Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
12/2008
12/31/2008EP2007760A1 Novel substituted-1, 1-dioxo-benzo[1,2,4]thiadizin-3-ones, preparation method thereof, and pharmaceutical composition containing the same
12/31/2008EP2007748A2 Synthesis and regioselective substitution of 6-halo- and 6-alkoxy nicotine derivatives
12/31/2008EP2007747A1 Process for preparing heterocyclic derivatives
12/31/2008EP2007745A2 Fungicide n-cyclopropyl-sulfonylamide derivatives
12/31/2008EP2007729A1 Substituted tetrahydroisoquinoline compounds, their preparation and use in medicaments
12/31/2008EP2007720A1 Benzamide derivatives as inhibitors of histone deacetylase
12/31/2008EP2007717A1 Novel sulfonamide compounds
12/31/2008EP1546099B1 3,6-disubstituted azabicyclo 3.1.0 hexane derivatives useful as muscarinic receptor antagonists
12/31/2008EP1435785B1 Iminobenzoxazines, iminobenzothiazines and iminoquinazolines for controlling invertebrate pests
12/31/2008EP1309587B1 Cinnoline compounds
12/31/2008CN101336239A Substituted oxindol-derivatives, medicaments containing said derivatives and use thereof
12/31/2008CN101336235A 1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors
12/31/2008CN101333196A 1,2,4-triazole derivatives containing a sulphamate group as aromatase inhibitors
12/31/2008CN101333192A Biaryl substituted pyrazoles as sodium channel blockers
12/31/2008CN100447140C 7-([1,4]dioxan-2-yl)-benzothiazole derivatives as adenosine receptor ligands
12/31/2008CN100446767C Use of GAL3 receptor antagonists for treatment of. depression and/or anxiety and compounds useful in such methods
12/31/2008CA2690378A1 Phthalazine compounds, compositions and methods of use
12/31/2008CA2690176A1 Novel herbicides
12/31/2008CA2686224A1 Piperazine compounds having herbicidal action
12/30/2008US7470807 Suppress production of both prostaglandins and leukotrienes and have reduced side effects; treatment of various inflammatory diseases, autoimmune diseases, allergic diseases, pain and fibrosis; for example, methyl 3-[3-acetylamino-4-cyclopentyloxy-5-(naphthalen-2-yl)phenyl]propionate
12/30/2008US7470798 7,8-bicycloalkyl-chroman derivatives
12/30/2008US7470793 Thiazol-(bi)cycloalkyl-carboxanilides
12/30/2008US7470792 Process for the preparation of epothilone derivatives, new epothilone derivatives as well as new intermediate products for the process and the methods of preparing same
12/30/2008US7470790 for treatment of various neurodegeneration, including that from stroke, Alzheimer's disease, Parkinson's disease, and Huntington's disease; [6-(1-benzyl-4-hydroxy-pyrrolidin-3-ylmethyl)-pyridin-2-yl]-carbamic acid tert-butyl ester
12/30/2008US7470712 Amino-benzazoles as P2Y1 receptor inhibitors
12/30/2008US7470710 Such as 2-Benzofuranylmethyl-1-((5-(4-fluorophenyl)-2-methyl-thiazolyl) carbonyl)piperidine; obesity, type 2 diabetes, sleep disorders; strokes, blocking emetic response
12/30/2008US7470708 Acidic quinoline derivatives and their use for the prevention and/or treatment of hyperglycaemia-related pathologies
12/30/2008US7470701 e.g. 3-(4-fluorophenyl)-N-{5-[2-(methylamino)pyrimidin-4-yl]thien-2-yl}propanamide; PKB/Akt kinase inhibitor; anticarcinogenic agent; carcinoma, cancer metastases, squamous cell carcinoma, esophageal squamous cell carcinoma, oral carcinoma, cutaneous T cell lymphoma, Hodgkin's lymphoma
12/30/2008US7470700 Such as 2-[2-(3-Amino-piperidin-1-yl)4-oxo-4H-quinazolin-3-ylmethyl]-benzonitrile; type 2 diabetes mellitus, diabetic dislipidemia, impaired glucose tolerance
