Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773) |
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10/15/2008 | CN101284819A Fused pyridazine derivative compounds and drugs containing these compounds as the active ingredient |
10/15/2008 | CN101284810A Cyano-pyrrolidine and cyano-tetrahydrothiazole derivates |
10/15/2008 | CN100425600C Benzothiazole- and benzoxazole-4,7-dione derivatives and their use as CDC25 phosphatase inhibitors |
10/15/2008 | CN100425592C Indole derivatives |
10/14/2008 | US7435829 Pyrazolyl-substituted heterocycles and their use as phytosanitary products |
10/14/2008 | US7435828 immunosuppressive agents; low dosages; 5-[4-(2-hydroxy-ethoxy)-benz[Z]ylidene]-2-([Z]-isopropylimino)-3-o-tolyl-thiazolidin-4-one |
10/14/2008 | US7435824 Prodrugs of potassium channel inhibitors |
10/14/2008 | US7435823 2,3-Dihydro-4H-1,4-benzoxazine derivatives containing an optionally fused pyridine or pyrimidine ring; 7-((6,7-bis(methyloxy)-4-quinolinyl)oxy)-N-phenyl-2,3-dihydro-4H-1,4-benzoxazine-4-carboxamide; kinase inhibitors; inflammation, angiogenesis and cancer |
10/14/2008 | US7435815 Sulfonylamino-acetic acid derivatives |
10/14/2008 | US7435814 N4-(1,4-Benzoxazin-6-yl)-5-fluoro-N2-[3-(N-methylamino)carbonylmethyleneoxyphenyl]-2,4-pyrimidinediamine or a salt, hydrate, solvate and/or N-oxide; inhibit the IgE and/or IgG receptor signaling cascades that lead to the release of chemical mediators; Syk kinase inhibitors |
10/14/2008 | US7435750 Method of using substituted 3-aryl-5-aryl-[1,2,4]-oxadiazoles and analogs as activators of caspases and inducers of apoptosis and the use thereof |
10/14/2008 | US7435748 Alzheimer's disease; bridged bicycloalkyl spirocyclic sulphonamide derivatives; oral administration |
10/14/2008 | US7435744 Brain disorders; central nervous system disorders; viricides |
10/14/2008 | US7435737 4-(1-Piperazinyl)-2(1H)-quinolone and 4-(1-piperazinyl)quinoline derivatives, e.g., 3-nitro- or 3-alkoxycarbonyl-1-methyl-4-[4-thiophene-2-carbonyl)-piperazine-1-yl]-1H-quinolin-2-one; antitumor and angiogenesis inhibitor, antiinflammatory, antidiabetic agent, autoimmune disorder |
10/14/2008 | US7435736 e.g. (2R-trans) [4-(4-azetidin-3-yl-piperazin-1-yl)-2-benzyl-piperidin-1-yl]-(3,5-bis-trifluoromethyl-phenyl)-methanone;tachykinins, substance P inhibitor; antidepressant, anxiolytic, antiinflammatory agent, cognition activator; neurodegenerative diseases; addiction, sleep, eating disorders |
10/14/2008 | US7435734 Such as N-(2-ethoxybenzyl)-5-hydroxy-1-methyl-2-(4-methylphenyl)-6-oxo-1,6-dihydropyrimidine-4-carboxamide; inhibitors of HIV replication; with other HIV/AIDS antivirals, anti-infectives, immunomodulators, antibiotics or vaccines; AIDS |
10/14/2008 | US7435729 using estrogen antagonist ; anticancer agents |
10/14/2008 | CA2497345C Novel quaternary ammonium compounds |
10/14/2008 | CA2382880C N-cyclopentyl modulators of chemokine receptor activity |
10/14/2008 | CA2309328C Cyclic amine derivatives and their use as drugs |
10/14/2008 | CA2222138C Method of preparing 3-haloalkyl-1h-pyrazoles |
10/09/2008 | WO2008121877A2 Cftr inhibitor compounds and uses thereof |
10/09/2008 | WO2008121861A2 Pyrazole and pyrrole compounds useful in treating iron disorders |
10/09/2008 | WO2008121670A1 Pyrimidine hydrazide compounds as pgds inhibitors |
10/09/2008 | WO2008121592A2 Acetyl coenzyme a carboxylase inhibitors |
10/09/2008 | WO2008121558A1 1, 3-thiazol-2 (3h) -ylidene compounds as cannabinoid receptor ligands |
10/09/2008 | WO2008121415A2 Improved process for preparing quetiapine fumarate |
10/09/2008 | WO2008120759A1 Urea compound and use thereof |
10/09/2008 | WO2008120754A1 Picolinamide compound |
10/09/2008 | WO2008120744A1 Five-membered cyclic amide compound and use thereof |
10/09/2008 | WO2008120725A1 Novel pyrrolinone derivative and medicinal composition containing the same |
10/09/2008 | WO2008120661A1 Novel fused pyrrole derivative |
10/09/2008 | WO2008119694A1 Benzimidazole cannabinoid agonists |
10/09/2008 | WO2008119657A1 Imidazolidinone derivatives |
