Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
04/2008
04/23/2008CN101166723A New compound for the treatinginflammatory disease
04/22/2008US7361787 Prophylaxis of respiratory disorders and therapy, also metod of synthesis and composition with PDE4 inhibitor, corticosteroid hibitor or anticholinergic agent
04/22/2008US7361771 Process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1H-pyrrole-3-carboxylic acid phenylamide
04/22/2008US7361685 Compounds for use in the treatment of skin conditions
04/22/2008US7361682 Indole derivatives as H3 inverse agonists
04/22/2008US7361678 Azole derivatives and fused bicyclic azole derivatives as therapeutic agents
04/22/2008US7361677 Polycyclic sulphamate compounds suitable for use as inhibitors of aromatase and/or sulphatase
04/22/2008US7361669 particularly useful for treating cardiovascular disease
04/22/2008US7361665 For therapy of inflammatory disease, autoimmune disease, destructive bone disorder, proliferative disorder, infectious disease, neurodegenerative disease, allergy, reperfusion/ischemia in stroke, heart attack, hypoxia
04/22/2008US7361657 Drugs for treatment of respiratory syncytial virus and salt formation
04/22/2008US7361655 Pharmaceutically effective compounds
04/22/2008US7361648 1-(4-{ethyl-[2-(4-methanesulfonylphenyl)-1-methylethyl]amino}butyl)-4-methanesulfonyl-[1,4]diazepan-2-one; repiratory system disorders: asthma and chronic obstructive pulmonary disease; nervous system, muscular,urogenital, gastrointestinal disorders; antiallergens; side effect reduction
04/22/2008CA2400447C Kinase inhibitors
04/22/2008CA2350137C New piperazine and di-dehydropiperidine compounds
04/22/2008CA2302669C Piperidinylmethyloxazolidinone derivative
04/22/2008CA2270777C Quinoline and quinazoline derivatives having corticotropin releasing factor (crf) antagonist activity
04/22/2008CA2210693C Pyrazol-4-yl-benzoyl derivatives and their use as herbicides
04/17/2008WO2008045978A1 Pinane-substituted pyrimidinediamine derivatives useful as axl inhibitors
04/17/2008WO2008045564A2 Carboxamide compounds and their use as antagonists of the chemokine ccr2 receptor
04/17/2008WO2008044767A1 Aromatic amine derivative and use thereof
04/17/2008WO2008044700A1 GSK-3β INHIBITOR
04/17/2008WO2008044102A1 Polymorph form of aprepitant and process for the preparation thereof
04/17/2008WO2008043788A2 Novel compounds
04/17/2008WO2008043544A1 Sulfonamide substituted pyrazoline compounds, their preparation and use as cb1 modulators
04/17/2008WO2008043183A1 Cyclopropyl-piperazine compounds as calcium channel blockers
04/17/2008WO2008027542A3 5-substituted isoindoline compounds
04/17/2008WO2008024337A3 Compounds and methods for inhibiting the interaction of bcl proteins with binding partners
04/17/2008WO2008022164A3 Pyrazine compounds, their use and methods of preparation
04/17/2008WO2008022046A3 Dicer substrate rna peptide conjugates and methods for rna therapeutics
04/17/2008WO2008019372A3 2-aminobenzoxazole carboxamides as 5ht3 modulators
04/17/2008WO2008008887A3 Gpr119 agonists for treating metabolic disorders
04/17/2008WO2008007390B1 An improved process for purification of zolmitriptan
04/17/2008WO2008002570B1 Human protein tyrosine phosphatase inhibitors and methods of use
04/17/2008WO2007144785A3 Ryanodine receptor inhibitors and methods relating thereto
04/17/2008US20080091026 Alpha crystal oxazolidone derivative; powder X-ray diffraction peaks at about 4.3, 8.9, 11.7, 15.6, and 16.3 degrees 2-theta; treatment or prevention of diseases, bacterial infections resistant to antibiotics
04/17/2008US20080091011 Novel crystalline form of linezolid
