Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
05/2001
05/09/2001EP1097921A1 Phenylhydrazines
05/09/2001EP1097147A1 Novel angiogenesis inhibitors
05/09/2001EP1097142A1 Phthalazine derivatives phosphodiesterase 4 inhibitors
05/09/2001EP1097137A1 N-substituted naphthalene carboxamides as neurokinin-receptor antagonists
05/09/2001EP1096934A1 Oxazolidinones to treat eye infections
05/09/2001EP1096925A2 Use of inhibitors of prenyltransferases for for inhibiting fungal growth
05/09/2001CN1294588A Spiropiperidine derivatives
05/09/2001CN1294583A Herbicidal 2-(5-isoxazolinyl methyloxyphenyl)-4,5,6,7-tetrahydro-2h-indazole derivatives
05/09/2001CN1294580A Indole derivatives with antiviral activity
05/09/2001CN1065532C Thiazolidine and oxaxoliding derivatives, their prepn. and their medical use
05/08/2001US6229011 N-aroylphenylalanine derivative VCAM-1 inhibitors
05/08/2001US6229010 Recovering form i of 2-(r)-(1-(r)-(3,5-bis(trifluoromethyl) -phenyl)ethoxy)-3-(s)-(4-fluoro)phenyl-4-(3-(5-oxo-1h,4h-1,2,4 -triazolo)methylmorpholine from form ii equilibrated in ethanol, isopropanol, acetonitrile or isopropyl acetate
05/08/2001US6228871 Angiogenesis inhibitors
05/08/2001US6228870 Oxazolidinones useful as alpha 1a adrenoceptor antagonists
05/08/2001US6228868 Anticarcinogenic and antitumor agents
05/08/2001US6228810 Outstanding efficacy against broad spectrum of phytopathogenic fungi; effective control of pests from classes of insects, arachnids and nematodes
05/03/2001WO2001030795A1 Hygromycin derivatives
05/03/2001WO2001030780A2 Pyridyl-containing spirocyclic compounds as inhibitors of fibrinogen-dependent platelet aggregation
05/03/2001WO2001030762A1 Imidazol-4-ylmethanols use as inhibitors of steroid c17-20 lyase
05/03/2001WO2001030749A1 Novel compounds
05/03/2001CA2389191A1 Hygromycin derivatives
05/03/2001CA2389034A1 Pyridyl-containing spirocyclic compounds as inhibitors of fibrinogen-dependent platelet aggregation
05/03/2001CA2387869A1 Imidazol-4-ylmethanols use as inhibitors of steroid c17-20 lyase
05/02/2001EP1095937A1 Process for the preparation of trisubstituted oxazoles
05/02/2001EP1095936A1 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses, and methods and intermediates useful for their preparation
05/02/2001EP1095935A1 6-Hydroxy-5,6-dihydrouracils as herbicides
05/02/2001EP1095275A2 Endogenous constitutively activated g protein-coupled orphan receptors
05/02/2001EP1095040A1 New benzoxazoles with pde-inhibiting activity
05/02/2001EP1095038A1 Antagonists of gonadotropin releasing hormone
05/02/2001EP1095025A2 Benzimidazoles, production thereof and use thereof as medicaments
05/02/2001EP1095016A1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them
05/02/2001EP1094826A1 Novel therapeutic agents that modulate alpha-1a adrenergic receptors
05/02/2001EP1094816A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
05/02/2001EP1094815A1 Farnesyl protein transferase inhibitors for treating arthropathies
05/02/2001EP0984959A4 Aromatic sulfonyl alpha-hydroxy hydroxamic acid compounds
05/02/2001EP0983257A4 Aromatic sulfonyl alpha-cycloamino hydroxamic acid compounds
05/02/2001EP0973392A4 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
05/02/2001EP0885218B1 Oxa- and thia-diazole muscarinic receptor antagonists
05/02/2001EP0769947B1 Indolinone compounds for the treatment of disease
05/02/2001CN1293673A 1-(3-heteroarylpropyl-or-prop-2-enyl)-4-benzylpiperidines used as NMDA receptor antagonists
05/02/2001CN1293672A Process for preparation of nitrofuanidine derivatives
05/02/2001CN1293669A Benzylpiperazingl-and benzylipeeridinyl ethanone derivatives, their preparation method and their use as dopamine D receptor antagonists
05/01/2001US6225335 3-(4′-bromobenzylindenyl)-2-indolinone and analogues thereof for the treatment of disease
05/01/2001US6225312 Piperazine and piperidine compounds
04/2001
04/27/2001CA2324433A1 Process for the preparation of trisubstituted oxazoles
04/26/2001WO2001029029A1 Tetrahydrobenzindolone derivatives, their preparation and their use as 5-ht7 receptor antagonists
04/26/2001WO2001029028A1 9- (piperazinylalkyl) carbazoles as bax-modulators
04/26/2001WO2001029025A2 Tyrosine kinase inhibitors