10/09/2008 | WO2008119563A2 Method for producing epothilone derivatives by means of selective catalytic epoxidation |
10/09/2008 | WO2008101682A3 Iminipyridine derivatives and their uses as microbiocides |
10/09/2008 | WO2008022002A3 2-amido-4-isoxazolyl thiazole compounds exhibiting atp-utilizing enzyme inhibitory activity, and compositions, and uses thereof |
10/09/2008 | WO2007149478A3 Pyrazine derivatives with extended conjugation and uses thereof |
10/09/2008 | US20080249148 For contraception, treating or preventing fibroids, uterine leiomyomata, endometriosis, dysfunctional bleeding, polycystic ovary syndrome, and hormone-dependent carcinomas, providing hormone replacement therapy, stimulating food intake, and synchronizing estrus |
10/09/2008 | US20080249111 Piperdine Derivatives as CCR5 Inhibitors |
10/09/2008 | US20080249095 tyrosine kinase inhibitors, in particular Met kinase; antitumor agents;1-(Benzo-1,2,5-thiadiazol-5-ylmethylcarbonyl)-3-(2,4-dimethoxyphenyl)-4,5-dihydro-1H-pyrazole; leukemia, carcinomas |
10/09/2008 | US20080249093 immunosuppressive, anti-inflammatory and hemostatic agents to modulate leukocyte trafficking, sequestering lymphocytes in secondary lymphoid tissues, and enhancing vascular integrity; safer and more effective; 3-(4-(5-(3-Cyano-4-isopropyloxyphenyl)-1,2,4-oxadiazol-3-yl)-3-methylphenyl)propanoic acid |
10/09/2008 | US20080249084 For diabetes, obesity or metabolic syndrome; improve physicochemical (like stability) and biological (inhibitor activity, specificity, bioavailability, metabolism) profiles; 11Beta-hydroxysteroid dehydrogenase 1 inhibitors; 3-chloro-4-[4-methyl-5-(1-phenyl-cyclopropyl)-4H-[1,2,4]triazol-3-yl]-benzamide |
10/09/2008 | CA2682629A1 Pyrimidine hydrazide compounds as pgds inhibitors |
10/09/2008 | CA2682473A1 Novel pyrrolinone derivative and pharmaceutical composition comprising the same |
10/09/2008 | CA2681806A1 Process for preparing epothilone derivatives by selective catalytic epoxidation |
10/09/2008 | CA2681586A1 1, 3-thiazol-2 (3h) -ylidene compounds as cannabinoid receptor ligands |
10/08/2008 | EP1978023A1 Pyridazines as fungicides |
10/08/2008 | EP1978019A1 3-phenyl-pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto |
10/08/2008 | EP1977749A1 Use of cyclooxygenase-2 inhibitors in the treatment and prevention of neoplasia |
10/08/2008 | EP1976851A2 Phenoxy-substituted pyrimidines as adenosine receptor antagonists |
10/08/2008 | EP1976849A2 Compounds for the treatment of inflammatory disorders |
10/08/2008 | EP1976836A2 Nitrogen-containing bicyclic heteroaryl compounds for the treatment of raf protein kinase-mediated diseases |
10/08/2008 | EP1976829A2 N-(6-membered aromatic ring)-amido anti-viral compounds |
10/08/2008 | EP1881830B1 4-phenyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline derivatives the treatment of infertility |
10/08/2008 | EP1660493B1 Peptidyl heterocyclic ketone derivatives and preparation processes |
10/08/2008 | EP1633348B1 4- BROMO - 5 - (2- CHLORO - BENZOYLAMINO) - 1H - PYRAZOLE - 3 - CARBOXYLIC ACID AMIDE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ B sb 1 /sb RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES |
10/08/2008 | EP1569931B1 Heterocyclic compounds as ccr5 antagonists |
10/08/2008 | EP1478628B1 2-amino-4-bicyclyl amino-6h-1.3.5-triazines, method for the production and use thereof as herbicides and plant growth regulators |
10/08/2008 | CN101282979A Composition containing chloromethyl phosphate derivative with improved stability and process for producing the same |
10/08/2008 | CN101282972A Piperidine and piperazine derivatives as P2X3 antagonists |
10/08/2008 | CN101282971A Chemical process for the preparation of benzoxazole derivatives used as pesticides |
10/08/2008 | CN101282970A Chemical process |
10/08/2008 | CN101282969A Bicyclic aryl-sulfonic acid [1,3,4]-thiadiazol-2-yl-amides, processes for their preparation and their use as pharmaceuticals |
10/08/2008 | CN101282951A N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, processes for their preparation and their use as pharmaceuticals |
