Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
04/2008
04/30/2008EP1916249A1 3-(benzo[d][1,3]dioxol-5-ylmethyl)-4-(thio)oxo-2-(thio)oxo-azolidin-5-ylidene derivatives as antibacterial agents
04/30/2008EP1916248A1 Furanone derivatives as cysteine protease inhibitors
04/30/2008EP1916240A1 Pyridazine derivatives
04/30/2008EP1915907A2 An agricultural and horticultural disease controller
04/30/2008EP1915366A2 Piperazine derivative renin inhibitors
04/30/2008EP1915354A1 Novel benzothiazolone derivatives
04/30/2008EP1915352A1 Compounds for the treatment of alzheimer's disease
04/30/2008EP1915350A1 Amide derivatives
04/30/2008EP1915339A1 Beta-secretase inhibitors for use in the treatment of alzheimer's disease
04/30/2008EP1601664B1 Biaryltetrahydroisoquinoline piperidines as selective mch receptor antagonists for the treatment of obesity and related disorders
04/30/2008DE102006050516A1 New pyrazol-3-one compounds are hypoxia-inducible transcription factor-prolyl-4-hydroxylase inhibitors useful e.g. to treat and/or prophylaxis heart-circulation diseases, heart failure, anemia, chronic kidney diseases and renal failure
04/30/2008DE102006050513A1 New substituted dihydropyrazolone derivatives are hypoxia-inducible transcription factor-prolyl-4-hydroxylase inhibitors useful to treat/prevent e.g. cardiovascular diseases, heart-circulation diseases, heart failure and anemia
04/30/2008DE102006050512A1 New substituted dihydropyrazole- and dihydrotriazole derivatives are hypoxia-inducible transcription factor-prolyl-4-hydroxylase inhibitors useful to treat/prevent e.g. cardiovascular diseases, heart-circulation diseases and anemia
04/30/2008DE102006050511A1 New substituted dihydrotriazolone compounds are hypoxia-inducible transcription factor-prolyl-4-hydroxylase inhibitors useful to treat or prophylaxis e.g. heart insufficiency, anemia, chronic kidney diseases and renal failure
04/30/2008DE102006050510A1 New substituted dihydropyrazolthione compounds are hypoxia-inducible transcription factor-prolyl-4-hydroxylase inhibitors useful to treat or prevent e.g. heart insufficiency, anemia, chronic kidney diseases and renal failure
04/30/2008CN101171251A Process for making aztreonam
04/30/2008CN101171250A Tricyclic derivatives of azetidine and pyrrole with antibacterial activity
04/30/2008CN101171249A Method for producing indole derivative having piperidine ring
04/30/2008CN101171248A 3-mono- and 3,5-disubstituted piperidine derivatives as renin inhibitors
04/30/2008CN101171247A Pyrrole derivatives as DNA gyrase and topoisomerase inhibitors
04/30/2008CN101171245A Indolylamino quinazoline derivatives as antitumor agents
04/30/2008CN101171244A Indazolylamino quinazoline derivatives as antitumor agents
04/30/2008CN100384851C Epothilone derivatives
04/30/2008CN100384843C CGRP receptor antagonists
04/30/2008CN100384838C Novel benzylpiperidine compound
04/30/2008CN100384834C Epothilone derivatives
04/30/2008CN100384833C Therapeutic chroman compounds
04/30/2008CN100384825C Benzheterocyclic derivatives
04/30/2008CN100384823C Bicyclic androgen and progesterone receptor modulator compounds and methods
04/30/2008CN100384424C Synergistic methods and compositions for treating cancer
04/30/2008CN100384421C N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines
04/29/2008US7365211 Heterocyclic GABAA subtype selective receptor modulators
04/29/2008US7365205 Diamine derivatives
04/29/2008US7365196 Sulphonamido-substituted bridged bicycloalkyl derivatives
04/29/2008US7365087 Oxazole derivatives of tetracyclines
04/29/2008US7365083 NMDA (N-methyl-D-aspartate) receptors; eg 6-(4-benzylpiperidin-1-carbonyl)-1,5-dihydro-oxazolo[4,5-f]indole-2-one
04/29/2008US7365082 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines
04/29/2008US7365077 Obesity, type 2 diabetes, sleep disorders, ischaemic or haemorrhagic strokes, antiemetic; toxicity; side effect reduction; 2-((benzofuran-4-yl)carbonylaminomethyl)-1-((4-(5-(4-fluorophenyl)-2-methyl)thiazolyl)carbonyl)-4-methylpiperazine
