Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
06/2000
06/28/2000CN1258283A Cyclic diamine compounds and medicine contg. same
06/28/2000CN1053905C Oxadiazine derivs., their preparing process and use, intermediates for preparing same
06/28/2000CN1053904C N-pyridyl carboxamides and derivs. processes for their preparation and pharmaceutical compositions contg. them
06/27/2000US6080873 Fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
06/27/2000US6080868 As a quencher in a reporter-quencher energy-transfer dye pair for nucleic acid hybridization assays
06/27/2000US6080860 Urea compound where one of the urea nitrogens is part of an (un)substituted 5 or 6 membered ring and/or the other urea nitrogen is substituted with a 2-cyano-4,5-dialkoxyphenyl group; reacting with electrophile to form a leaving group
06/27/2000US6080776 Used as a microbiocide for crop protection
06/27/2000US6080774 Substituted biphenylsulfonamide endothelin antagonists
06/27/2000US6080773 Benzylamine derivatives which are useful in treating psychiatric disorders
06/27/2000US6080764 Superoxide radical inhibitor
06/27/2000US6080760 Treating benign prostatic hyperplasia; complement slower-acting therapeutics by providing acute relief; induce relaxation of the lower urinary tract to decrease difficulty in urination and sexual dysfunction
06/27/2000US6080745 For treating or preventing disorders of dopamine system, such as schizophrenia
06/27/2000US6080743 2,3-dioxo-1,2,3,4-tetrahydro-quinoxalinyl derivatives
06/27/2000US6080738 Heterocyclic amide compounds and medicinal uses thereof
06/27/2000US6080702 Herbicidal heterocyclic benzisoxazoles and benzisoxazolidinones
06/27/2000CA2188427C Neurotransmitter release enhancers
06/27/2000CA2017193C N-(aryloxyalkyl)heteroarylpiperidines and-heteroarylpiperazines, a pro cess for their preparation and their use as medicaments
06/22/2000WO2000035917A1 1,4-benzodiazepinone derivatives and their use as integrin antagonists
06/22/2000WO2000035916A1 Herbicidal 4-benzoylisoxazoles
06/22/2000WO2000035915A1 Piperazine derivatives
06/22/2000WO2000035914A1 Optically active pyridyl-4h-1,2,4-oxadiazine derivative and its use in the treatment of vascular diseases
06/22/2000WO2000035913A1 4-trifluoromethyl-3-oxadiazolyl pyridines, methods for the production thereof, agents containing these compounds, and their use as pesticides
06/22/2000WO2000035912A1 4-trifluoromethyl-3-oxazolylpyridines, method for producing them, products containing the same, and their use as pesticides
06/22/2000WO2000035911A1 Heteroaryl-cyclic acetals
06/22/2000WO2000035908A1 4-alkenyl (and alkynyl) oxindoles as inhibitors of cyclin-dependent kinases, in particular cdk2
06/22/2000WO2000035891A1 Morpholinone and morpholine derivatives and uses thereof
06/22/2000WO2000035890A1 Novel heterocyclic compounds and drug compositions containing the same
06/22/2000WO2000035886A2 (hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors
06/22/2000WO2000035877A1 Heterocyclic piperidines as modulators of chemokine receptor activity
06/22/2000WO2000035864A1 New biphenyl and biphenyl-analogous compounds as integrin antagonists
06/22/2000WO2000035454A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000WO2000035453A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000WO2000035452A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000WO2000035451A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000WO2000035449A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000WO2000035285A1 4-haloalkyl-3-heterocyclylpyridines and 4-haloalkyl-5-heterocyclyl-pyrimidines and their use as repellents
06/22/2000CA2355249A1 Protease inhibitors
06/22/2000CA2355201A1 Morpholinone and morpholine derivatives and uses thereof
06/22/2000CA2355161A1 Biphenyl and biphenyl-analogous compounds as integrin antagonists
06/22/2000CA2355079A1 Novel heterocyclic compounds and drug compositions containing the same
06/22/2000CA2354875A1 Piperazine derivatives
06/22/2000CA2354873A1 4-alkenyl (and alkynyl) oxindoles as inhibitors of cyclin-dependent kinases, in particular cdk2
06/22/2000CA2353897A1 1,4-benzodiazepinone derivatives and their use as integrin antagonists
06/22/2000CA2350730A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000CA2348923A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000CA2347912A1 Heterocyclic piperidines as modulators of chemokine receptor activity
06/22/2000CA2347909A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000CA2347770A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/22/2000CA2346933A1 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/21/2000EP1009742A1 5,5-disubstituted-1,5-dihydro-4,1-benzoxazepin-2(3h)-ones useful as hiv reverse transcriptase inhibitors
06/21/2000EP1009738A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
06/21/2000EP1009405A1 Pyrrolidine and piperidine modulators of chemokine receptor activity
