Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
09/2000
09/19/2000US6121282 3-(carboxy, amido, cyano, or hydroxyaminocarbonyl)-6 or 7-substituted-1,2,3,4-tetrahydroisoquinoline compounds
09/19/2000US6121260 Appetite stimulation with dosage of neuropeptide y (npy) receptor agonist
09/19/2000US6121258 For treatment of arthritis, cancer, cardiovascular disorders, skin disorders, ocular disorders, inflammation, gum disease
09/14/2000WO2000053599A1 Pesticidal hetero-substituted oxadiazine compounds
09/14/2000WO2000053582A1 HETEROCYCLIC COMPOUNDS HAVING EFFECT OF ACTIVATING NICOTINIC ACETYLCHOLINE α4β2 RECEPTOR
09/14/2000WO2000053573A1 Medicinal compositions with [2.2.1] and [3.1.1] bicycloskeleton antagonistic to both of pgd2/txa2 receptors
09/14/2000WO2000037422A3 Ion channel modulating agents
09/14/2000WO1999063999A8 H1-histamine receptor antagonists
09/14/2000CA2366612A1 Pesticidal hetero-substituted oxadiazine compounds
09/14/2000CA2366260A1 Heterocyclic compounds having effect of activating .alpha.4.beta.2 nicotinic acetylcholine receptors
09/13/2000EP1035122A1 Heterocyclic subsituted isoxazolidines and their use as fungicides
09/13/2000EP1035115A1 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists
09/13/2000EP1034176A1 Thiophene-sulfonamide compounds
09/13/2000EP1034175A1 Substituted phenyloxazolidinones and their use as antibiotics
09/13/2000EP1034167A1 Alpha-alkylthio substituted pyrimidine ethers and thioethers as viral reverse transcriptase inhibitors
09/13/2000EP1034164A1 Substituted beta-alanine derivatives as cell adhesion inhibitors
09/13/2000EP0691962B1 1-amino-3-phenoxy propane derivatives as modulators of multi-drug resistance
09/13/2000CN1266431A Aroyl-piperazine derivatives, their preparation and their use as tachykinin antagonists
09/13/2000CN1266428A Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
09/13/2000CN1056372C Thiazolidinedione derivatives, their production and use
09/13/2000CN1056370C 4-aryloxy (arylthio or arylamino) pyrimidine derivative with herbicide active, and preparation process thereof
09/12/2000US6117999 Chemical intermediate for nelfinavir
09/12/2000US6117893 Heterocyclic compounds having anti-diabetic activity and their use
09/12/2000CA2105384C Treatment of addiction to drugs and substances of abuse
09/08/2000WO2000052032A1 Heterocyclic compounds, intermediates thereof and elastase inhibitors
09/08/2000WO2000052003A1 A process for the preparation of taxanes from 10-deacetylbaccatin iii
09/08/2000WO2000051998A1 Compounds useful as reversible inhibitors of cathepsin s
09/08/2000WO2000051993A2 Dihetero-substituted metalloprotease inhibitors
09/08/2000WO2000051991A1 4-AMINO-QUINAZOLINE AND QUINOLINE DERIVATIVES HAVING AN INHIBITORY EFFECT ON SIGNAL TRANsSDUCTION MEDIATED BY TYROSINE KINASES
09/08/2000WO2000051989A1 Pyrazole-3-on-derivative as factor xa inhibitors
09/08/2000WO2000051986A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
09/08/2000WO2000051975A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors
09/08/2000WO2000051608A1 3-thienyl and 3-furanyl pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000023060A3 Method of treating immunological disorders mediated by t-lymphocytes
09/08/2000CA2366954A1 Dihetero-substituted metalloprotease inhibitors
09/08/2000CA2364908A1 Pyrazol-3-one derivatives
09/08/2000CA2364878A1 Alkenyl- and alkynyl-containing metalloprotease inhibitors
09/08/2000CA2362911A1 Heterocyclic compounds, intermediates thereof and elastase inhibitors
09/08/2000CA2360740A1 Compounds useful as reversible inhibitors of cathepsin s
09/08/2000CA2330541A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
09/07/2000DE19909785A1 New 1-heterocyclyl-5-carbonylaminomethyl-isoxazoline and 1-heterocyclyl-5-thionocarbonylaminomethyl-isoxazoline derivatives useful as antibacterial agents in human and veterinary medicine
09/07/2000DE19909237A1 Pyrazol-3-on-derivate Pyrazol-3-one derivatives
09/06/2000EP1032393A1 QUINOLINE-CONTAINING $g(a)-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS
09/06/2000CN1265652A 2-acrylaminopropanamines as tachykinin receptor antagonists
09/06/2000CN1265591A Coumpound
09/06/2000CN1265590A Substituted alkanohydroxamic acid and method of reducing TNF 'alpha' levels
09/06/2000CN1265585A (Imidazol-5-yl) methyl-2-quinolinone derivatives as inhibitors of smooth muscle cell proliferation
09/06/2000CN1265394A Compound as intermediates for use in preparation of optically active 2-imidazoline-5-one or 2-imidazoline-5-thionone derivatives
09/06/2000CN1056144C New use of 6-heterocyclic-4-amino-3,4,5-tetrahydrobenz (CD) indoles compound
09/05/2000US6114538 2-position of benzoy ring of 4-benzoylisoxazole derivative is substituted and particularly used against monocotyledonous weeds by post-emeregenece application
09/05/2000US6114534 Reacting a ketone derivative of carbamoyl substituted heterocycle with phosphorane, followed by acidification to form an anticoagulant
09/05/2000US6114526 Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
