Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
12/2008
12/02/2008US7459558 Enzyme inhibitor on NO-synthase enzymes; treating STROKE, NEURODEGENERATIVE DISEASES, preventing ISCHEMIC OR HEMORRAGIC CARDIAC OR CEREBRAL INFARCTIONS; inhibiting lipidic peroxidation
12/02/2008US7459556 Process for preparing substituted 8-azabicyclo[3.2.1]octan-3-ols
12/02/2008US7459552 Reacting N-[2,4-bis(methylthio)-6-methylpyridin-3-yl]-2-[4-(2-hydroxyethyl)piperazin-1-yl]acetamide with 5-benzyloxy-2-mercaptobenzimidazole in presence of triphenylphosphine and diethyl azodicarboxylate; acyl-coenzyme A cholesterol acyltransferase (ACAT) inhibitor
12/02/2008US7459473 1-(phenylmethyl)sulfonyl-2-hydroxymethyl pyrrolidine for example; use treating neurological disorders including physically damaged nerves and neurodegenerative diseases; treating alopecia and promoting hair growth
12/02/2008US7459456 e.g. 3-(3-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}phenyl)-1,3-oxazolidin-2-one; serotonin receptor antagonist and inverse agonists, agonists or partial agonists, serotonin reuptake inhibitor; antidepressant, anxiolytic agent
12/02/2008US7459454 Aminopyrazine derivatives and compositions
12/02/2008US7459452 Dihydroxypyrimidine carboxamide inhibitors of HIV integrase
12/02/2008US7459450 metabolic and eating disorders, symptoms of hepatitis C, pain, sexual dysfunction, congestive heart failure, cerebral hemorrhage, anxiety, depression, epileptic seizures, sleep disorders, migraine and allergic rhinitis.
12/02/2008US7459414 Herbicides
12/02/2008CA2424600C Aliphatic nitrogenous five-membered ring compounds
12/02/2008CA2305548C Prostaglandin agonists and their use to treat bone disorders
12/02/2008CA2248300C Sulfonamide-substituted chromans, processes for their preparation, their use as a medicament, and pharmaceutical preparations comprising them
12/02/2008CA2186380C Novel carbamates and ureas as modifiers of multi-drug resistance
11/2008
11/27/2008WO2008144305A1 Diaryl-substituted tetrahydroisoquinolines as histamine h3 receptor and serotonin transporter modulators
11/27/2008WO2008144062A1 Csf-1r inhibitors, compositions, and methods of use
11/27/2008WO2008143759A1 Pyrimidinones as casein kinase ii (ck2) modulators
11/27/2008WO2008143254A1 Pharmaceutical containing pparδ agonist
11/27/2008WO2008142706A2 Novel process for the synthesis of pioglitazone and its salts thereof
11/27/2008WO2008141976A1 Diacylglycerol acyltransferase inhibitors
11/27/2008WO2008141462A1 Novel case of renin inhibitors
11/27/2008WO2008109731A3 Substituted phenoxy n-alkylated thiazoledinedione as estrogen related receptor-alpha modulators
11/27/2008WO2008083367A3 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors
11/27/2008WO2008046072A3 Chemical inducers of neurogenesis
11/27/2008US20080293784 Epothilones c, d, e and f, preparation and compositions
11/27/2008US20080293776 1,2,5-Thiazolidine Derivatives Useful for Treating Conditions Mediated by Protein Tyrosine Phosphatases (Ptpase)
11/27/2008US20080293747 Chemical Synthesis of a Highly Potent Epothilone
11/27/2008US20080293727 Amine hydroxyalkyl sulfonamides as enzyme inhibitors; for example, N-1-(3-((3-acetylamino-4-fluoro-benzenesulfonyl)-benzyl-amino)-(1S,2 syn)-1-benzyl-2-hydroxy-propyl)-2-((quinoline-2-carbonyl)-amino)-succinamide; may be used as anti-viral agents against the HIV-1 and HIV-2 viruses