04/17/2008US20080091010 Induce the biosynthesis of cytokines such as interferon and tumor necrosis factor; antiviral and antitumor agents
04/17/2008US20080090884 Antimicrobial [3.1.0] bicyclohexylphenyl- oxazolidinone derivatives and analogues
04/17/2008US20080090863 Melanin Concentrating Hormone (MCH) receptor antagonists; eating disorder, obesity, psychological disorders, drug addiction, diabetes, cardiovascular disorders; 2-(cyclohexyl(alkyl)amino)pyridines such as 3-chloro-4-fluoro-N-(cis-4-[(4-methoxypyridin-2-yl)amino]cyclohexyl)benzamide
04/17/2008US20080090846 Chemokine receptor binding heterocyclic compounds
04/17/2008US20080090840 Heterocyclic GPR40 Modulators
04/17/2008US20080090830 thrombosis, atherosclerosis, restenosis, hypertension, angina pectoris, arrhythmia, heart failures and cancer
04/17/2008US20080090828 insecticides for soil-borne insects, such as termites and white grubs; less costly and safer to use on crops; N-{4-[(4-{bis[4-(trifluoromethyl)phenyl]methylene}piperidyl)methyl]phenyl}ethoxycarboxamide, N-oxide
04/17/2008US20080090824 Novel crystalline form of linezolid
04/17/2008US20080090821 Improved solubility, lower tendency to bind to plasma proteins and greater activity especially in serum-based assay systems; remodeling of heart after myocardial infarction; atherosclerosis; 2-[4-(4-Fluorophenoxy)benzenesulfonyl]-6-(2-piperidin-1-ylethoxy)-1,2,3,4-tetrahydroisoquinoline-1-carboxylic acid
04/17/2008US20080090820 Novel crystalline form of linezolid
04/17/2008US20080090818 (4-Morpholin-4-yl-phenyl)-[5-(1H-pyrazol-4-yl)-[1,2,4]triazolo[1,5-a]pyrazin-8-yl]-amine; mitogen-activated protein kinase and matrix metallo proteinase inhibitor; antiinflammatory and analgesic agent; rheumatoid arthritis
04/17/2008US20080090816 Anti-infective biaryl compounds
04/17/2008US20080090815 Anticoagulates for treating cardiovascular disorders, such as myocardial infarct, angina pectoris, restenoses after angioplasty, bypass, stroke; treatment of atherosclerosis, arthritis, Alzheimer's disease or cancer
04/17/2008US20080090813 4-(3-hydroxy-1-propyl)-6-(3-trifluoromethylphenyl)-pyrimidine-2-carbonitrile; cysteine proteases (cathepsin K and S) inhibitor; antiinflammatory and analgesic agent; rheumatoid arthritis, multiple sclerosis, chronic and neuropathic pain
04/17/2008US20080090807 Lactam-containing compounds and derivatives thereof as factor xa inhibitors
04/17/2008US20080090802 2-[2-(3-Chlorophenyl)-4-oxo-6-perhydro-1,4-diazepin-1-yl-4H-quinazolin-3-yl]-N-isopropylacetamide; hypothalamo-pituitary-adrenal (HPA) axis stress relieving agent; adrenocorticotropic hormone (ACTH)/ glucocorticoid antagonist; psychological and bipolar disorders, schizophrenia, psychosis, hyperactivity
04/17/2008US20080090800 Mandelic acid derivatives and their use as thrombin inhibitors
04/17/2008US20080090797 tert-Butyl[3-(4-phenyloxazolidin-2-on-3-yl)-4-(2-styryl)azetidin-2-on-1-yl]acetate; known as synthetic intermediates for the preparation of beta -lactam antibiotics; diuretic
04/17/2008US20080090794 Potassium Channel Inhibitors
04/17/2008US20080090782 Inhibit DNA-dependent protein kinase; reduced side effects caused by radiation and chemotherapy drugs
04/17/2008CA2666275A1 Cyclopropyl-piperazine compounds as calcium channel blockers
04/16/2008EP1911758A1 Phenyl piperidine derivatives for use as renin inhibitors
04/16/2008EP1911756A2 Substituted pyridinyl and pyrimidinyl derivatives as modulators of metabolism and the treatment of disorders related thereto
04/16/2008EP1911755A1 Benzoimidazole compound capable of inhibiting prostaglandin d synthetase