10/08/2008 | CN101282950A Novel benzothiazolone derivatives |
10/08/2008 | CN101282948A Phosphatidylinositol 3-kinase inhibitors and methods of their use |
10/08/2008 | CN101282942A Imidazole derivatives for the treatment of anxiety and related diseases |
10/08/2008 | CN101279971A 4,4-difluoro-1,2,3,4-tetrahydro-5h-1-benzoazepine derivative or salt of the same |
10/08/2008 | CN100423721C Thrombopoietin mimetics |
10/07/2008 | US7432379 3-Amido-5-substituted pyrazole derivatives and related compounds useful as bradykinin B1 receptor antagonists to relieve adverse symptoms in mammals mediated, at least in part, by bradykinin B1 receptor including pain, inflammation, septic shock, scarring process |
10/07/2008 | US7432374 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same |
10/07/2008 | US7432292 Anticancer agents; autoimmune diseases; antiinflammatory agents; ; graft versus host disease; Crohn's diseases; skin disorders |
10/07/2008 | US7432291 Anticancer, antitumor agents; compounds are 1-(2-(phenethenyl)oxazol-4-ylmethoxy)-4-(1,2,3-triazolylethoxymethyl)-benzenes or corresponding derivatives where oxazole is replaced by thiazole |
10/07/2008 | US7432290 Claimed is 1-Cyanobutan-2-yl-1-[3-[3-[3-methoxy-4-(oxazol-5-yl)phenyl]ureido]phenyl] ethylcarbamate, AVN 944, VX-944 |
10/07/2008 | US7432289 5-Acylamino-1,1′-biphenyl-4-carboxamide derivatives and their use as P38 kinase inhibitors |
10/07/2008 | US7432287 e.g. 3-(6-ethanesulfonylpyridin-3-yloxy)-5-(2-hydroxy-1-methyl-ethoxy)-N-(1-methyl-1H-pyrazol-3-yl)benzamide; glucokinase activator; antidiabetic agent; obesity, insulin resistance |
10/07/2008 | US7432286 Pharmaceutically active sulfonyl hydrazide derivatives |
10/07/2008 | US7432275 Carboxylic acid, phosphate or phosphonate substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators |
10/07/2008 | US7432270 N-aroyl cyclic amines |
10/07/2008 | US7432269 Arylpiperaszine derivatives, to the process for the production thereof and to the use thereof as therapeutic agents |
10/07/2008 | US7432268 17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases |
10/07/2008 | US7432264 Antibacterial compounds such as (S)-2-cyano-1-(trans-4-(5-nitro-2-pyridylamino)cyclohexylamino )acetylpyrrolidine; activity against Gram-negative and Gram-positive pathogens, including a methicillin-resistant S. aureus strain |
10/07/2008 | US7432260 Pyrimidine compounds |
10/07/2008 | US7432257 Piperdinyl-phenoxazine and phenothiazine derivatives as δ-opioid modulators |
10/07/2008 | CA2435946C Piperidine derivatives as neurokinin 1 antagonists |
10/07/2008 | CA2433772C Pyrimidine matrix metalloproteinase inhibitors |
10/07/2008 | CA2426009C Cholesterol lowering benzo[b]thiophenes and benzo[d]isothiazoles |
10/07/2008 | CA2392971C 2,4-diaminopyrimidine compounds useful as immunosuppressants |
10/07/2008 | CA2248143C Process to prepare oxazolidinones |
10/02/2008 | WO2008118718A2 2-aminopyridine analogs as glucokinase activators |
10/02/2008 | WO2008117982A1 Heterocyclic carboxylic acid derivatives and pharmaceutical composition for inhibiting lipid accumulation containing same |
10/02/2008 | WO2008117862A1 Novel (2-aminophenyl)pyridinecarboxamide derivative having urea structure |
10/02/2008 | WO2008117050A1 Pyrazolyl-amino-substituted pyrazines and their use for the treatment of cancer |
10/02/2008 | WO2008116881A1 Substituted pyrrolidine amides, the production thereof, and the use thereof as medications |
10/02/2008 | WO2008116831A1 Quinoline compounds suitable for treating didorders that respond to modulation of the serotonin 5-ht6 receptor |
10/02/2008 | WO2008116620A1 8-oxy-quinoline derivatives as bradykinin b2 receptor modulators |
10/02/2008 | WO2008098949A3 Process for the synthesis of 2-aminothiazole compounds as kinase inhibitors |
10/02/2008 | WO2008097640A3 Triazole compounds that are useful in the treatment of proliferative disorders, such as cancer |
10/02/2008 | WO2008092954A3 Polymorphic forms of a macrocyclic inhibitor of hcv |