Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
11/2000
11/30/2000CA2382751A1 Inhibitors of factor xa
11/30/2000CA2374820A1 Inhibitors of factor xa
11/30/2000CA2374788A1 Inhibitors of factor xa
11/30/2000CA2372743A1 New pharmaceutically active compounds
11/30/2000CA2371904A1 Inhibitors of factor xa
11/29/2000EP1055668A1 New 4-arylpiperidine derivatives for the treatment of pruritus
11/29/2000EP1054886A1 Heteroaryl amidines, methylamidines and guanidines as protease inhibitors, in particular as urokinase inhibitors
11/29/2000EP1054885A2 Benzisoxazole derivatives having d4-antagonistic activity
11/29/2000EP1054884A1 Benzofuran-4-carboxamides and their therapeutic use
11/29/2000EP1054882A1 Condensed heterocyclic system derivatives, preparation, pharmaceutical compositions containing them
11/29/2000EP1054875A1 Insecticidal dihydro-oxadiazines, -thiadiazines and -triazines
11/29/2000EP1054874A1 Substituted aminophenyl isoxazoline derivatives useful as antimicrobials
11/29/2000EP1054871A2 Pyrimidines and triazines as integrin antagonists
11/29/2000CN1275123A Prostaglandin agonists and their use to treat bone disorders
11/29/2000CN1275122A Process to produce oxazolidinones
11/29/2000CN1274718A Novel benzo-[3,4] cyclobutano [1,2-C] pyrroles compound, its prepn. and medicine composition containing the same
11/29/2000CN1058841C Fungicidal oxazolidinones
11/28/2000US6153759 Herbicide comprising a 5-membered or 6-membered heterocyclic, saturated or unsaturated radical containing one to three hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen
11/28/2000US6153640 For treating depression, panic attacks, obsessive-compulsive disorders, phobias, impulsive disorders, drug abuse or anxiety
11/28/2000US6153628 1,3,4-thiadiazoles and 1,3,4-Oxadiazoles as αv β3 antagonists
11/28/2000CA2309505A1 New 4-arylpiperidine derivatives for the treatment of pruritus
11/23/2000WO2000069923A1 Transition metal complexes and olefin polymerization process
11/23/2000WO2000069847A1 Substituted 3-pyridyl-4-arylpyrroles, and related therapeutic and prophylactic methods
11/23/2000WO2000069842A1 Benzofuranylsulfonates
11/23/2000WO2000069834A1 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade
11/23/2000WO2000069821A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
11/23/2000WO2000069810A1 Glucagon antagonists/inverse agonists
11/23/2000WO2000034247A3 Method for producing pyrazolylbenzoyl derivatives and novel pyrazolylbenzoyl derivatives
11/23/2000CA2374559A1 Substituted 3-pyridyl-4-arylpyrroles, and related therapeutic and prophylactic methods
11/23/2000CA2373892A1 Glucagon antagonists/inverse agonists
11/23/2000CA2373666A1 Benzofuranylsulfonates
11/23/2000CA2372934A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
11/23/2000CA2372617A1 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade
11/23/2000CA2372224A1 Transition metal complexes and olefin polymerization process
11/22/2000EP1054005A1 Sulfonamide derivatives, process for producing the same and utilization thereof
11/22/2000EP1053235A1 Oxazole derivatives as serotonin-1a receptor agonists
11/22/2000EP1053227A1 Ppar-gamma modulators
11/22/2000EP1053224A1 Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament
11/22/2000EP0693061B1 Fungicidal oxazolyl and oxadiazolyl derivatives
11/22/2000CN1274350A Efficient method for conversion of nitriles to amidines
11/22/2000CN1274288A Peptide-containing & alpha; -ketoamide cysteine and serine protease inhibitors
11/22/2000CN1274283A Quinoline-containing & Alpha;-ketoamide cysteine and serine protease inhibitors
11/22/2000CN1058709C Amide compounds for medical treatment
11/21/2000US6150557 Compounds
11/21/2000US6150537 Methods for the esterification of alcohols and compounds useful therefor as potential anticancer agents
11/21/2000US6150532 Modulators of proteins with phosphotyrosine recognition units
11/21/2000US6150531 Benzoxazolylisoindolenines
11/21/2000US6150530 Amidation of amine with acid
11/21/2000US6150526 Piperidine derivative having renin inhibiting activity
11/21/2000US6150416 2-hydroxy-3-(substitued benzyl)-n,n'-bis(substituted carbonyl)-n-(substituted)-1,3-propanediamine based compounds; use in the detection, labelling and inhibition of cathepsin d
11/21/2000US6150394 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
11/21/2000US6150389 Antidepressants; treating elevated intraocular pressure, e.g., glaucoma; antidiabetic agents for non-insulin dependent diabetes, sexual disorders, e.g., male impotence and obesity; e.g. trans-2-(3-phenyl-bicyclo(2.2.1)heptyl)-2-aminooxazoline
11/21/2000US6150388 Indole derivatives as 5-HT1 agonists
