Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
06/2008
06/19/2008US20080146533 Containing tertiary amine linked pyrrolidine, azetidine, morpholine or piperidine group; inhibiting GlyCer synthase, lowering glycosphingolipid levels; collagen vascular diseases, atherosclerosis, diabetic renal hypertrophy
06/19/2008US20080146523 Imidazole derivatives
06/19/2008US20080146458 Process for the preparation of oxazolidinones and method of use thereof
06/19/2008US20080145356 Administering glutenase to Celiac or dermatitis herpetiformis patient reduces levels of toxic gluten oligopeptides
06/19/2008CA2672601A1 Polycyclic acid compounds useful as crth2 antagonists and antiallergic agents
06/19/2008CA2672347A1 Sulfonyl-phenyl-2h-[1,2,4]oxodiazol-5-one derivatives, processes for their preparation and their use as pharmaceuticals
06/19/2008CA2672233A1 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds and methods of their use
06/19/2008CA2672167A1 Dihydropyridine derivatives as useful as protein kinase inhibitors
06/19/2008CA2672101A1 Compounds and compositions as kinase inhibitors
06/19/2008CA2672023A1 Process for the preparation of valsartan and intermediate products
06/19/2008CA2671970A1 4-phenyl-pyrane-3,5-diones, 4-phenyl-thiopyrane-3,5-diones and cyclohexanetriones as novel herbicides
06/19/2008CA2670728A1 Pyridine derivatives used as xiap inhibitors
06/18/2008EP1932843A1 Sulfonyl-phenyl-2H-(1,2,4) oxadiazole-5-one derivatives, processes for their preparation and their use as pharmaceuticals
06/18/2008EP1932842A1 Compound having oxadiazole ring structure bonded with aromatic heterocyclic ring and organic electroluminescent device
06/18/2008EP1932840A1 Nitrogen-containing heterocyclic compound and pharmaceutical application thereof
06/18/2008EP1932837A1 Bicyclo heterocyclic compound having antifungal action
06/18/2008EP1932836A1 Isoxazoline-substituted benzamide compound and harmful organism-controlling agent
06/18/2008EP1931681A1 Substituted benzofused derivatives and their use as vanilloid receptor ligands
06/18/2008EP1931662A1 Pyrimidine derivatives for the inhibition of igf-ir tyrosine kinase activity
06/18/2008EP1931661A1 Isoxazolo derivatives as gaba a alpha5 inverse agonists
06/18/2008EP1931660A2 Phenyl-[1,2,4]-oxadiazol-5-one derivatives with phenyl group, processes for their preparation and their use as pharmaceuticals
06/18/2008EP1931659A1 Derivatives of 2 -aminthiazoles and 2-aminooxazoles, processes for their preparation and their use as pharmaceuticals
06/18/2008EP1931657A2 Novel high affinity quinoline-based kinase ligands
06/18/2008EP1931645A2 N- (3-amino-quinoxalin-2-yl) -sulfonamide derivatives and their use as phosphatidylinositol 3-kinase inhibitors
06/18/2008EP1931643A1 2-substituted hydroxylaminopyrimidine, method for the production and the use thereof in the form of pesticides
06/18/2008EP1931640A2 Substituted-3-sulfonylindazole derivatives as 5-hydroxytryptamine-6 ligands
06/18/2008EP1931637A2 Methods of modulating neurotrophin-mediated activity
06/18/2008EP1931627A1 Amino-alkyl-amide derivatives as ccr3 receptor ligands
06/18/2008EP1931337A2 Phenyl- and pyridinyl- 1, 2 , 4 - oxadiazolone derivatives, processes for their preparation and their use as pharmaceuticals
06/18/2008EP1931205A2 Transglutaminase inhibitors and methods of use thereof
06/18/2008EP1585521B1 Derivatives of aryl-quinazoline/aryl-2amino-phenyl methanone which promote the release of parathyroid hormone
06/18/2008EP1485378B1 Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase
