Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
07/2000
07/13/2000WO2000040548A1 Arylalkanoyl derivatives, processes for their preparation, their use and pharmaceutical compositions containing them
07/13/2000WO2000040247A1 2-oxy-benzoxazinone derivatives for the treatment of obesity
07/13/2000WO2000021927A3 Pyrrole-2,5-diones as gsk-3 inhibitors
07/13/2000WO2000006597A9 Endogenous constitutively activated g protein-coupled orphan receptors
07/13/2000DE19900519A1 Substituierte Guanidin-Derivate Substituted guanidine derivatives
07/13/2000DE19900355A1 New 2-(naphthalen-2-ylmethyl)-benzimidazole derivatives are Factor VIIa, IXa, Xa and thrombin inhibitors useful for treating thrombosis and other cardiovascular disorders, inflammation and apoplexy
07/13/2000DE19845405C2 Arylsubstituierte Propanolaminderivate und deren Verwendung Aryl-substituted Propanolaminderivate and their use
07/13/2000CA2358576A1 Cyclic guanidine derivatives and their use as pesticides
07/13/2000CA2355308A1 3,4-dihydro-2h-benzo¬1,4|oxazinyl-methyl¬3-(1h-indol-3-yl)-alkyl|-amines
07/13/2000CA2353636A1 Quinolinecarboxamides as antiviral agents
07/12/2000EP1018008A2 Method of identification of leads or active compounds
07/12/2000EP1017691A1 Bisethers of 1-oxa, aza and thianaphthalen-2-ones as phospholamban inhibitors
07/12/2000EP1017395A1 Method for treating premenstrual or late luteal phase syndrome
07/12/2000EP0745073B1 5-substituted derivatives of mycophenolic acid
07/12/2000EP0628041B1 Heterocyclic compounds and their preparation and use
07/12/2000CN1259943A Substituted aryluracils
07/12/2000CN1259942A Novel guanidine mimics as factor Xa inhibitors
07/12/2000CN1259935A Substituted naphthopyrans
07/11/2000US6087502 Acridinium compound having a plurality of luminescent groups and binding groups, and conjugate thereof
07/11/2000US6087496 Enzyme inhibitors
07/11/2000US6087384 Treating prophylaxis and treatment of a disease associate with death of cells caused by viral diseases, myelodysplasis, neurodegenerative, ischemic and hepatic diseases with a compound having an insulin sensitivity enhancing activity
07/11/2000US6087365 Treating drug-resistant malaria in a mammal
07/11/2000US6087357 Piperazine derivatives as tachykinin antagonists
07/06/2000WO2000039126A1 Method for preparing (r)- (+) -3 {1- [2-( 4-benzoyl- 2-(3,4- difluorophenyl)morpholin- 2-yl)ethyl]- 4-phenylpiperidin -4-yl}-1,1- dimethylurea, its salts solvates and/or hydrates
07/06/2000WO2000039125A1 Piperidines as ccr5 modulators
07/06/2000WO2000039124A1 Thrombin inhibitors
07/06/2000WO2000039114A2 Substituted oximes and hydrazones as neurokinin antagonists
07/06/2000WO2000039108A1 Thrombin or factor xa inhibitors
07/06/2000WO2000039102A1 THROMBIN OR FACTOR Xa INHIBITORS
07/06/2000WO2000039101A1 Pyrimidine compounds
07/06/2000WO2000039091A1 3,3-biarylpiperidine and 2,2-biarylmorpholine derivatives
07/06/2000WO2000039089A1 3-azabicyclo[3.1.0.] hexane derivatives as opiate receptors ligands
07/06/2000WO2000039087A2 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds as factor xa inhibitors
07/06/2000WO2000039081A2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
07/06/2000WO2000038786A2 Use of cyclooxygenase 2 inhibitor and an integrin antagonist as a combination therapy in the treatment of neoplasia
07/06/2000WO2000038730A2 Use of a cyclooxygenase-2 inhibitor and one or more antineoplastic agents for combination therapy in neoplasia
07/06/2000WO2000038719A1 Use of a matrix metalloproteinase inhibitor and an integrin antagonist in the treatment of neoplasia
07/06/2000WO2000038718A2 Use of matrix metalloproteinase inhibitor together with an antineoplastic agents, optionally also together with radiation, in the treatment of neoplasia
07/06/2000WO2000038717A2 Use of a matrix metalloproteinase inhibitor and radiation as a combined treatment of neoplasia
07/06/2000WO2000038715A2 Use of an integrin antagonist and radiation in the treatment of neoplasia
07/06/2000WO2000038687A1 Protease inhibitors
07/06/2000WO2000038683A1 THROMBIN OR FACTOR Xa INHIBITORS
07/06/2000WO2000038680A1 Azabicycloalkanes as ccr5 modulators
07/06/2000WO2000038665A2 Use of an integrin antagonist and one or more antineoplastic agents as a combination therapy in the treatment of neoplasia
07/06/2000WO1999064035A9 β2-ADRENERGIC RECEPTOR AGONISTS
07/06/2000CA2358047A1 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds
07/06/2000CA2356929A1 Method of using a matrix metalloproteinase inhibitor and one or more antineoplastic agents as a combonation therapy in the treatment of neoplasia
07/06/2000CA2356748A1 Method of using an integrin antagonist and radiation therapy as combination therapy in the treatment of neoplasia
07/06/2000CA2356671A1 Protease inhibitors
