Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
12/1999
12/29/1999WO1999067252A2 Epothilone derivatives and their synthesis and use
12/29/1999WO1999067237A1 4,5,6 and 7-indole and indoline derivatives, their preparation and use
12/29/1999WO1999067230A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION
12/29/1999WO1999067229A1 New 2-aminocarbonyl-5(2h)-isoxazolones as ligands of a dfp-binding site for treatment of cns-diseases
12/29/1999WO1999066944A1 Methods for identifying novel multimeric agents that modulate receptors
12/29/1999WO1999031079A3 Methods for the esterification of alcohols and compounds useful therefor as potential anticancer agents
12/29/1999EP0966465A1 Inhibitors of impdh enzyme
12/29/1999EP0966452A1 Process for preparing sulphurous 2-chloro-3-(4,5-dihydroisoxazol-3-yl)-benzoic acids
12/29/1999EP0966440A1 Method of production and method of separation of 2,4'-dipyridyl derivatives and methods of production of benzoxazepine derivatives and salts thereof
12/29/1999EP0966283A2 Pharmaceutical products for curing and preventing illnesses connected with the malfunction of vascular endothelial cells
12/29/1999CN1239960A Thienylsulfonylamino (THIO) carbonyl compounds
12/29/1999CN1239952A 6-phenylpyridyl-2-amine derivatives useful as NOS inhibitors
12/29/1999CN1239950A New derivates from piperidine-keto acid, their preparation and use
12/29/1999CN1239889A Novel compounds useful as neuro-protective agents
12/29/1999CA2342778A1 Inhibitors of .alpha.4.beta.1 mediated cell adhesion
12/29/1999CA2335711A1 4,5,6 and 7-indole and indoline derivatives, their preparation and use
12/29/1999CA2335190A1 New 2-aminocarbonyl-5(2h)-isoxazolones as ligands of a dfp-binding site for treatment of cns-diseases
12/29/1999CA2319650A1 Methods for identifying novel multimeric agents that modulate receptors
12/28/1999US6008353 Pesticide, insecticide, nematocide, paracitiside
12/28/1999US6008350 Process for the production of cyanine dyes
12/28/1999US6008348 Treating a 1-tosylated indazol-3-yl piperazine derivative with concentrated hydrochloric acid to produce the detosylated indazol-3-yl piperazine compound of given formula
12/28/1999US6008230 Treating bone diseases caused by abnormal bone metabolism in human being or animals as the inhibitors of bone resorption or the inhibitors of bone metastasis
12/28/1999US6008229 Treating allergy, inflammation, autoimmune disease, shock, pain
12/23/1999WO1999065913A2 Epothilone minor constituents
12/23/1999WO1999065901A1 1,3-oxazoline and 1,3-thiazoline derivatives, method for producing the same and their use as pesticides
12/23/1999WO1999065900A1 Chemical synthesis of morpholine derivatives
12/23/1999WO1999065899A1 New oxazinylazole derivatives as fungicides
12/23/1999WO1999065897A1 Inhibitors of glycogen synthase kinase 3
12/23/1999WO1999065896A1 Preparation of heteroaryl compounds
12/23/1999WO1999065893A1 Novel benzopyran or thiobenzopyran derivatives
12/23/1999WO1999065882A1 2,4-diamino-1,3,5-triazine, method for the production and use of the same as herbicides and plant growth regulators
12/23/1999WO1999065878A1 Synthesis of benzo[f]quinolinones
12/23/1999WO1999065870A2 Sulfonamide inhibitors of aspartyl protease
12/23/1999WO1999065487A1 Inhibitors of serotonin reuptake
12/23/1999WO1999055156A3 The use of derivatives of iminotriazole as crop protection agents and novel iminotriazoles
12/23/1999DE19925329A1 New triazine derivatives useful as selective herbicides and plant growth regulators
12/23/1999DE19827387A1 Use of ligands of the high affinity binding site of diisopropyl-fluorophosphate in treatment of central nervous system disorders
12/23/1999DE19826988A1 Epothilon-Nebenkomponenten Epothilone secondary components
12/23/1999DE19826671A1 1,3-Oxazolin- und 1,3-Thiazolin-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel 1,3-oxazoline and 1,3-thiazoline derivatives, processes for their preparation and their use as pesticides
12/23/1999CA2336189A1 Epothilone minor constituents
12/23/1999CA2335352A1 1,3-oxazoline and 1,3-thiazoline derivatives, their preparation, and their use as pesticides
12/23/1999CA2335327A1 2,4-diamino-1,3,5-triazines, their preparation, and their use as herbicides and plant growth regulators
12/23/1999CA2335322A1 Inhibitors of serotonin reuptake