12/30/2008US7470699 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
12/30/2008US7470686 e.g. 1,3-benzothiazol-2-yl (2-chloral -4-pyrimidinyl)acetonitrile; Jun N -terminal kinase inhibitor; anticarcinogenic agent; neuronal disorders, autoimmune diseases, cardiovascular disordres
12/30/2008US7470685 e.g. 1-(2-(4-(N'-(3-Methyl-benzylidene)-hydrazino)-6-morpholin-4-yl-pyrimidin-2 -yloxy)-ethyl)-1H-pyridin-2-one; control interleukin production; antiinflammatory, antidiabetic agent; interleukin IL-12 overproduction-related disorder: rheumatoid arthritis, sepsis, Crohn's disease, multiple sclerosis
12/30/2008US7470681 Pyrimidine compounds
12/30/2008CA2441771C Dihydro-benzo[b][1,4]diazepin-2-one derivatives as mglur2 antagonists i
12/30/2008CA2429850C Ep4 receptor selective agonists in the treatment of osteoporosis
12/30/2008CA2356300C 3-azabicyclo[3.1.0]hexane derivatives useful in therapy
12/30/2008CA2312098C A process for the preparation of ring-opened epothilone intermediates which are useful for the preparation of epothilone analogs
12/30/2008CA2245587C Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
12/25/2008US20080319188 Novel pyridine derivatives and pyrimidine derivatives (3)
12/25/2008US20080319033 3-{3-[5-(4-acetylphenyl)-4-methylthiazol-2-yl]-ureido}-N-tert-butylpropionamide, exhibiting phosphatidylinositol 3-kinase inhibitory activity and used for treating respiratory system disorders, such as asthma
12/25/2008US20080319024 Rosiglitazone Phosphate and Polymorphic Forms
12/25/2008US20080319017 Non-Anilinic Derivatives of Isothiazol-3(2H)-Thione 1,1-Dioxides As Liver X Receptor Modulators
12/25/2008US20080319011 Protein tyrosine kinase enzyme inhibitors
12/25/2008US20080318984 Compounds Having Activity in Correcting Mutant-Cftr Processing and Uses Thereof
12/25/2008US20080318978 Hyperaldosteronism; 4-(5,6,7,8-Tetrahydroimidazo[1,5-a]phyridin-5-yl)cyclohexanecarbonitrile; 1-[3-(5,6,7,8-Tetrahydroimidazo[1,5-a]pyridin-8-yl)pyrrolidin-1-yl]ethanone
12/25/2008US20080318954 Compounds
12/25/2008US20080318944 N-aroyl cyclic amine derivatives as orexin receptor antagonists
12/25/2008US20080318937 Tricyclic delta-opioid modulators
12/25/2008US20080318936 Substituted 5-Phenyl-3,6-Dihydro-2-Oxo-6H-1,3,4-Thiadiazines
12/25/2008US20080318933 5-Sulfonyl-1-Piperidinyl Substituted Indole Derivatives as 5-Ht6 Receptor Antagonists for the Treatment of Cns Disorders
12/25/2008US20080318927 Substituted monocyclic CGRP receptor antagonists
12/25/2008US20080317671 Non-imidazole heterocyclic compounds
12/24/2008WO2008157575A1 Protein kinase inhibitors and methods for using thereof
12/24/2008WO2008157500A1 Aminoquinazoline cannabinoid receptor modulators for treatment of disease
12/24/2008WO2008157407A2 Thiadiazole, oxadiazole and triazole derivatives for treating leukemia
12/24/2008WO2008157162A1 Dipeptide analogs as coagulation factor inhibitors
12/24/2008WO2008156208A1 5-phenyl-3-pyridazinone derivative
12/24/2008WO2008156174A1 Pyrazinamide compound
12/24/2008WO2008156102A1 Pyrazolone derivative and pde inhibitor containing the same as active ingredient
12/24/2008WO2008156094A1 Pyridazinone derivative and pde inhibitor containing the same as active ingredient
12/24/2008WO2008156092A1 Azolylmethylidenehydrazine derivative and use thereof
12/24/2008WO2008154817A1 Bromo-phenyl substituted thiazolyl dihydropyrimidines
