Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
08/2000
08/22/2000US6107519 Amido-substituted secondary alcohol intermediates and preparation thereof
08/22/2000US6107329 Hypotensive agents; cardiovascular disorders
08/22/2000US6107323 Preventing or treating angiotensin diseases by administering an antagonist and compound which increases insulin sensitivity
08/22/2000US6107314 Pesticides
08/22/2000US6107313 Nervous system disorders; psychological disorders
08/22/2000US6107295 Arylalkanoyl pyridazines
08/22/2000US6107251 Oxazole derivative, process for producing the same, and herbicide
08/22/2000CA2176973C Phenyl heterocycles as cyclooxygenase-2 inhibitors
08/22/2000CA2085987C Piperidyl-substituted indoles
08/22/2000CA2020554C Process for the control of sea lice
08/17/2000WO2000047584A2 Epothilon derivatives, method for the production and the use thereof as pharmaceuticals
08/17/2000WO2000047578A1 Heteroaryl amidines, methylamidines and guanidines as protease inhibitors
08/17/2000WO2000047577A1 Phenyl urea and phenyl thiourea derivatives as orexin receptor antagonists
08/17/2000WO2000047572A1 (1-phenacy-3-phenyl-3-piperidylethyl)piperidine derivatives, method for the production thereof and pharmaceutical compositions containing the same
08/17/2000WO2000047567A1 Heterodiazinone derivatives
08/17/2000WO2000047212A1 Quinazoline derivatives as angiogenesis inhibitors
08/17/2000WO2000047194A2 METHODS OF TREATING C1s-MEDIATED DISEASES AND CONDITIONS, AND COMPOUNDS AND COMPOSITIONS THEREFOR
08/17/2000WO2000027819A3 Antrhranilic acid amides and the use thereof as medicaments
08/17/2000DE19907480A1 New epothilone derivatives, useful for treating malignant tumors such as ovarian, stomach, colon, breast and lung carcinoma, acute lymphocytic and myelocytic leukemia and chronic inflammatory diseases such as psoriasis
08/17/2000CA2362390A1 Heteroaryl amidines, methylamidines and guanidines as protease inhibitors
08/17/2000CA2360952A1 Epothilon derivatives, method for the production and the use thereof as pharmaceuticals
08/17/2000CA2360233A1 Methods of treating c1s-mediated diseases and conditions, and compounds and compositions therefor
08/16/2000EP1027347A2 3-aminoalkylamino-2h-1,4-benzoxa(thia-)zines and pharmaceutical compositions containing them
08/16/2000EP1027340A1 4, 5-diaryloxazole compounds
08/16/2000EP1027337A1 Integrin receptor antagonists
08/16/2000EP1027332A1 Novel lactam metalloprotease inhibitors
08/16/2000EP1027051A1 Antithrombotic agents
08/16/2000EP1026950A1 Treatment of schizophrenia with ampakines and neuroleptics
08/16/2000CN1263528A N-triazolyl-2-indolecarboxamides and their use as CCK-A agonists
08/16/2000CN1263526A Triazine derivatives, their production and use
08/16/2000CN1055467C Taxoids compound, their preparation and pharmaceutical compositions containing them
08/16/2000CN1055465C Optical active 2-imidazoline-5-thione derivatives and preparating method and use thereof
08/15/2000US6103936 Reacting aldehyde, sulfide, sulfone, or sulfoxide with formamide in presence of acid catalyst, and optionally a dehydrating agent
08/15/2000US6103910 D-proline derivatives
08/15/2000US6103752 Therapeutic heterocyclic compounds
08/15/2000US6103717 Strong fungicides; bactericides; microbiocides; nonphytotoxic; crops, cereals, fruits, vegetables
08/15/2000US6103715 Compounds that bind to the dopamine d4 receptor and their use as anxiolytic agents, treatment for schizophrenia, and drug screening; side effect reductioon
08/15/2000CA2105385C Treatment of cognitive disorders
08/15/2000CA2046883C Heterocyclic derivatives, method for preparing same, and their therapeutic applications
08/10/2000WO2000046222A1 Heteroaromatic compounds with neuronal activity
08/10/2000WO2000046221A1 Sulfamato hydroxamic acid metalloprotease inhibitor
08/10/2000WO2000046214A1 Substituted 4-amino-2-aryltetrahydroquinazolines, their preparation, their use and pharmaceutical compositions comprising them
08/10/2000WO2000046199A2 Indole derivatives as anti-inflammation agents
08/10/2000WO2000046197A1 Indole derivatives and their use as mcp-1 receptor antagonists
08/10/2000WO2000046189A1 Sulfonamide derivatives having cyclic structures
08/10/2000WO2000027822A3 Tricyclic pyrazole derivatives
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/10/2000DE19905256A1 New heteroaromatic compounds, useful e.g. in the treatment of Parkinson's, Alzheimer's and Huntington's diseases, stimulate neurite growth
08/10/2000DE19904710A1 Substituierte 4-Amino-2-aryl-tetrahydrochinazoline, ihre Herstellung, ihre Verwendung und sie enthaltende pharmazeutische Präparate Substituted 4-amino-2-aryl-tetrahydroquinazolines, their preparation, their use and pharmaceutical compositions containing them