04/29/2008US7365073 3-(heteroaryl) alanine derivatives-inhibitors of leukocyte adhesion mediated by VLA-4
04/29/2008US7365068 Hepatitis C virus infections; -(3-cyclopropyl-4-(pentyloxy)phenyl)-3-nicotinoylthiourea;methyl 2-oxo-2-(5-((3-(4-(pentyloxy)-3-(trifluoromethyl)phenyl)thioureido)carbonyl)pyridin-2-ylamino)acetate
04/29/2008US7365065 Antigonadotrophins; Breast and prostate cancer, endometriosis and benign prostate hyperplasia; regulation of fertility; in-vitro fertilisation; oral administration; inexpensive; 3-Amino-4-chloro-N-[4-chloro-5-(2,3-dihydro-benzo[1,4]oxazine-4-carbonyl)-thiophen-3-ylmethyl]-N-methyl-benzenesulfonamide
04/29/2008US7365063 5-HT6 receptor and/or 5-HT2A receptor modulators; CNS disorders such as Parkinson's disease, Huntington's disease, anxiety, depression, manic depression, psychoses, epilepsy, obsessive compulsive disorders, mood disorders, migraine, Alzheimer's disease, sleep disorders, feeding disorders
04/29/2008US7364804 Pyran derivative, method for manufacturing the same, and light-emitting element containing the pyran derivative
04/29/2008CA2394037C New derivatives of benzene sulfonamide, their preparation process and pharmaceutical compositions that contain them
04/29/2008CA2218887C Piperazino derivatives as neurokinin antagonists
04/28/2008CA2666880A1 Organic compounds
04/24/2008WO2008049123A2 2,4-pyrimidinediamine derivatives as inhibitors of jak kinases for the treatment of autoimmune diseases
04/24/2008WO2008048609A1 Biphenyl sulfonyl and phenyl-heteroaryl sulfonyl modulators of the histamine h3-receptor useful for the treatment of disorders related thereto
04/24/2008WO2008048171A1 N- (2 -hydroxyethyl) -n-methyl- 4- (quinolin- 8-yl (1- (thiazol-4- ylmethyl) piperidin- 4 -ylidene) methyl) benzamide, the process of making it as well as its use for the treatment of pain, anxiety and depression.
04/24/2008WO2008047883A1 Piperazine-substituted benzothiophenes for treatment of mental disorders
04/24/2008WO2008047109A1 Thiazole derivatives as kinase inhibitors
04/24/2008WO2008046226A1 Azacycloalkane derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase
04/24/2008WO2008024765A3 Therapeutic substituted thiazolidinones, oxazolidinones, and related compounds
04/24/2008WO2008020227A3 Antibacterial pyrrolecarboxamides
04/24/2008WO2007032028A8 Thiazolinones and oxazolinones and their use as ptp1b inhibitors
04/24/2008US20080097109 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
04/24/2008US20080097105 Biphenyl-2-ylcarbamic Acid 1-{9-[2-(4-Hydroxy-2-oxo-2,3-dihydrobenzothiazol-7-yl)-ethylamino]nonyl}piperidin-4-yl Ester Bis(trifluoroacetate) Salt; chronic obstructive pulmonary disease, asthma; bronchodilators
04/24/2008US20080097099 Insecticides; for human or veterinary medicine; preparing heterocyclic amide and imine derivatives
04/24/2008US20080096925 Analgesics for neuropathy, surgery, nervous system disorders, headaches, arthritis, psoriasis, respiratory system disorders, and gastrointestinal disorders; ethyl 4-phenyl-4-[1-(phenylmethyl)-1H-imidazol-2-yl]-1-piperidinecarboxylate;
04/24/2008US20080096924 (2R) N-(1-benzylpiperidin-4-yl)-3-cyclohexylmethylthio-2-[(4R)-3-tert-butoxycarbonylthiazolidin-4-ylcarbonylamino]propanamide and hydroxypropyl methylcellulose acetate succinate or hydroxypropyl cellulose; N-type calcium channel blockers; analgesics; oral and nasal formulations; storage stability
04/24/2008US20080096922 N-{[cis-1-(3-methoxyphenyl)-4-(piperidin-4-ylamino)-cyclohexyl]methyl}sulfamide diHCL; tert-butyl [({[cis-4-[(biphenyl-4-ylmethyl)amino]-1-(3-methoxyphenyl)cyclohexyl]methyl}amino)sulfonyl]carbamate; for potentiating expression of low density lipoprotein recepotr; arteriosclerosis; hyperlipidemia
04/24/2008US20080096920 3-{4-[Bis-(quinolin-8-ylcarbamoylmethyl)-amino]-phenyl}-N-hydroxy-acrylamide; 4-(2-Hydroxycarbamoyl-vinyl)-N,N-bis-phenylcarbamoylmethyl-benzamide; useful in treatment of cellular proliferative diseases, for example cancer, autoimmune, allergic and inflammatory diseases, and neurdegenerative disorders