04/16/2008EP1911749A1 New long-working Beta-2 agonists and their use as medicine
04/16/2008EP1911747A1 Sulfonamide substituted pyrazoline compounds, their preparation and use as CB1 modulators
04/16/2008EP1911350A1 Amidine compound and herbicide
04/16/2008EP1910378A1 Hepatitis c inhibitor peptide analogs
04/16/2008EP1910352A1 Heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase
04/16/2008EP1910351A1 Colourless water-soluble organic luminophores and intermediates thereof
04/16/2008EP1910346A2 Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonist
04/16/2008EP1910342A1 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease
04/16/2008EP1910338A2 Heterotetracyclic compounds as tpo mimetics
04/16/2008EP1910335A1 N-(heteroaryl)-1-heteroarylalkyl-1h-indole-2-carboxamide derivatives, preparation and use thereof
04/16/2008EP1910321A1 New compounds, process for their preparation, intermediates, pharmaceutical compositions and their use in the treatment of 5-ht6 mediated disorders such as alzheimer's disease, cognitive disorders, cognitive impairment associated with schizophrenia, obesity and parkinson's disease
04/16/2008EP1910290A2 Gpcr agonists
04/16/2008EP1909792A1 Substituted piperidine derivatives as somatostatin sst1 receptor antagonists
04/16/2008EP1909791A1 G-protein coupled receptor agonists
04/16/2008EP1909789A2 Antidiabetic oxazolidinediones and thiazolidinediones
04/16/2008EP1909572A2 Potassium channel inhibitors
04/16/2008EP1711492B1 Substituted quinolines and their use as mycobacterial inhibitors
04/16/2008CN101163700A 三胺衍生物 Triamine derivative
04/16/2008CN101163699A Methods for synthesis of dicarbamate compounds and intermediates in the formation thereof
04/16/2008CN101163692A Heterocyclic substituted piperazines with cxcr3 antagonist activity
04/16/2008CN101163683A 4-0x0quinaz0lin-3-yl benzamide derivatives for the treatment of cytokine diseases
04/16/2008CN101163478A Compounds for inflammation and immune-related uses
04/16/2008CN100381441C 5,5' bit connected 1,1'-diphenyl kind axle chirality ligand
04/16/2008CN100381437C Compounds, compositions and methods
04/15/2008USRE40245 Gyrase inhibitors and uses thereof
04/15/2008US7358386 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation
04/15/2008US7358376 Substituted Thiophene compounds
04/15/2008US7358276 2-Oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
04/15/2008US7358268 Imidazole derivatives as factor Xa inhibitors
04/15/2008US7358265 Oxa-and thiadiazoles and their use as metalloproteinase inhibitors
04/15/2008US7358263 Fused bicyclic-substituted amines as histamine-3 receptor ligands
04/15/2008US7358254 Method for treating atherosclerosis employing an aP2 inhibitor and combination
04/15/2008US7358251 Bcl-XL inhibitors; N-{[4-({(1R)-5-(dimethylamino)-1-[(phenylthio)methyl]pentyl}amino)-3-nitrophenyl]sulfonyl}-4-(4-fluorophenyl)piperidine-1-carboxamide; useful for promoting apoptosis; Anticancer agents; autoimmune diseases; antiinflammatory agents
04/15/2008US7358250 Pyrrolo[2,3-d]pyrimidines that modulate ACK1 activity
04/15/2008US7358249 Heterocyclic compounds having inhibitory activity against HIV integrase
04/15/2008US7358247 Mycophenolate mofetil impurity
04/15/2008US7358246 5-(4,4-dimethyl-2-oxo-1,4-dihydro-2H-3,1-benzoxazin-6-yl)-1-methyl-1H-pyrrole-2-carbothioamide; contraceptive, menopause; reduces risk of uterine cancers coused by treating with estrogen receptor (ER) agonists
04/10/2008WO2008042928A2 Oxadiazole and thiadiazole derivatives as mitotic kinesin inhibitors and methods of use thereof
04/10/2008WO2008041075A1 Mglur5 modulators
04/10/2008WO2008040979A1 Arginine derivatives with np-i antagonistic activity