11/27/2008US20080293720 Pyridinyl Sulfonamide Modulators of Chemokine Receptors
11/27/2008US20080293716 Benzamide rho-kinase (ROCK-1) inhibitors; N-(2-phenylethyl)-5-(4-pyridinyl)-2-thiophenecarboxamide
11/27/2008US20080293711 Chemokine receptor modulators
11/27/2008US20080293684 Heterocyclic Acetophenone Potentiators of Metabotropic Glutamate Receptors
11/27/2008US20080293573 Use as pesticide, microbiocide, or herbicide
11/27/2008US20080292608 Compounds and Compositions as Ppar Modulators
11/27/2008CA2688057A1 Novel case of renin inhibitors
11/27/2008CA2687957A1 Pharmaceutical containing ppar.delta. agonist
11/27/2008CA2686951A1 Diacylglycerol acyltransferase inhibitors
11/27/2008CA2683276A1 Ziprasidone formulations
11/26/2008EP1995246A1 Nitrogenated heterocyclic derivative, and pharmaceutical agent comprising the derivative as active ingredient
11/26/2008EP1995242A1 Novel 1,2,3,4-tetrahydroquinoxaline derivative having glucocorticoid receptor binding activity
11/26/2008EP1995241A1 Inhibitors of ion channels
11/26/2008EP1995240A1 Quinolone derivative or pharmaceutically acceptable salt thereof
11/26/2008EP1994031A1 Use of adenosine a1 and/or dual a1/a2b agonists for production of medicaments for treating diseases
11/26/2008EP1994030A1 Multi-cyclic compounds and method of use
11/26/2008EP1994017A2 Novel heterocyclic nf-kb inhibitors
11/26/2008EP1994015A1 Dibenzyl amine derivatives as cetp inhibitors
11/26/2008EP1993551A2 Potassium channel inhibitors
11/26/2008EP1756084B1 Substituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
11/26/2008EP1740568B1 Benzofuran and benzothiophene derivatives useful for the treatment of cardiovascular disease.
11/26/2008EP1480642B1 Peroxisome proliferator activated receptor modulators
11/26/2008EP1421070B1 New piperidinyl derivates as modulators of chemokine receptor activity
11/26/2008EP1330452B1 Pyrazine derivatives as modulators of tyrosine kinases
11/26/2008EP0945448B1 5-alkoxy-2(3h)-oxazolone compounds and process for the preparation thereof
11/26/2008CN101312966A Benzothiazole cyclobutyl amine derivatives and their use as histamine-3 receptors ligands
11/26/2008CN101312958A 3, 6-dihydro-2-oxo-6H-(1,3,4)thiadiazine derivatives
11/26/2008CN101312956A Substituted 5-phenyl-3,6-dihydro-2-oxo-6H-[1,3,4]thiadiazines
11/26/2008CN100436456C Imidazo [4,5-b] pyridiniummethyl-containing cephem compounds having broad antibacterial spectrum
11/26/2008CN100436452C Pyrazole compounds useful as protein kinase inhibitors
11/26/2008CN100436445C Pyrazole derivative
11/26/2008CN100436421C Dual binding site acetylcholinesterase inhibitors for the treatment of alzheimer's disease
11/25/2008US7456288 Heterocyclic compounds and methods of making and using thereof
11/25/2008US7456211 Enzyme inhibitors as bactericides for infections and as enzyme inhibitors
11/25/2008US7456206 Biaryl heterocyclic compounds and methods of making and using the same
11/25/2008US7456200 Compounds
11/25/2008US7456196 Alzheimer's disease; antihistamine; attention deficit disorder; hyperactivity; bipolar disorder; cognition activators; psychological disorder; anticancer agent; antidepressants; antiepileptic agents; gastrointestinal disorder; analgesics; 6-{2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl}-2-(3-pyridinyl)quinoline
11/25/2008US7456182 Phenylpiperazines
11/25/2008US7456176 Benzotriazine inhibitors of kinases