12/23/1999CA2334701A1 Synthesis of benzo¬f|quinolinones
12/23/1999CA2334677A1 Preparation of heteroaryl compounds
12/23/1999CA2334634A1 Novel benzopyran or thiobenzopyran derivatives
12/22/1999EP0965587A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake
12/22/1999EP0964863A1 Oxazolidines as 5-ht2a-antagonists
12/22/1999EP0964862A1 Insecticidal oxadiazine compounds
12/22/1999EP0964860A1 Atropisomers of 3-heteroaryl-4(3h)-quinazolinones for the treatment of neurodegenerative and cns-trauma related conditions
12/22/1999EP0964856A1 Bicyclic amino acids
12/22/1999EP0904077A4 Methods for the preparation of biphenyl isoxazole sulfonamides
12/22/1999EP0731795B1 Substituted pyrazolyl benzenesulfonamides for the treatment of inflammation
12/22/1999CN1239474A Substituted pyridines and biphenyls as anti-hypercholesterinemic, anti-hyperlipoproteinemic and anti-hyperglycemic agents
12/22/1999CN1047595C Prepn. method of aminocoumaran derivatives
12/21/1999US6005116 Isoxazole compounds useful for the prophylaxis or treatment of nervous diseases
12/21/1999US6005106 Naphthalene derivatives, process for the preparation therof, and intermediates thereof
12/21/1999US6005103 Pyrone derivatives as protease inhibitors and antiviral agents
12/21/1999US6005000 5,5-Disubstituted-3, 4-dihydroxy-2(5H)-furanones and methods of use therefor
12/21/1999US6004963 Tumor necrosis factor release inhibitors; immunomodulators
12/21/1999US6004961 1,4-disubstituted piperazines
12/21/1999US6004955 Cyclic carbamates and isoxazolidines as IIb/IIIa antagonists
12/21/1999US6004903 2-Anylocyclohexanediones having improved herbicidal properties
12/21/1999US6004536 Lipophilic cyanine dyes with enchanced aqueous solubilty
12/16/1999WO1999064519A1 Energy transfer assay method and reagent
12/16/1999WO1999064417A2 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
12/16/1999WO1999064416A2 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
12/16/1999WO1999064415A1 Sulfonylbenzene compounds as anti-inflammatory/analgesic agents
12/16/1999WO1999064401A2 Imidazolyl derivatives and their use as somatostatin receptor ligands
12/16/1999WO1999064399A1 Protease inhibitors
12/16/1999WO1999064055A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht4 receptors
12/16/1999WO1999064054A1 Multibinding inhibitors of topoisomerase
12/16/1999WO1999064053A1 β3-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064052A1 Novel leukotriene receptor antagonists and their uses
12/16/1999WO1999064051A1 Novel antibacterial compounds
12/16/1999WO1999064049A1 Novel antibacterial agents
12/16/1999WO1999064048A1 Inhibitors of hiv reverse transcriptase
12/16/1999WO1999064047A1 Novel antiviral compounds
12/16/1999WO1999064042A1 Novel therapeutic agents that modulate alpha-1a adrenergic receptors
12/16/1999WO1999064041A1 Multibinding agents that modulate nmda receptors
12/16/1999WO1999064038A1 Novel analgesic agents
12/16/1999WO1999064037A1 Novel therapeutic agents that modulate enzymatic processes
12/16/1999WO1999064035A1 β2-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064034A1 β2-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064033A1 Phosphodiesterase-v modulator drugs and their uses
12/16/1999WO1999064032A1 Combinatorial synthesis of multibinding libraries
12/16/1999WO1999064031A1 β2-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064010A1 Use of a nk-1 receptor antagonist for treating psychiatric disorders
12/16/1999WO1999064000A1 Novel therapeutic agents that modulate neurokinin receptors
12/16/1999WO1999063999A1 H1-histamine receptor antagonists
12/16/1999WO1999063996A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
12/16/1999WO1999063994A1 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE
12/16/1999WO1999063993A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the d1 receptors
12/16/1999WO1999063988A1 Inhibitors of nitric oxide synthase
12/16/1999WO1999063983A1 MULTIBINDING AGENTS THAT MODULATE PPARη AND RXR RECEPTORS
12/16/1999WO1999063944A2 Novel therapeutic agents that modulate estrogen receptors
12/16/1999WO1999063940A2 INHIBITORS OF H+K+-ATPase
12/16/1999WO1999063939A2 Multibinding inhibitors of cyclooxygenase-2
12/16/1999WO1999063937A2 Multivalent macrolide antibiotics
12/16/1999WO1999063936A2 Novel therapeutic agents that modulate endothelin receptors