06/21/2000DE19858193A1 4-Trifluormethyl-3-oxadiazolylpyridine, Verfahren zu ihrer Herstellung, sie enthaltende Mittel und ihre Verwendung als Schädlingsbekämpfungsmittel 4-trifluoromethyl-3-oxadiazolylpyridine, processes for their preparation, compositions containing them and their use as pesticides
06/21/2000DE19858192A1 4-Trifluormethyl-3-oxazolylpyridine, Verfahren zu ihrer Herstellung, sie enthaltende Mittel und ihre Verwendung als Schädlingsbekämpfungsmittel 4-trifluoromethyl-3-oxazolylpyridine, processes for their preparation, compositions containing them and their use as pesticides
06/21/2000DE19858191A1 4-Haloalkyl-3-heterocyclylpyridine und 4-Haloalkyl-5-heterocyclyl-pyrimidine und ihre Verwendung als Repellentien 4-haloalkyl-3-heterocyclylpyridine and 4-haloalkyl-5-heterocyclyl-pyrimidines and their use as repellents
06/21/2000CN1257486A Oxazolidinone antibacterial agents having a thiocarbonyl functionality
06/21/2000CN1053666C Benzoheterocylic compounds and process for preparing medicated salt thereof
06/21/2000CN1053661C Method for the preparation of 2-perflouoroalkyl-3-oxazolin-5-one
06/21/2000CN1053657C Didepside phthaleins based internal parasite compositions, novel didepside phthaleins and preparation process thereof
06/20/2000US6077861 Modulators of the large-conductance calcium-activated potassium (bk) channels, therefore, useful in the treatment of ischemic stroke
06/20/2000US6077850 Useful for treating cyclooxygenase-2 mediated disorders, such as inflammation and inflammation-related disorders
06/20/2000US6077813 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
06/20/2000US6077812 Cycloimido-substituted benzofused heterocyclic herbicides
06/15/2000WO2000034437A2 Inhibitors of prenyl-protein transferase
06/15/2000WO2000034274A1 Cyclohexylpiperidine derivatives
06/15/2000WO2000034273A2 3-(heterocyclyl)-substituted benzoylpyrazols
06/15/2000WO2000034272A2 3-(heterocyclyl)-benzoylpyrazole-derivatives
06/15/2000WO2000034255A1 Substituted thiazoles for treatment of human diseases involving modulators of p-, l- and e- selectin
06/15/2000WO2000034252A2 Process for the preparation of cryptophycin derivatives
06/15/2000WO2000034247A2 Method for producing pyrazolylbenzoyl derivatives and novel pyrazolylbenzoyl derivatives
06/15/2000WO2000033836A1 5-membered heterocycles for the treatment of human diseases involving modulators of selectins
06/15/2000DE19857202A1 New benzimidazolyl amidine or nitrile compounds, useful as thrombin inhibitors or antithrombotic agents, for treating deep leg vein thrombosis
06/15/2000CA2353573A1 3-(heterocyclyl)-benzoylpyrazole-derivatives
06/14/2000EP1007525A1 Aminometyl oxooxazolidinyl benzene derivatives
06/14/2000EP1007524A1 Indole derivatives as 5-ht1b and 5-ht1d agonists
06/14/2000EP1007520A1 2-aminopyridines containing fused ring substituents as nos inhibitors
06/14/2000EP1007518A1 Solid and liquid-phase synthesis of benzoxazoles and benzothiazoles and their use
06/14/2000EP1007042A1 Novel heteroaryl compounds for the modulation of protein tyrosine enzyme related cellular signal transduction
06/13/2000US6075147 Carbamoyl substituted heterocycles
06/13/2000US6075040 Obesity and diabetes
06/13/2000US6075039 5HT receptor binding benzimidazolylpiperidines
06/13/2000US6075016 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity
06/13/2000CA2014062C Pyridine derivatives
06/08/2000WO2000032599A1 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
06/08/2000WO2000032588A2 Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
06/08/2000WO2000032575A1 β-ALANINE DERIVATIVES AS α4 INTEGRIN INHIBITORS
06/08/2000WO2000032216A1 Peptoid and nonpeptoid containing alpha-keto oxadiazoles as serine protease inhibitors
06/08/2000WO2000032190A1 Compositions and methods for the treatment of alzheimer's disease, central nervous system injury, and inflammatory diseases
06/08/2000WO2000009103A9 N-linked sulfonamides of n-heterocyclic carboxylic acids or isosteres for vision and memory disorders
06/08/2000CA2351062A1 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
06/08/2000CA2347701A1 .beta.-alanine derivatives as .alpha.4 integrin inhibitors
06/07/2000EP1006114A1 Pyrazole derivatives and cox inhibitors containing them
06/07/2000EP1005469A1 Oxazolidinone derivatives and their use as antibacterial agents
06/07/2000EP1005468A1 Antibiotic oxazolidinone derivatives
06/07/2000EP1005467A1 Benzothiophene derivatives as herbicides
06/07/2000EP1005459A1 Substituted isoquinolines as anticonvulsivants
06/07/2000EP1005455A1 Method for producing substituted-2-nitroguanidine derivatives
06/07/2000EP1005448A2 Novel inhibitors of aggrecanase and matrix metalloproteinases for the treatment of arthritis
06/07/2000EP1005445A1 N-alkanoylphenylalanine derivatives
06/07/2000EP1005356A1 Novel antibacterial agents