Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
06/2008
06/11/2008EP1928866A1 Substituted indazoles as inhibitors of phosphodiesterase type-iv
06/11/2008EP1928864A1 Novel cycloalkane carboxamides as factor xa inhibitors
06/11/2008EP1928861A1 4- (ih-indazol-s-yl-amino)-quinazoline compounds as erbb receptor tyrosine kinase inhibitors for the treatment of cancer
06/11/2008EP1928859A1 Pyrazole derivates as cannabinoid receptor modulators
06/11/2008EP1928846A2 Triazole compounds that modulate hsp90 activity
06/11/2008EP1928829A1 Piperidine derivatives as antagonists of the cc chemokine receptor ccr1 and their use as anti-inflammatory agents
06/11/2008EP1928821A1 Carboxamide derivatives as muscarinic receptor antagonists
06/11/2008EP1727809B1 Substituted morpholine and thiomorpholine derivatives
06/11/2008EP1485348B1 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
06/11/2008EP1255739B1 3-aminoquinazolin-2,4-dione antibacterial agents
06/11/2008CN101198604A NPY antagonists, preparation and use
06/11/2008CN101198603A 4-(pyrid-2-yl) amino substituted pyrimidine as protein kinase inhibitors
06/11/2008CN101198598A Compounds, compositions and methods for stabilizing transthyretin and inhibiting transthyretin misfolding
06/11/2008CN101198596A 2-amino-quinaz0lin-5-ones as HSP90 inhibitors useful in treating proliferation diseases
06/11/2008CN101195601A 2-dihydro indolone derivant, preparation method and application thereof
06/11/2008CN100393741C Compounds with anti-inflammatory activity
06/11/2008CN100393717C Benzoxazine containing maleimide and allyl ether and its preparing method
06/11/2008CN100393714C Gyrase inhibitors and uses thereof
06/10/2008US7385063 Method for preparing imidazole derivatives
06/10/2008US7385061 Furazanobenzimidazoles
06/10/2008US7385059 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators
06/10/2008US7384970 Inhibitors of cathepsin S
06/10/2008US7384965 Fused heterocyclic derivatives as PPAR modulators
06/10/2008US7384964 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
06/10/2008US7384963 2′-Methyl-5-(1,3,4-oxadiazol-2-yl)1, 1′-biphenyl-4-carboxaide derivatives and their use as p38 kinase
06/10/2008US7384957 3,4-dihydro-1H-isoquinolin-2-yl-derivatives
06/10/2008US7384947 Treating cancer with anticarcinogenic agents 3-Amino-9-chloro-5,6,7,8-tetrahydro-naphtho[2,3-b]furan-2-yl))-(2-methyl-pyridin-3-yl)-methanone; antiproliferative agents
06/10/2008US7384944 Organ grafting; antiarthritic agents; inflammatory bowel disease
06/10/2008US7384936 Carboxamidine derivatives and their use in the treatment of vascular diseases
06/10/2008US7384929 N-aryl azaspiroalkene and azaspiroalkane compounds and methods of preparation and use thereof
06/10/2008CA2393995C Novel benzene sulfonamide derivatives, their preparation and pharmaceutical compositions containing them
06/10/2008CA2238889C Method for selective protection of baccatin derivatives and its application to taxane synthesis
06/05/2008WO2008066131A1 Novel phenyl-isoxazol-3-ol derivative
06/05/2008WO2008066097A1 Carboxylic acid derivative
06/05/2008WO2008065500A2 Heteroaryl amides as type i glycine transport inhibitors
06/05/2008WO2008065141A1 Novel inhibitors of glutaminyl cyclase
06/05/2008WO2008064789A1 Substituted 4-amino-3,5-dicyano-2-thiopyridines and use thereof
06/05/2008WO2008064788A1 Cyclically substituted 3,5-dicyano-2-thiopyridines and use thereof
06/05/2008WO2008064474A1 Azacycloalkane derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase
06/05/2008WO2008043788A3 Novel compounds
06/05/2008WO2008033857A3 Substituted amides, method of making, and method of use thereof
06/05/2008WO2007112322A3 Indole compounds having sphingosine-1-phosphate (s1p) receptor agonist and/or antagonist biological activity
06/05/2008US20080132706 Compounds as PDE IV and TNF Inhibitors
06/05/2008US20080132699 Process For the Preparation of Diazine Derivatives
06/05/2008US20080132551 Positive allosteric modulators of the nicotinic acetylcholine receptor
06/05/2008US20080132548 Certain chemical entities, compositions, and methods
06/05/2008US20080132546 e.g. Methyl 2-(6-{[(ethylamino)carbonyl]amino}pyridin-3-yl)-1,3-thiazole-5-carboxylate; bacterial DNA gyrase or bacterial topoisomerase IV inhibitor; antibacterial agent; antibiotic resistance; skin structure infections, pneumoniae, bronchitis, acute sinusitis, otitis media, sepsis, osteomyelitis
06/05/2008US20080132540 Such as trans-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-N-(1-benzyl-piperidin-4-yl)-3-phenyl-acrylamide; for treating/preventing anxiolytic disorders/depression, injured mammalian nerve tissue, conditions, neurological disorders, bone loss, substance related disorders, and obesity; neuropeptide y (NPY Y2)
06/05/2008US20080132524 Ortho-heterocyclic substituted aryl amides for controlling invertebrate pests
06/05/2008US20080132523 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/05/2008US20080132520 Compositions, kits and methods for administering a titration schedule comprising bifeprunox compounds
06/05/2008US20080132516 Viricides, immunomodulators or HIV entry inhibitors; lymphadenopathy associated virus, human T-cell leukemia/lymphoma virus; AIDS