04/26/2001WO2001029013A1 Process for preparing oxazolines from tetrahydrofurans
04/26/2001WO2001029012A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
04/26/2001WO2001029011A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
04/26/2001WO2001029006A1 Synthesis of 1,3,5-trisubstituted pyrazoles and intermediates therefore
04/26/2001WO2001028996A2 Pyrrolidine derivatives, their preparation and their use as inhibitors of neuraminidases
04/26/2001WO2001028987A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/26/2001WO2001028537A2 Bissulfonamide derivatives as enzyme inhibitors
04/26/2001WO2000059902A3 Aryl sulfonyls as factor xa inhibitors
04/26/2001WO2000055139A3 Heterocyclic urea and related compounds useful as anti-inflammatory agents
04/26/2001DE19932621A1 Neue substituerte alpha, beta-anellierte Butyrolactone New substituerte alpha, beta-fused butyrolactones
04/26/2001CA2388859A1 Inhibitors of neuraminidases
04/26/2001CA2387593A1 Enzyme inhibitors
04/26/2001CA2384240A1 Benzylcycloalkyl amines as modulators of chemokine receptor activity
04/26/2001CA2382212A1 Synthesis of 1,3,5-trisubstituted pyrazoles and intermediates therefore
04/25/2001EP1094063A1 9-(Piperazinylalkyl)carbazoles as Bax-modulators
04/25/2001EP1093368A1 INDOLE AND TETRAHYDROISOQUINOLINE CONTAINING $g(a)-KETO OXADIAZOLES AS SERINE PROTEASE INHIBITORS
04/25/2001EP0885263B1 Benzophenoxazine dyes
04/25/2001CN1292791A Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
04/25/2001CN1292787A Fungicidal benzoheterocyclyloxime
04/25/2001CN1064965C Novel sulfonamides compound and its use as medicine
04/25/2001CN1064964C Novel benzobiukyl, preparation of same and parmaceutical composition of same
04/24/2001US6222036 Reacting 2-thio-4-dimethyoxymethyl-pyrimidine with acetic acid and catalytic amount of concetrated sulfuric acid to produce 2-thiopyrimidine aldehyde
04/24/2001US6221863 Treating depression in a patient
04/24/2001US6221862 Microbicide 1,4,2-dioxazine derivatives
04/24/2001US6221574 Spectral sensitizers
04/24/2001CA2220055C Dipeptides which promote release of growth hormone
04/19/2001WO2001027108A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
04/19/2001WO2001027107A2 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001WO2001027091A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
04/19/2001WO2001027089A1 Pyrimidine derivatives
04/19/2001WO2001027085A1 Nicotinyl aspartyl ketones as inhibitors of caspase-3
04/19/2001WO2001026656A2 5-membered heterocycle derivatives and use thereof as monoamine oxidase inhibitors
04/19/2001WO2000018767A9 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
04/19/2001CA2388813A1 Heterocyclic sodium/proton exchange inhibitors and method
04/19/2001CA2388505A1 5-membered heterocycle derivatives, their preparation and application as medicine
04/19/2001CA2387493A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production
04/19/2001CA2386411A1 Nicotinyl aspartyl ketones as inhibitors of caspase-3
04/19/2001CA2384544A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production
04/19/2001CA2382605A1 Pyrimidine derivatives
04/18/2001EP1092711A1 Retinoid-associated receptor regulators
04/18/2001EP1091957A1 Pyrimidin-aminomethyl-pyridine derivatives, their preparation and their use in the control of helicobacter bacteria
04/18/2001EP1091955A1 Quinolones as serine protease inhibitors
04/18/2001EP1091945A1 Cyclic carbamates and isoxazolidines as iib/iiia antagonists
04/18/2001EP1091943A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
04/18/2001EP0765321B1 2-amino-3-aroyl-benzo beta thiophenes and method of making the same
04/18/2001EP0740661B1 Diphenyl oxazoline derivatives
04/18/2001EP0682663B1 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b]pyran-2-ones useful to treat retroviral infections
04/18/2001CN1291984A Glycine transport inhibitors
04/18/2001CN1291892A Substituted oxoazaheterocyclyl factor Xa inhibitors
04/18/2001CN1064679C Herbicidal thiocarbamoyltetrazolinones
04/17/2001US6218550 Intermediates useful for the manufacture of carbapenem and a stereoselective manufacturing method therefor
04/17/2001US6218547 1-phenyl-benzimidazole compounds and their use as GABA-a receptor modulators