piperazinyl]propan-2-ol; fatty acid oxidation inhibitor; cardiovascular diseases: atrial and ventricular arrhythmias, intermittent claudication, Prinzmetal's angina, stable and unstable angina, and diabetes
11/18/2008US7452883 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses
11/18/2008US7452881 Such as N-[3-(2-diethylaminoethyl)-1H-indol-5-yl]-5-chloro-3-methylbenzo[b]thiophene-2-sulphonamide; serotonin receptors antagonist; anxiolytic, antidepressant, cognitive activator, senile dementia, psychosis, attention deficit/hyperactivity disorder
11/18/2008US7452879 Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds
11/18/2008US7452874 Thrombopoietin mimetics
11/18/2008CA2422379C Pyrazole compounds useful as protein kinase inhibitors
11/18/2008CA2383630C Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
11/18/2008CA2352430C New pharmaceutical composition and the process for its preparation
11/18/2008CA2352275C Il-5 inhibiting 6-azauracil derivatives
11/18/2008CA2331187C Water soluble azoles as broad-spectrum antifungals
11/18/2008CA2278331C 3-heterocyclyl-substituted benzoyl derivatives
11/18/2008CA2230516C Pyrimidine derivatives
11/13/2008WO2008137794A1 Compounds and compositions as c-kit and pdgfr kinase inhibitors
11/13/2008WO2008137622A2 Aminopyrimidines useful as kinase inhibitors
11/13/2008WO2008137621A1 Aminopyrimidines useful as kinase inhibitors
11/13/2008WO2008137619A2 Thiazoles and pyrazoles useful as kinase inhibitors
11/13/2008WO2008136428A1 Nitrogen-containing five-membered heterocyclic compound
11/13/2008WO2008135786A1 Amino-thiazolyl- pyrimidine derivatives and their use for the treatment of cancer
11/13/2008WO2008118718A3 2-aminopyridine analogs as glucokinase activators
11/13/2008WO2008115369A3 Inhibitors of focal adhesion kinase
11/13/2008WO2008114023A3 Phthalazinone derivatives
11/13/2008WO2008099072A3 New 2, 4-dianilinopyrimidines, preparation thereof as drugs, pharmaceutical compositions and use thereof essentially as ikk inhibitors
11/13/2008WO2008097640A8 Triazole compounds that are useful in the treatment of proliferative disorders, such as cancer
11/13/2008WO2007145563A8 Benzimidazole derivatives which are to be used as antagonist for the cb1-receptor
11/13/2008US20080281095 Asparatyl protease inhibitor
11/13/2008US20080280962 Novel thiazolidin-4-one derivatives
11/13/2008US20080280948 Modulators of amyloid beta
11/13/2008US20080280919 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors
11/13/2008US20080280905 Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
11/13/2008US20080280895 5-Amino-4-Hydroxy-7-(1H-Indolmethyl)-8-Methylnonamide Derivatives as Renin Inhibitors for the Treatment of Hypertension
11/13/2008US20080280891 effective against a broad range of cancers, especially leukemia, non-small cell lung and colon; (6-chloropyridin-3-yl)-[3-hydroxy-5-(1H-indol-4-yl)-phenyl]-methanone; antimitotic agents that can block cell cycle progression
11/13/2008US20080280890 Hydroxylamine compounds and methods of their use
11/13/2008US20080280889 Cancer; N,N-dimethyl-5-phenyl-6-(4-{[4-(5-pyridin-2-yl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}phenyl) pyridazin-3-amine;; serine/threonine kinase (Akt) suppression; increased cellular potency or solubility, enhanced pharmacokinetic properties
11/13/2008US20080280888 Antibiotics Derivatives
11/13/2008US20080280873 Biaryl Substituted Pyrazinones as Sodium Channel Blockers
11/13/2008US20080280872 Benzamide Derivatives and Their Use as Glucokinase Activating Agents
11/13/2008US20080280871 5-Phenyl-4-Methyl-Thiazol-2-Yl-Amine Derivatives as Inhibitors of Phosphatidylin Ositol 3 Kinase Enzymes (PI13) For Treatment of Inflammatory Diseases