06/05/2008US20080132506 Anti-inflammatory medicaments
06/05/2008US20080132504 2, 4-Pyrimidinediamines Useful In The Treatment Of Neoplastic Diseases, Inflammatory And Immune System Disorders
06/05/2008US20080132503 Inhibitors of Histone Deacetylase
06/05/2008US20080132502 Phosphatidylinositol (PI) 3-kinase (PI3K); N-[5-(5-Benzylamino-6-chloropyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]acetamide, for example; anticancer agents, cardiovascular disorders, autoimmune disorders, rheumatic diseases
06/05/2008US20080132501 Indazole compounds
06/05/2008US20080132496 Anticoagulants; factor Xa inhibitors; compounds are N-(benzimidazolyl, imidazo(4,5-b)pyridyl- or indolyl)-substituted benzamides
06/05/2008US20080132495 Pyrazole Compounds that Modulate the Activity of Cdk, Gsk and Aurora Kinases
06/05/2008US20080132487 5-aminopyrazole derivatives as pesticidal compounds
06/05/2008US20080132483 Administering (3R,5S)-N-propanesulfonyl-7-chloro-5-(2,3-dimethoxyphenyl)-1-(3-hydroxy-2,2-dimethylpropyl)-1,2,3,5-tetrahydro-4,1-benzoxazepine-3-acetamide; cerebral infarction
06/05/2008DE60129697T2 Kondensierte azepinderivate und ihre verwendung als antidiuretisches mittel Condensed azepine derivatives and their use as antidiuretic agent
06/05/2008CA2671080A1 Carboxylic acid derivatives
06/05/2008CA2668713A1 Novel phenyl-isoxazol-3-ol derivative
06/04/2008EP1927594A1 1,2,3-Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
06/04/2008EP1926826A2 Class iia histone deacetylase (hdac) substrate
06/04/2008EP1926728A1 Dioxazine- and oxadiazine-substituted arylamides
06/04/2008EP1926725A1 Alkoxy indolinone based protein kinase inhibitors
06/04/2008EP1926724A1 Analogs of dehydrophenylahistins and their therapeutic use
06/04/2008EP1926721A2 Thiophene and thiazole substituted trifluoroethanone derivatives as histone deacetylase (hdac) inhibitors
06/04/2008EP1926711A1 Novel heterobicyclic derivatives useful as inhibitors of liver carnitine palmitoyl transferase
06/04/2008EP1926708A1 Biaryl substituted heterocycle inhibitors of lta4h for treating inflammation
06/04/2008EP1343775B1 Piperazine derivatives
06/04/2008EP1237887B1 9-(piperazinylalkyl)carbazoles as bax-modulators
06/04/2008EP1204643B1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
06/04/2008EP0931071B1 Methods of making hiv-protease inhibitors and intermediates for making them
06/04/2008CN101193880A Exo- and diastereo- selective syntheses of himbacine analogs
06/04/2008CN101193869A Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/04/2008CN101193868A Pyrimidine derivatives for the treatment of GABA B mediated nervous system disorders
06/04/2008CN101193867A N-substituted benzimidazolyl c-Kit inhibitors and combinatorial benzimidazole library
06/04/2008CN101190917A 3,4-dihydro-3-methyl-4-oxomidazo[5,1-d]-1,2,3,5-tetrazine-8-formic acid benzenesulfonyl furoxan esters compound, preparation method and use thereof
06/04/2008CN100391954C Enantiomers of thiophene hydroxamic acid derivatives and their use as hdac inhibitors
06/04/2008CN100391944C Indoles useful in the treatment of androgen-receptor related diseases
06/04/2008CN100391338C Arthropodicidal anthranilamides
06/03/2008US7381825 Antiinflammatory agents; skin disorders; inflammatory bowel disorders
06/03/2008US7381738 Substituted bicycloalkylamine derivatives as modulators of chemokine receptor activity
06/03/2008US7381726 Polymorphic forms of 1-′4-(5-cyanoindol-3-yl)butyl-4-(2-carbamoylbenzofuran-5-yl)piperazine hydrochloride
06/03/2008US7381723 Antiserotonine agents; stroke, brain disorders;trauma; Alzheimer's disease; neurodegenerative disease; schizophrenia; psychological disorders; anxiolytic agents; controlling stresses; eating disorders; sleep disorders; sexual disorders
06/03/2008US7381722 poly (ADP-ribose) synthetase inhibitors; synergistic; indeno[1,2-c]isoquinoline derivatives; inflammatory disease, a reperfusion injury, diabetes or its complications, reoxygenation injury resulting from organ transplantation, an ischemic condition, Parkinson's disease, renal failure, a vascular disease
06/03/2008US7381721 Substituted piperidine compounds
06/03/2008US7381719 To treat obesity and Related Diseases; oral bioavailablility, oral administration; inhibition of orexigenic effects; side effects reduction; weight loss while maintaining or minimizing the loss of lean muscle mass; 6-[4-(2-Benzylamino-ethyl)-phenoxy]-nicotinamide
06/03/2008US7381687 3-heteroaryl substituted 5-methyloxymethyl isoxazolines used as herbicides
06/03/2008CA2401711C Cyclic amide derivatives
06/03/2008CA2389360C Urea derivatives as anti-inflammatory agents
05/2008
05/29/2008WO2008064315A1 Tetralin analogs having sphingosine 1-phosphate agonist activity
05/29/2008WO2008063912A1 Substituted pyrazole and triazole compounds as ksp inhibitors
05/29/2008WO2008063667A1 Heterotricyclic metalloprotease inhibitors
05/29/2008WO2008063625A2 Pyridine compounds and methods of their use
05/29/2008WO2008062905A2 Heteromonocyclic compound and use thereof
05/29/2008WO2008062878A1 Novel pyrazole derivative, harmful organism control agent, and use of the control agent