07/06/2000CA2356606A1 Method of using a cyclooxygenase-2 inhibitor and one or more antineoplastic agents as a combination therapy in the treatment of neoplasia
07/06/2000CA2356462A1 Method of using an integrin antagonist and one or more antineoplastic agents as a combination therapy in the treatment of neoplasia
07/06/2000CA2356459A1 Method of using a matrix metalloproteinase inhibitor and radiation therapy as combination therapy in the treatment of neoplasia
07/06/2000CA2356402A1 Use of a matrix metalloproteinase inhibitor and an integrin antagonist in the treatment of neoplasia
07/06/2000CA2356302A1 Method of using a cyclooxygenase-2 inhibitor and an integrin antagonist as a combination therapy in the treatment of neoplasia
07/06/2000CA2355281A1 Thrombin inhibitors
07/06/2000CA2352896A1 Pyrimidine compounds
07/06/2000CA2351539A1 Method for preparing (r)- (+) -3 {1- ¬2-( 4-benzoyl- 2-(3,4- difluorophenyl)morpholin- 2-yl)ethyl|- 4-phenylpiperidin -4-yl}-1,1- dimethylurea, its salts solvates and/or hydrates
07/06/2000CA2350589A1 3,3-biarylpiperidine and 2,2-biarylmorpholine derivatives
07/06/2000CA2349557A1 Thrombin or factor xa inhibitors
07/06/2000CA2348740A1 Thrombin or factor xa inhibitors
07/06/2000CA2320730A1 Thrombin or factor xa inhibitors
07/05/2000EP1015447A1 Piperidinylmethyloxazolidinone derivative
07/05/2000EP1015446A1 (4-piperidinyl)-1h-2-benzopyran derivatives useful as antipsychotic agents
07/05/2000EP1015437A1 Benzoxazine and benzothiazine derivatives and their use in pharmaceuticals
07/05/2000EP1015436A1 Morpholinones as light stabilizers
07/05/2000EP1015429A1 Benzimidazolinones, benzoxazolinones, benzopiperazinones, indanones, and derivatives thereof as inhibitors of factor xa
07/05/2000EP1014982A1 Troglitazone compounds for treating climacteric
07/05/2000EP1014973A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
07/05/2000EP0882138B1 Stereoselective preparation of 2-substituted succinic derivatives
07/05/2000EP0734381B1 Morpholine tachykinin receptor antagonists
07/05/2000EP0692982B1 RADIOLABELED PLATELET GPIIb/IIIa RECEPTOR ANTAGONISTS AS IMAGING AGENTS FOR THE DIAGNOSIS OF THROMBOEMBOLIC DISORDERS
07/05/2000EP0686151B1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
07/05/2000EP0675886B1 Aminomethylene substituted non-aromatic heterocycles and use as substance p antagonists
07/05/2000CN1259129A Desoxycyclodepsipeptides and their use for combatting endoparasites
07/05/2000CN1259128A Thiodepsipeptides for combating endoparasites and a method for producing the same
07/05/2000CN1259125A Substituted 3-cyano quinolines
07/05/2000CN1259122A Method for producing chiral 3,4-dehydroprolines
07/04/2000US6084130 For treatment of central nervous system disorders
07/04/2000US6084103 Forming a carbamate from methyl 4-nitro-(l)-phenylalaninate hydrochloride; reducing the nitro and ester groups; ring closure free of phosgene; forming a diazonium salt without using tin chloride; fischer reaction; migraines; 5ht1-agonist
07/04/2000US6083967 Antimicrobial agents; assay for determining the inhibitory activity of oxazolidinones to human monoamine oxidase
07/04/2000US6083965 Antiparasitic agents
07/04/2000US6083961 For prevention and/or treatment of bradykinin or its analogues mediated diseases such as allergy, inflammation, autoimmune disease, shock, pain
07/04/2000US6083944 Enzyme inhibitors; treatment of various debilitating disorders
07/04/2000US6083942 Pesticidal hetero-substituted oxadiazine compounds
07/04/2000US6083881 Pyrazole derivatives as herbicides
06/2000
06/29/2000WO2000037473A1 Epothilone derivatives and their use as antitumor agents
06/29/2000WO2000037464A2 4-(aminoalkoxy)benzofurans as n-myristoyltransferase inhibitors
06/29/2000WO2000037462A1 Non-peptide nk1 receptors antagonists
06/29/2000WO2000037458A1 Farnesyl protein transferase inhibitors
06/29/2000WO2000037422A2 Ion channel modulating agents
06/29/2000WO2000037107A2 Use of cyclooxygenase-2 inhibitor, a matrix metallaproteinase inhibitor, an antineoplastic agent and optionally radiation as a combination treatment of neoplasia
06/29/2000WO1999064034A9 β2-ADRENERGIC RECEPTOR AGONISTS
06/29/2000CA2356426A1 Method of using a cyclooxygenase-2 inhibitor and a matrix metalloproteinase inhibitor as a combination therapy in the treatment of neoplasia
06/29/2000CA2355694A1 Novel bicyclic compounds
06/29/2000CA2355137A1 Non-peptide nk1 receptors antagonists
06/28/2000EP1014186A1 Photographic yellow dye-forming couplers
06/28/2000EP1013276A1 Aminoazacycloalkanes as CCR5 modulators
06/28/2000EP1012150A1 Heteroarylcarboxamide compounds active against protein tyrosine kinase related disorders
06/28/2000EP1011667A1 Antagonists of gonadotropin releasing hormone
06/28/2000CN1258296A Pyridine derivatives and pharmaceutical compositions contg. them