11/13/2008US20080280857 ligands for Calcitonin gene related peptide; azepinone ligands; migranes; N-[5-(2,3-Difluorophenyl)-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]-4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxamide
11/13/2008CA2694381A1 Aminopyrimidines useful as kinase inhibitors
11/13/2008CA2688584A1 Aminopyrimidines useful as kinase inhibitors
11/13/2008CA2686382A1 Phenylaminopyrimidine derivatives and compositions thereof as c-kit and pdgfr kinase inhibitors
11/13/2008CA2685876A1 Thiazoles and pyrazoles useful as kinase inhibitors
11/13/2008CA2685389A1 Tricyclic compounds as matrix metalloproteinase inhibitors
11/12/2008EP1990335A1 17 beta hsd type 5 inhibitor
11/12/2008EP1990053A1 Pharmaceutical composition for enhancing adiponectin production
11/12/2008EP1989201A1 Pi-3 kinase inhibitors and methods of their use
11/12/2008EP1989185A1 Therapeutic compounds
11/12/2008EP1756099B1 Synthesis of antidiabetic rosiglitazone derivatives
11/12/2008EP1732918B1 Novel pyrrolidine-3,4-dicarboxamide derivatives
11/12/2008EP1727808B1 Biaryl amino acids and their use in dna binding oligomers
11/12/2008EP1606282B1 Phenyl- and pyridylpipereidinye-derivatives as modulators of glucose metabolism
11/12/2008EP1343503B1 Heteroaryl urea neuropeptide y y5 receptor antagonists
11/12/2008EP1261607B1 2,4-disubstituted thiazolyl derivatives
11/12/2008CN101304995A Thiazole derivatives and use thereof
11/12/2008CN101304989A Carbocyclic fused cyclic amines as inhibitors of the coagulation factor XA
11/12/2008CN101304985A Thiazole compounds and their use as PGD2 antagonists
11/12/2008CN101304983A Compounds and compositions as PPAR modulators
11/12/2008CN101304976A Inhibitors of viral replication
11/12/2008CN101302215A 5-[4-[2-(n-methyl-n-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione,maleic acid salt,hydrate as pharmaceutical
11/12/2008CN101302214A Aralkyl piperidine (piperazidine) derivate and use thereof in mental disease treatment
11/12/2008CN101302182A Virus polymerase inhibitors
11/12/2008CN101302180A 8-azaprostaglandin derivative compound and agent comprising the compound as active ingredient
11/12/2008CN100432070C Novel sulfamides and their use as endothelin receptor antagonists
11/11/2008US7449483 e.g. 2-(Ethyl-{4-[2-methyl-3-(4-trifluoromethyl-phenyl)-benzo[b]thiophen-6-yl]-butyl}-amino)-ethanol; 2,3-oxidosqualene-lanosterol cyclase inhibitor; antidiabetic, antitumor, antiproliferative agent; hypercholesterolemia, hyperlipemia, arteriosclerosis, vascular diseases, mycoses, gallstones
11/11/2008US7449482 Piperidine compounds useful as malonyl-CoA decarboxylase inhibitors
11/11/2008US7449479 Hepatitis C virus inhibitors
11/11/2008US7449468 Thiazole and oxazole derivatives as activators of human peroxisome proliferator activated receptors
11/11/2008US7449464 4-{3-[4-(6-Chlorobenzothiazol-2-yl)-1,4-diazepan-1-ylcarbonyl]benzyl}-1(2H)-phthalazinone; Cancer, BRCA deficient
11/11/2008US7449457 Substituted heterocyclic carboxamides with antithrombotic activity
11/11/2008US7449456 signal transducer and activator of transcription-6 inhibitors; asthma, COPD, respiratory, inflammatory and allergic diseases; compounds have less suppressive effect on immunological functions; 4-[(2,5 -difluorobenzyl) amino]-2-[(4-morpholin-4-ylphenyl)amino]pyrimidine-5 -carboxamide
11/06/2008WO2008134693A1 Inhibitors of diacylglycerol o-acyltransferase type 1 enzyme
11/06/2008WO2008133973A1 Therapeutic agents useful for treating pain
11/06/2008WO2008133288A1 Tricyclic aryl compounds
11/06/2008WO2008133274A1 Aminodihydrothiazine derivatives substituted with cyclic groups