06/18/2008CN101203512A Heterocyclic compound
06/18/2008CN101203511A New azetidine derivatives as neurokinin receptor antagonists for the treatment of gastrointestinal diseases
06/18/2008CN101203510A Carbon-linked substituted piperidines and derivatives thereof used as histamine H3 antagonists
06/18/2008CN101203509A Amine-linked pyridyl and phenyl substituted piperazine-piperidines with CXCR3 antagonist activity
06/18/2008CN101203498A Heterocyclic anti-viral compounds comprising metabolizable moieties and their uses
06/18/2008CN101203243A Remedy for xanthoma
06/18/2008CN101203134A Substituted arylpyrazoles as parasiticidal pharmaceutical product
06/18/2008CN101200456A Bromine difluoro methyl substituted isoxazole derivatives
06/18/2008CN101200454A Crystalline modifications of triazinylaminostilbenes
06/17/2008US7388095 modulation of H3 Histamine receptors; e.g. 5-(4-isopropyl-morpholin-2-ylmethoxy)-1-(2,2,2-trifluoro-ethyl)-1H-indol-2-yl]-morpholin -4-yl-methanone; antagonists/inverse agonists
06/17/2008US7388025 3-aryl-isoxazole-4-carbonyl-benzofuran derivatives
06/17/2008US7388021 Novel pyridyl or phenyl ureas and analogues; Purinoreceptors inhibitors; 1-(4-tert-butylphenyl)-3-(2-(3-isopropylphenoxy)pyridin-3-yl)urea; for the treatment of a thromboembolic disorders
06/17/2008US7388020 Compounds for chronic obstructive pulminary disorders for breathingand respiratory system diorders
06/17/2008US7388013 Capped pyrazinoylguanidine sodium channel blockers
06/17/2008US7388007 2-(3-acetamido-3-isobutyl-2-oxopyrrolidin-1-yl)-N-(3-(3,5-difluorophenyl)-1-hydroxy-1-(4-propoxypyrrolidin-2-yl)propan-2-yl)-4-phenylbutanamide; beta-amyloid peptide inhibitors; neurodegenerative diseases; Alzheimer's Disease, cerebral amyloid angiopathy and Down's Syndrome
06/17/2008CA2501799C Pyrazole compounds for treatment of neurodegenerative disorders
06/17/2008CA2439152C Acylated piperidine derivatives as melanocortin-4 receptor agonists
06/17/2008CA2395193C Pyrrolidine derivatives as cyclic amp-specific phosphodiesterase inhibitors
06/17/2008CA2393749C Substituted 8-arylquinoline phosphodiesterase-4 inhibitors
06/17/2008CA2286772C Fungicide active substance combinations
06/12/2008WO2008070831A2 Bisbenzamidines and bisbenzamidoximes for the treatment of human african trypanosomiasis
06/12/2008WO2008070661A1 Substituted pyrimidines as adenosine receptor antagonists
06/12/2008WO2008070447A2 Anti-viral compounds
06/12/2008WO2008069997A1 Substituted diazepan compounds as orexin receptor antagonists
06/12/2008WO2008069242A1 Novel bicyclic heterocyclic compound
06/12/2008WO2008068270A1 Antibacterial quinoline derivatives
06/12/2008WO2008068267A1 Antibacterial quinoline derivatives
06/12/2008WO2008068183A1 Indoles
06/12/2008WO2008068157A1 2-aminoquinolines as 5-ht(5a) receptor antagonists
06/12/2008WO2008067871A1 Substituted dihydropyrazolones for treating cardiovascular and haematological diseases
06/12/2008WO2008067644A1 Inhibitors of hiv replication
06/12/2008WO2008033389A3 Macrocyclic hcv inhibitors and their uses
06/12/2008WO2008017361A3 2-(heterocyclylbenzyl)pyridazinone derivatives
06/12/2008WO2007118323A8 Isoxazole derivatives as calcium channel blockers
06/12/2008WO2007110237A3 Amide derivatives and their application for the treatment of g protein related diseases
06/12/2008US20080139811 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection
06/12/2008US20080139627 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides
06/12/2008US20080139617 Indoles
