Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/2001
01/11/2001CA2376619A1 Detection using dendrimers bearing labels and probes
01/11/2001CA2373883A1 Method of reducing neuronal injury or apoptosis
01/10/2001EP1067128A1 Fused thiophene derivatives and drugs containing the same as the active ingredient
01/10/2001EP1067109A1 Carboxylic acid derivatives and drugs containing the same as the active ingredient
01/10/2001EP1066281A1 Cationic methylenedioxy benzenes, their use for oxidation dyeing of keratin fibres, dyeing compositions and methods
01/10/2001EP1066279A1 Imidazolone anorectic agents: ii. phenyl derivatives
01/10/2001EP1066278A1 Imidazolone anorectic agents: iii. heteroaryl derivatives
01/10/2001EP1066262A1 Imidazolone anorectic agents: i. acyclic derivatives
01/10/2001EP1066256A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
01/10/2001CN1279680A Imidazole derivatives with inhabiting activity to transterasa and preparing method thereof
01/10/2001CN1279674A 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analoguse), their preparation and their use in the treatment of neurological disorders
01/10/2001CN1279673A ((Cyclo) alkyl substituted-.gamma.-aminobutyric acid derivatives (=GABA analogurs), their preparation and their use in the treatment of neurolog disorders
01/10/2001CN1279669A Aromatic sulfone hydroxamic acid metalloprotease inhibitor
01/10/2001CN1279667A 4(3)-substituted-4(3)-aminonethyl-(thioxo)pyran(thiapyran)or-piperidine derivatives(=gabapendin analogues), their preparation and their use in treatment of neurological disorders
01/10/2001CN1060479C Preparation method for inidazole derivatives
01/10/2001CN1060472C Hydroxamic acid derivatives with tricylic substitution, their preparing methods, medicines containing them and uses thereof
01/09/2001US6172239 Psychological, nervous system disorders
01/09/2001US6172235 Endothelian antagonist
01/09/2001US6172092 Fungicides, bactericides for crops; treating plant diseases; applying to wood, leather, plastic
01/09/2001US6172073 Benzimidazolyloxy alkanamines as serotonin reuptake inhibitors; nicotine and tobacco withdrawal; psychological, eating, brain, gastrointestinal, sleep, and sexual disorders
01/09/2001US6172067 Analgesics, antiinflammatory agents
01/09/2001CA2031766C 2-substituted phenyl-2-oxazoline or thiazoline derivatives, process for producing the same and insecticides and acaricides containing the same
01/04/2001WO2001000622A1 Prodrugs of carbamate inhibitors of impdh
01/04/2001WO2001000615A1 Respiratory syncytial virus replication inhibitors
01/04/2001WO2001000611A1 Respiratory syncytial virus replication inhibitors
01/04/2001WO2001000610A1 Substituted benzimidazole
01/04/2001WO2001000603A1 Thiazole and oxazole derivatives and their pharmaceutical use
01/04/2001WO2001000601A1 Novel 4-(2-oxodihydrooxadiazinylphenyl)amides and the use thereof for treating anemia
01/04/2001WO2001000600A1 N-substituted perhydro diazine
01/04/2001WO2001000586A1 Compounds as selective agonists at alpha 2b or 2b/2c adrenergic receptors
01/04/2001WO2001000583A1 Ucf116 derivatives as antitumor agents
01/04/2001WO2001000579A1 COMPOUNDS FOR THE MODULATION OF PPARη ACTIVITY
01/04/2001WO2001000578A1 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
01/04/2001WO2001000214A1 Src kinase inhibitor compounds
01/04/2001WO2001000213A1 Src kinase inhibitor compounds
01/04/2001WO2001000206A1 Vla-4 inhibitor compounds
01/04/2001WO2000038715A3 Use of an integrin antagonist and radiation in the treatment of neoplasia
01/04/2001DE19929787A1 Neue 4-(2-Oxodihydrooxadiazinylphenyl)amide und ihre Verwendung New 4- (2-Oxodihydrooxadiazinylphenyl) amides and their use
01/04/2001CA2383546A1 Src kinase inhibitor compounds
01/04/2001CA2377137A1 N-substituted perhydro diazine
01/04/2001CA2376951A1 Src kinase inhibitor compounds
01/04/2001CA2376785A1 Benzimidazoles and imidazopyridines as respiratory syncytial virus replication inhibitors
01/04/2001CA2376781A1 Benzimidazoles and imidazopyridines as respiratory syncytial virus replication inhibitors
01/04/2001CA2370500A1 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
01/04/2001CA2369308A1 Vla-4 inhibitor compounds
01/03/2001EP1064289A1 Heterocyclic signal transduction inhibitors, compositions containing them
01/03/2001CN1278817A S-oxide and S,S-dioxide tetrahydrothiopyran phenyloxazolidinones
01/03/2001CN1278816A 5,11-Dihydrodibenz [b,e] [1,4] oxazepine derivaties and medicinal composition containing the same
01/03/2001CN1278805A Novel heterocyclioally substituted and a-hydroxycarboxlic acid derivatives, method for producing the same and their use as endothelin receptor antagonists