11/25/2008US7456169 Heterocyclic kinase inhibitors
11/25/2008CA2219747C Aminothiazole derivative, medicament containing the same, and intermediate for preparation of said compound
11/21/2008CA2685967A1 Csf-1r inhibitors, compositions, and methods of use
11/20/2008WO2008141227A1 Novel peptide inhibitors of hepatitis c virus replication
11/20/2008WO2008141020A1 2-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-3-phenyl pyrazines and pyridines and 3-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-2-phenyl pyridines as 5-ht7 receptor antagonists
11/20/2008WO2008140099A1 Tetrazoyloxime derivative and plant disease control agent
11/20/2008WO2008139941A1 Substituted imidazole compound and use thereof
11/20/2008WO2008139416A1 2-cyclopropyl-thiazole derivatives
11/20/2008WO2008139288A2 Substituted heterocyclic derivatives and compositions and their pharmaceutical use as antibacterials
11/20/2008WO2008139287A1 Azetidine derivatives and their use as prostaglandin e2 antagonists
11/20/2008WO2008139152A1 N-oxide-containing pharmaceutical compounds
11/20/2008WO2008138939A1 Pyrazolone derivatives as pde4 inhibitors
11/20/2008WO2008138917A1 Novel aromatic heterocyclic carboxylic acid amide derivatives useful as potassium channel modulators
11/20/2008WO2008138753A1 Hetarylanilines as modulators for amyloid beta
11/20/2008WO2008138733A1 Oxime ester photoinitiators
11/20/2008WO2008138591A2 Bicyclic and heterobicyclic derivatives,processes for preparing them and their uses
11/20/2008WO2008090048A3 3-amino-1,2-benzisothiazole compounds for combating animal pest ii
11/20/2008WO2007110418A3 Substituted 5-hetaryl-4-aminopyrimidines
11/20/2008US20080287504 Such as N-(4-Fluoro-benzyl)-4-(3-phenyl-indole-1-sulfonyl)-benzamide; Cannabinoid-1 (CB1) receptor; dietetics
11/20/2008US20080287449 Aza-tripeptide hepatitis c serine protease inhibitors
11/20/2008US20080287444 Pyrazole compounds useful as protein kinase inhibitors
11/20/2008US20080287439 Pyrimidine compounds
11/20/2008US20080287438 Agent for preventing or treating neuropathy
11/20/2008US20080287424 e.g. N-[amino(imino)methyl]-2-[2-(4-phenoxyphenyl)-5-phenyl-1H-pyrrol-1-yl]acetamide; beta -amyloid deposits and neurofibrillary tangles; cognition activator, neurodegenerative diseases; Alzheimer's disease, Down's syndrome
11/20/2008US20080287409 Phenyl and pyridinyl-1,2,4-oxadiazolone derivatives, processes for their preparation and their use as pharmaceutical compositions
11/20/2008US20080287394 hydroxy-substituted pyrazinopyrrolopyridazine dione compounds; viricide; infection by HIV, AIDS; with other HIV/AIDS antivirals, immunomodulators, antibiotics or vaccines; 2-(2-fluorobenzyl)-10-hydroxy-4,8-dimethyl-7,8-dihydropyrazino[1',2':1,5]-pyrrolo[2,3-d]pyridazine-1,9(2H,6H)-dione
11/20/2008US20080286265 Substituted phenoxy n-alkylated thiazolidinediones as estrogen related receptor-alpha modulators
11/20/2008CA2686909A1 Pyrazolone derivatives as pde4 inhibitors
11/20/2008CA2686754A1 Hetarylanilines as modulators for amyloid beta
11/20/2008CA2686546A1 Novel peptide inhibitors of hepatitis c virus replication
11/20/2008CA2686517A1 Azetidine derivatives and their use as prostaglandin e2 antagonists
11/20/2008CA2685888A1 Substituted heterocyclic derivatives and their pharmaceutical use and compositions
11/20/2008CA2685743A1 2-cyclopropyl-thiazole derivatives
11/20/2008CA2684931A1 Oxime ester photoinitiators