06/12/2008US20080139563 Oxazolidinone derivatives and methods of use
06/12/2008US20080139562 e.g. {-[3-Cyclopentyl-2-(4-methane sulfonyl-phenyl)-propionylamino]-5-methyl-thiazol-4-yl}-acetic acid ethyl ester; antidiabetic and hypoglycemic agent; non-insulin dependent diabetis, obesity, impaired glucose tolerance, eating disorder, dyslipidemia, hyperlipidemia, hypertension
06/12/2008US20080139561 e.g. 6-(5-Cyclopropyl-1H-pyrazol-3-ylamino)-5-fluoro-2-(1-(4-fluorophenyl)ethylamino) nicotinonitrile; tropomyosin-related kinases (Trk's) inhibitor; anticarcinogenic agent; hormone related cancer, leukemia; antiinflammatory agent; arthritis, restenosis; autoimmune diseases
06/12/2008US20080139560 Ion Channel Modulators
06/12/2008US20080139557 [5-(Pyridin-2-ylamino)-6-oxo-1,6-dihydro-pyridin-3-yl]-(3-amido)-benzene derivatives; anticarcinogenic, antiproliferative, antiallergen, and antiinflammatory agents; lymphoma, leukemia, autoimmune diseases; Bruton's tyrosine kinase inhibitors
06/12/2008US20080139555 1-[(4-{[4-(3-amino-6-methylphenyl)piperidyl]methyl}phenyl)sulfonyl]-4; melatonin-concentrating hormone (MCH1) receptor ligand; antidepressant, anxiolytic, antidiabetic agent
06/12/2008US20080139553 Spiro-piperidine derivatives
06/12/2008US20080139552 Indoles
06/12/2008US20080139550 e.g. {5-Chloro-2-[4-(2-oxo-2,3-dihydro-benzooxazol-7-yl)-piperidine-1-carbonyl]-1H-indol-7-yl}-acetonitrile; vasopressin receptors antagonist; antidepressant, anxiolytic agent; dysmenorrhea, hypertension, inappropriate secretion of vasopressin, liver cirrhosis, obsessive compulsive disorder
06/12/2008US20080139549 Indoles
06/12/2008US20080139548 Indoles
06/12/2008US20080139547 N-Hydroxyalkynylbenzamide (or hydroxamate) derivatives; anticarcinogenic and antiproliferative agents
06/12/2008US20080139546 e.g. 3-(3,4-dihydroquinolin-1(2H)-yl)-N-{[8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}propan-1-amine; modulators of serotonin 5-HT1A receptor activity and/or serotonin reuptake; antidepressant, anxiolytic agent, cognition activator; schizophrenia, sexual disorders
06/12/2008US20080139536 Benzodiazepines for Treating or Preventing Rsv Infection
06/12/2008US20080139534 Bisbenzamidines and bisbenzamidoximes for the treatment of human African trypanosomiasis
06/12/2008US20080139533 Substituted 4-imidazoles
06/12/2008US20080139532 Tetrahydrobenzazepine Derivatives as Modulators of Dopamine D3 Receptors (Antipsychotic Agents)
06/12/2008US20080139530 7-Aryl 1,5-Dihydro-4,1-Benzoxazepin-2(3H)-One Derivatives And Their Use As Progesterone Receptor Modulators
06/12/2008US20080139390 Isoxazoline Derivatives and Their Use as Herbicides
06/12/2008US20080138740 Cyanine Compound, Optical Recording Material Using the Same and Optical Recording Medium
06/12/2008CA2671749A1 Bicyclic compounds and uses as antidiabetics
06/12/2008CA2670892A1 Substituted diazepan compounds as orexin receptor antagonists
06/12/2008CA2670139A1 Indoles
06/12/2008CA2669829A1 Antibacterial quinoline derivatives
06/12/2008CA2669819A1 Antibacterial quinoline derivatives
06/12/2008CA2669590A1 2-aminoquinolines as 5-ht(5a) receptor antagonists
06/11/2008EP1930322A1 1-(4-piperidinyl)-1,3-dihydro-2H-benzoxazole-2-one derivatives and related compounds as nociceptin analogs and ORL1 ligands for the treatment of pain
06/11/2008EP1930319A1 Proline derivatives and use thereof as drugs
06/11/2008EP1928868A1 Iminooxazolidine derivatives and use thereof
06/11/2008EP1928867A1 2-aminoethoxyacetic acid derivatives and their use in treating thromboembolic disorders