11/21/2000US6150386 Pest control, in particular, as microbicides, insecticides and acaricides in agriculture, in horticulture and hygiene sector; crop storage; fungicides
11/21/2000US6150378 Peptidyl-containing α-ketoamide cysteine and serine protease inhibitors
11/21/2000US6150375 Inhibitors of both of the human 5ar isozymes; benign prostate hyperplasia, male pattern baldness, acne vulgaris, seborrhea, androgenic alopecia, hirsutism and prostate cancer; blocks the conversion of testosterone to 5-alpha-dihydrotestosterone
11/21/2000US6150372 Immunoinflammatory and autoimmune diseases; blocking intracellular signal transduction and activation of transcription factors; kinase inhibitors; antiarthritic, ischemic agents, multiple sclerosis, transplant rejection
11/21/2000US6150371 Method for preventing and for treating autoimmune disease
11/21/2000US6150370 1,3-dinitrocyclic compound treats numerous diseases caused by undesired metalloprotease activity, such as tumor metastasis, osteoarthritis, rheumatoid arthritis, skin inflammation, ulcerations, and periodontitis
11/21/2000US6150362 Administering 1,3,5-substituted triazine compounds to the patient suffering from angiogenic diseases
11/21/2000US6150356 Potassium channel inhibitors and method
11/21/2000US6150352 Antagonists of gonadotropin releasing hormone
11/21/2000US6150334 Serine protease inhibitors-tripeptoid analogs
11/16/2000WO2000068228A1 4-(3',4'-heterocyclyl benzoyl) pyrazoles as herbicidal agents
11/16/2000WO2000068227A1 Substituted benzoylisoxazoles and the use thereof as herbicides
11/16/2000WO2000068224A1 Substituted benzolactam compounds
11/16/2000WO2000068213A1 Substituted bicyclic compounds
11/16/2000WO2000068206A1 Heterocyclically substituted benzimidazoles, the production and application thereof
11/16/2000WO2000068204A1 Substituted benzoyl ketones, methods for producing them and their use as herbicides
11/16/2000WO2000068202A1 Substituted 4-oxo-quinoline-3-carboxamides: gaba brain receptor ligands
11/16/2000WO2000068201A1 Quinoline derivatives as inhibitors of mek enzymes
11/16/2000WO2000068195A2 Substituted pyrrolidines as cell adhesion inhibitors
11/16/2000WO2000038665A3 Use of an integrin antagonist and one or more antineoplastic agents as a combination therapy in the treatment of neoplasia
11/16/2000WO2000034437A3 Inhibitors of prenyl-protein transferase
11/16/2000WO2000028822A3 Herbicidal 3-(benzo(ox/thi)azol-7-yl)-1h-pyrimidine-2,4-diones
11/16/2000WO2000015634A3 Hiv protease inhibitors
11/16/2000WO2000009103A3 N-linked sulfonamides of n-heterocyclic carboxylic acids or isosteres for vision and memory disorders
11/16/2000DE19923001A1 New epothilone derivatives, used as mitosis regulators e.g. for treating malignant tumors, psoriasis or arthritis
11/16/2000DE19920247A1 Arzneimittel mit einem Gehalt an Verbindungen mit einem Stickstoff-Sauerstoff-Heterocyclus als Wirkstoff und ihre Verwendung Medicaments with an amount of compounds having a nitrogen-oxygen heterocycle as active ingredient and their use
11/16/2000CA2373293A1 4-(3',4'-heterocyclyl benzoyl) pyrazoles as herbicidal agents
11/16/2000CA2373079A1 Substituted benzolactam compounds
11/16/2000CA2373076A1 Substituted benzoyl ketones, methods for producing them and their use as herbicides
11/16/2000CA2372963A1 Substituted benzoylisoxazoles and the use thereof as herbicides
11/16/2000CA2372663A1 Quinoline derivatives as inhibitors of mek enzymes
11/16/2000CA2371472A1 Substituted 4-oxo-quinoline-3-carboxamides: gaba brain receptor ligands
11/15/2000EP1052261A1 Pyran derivatives and use thereof
11/15/2000EP1052255A1 Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics.
11/15/2000EP1051415A1 Benzamide derivatives as vasopressin antagonists
11/15/2000EP1051176A1 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS
11/15/2000EP1051169A1 Compounds, compositions and methods for treating or preventing pneumovirus infection and associated diseases
11/15/2000CN1273585A Substituted 3-(1,2-benzisothiazol or isoxazel-5-yl)-substituted pyrimidine as heribicides
11/15/2000CN1273584A Imidazolyl-cyclic acetals
11/15/2000CN1058490C Tetrazolinone derivatives
11/14/2000US6147220 Process to 5-methyleneoxazolines
11/14/2000US6147100 Antiinflammatory agents
11/14/2000US6147099 Oxazolidinedione derivatives, their production and use
11/14/2000US6147088 Antagonists of gonadotropin releasing hormone
11/14/2000US6147031 Benzoylpyrazole compounds, intermediate preparing therefor and herbicides
11/14/2000CA2012432C N-(3-hydroxy-4piperidinyl)(dihydrobenzofuran, dihydro-2h-benzopyran or dihydrobenzodioxin) carboxamide derivatives
11/09/2000WO2000066618A1 Integrin receptor antagonists