12/24/2008WO2008125839A3 Pyrimidine derivatives as inhibitors of phosphatidylinositol-3-kinase
12/24/2008WO2008121861A3 Pyrazole and pyrrole compounds useful in treating iron disorders
12/24/2008WO2008057856A3 Modulators of glucocorticoid receptor, ap-1 and/or nf-kappab activity and use thereof
12/24/2008WO2008033455A3 Biphenyl and heteroaryl phenyl derivatives as protein tyrosine phosphatases inhibitors
12/24/2008WO2008010089A3 Process for preparation of intermediates of rosiglitazone, rosiglitazone and polymorphic forms thereof
12/24/2008EP2004641A1 Hiv inhibiting 5-(hydroxymethylene and aminomethylene) substituted pyrimidines
12/24/2008EP2004639A2 Processes for the synthesis of azetidinone
12/24/2008EP2004635A1 Substituted enaminocarbonyl compounds
12/24/2008EP2004632A1 Hiv inhibiting 5-amido substituted pyrimidines
12/24/2008EP2004625A2 C-met protein kinase inhibitors for the treatment of proliferative disorders
12/24/2008EP2004601A1 Novel dipeptidyl peptidase iv inhibitors and processes for their preparation and pharmaceutical compositions containing them
12/24/2008EP2003975A1 3-amino-1,2-benzisothiazole compounds for combating animal pest
12/24/2008EP1805169B1 Histamine h3 receptor inhibitors, their preparation and therapeutic uses
12/24/2008EP1554274B1 1-acyl-pyrrolidine derivatives for the treatment of viral infections
12/24/2008EP1551804B1 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
12/24/2008CN101331125A N-(5-membered aromatic ring)-amido anti-viral compounds
12/24/2008CN101328171A Bromophenyl-substituted thiazole dihydropyrimidine
12/24/2008CN101328170A Fluorophenyl-substituted thiazole dihydropyrimidine
12/24/2008CN101328169A Diethylcarbamyl-substituted thiazole dihydropyrimidine
12/24/2008CN101328168A Diethylcarbamyl-substituted thiazole dihydropyrimidine
12/24/2008CN101328163A Compounds, compositions and methods
12/24/2008CN101328150A 新的苯并咪唑衍生物 New benzimidazole derivatives
12/24/2008CN100445274C 2,1,3-benzothiadiazoles for use as electronic active components
12/24/2008CN100445271C Amide derivative
12/24/2008CN100445270C Pyrimidine compounds
12/24/2008CA2692249A1 Pyrazolone derivative and pde inhibitor containing the same as active ingredient
12/24/2008CA2692248A1 Pyridazinone derivative and pde inhibitor containing the same as active ingredient
12/24/2008CA2692170A1 Azolylmethylidenehydrazine derivative and use thereof
12/24/2008CA2691100A1 Protein kinase inhibitors and methods for using thereof
12/24/2008CA2691056A1 Bromo-phenyl substituted thiazolyl dihydropyrimidines for treating and preventing hepatitis b infections
12/24/2008CA2687255A1 Heteroarylamide pyrimidone derivatives
12/23/2008US7468380 Nitrogen-containing aromatic derivatives
12/23/2008US7468368 Piperazinylacylpiperidine derivatives, their preparation and therapeutic use thereof
12/23/2008US7468367 depression; anxiety; addictions; obsessive compulsive disorder; affective neurosis/disorder; depressive neurosis/disorder, anxiety neurosis; dysthymic disorder; behaviour disorder; mood disorder; sexual dysfunction; psychosexual dysfunction; sex disorder, sexual disorder; schizophrenia; manic depression;
12/23/2008CA2560580C Imidazole compounds for inhibition of a.beta.-peptide production and for modulation of the notch signaling pathway
12/23/2008CA2442557C Dihydro-benzo¬b|¬1,4|diazepin-2-one derivatives as mglur2 antagonists ii
12/23/2008CA2424664C Novel non-imidazole compounds
12/18/2008WO2008154642A2 Antibacterial agents