09/05/2000US6114522 Process of production of 4-substituted-3-halogeno-1,4-benzoxazepine derivative and salts thereof
09/05/2000US6114367 Such as 3-(3-cyclopentyloxy-4-methoxy)phenyl-2-isoxazoline-5-hydroxamic acid; treating sepsis, septic shock, inflammatory bowel disease, tuberculosis, graft versus host disease or cachexia associated with aids or cancer in a mammal
09/05/2000US6114328 Isoxazoline and isoxazole fibrogen receptor antagonists
09/05/2000CA2039399C Dual functioning excipient for metal chelate contrast agents
08/2000
08/31/2000WO2000050414A1 Novel tricyclic compounds and their use in medicine; process for their preparation and pharmaceutical composition containing them
08/31/2000WO2000050407A1 Herbicidal 2-(5-isoxazolinyl methyloxyphenyl) -4,5,6,7-tetrahydro -2h-indazole derivatives
08/31/2000WO2000050397A1 Substituted piperidinedione derivatives and herbicide
08/31/2000WO2000007996A3 Pyrazoles as estrogen receptor modulators
08/31/2000DE19908567A1 New 4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors, polyps or respiratory or gastrointestinal diseases
08/31/2000DE10008042A1 Neurokinin-1-Rezeptorantagonisten Neurokinin-1 receptor antagonists
08/31/2000CA2365793A1 Novel tricyclic compounds and their use in medicine; process for their preparation and pharmaceutical composition containing them
08/30/2000EP1031573A1 Novel benzoylpyrazole compounds, intermediates, and herbicides
08/30/2000EP1030852A1 Oxazolidinone derivatives and pharmaceutical compositions
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000EP1030835A2 Urea derivatives and their use as integrin inhibitors
08/30/2000EP0821680B1 Novel taxoids, preparation thereof, and pharmaceutical compositions containing same
08/30/2000EP0787141B1 Cyclic depsipeptide sulfonylation, sulfenylation and phosphorylation process
08/30/2000CN1265102A Benzothia (oxa) diazol derivatives and their use as endothelin-receptor antagonists
08/30/2000CN1265033A Certain diarylimidaozle derivatives, new class of NPY speific ligands
08/30/2000CN1055925C Synthesizing of ammonia-carboxylic acids chelating agent of inner-acid anhydride by homogeneous phase method
08/30/2000CN1055924C Novel aminoalkyl benzoxazolinones and benzothizolinones and pharmaceutical compsns. and method for preparing same
08/29/2000US6110963 Aryl-oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
08/29/2000US6110958 Pyrrole compounds having parasiticidal properties
08/29/2000US6110952 Preventing or treating nasal congestion, otitis media and sinusitis without undesired side effects, also asthma, pain, migraine, substance abuse and addiction, gastrointestinal disorder, ulcer, stomach hyperacidity
08/29/2000US6110948 Treating of malignant tumor, tuberculosis, diabetes, blood dyscrasia, endocrine disease, infectious disease, or acquired immunodeficiency syndrome
08/29/2000US6110939 As a substance p antagonists treating tachykinin-mediated disease, asthma, central nervous system disorder
08/29/2000US6110938 1-(arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-4-(heteroaryl)piperidines and related compounds useful as antipsychotics and analgesics
08/29/2000US6110935 A promoter for n-methyl-d-aspartic acid (nmda) receptors, useful for such therapeutic purposes as facilitating the learning of behaviors, treating schizophrenia, memory impairment
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/29/2000US6110909 Squalene synthetase inhibiting antilipemic agents
08/24/2000WO2000049016A1 Process for the preparation of 6-(perfluoroalkyl)uracil compounds
08/24/2000WO2000049015A1 Pyridine compounds and their pharmaceutical use
08/24/2000WO2000049002A1 Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils
08/24/2000WO2000048603A1 DIBENZO-AZEPINE DERIVATIVES AS αV INTEGRIN RECEPTOR ANTAGONISTS
08/24/2000WO2000048446A2 Use of antagonists of pg-e for the treatment of neuropathic pain
08/24/2000CA2364281A1 Processes and intermediates for the preparation of 1,3-oxazin-6-ones and uracils
08/24/2000CA2362990A1 Process for the preparation of 6-(perfluoroalkyl)uracil compounds
08/24/2000CA2362334A1 Dibenzo-azepine derivatives as .alpha.v integrin receptor antagonists
08/23/2000EP1029861A1 Benzisothiazol-piperazinyl derivative and its use as neuroleptic
08/23/2000EP1029541A1 Therapeutic or prophylactic agent for glomerulopathy
08/23/2000EP1028945A1 Substituted pyridine compounds as anti-inflammatory agents
08/23/2000EP1028940A1 Process to produce oxazolidinones
08/23/2000EP1028730A1 Compositions of lipid lowering agents
08/23/2000EP0652882B1 Anellated (oxa)hydantoines and their use as herbicides
08/23/2000CN1264385A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same
08/23/2000CN1264377A Substituted pyrazoles as P38 kinase inhabitors
08/23/2000CN1055690C 4-aryloxy-and-4-arylthiopiperidine derivatives, method for preparation them, medicine compound containing them and use thereof
08/23/2000CN1055686C Substituted benzisoxazole and benzisothaazole herbicidal agents