04/24/2008US20080096911 Biphenyl-2-ylcarbamic Acid 1-{9-[2-(4-Hydroxy-2-oxo-2,3-dihydrobenzothiazol-7-yl)-ethylamino]nonyl}piperidin-4-yl Ester Bis(trifluoroacetate) Salt; chronic obstructive pulmonary disease, asthma; bronchodilators
04/24/2008US20080096899 N-Phenyl-2-Pyrimidine-Amine Derivatives and Process for the Preparation Thereof
04/24/2008US20080096885 Methyl 1-(2-fluorophenyl)-2-[(3-methoxy-2-phenylquinolin-4-yl)carbonyl]hydrazinecarboxylate; schizophrenia
04/24/2008US20080096878 CGRP (Calcitonin Gene-Related Peptide); migraine and cluster headaches; 2-(5-Bromo-1'1'-dioxido-2-oxo-2',3',5',6'-tetrahydrospiro[indole-3,4'-thiopyran]-1 (2H)-yl)-N-(2'-oxo-1,1',2',3-tetrahydrospiro[indene-2,3'-pyrrolo[2,3-b]pyridin]-5-yl)acetamide for example; use with other drugs
04/24/2008US20080096876 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia
04/24/2008US20080096874 Oxadiazole Derivative as Dgat Inhibitors
04/24/2008US20080096843 For crops; 3-(2,6-Dichlorophenyl)-4-[(3-pyridyl)hydroxymethyl]-5-trimethylsilylisoxazole for example
04/24/2008US20080096802 administering peroxisome proliferator-activated receptor agonists (PPAR) and sodium glucose co-transporters (SGLTs) inhibitors for the treatment of diabetes and Syndrome X
04/24/2008US20080096193 Quantitative analysis; optical properties; kits
04/24/2008US20080095739 Heterocyclic antiviral compounds
04/24/2008US20080095707 Inhibiting the growth of tumor cells overexpressing MN protein with enzyme inhibitors of carbonic anhydrase (CA 1X) (MN protein); pyridinium derivatives of aromatic heterocyclic sulfonamides; side-effect reduction; antitumor, -carcinogenic, -metastasis agents
04/24/2008DE102006048924A1 Acylaminopyrazole Acylaminopyrazole
04/24/2008CA2673125A1 Compositions and methods for inhibition of the jak pathway
04/24/2008CA2665204A1 Biphenyl sulfonyl and phenyl-heteroaryl sulfonyl modulators of the histamine h3-receptor useful for the treatment of disorders related thereto
04/24/2008CA2664849A1 Azacycloalkane derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase
04/23/2008EP1912983A2 Modulators of cystic fibrosis transmembrane conductance regulator
04/23/2008EP1912982A2 Novel heterocyclic nf- b inhibitors
04/23/2008EP1912981A2 Macrocyclic inhibitors of hepatitis c virus
04/23/2008EP1912980A2 Oxazolidinones bearing antimicrobial activity composition and methods of preparation
04/23/2008EP1912970A2 Acyltryptophanols for fertility control
04/23/2008EP1912966A2 2-oxo-1-pyrrolidine derivatives and their therapeutic use on the central nervous system
04/23/2008EP1912959A2 5-substituted thiazol-2-yl amino compounds and compositions as protein kinase inhibitors
04/23/2008EP1912957A1 Ep4 receptor agonist, compositions and methods thereof
04/23/2008EP1912948A1 Antibacterial quinoline derivatives
04/23/2008EP1912939A1 Metabotropic glutamate-receptor-potentiating isoindolones
04/23/2008EP1912706A2 Novel 5-substituted indole derivatives as dipeptidyl peptidase iv (dpp-iv) inhibitors
04/23/2008EP1597398B1 Method of diagnostic of mastocytosis
04/23/2008EP1333834B1 Antiinflammation agents
04/23/2008EP1305312B1 Tartrate salts of thiazolidinedione derivative
04/23/2008EP1219612B1 2-imino-1,3-thiazine derivatives
04/23/2008EP1216230B1 Fused cycloheptane and fused azacycloheptane compounds and their use as integrin receptor antagonists
04/23/2008CN101166737A Phosphodiesterase 4 inhibitors
04/23/2008CN101166726A Quinoline and quinoxaline derivatives as inhibitors of kinase enzymatic activity
04/23/2008CN101166725A Pyridylacetic acid compound
04/23/2008CN101166723A New compound for the treatinginflammatory disease
04/23/2008CN101166529A Benzotriazole derivatives as cannabinoid receptor antagonists
04/23/2008CN100383132C Azoles as malonyl-COA decarboxylase inhibitors useful as metabolic modulators
04/22/2008US7361682 Indole derivatives as H3 inverse agonists