01/03/2001CN1278802A Benzoxazine and Benzothiazine derivatives and their use in pharmaceuticals
01/03/2001CN1278794A Substituted di-hydroxyl-indol derivatives as protein tyrosine kinase and as protein serine/threenine kinase inhibitors
01/03/2001CN1278790A Chemical compound
01/03/2001CN1060173C Heterocyclic compound with activity against diabetes and preparation nad application of same
01/03/2001CN1060172C Substituted biphenyl sulfonamide endothelin antagonists
01/03/2001CN1060171C Substituted biphenyl isoxazole sulfonamides
01/02/2001US6169102 Oxazolone derivatives and their use as anti-Helicobacter pylori agent
01/02/2001US6169096 For inhibiting tumor growth in a mammal
01/02/2001US6169095 For prevention and/or treatment of bradykinin or its analogues mediated diseases in the eye, such as allergy, inflammation and pain of the eye
01/02/2001US6169093 Quinoline and quinazoline compounds useful in therapy, particularly in the treatment of benign prostatic hyperplasia
01/02/2001CA2161662C Process for preparing intermediates for the synthesis of antifungal agent
01/02/2001CA2026761C Preparation of isoxazole-4,5-dicarboxylic diesters
12/2000
12/28/2000WO2000078746A1 Antiviral agents
12/28/2000WO2000078735A1 Bicyclic heterocycles, medicaments containing these compounds, their use and methods for the production thereof
12/28/2000WO2000078733A1 Phenoxy fluoropyrimidines
12/28/2000WO2000078728A1 Novel benzimidazole derivatives and pharmaceutical compositions comprising these compounds
12/28/2000WO2000078716A1 α1B-ADRENERGIC RECEPTOR ANTAGONISTS
12/28/2000WO2000078708A1 Substituted benzamide inhibitors of rhinovirus 3c protease
12/28/2000WO2000078313A1 Arylthiazolidinedione and aryloxazolidinedione derivatives
12/28/2000WO2000047584A3 Epothilon derivatives, method for the production and the use thereof as pharmaceuticals
12/28/2000WO2000043373A3 Kinase inhibitors
12/28/2000WO1999052493A3 Compounds that inhibit the binding of integrins to their receptors
12/28/2000DE19928306A1 New 4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors, polyps or respiratory or gastrointestinal diseases
12/28/2000CA2377246A1 Arylthiazolidinedione and aryloxazolidinedione derivatives
12/28/2000CA2375356A1 Substituted benzamide inhibitors of rhinovirus 3c protease
12/28/2000CA2375211A1 Antiviral agents
12/28/2000CA2373921A1 Novel benzimidazole derivatives and pharmaceutical compositions comprising these compounds
12/28/2000CA2341542A1 .alpha.1b-adrenergic receptor antagonists
12/27/2000EP1063235A1 Benzofurylpyrone derivatives
12/27/2000EP1062218A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
12/27/2000EP1062217A1 Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
12/27/2000EP1062208A1 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
12/27/2000EP1062205A2 Inhibitors of phospholipase enzymes
12/27/2000EP1061921A1 Vitronectin receptor antagonists
12/27/2000EP0823900B1 Quinazoline derivatives
12/27/2000EP0821671B1 Arylsulfonyl hydroxamic acid derivatives as mmp and tnf inhibitors
12/27/2000CN1278259A Novel benzoylpyrazole compounds, intermediates and herbicides
12/27/2000CN1278252A 4,5-diaryloxazole compounds
12/27/2000CN1278175A Compositions of lipid lowering agents
12/26/2000US6166222 Reacting a pyrrolecarboxylic acid derivative in ammonia with an alkali metal or alkaline earth metal and then an aqueos salt solution of a alkyl- or silyl-leaving group compound
12/26/2000US6166216 Compounds useful as neuro-protective agents
12/26/2000US6166202 Benzophenoxazine dyes
12/26/2000US6166056 Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings
12/26/2000US6166041 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma
12/26/2000US6166027 Treatment of high blood pressure and cardiac insufficiency, angina pectoris, arrhythmias, thromboembolic diseases, ischaemias, myocardial infarction, cerebral stroke, restenoses, coronary angioplasties, arteriosclerosis
12/26/2000US6166023 1,5- and 3-O-substituted 1H-indazoles having anti-asthmatic, anti-allergic, anti-inflammatory, immunomodulating and neuroprotective action, process for their preparation and their use as medicaments
12/26/2000US6166020 Aryl and heteroaryl alkoxynaphthalene derivatives
12/26/2000US6166011 For treatment of disorders arising from neurodegenerative diseases or other disorders involving nerve damage
12/26/2000US6166010 For combating animal pests
12/26/2000US6166008 Treatment of schizophrenia with ampakines and neuroleptics
12/26/2000US6166005 Heterocyclic metalloprotease inhibitors