08/10/2000CA2362230A1 Sulfamato hydroxamic acid metalloprotease inhibitor
08/10/2000CA2355734A1 Indole derivatives as anti-inflammation agents
08/09/2000EP1026149A1 Amidocarboxylic acid derivatives
08/09/2000EP1025086A1 Benzamidine derivatives as factor xa inhibitors
08/09/2000EP1025085A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
08/09/2000CN1262679A IL-5 inhibiting 6-azauracil derivatives
08/09/2000CN1262678A Triazole compounds and use thereof as dopamine-D3-ligands
08/09/2000CN1262676A 吡啶衍生物 Pyridine derivatives
08/08/2000US6100399 Synthesis for 4-aryl-5-pyrimidine imidazole substituted compounds
08/08/2000US6100289 Indole derivatives
08/08/2000US6100284 Antiallergens
08/08/2000US6100260 Isoxazole derivatives
08/08/2000US6100259 Cannabinoid receptor modulators
08/08/2000US6100258 Aromatic amine compounds that antagonize the pain enhancing effects of prostaglandins
08/08/2000US6100257 2-haloalkyl,3-(haloalkyl, alkenyl, or alkynyl),5-(substituted phenyl or heterocycle),6-alkyl-pyrimidin-4-one compounds of given structure; use as herbicides
08/08/2000US6100255 Bind selectively with high affinity to the dopamine d4 receptor subtype; use in treating various neuropsychological disorders, including alzheimer's disease, schizophrenia, parkinson's disease, or tardive dyskinesia
08/08/2000US6100252 Specified compounds including methyl 2-butyl-1-((2'-(2-oxo-3h-1,2,3,5-oxathiadiazol-4-yl)biphenyl) methyl)-benzimidazole-7-carboxylate; use to treat circulatory diseases such as hypertensive diseases and heart diseases
08/08/2000US6100238 Indole and tetrahydroisoquinoline containing Alpha-keto oxadiazoles as serine protease inhibitors
08/08/2000CA2185019C Isoxazoline compounds as inhibitors of tnf release
08/08/2000CA2085796C 3(2h)-pyridazinone derivatives and process for the preparation thereof
08/08/2000CA2018438C Imidazolyl-alkenoic acids
08/03/2000WO2000044741A2 Process to prepare cyclic-sulfur fluorine containing oxazolidinones
08/03/2000WO2000044728A1 Substituted bicyclic derivatives useful as anticancer agents
08/03/2000DE19904310A1 Verfahren zur Herstellung heterocyclischer Verbindungen Process for the preparation of heterocyclic compounds
08/03/2000CA2359711A1 Process to prepare cyclic-sulfur fluorine containing oxazolidinones
08/03/2000CA2356313A1 Alkynyl containing hydroxamic acid derivatives, their preparation and their use as matrix metalloproteinase (mmp) inhibitors/tnf-alpha converting enzyme (tace) inhibitors
08/02/2000EP1024140A1 Process for N-alkylation of cyclic cyanoamidines
08/02/2000EP1024138A1 Pyrazole derivatives
08/02/2000EP1023276A1 Microbicide 1,4,2-dioxacine derivatives
08/02/2000EP1023275A1 Azines containing the 5,6-di-hydro-(1,4,2) dioxazine-3-yl group and the use thereof as fungicides
08/02/2000EP1023274A1 An efficient method for the conversion of nitriles to amidines
08/02/2000EP1023265A1 Azetidinone derivatives for the treatment of hcmv infections
08/02/2000EP1023072A1 Analgesic compositions
08/02/2000EP1023068A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
08/02/2000CN1261889A Thiadiazolyl and oxadiazolyl phenyl oxazolidinone antibacterial agent
08/02/2000CN1261884A Benzothiophene derivatives as herbicides
08/02/2000CN1261882A Polymorphic form of tachykinin receptor antagonist 2-(R)-(1-(R)-(3,5-bis(trifluoromethyl) phenyl) ethoxy)-3-(S)-(4-fluoro) phenyl-4-(3-5(oxo-1H,4H-1,2,4-triazolo methylmorpholine
08/02/2000CN1261795A Compounds and methods
08/02/2000CN1261688A 照相黄色成色剂 Photographic yellow couplers
08/01/2000US6096904 Discodermolides
08/01/2000US6096898 One pot synthesis of 1,2,4-triazoles
08/01/2000US6096895 Heterocyclic dihydrazole compounds and their use for controlling fungal plant diseases
08/01/2000US6096884 Method of production and method of separation of 2,4'-dipyridyl derivatives and methods of production of benzoxazepine derivatives and salts thereof
08/01/2000US6096773 Inhibitor of binding of integrin to its receptors, such as (vascular cell adhesion molecule-1) and fibronectin and useful for controlling the diseases induced by binding
08/01/2000US6096745 Imidazolone anorectic agents: III. heteroaryl derivatives
08/01/2000US6096742 Polymorphic form of a tachykinin receptor antagonist
08/01/2000US6096735 Benzoheterocyclic derivatives
08/01/2000US6096729 Use of NK-1 receptor antagonists for treating amnestic disorders
08/01/2000US6096689 5-pyrazolylbenzoic acid derivatives as herbicides
08/01/2000US6096688 Oxazole carboxamide herbicides
07/2000
07/27/2000WO2000043391A1 Substituted 1-(pieridin-4-yl)-3-(aryl) isothioureas their preparation and therapeutic application