Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
01/2008
01/24/2008WO2007094819A3 Triazole compounds that modulate hsp90 activity
01/24/2008WO2007001975A8 Piperidine derivatives useful as histamine h3 antagonists
01/24/2008US20080021222 Reacting an organic amine compound with a carbamyl-group-containing amide compound in the presence of a suitable polar or nonpolar aprotic, substantially anhydrous solvent or mixtures thereof; used as therapeutic agents for IMPDH-mediated diseases
01/24/2008US20080021217 Heterocyclic inhibitors of rho kinase
01/24/2008US20080021215 Reacting 3-fluoro-4-morpholinyl aniline derivative with epichlorohydrin; converting chloromethyl oxazolidinone to aminomethyl oxazolidinone; carbonylation ; reacting with potassium phthalimide, hydrazine hydrate, and acetic anhydride; cyclization, carbamylation; antibacterial agent
01/24/2008US20080021214 Novel process for the preparation of linezolid and related compounds
01/24/2008US20080021213 Intermediates for oxazolidinone antibacterials; N-[3-Chloro-2-(R)-hydroxypropyl]-3-fluoro-4-morpholinyl aniline
01/24/2008US20080021180 Chromium catalysts active in olefin polymerization
01/24/2008US20080021079 Compounds, Compositions, and Methods
01/24/2008US20080021071 3-{4-(Pyridin-3-Yl) Phenyl}-5-(1H-1,2,3-Triazol-1-Ylmethyl)-1,3-Oxazolidin-2-Ones as Antibacterial Agents
01/24/2008US20080021053 Heterocyclic Derivatives
01/24/2008US20080021030 Substituted Pyrazoles As Ppar Agonists
01/24/2008US20080021029 Substituted Cyclic Urea Derivatives, Preparation Thereof And Pharmaceutical Use Thereof As Kinase Inhibitors
01/24/2008US20080021028 ((2S,3S) N,2-dihydroxy-5-methyl-3-{[4-(2-pyridinyl)-1-piperazinyl]carbonyl}hexanamide; for treatment and/or prevention of disorders related to autoimmune disorders and/or inflammatory diseases, cardiovascular diseases, neurodegenerative diseases, stroke, cancer, pre-term labor, endometriosis
01/24/2008US20080021027 Novel benzimidazole derivatives
01/24/2008US20080021025 Inhibitors of cathepsin s
01/24/2008US20080021022 (5-(4-Chlorophenyl)isoxazol-4-yl)(3-(pyridin-3-yl)pyrrolidin-1-yl)methanone; enzyme inhibitor of Hydroxysteroid dehydrogenases; treatment of diabetes, obesity
01/24/2008US20080021012 3-[4-{6-Substituted Alkanoyl Pyridin-3-Yl}-3-Phenyl]-5-(1H-1,2,3-Triazol-1-Ylmethyl)-1,3-Oxazolidin-2-Ones As Antibacterial Agents
01/24/2008US20080021011 Therapeutic compounds
01/24/2008US20080021010 2,4-dichloro-N-{[1- (propylsulfonyl)-3-pyridin-2- ylazetidin-3- yl]methyl}benzamide; neurological and psychiatric disorders associated with glycinergic or glutamatergic neurotransmission dysfunction
01/24/2008US20080021009 1,2,4-Oxadiazole Derivatives as Dipeptidyl Peptidase-IV Inhibitors for the Treatment or Prevention of Diabetes
01/24/2008US20080019915 including cystic fibrosis transmembrane conductance regulator ("CFTR"); N[6-(2-hydroxymethylphenyl-1yl)-5-methylpyrimidine][(4-methoxophenyl-1-yl)cyclopopyl]-amide; genetic disorders; respiratory system disorders, cystic fibrosis, hereditary emphysema and hemochromatosis, coagulation-fibrinolysis
01/24/2008US20080017846 1,3-Bis[2-(2,2'-bipyridin-6-yl)-1,3,4-oxadiazol-5-yl]benzene; excellent electron injecting and transporting performances and hole blocking ability; high stability in a thin film state; high efficiency and high durability; organic electroluminescent devices
01/24/2008US20080016674 Method And Installation Means For Installing An Electrical Machine
01/24/2008CA2659524A1 Novel chromene and thiochromene carboxamide derivatives, methods for preparing same and therapeutic applications of same
01/24/2008CA2659155A1 Substituted azole aromatic heterocycles as inhibitors of 11.beta.-hsd-1
01/24/2008CA2658573A1 Cgrp receptor antagonists
01/24/2008CA2658190A1 Di-amino-substituted heterocyclic compounds and methods of use
01/24/2008CA2657850A1 Novel pyridazine derivatives
01/24/2008CA2657776A1 Triazolyl phenyl benzenesulfonamides
01/24/2008CA2657280A1 Macrocyclic compounds useful as bace inhibitors
01/24/2008CA2657258A1 Amino-piperidine derivatives as cetp inhibitors
01/24/2008CA2656715A1 Compounds and compositions as itpkb inhibitors
01/24/2008CA2644047A1 Heterobicyclic carboxamides as inhibitors for kinases
01/23/2008EP1880995A1 Method for producing indole derivative having piperidine ring
01/23/2008EP1879904A1 4" amino linked macrolides useful for the treatment of microbial infections
01/23/2008EP1879887A2 Npy antagonists, preparation and use
01/23/2008EP1879884A1 Azole-based phosphodiesterase inhibitors
01/23/2008EP1879882A1 3 -m0n0- and 3 , 5-disubstituted piperidine derivatives as renin inhibitors
01/23/2008EP1879881A2 Inhibitors of 11-beta hydroxysteroid dehydrogenase type i
01/23/2008EP1879879A1 Compounds and methods for the treatment or prevention of flavivirus infections
01/23/2008EP1879858A2 Processes for preparing biaryl ureas and analogs thereof
01/23/2008EP1879573A1 Modulators of indoleamine 2,3-dioxygenase and methods of using the same
01/23/2008EP1773825B1 Dioxazinyl-substituted thienylsulphonylaminocarbonyl compounds
01/23/2008EP1725232B1 (indol-3-yl)-heterocycle derivatives as agonists of the cannabinoid cb1 receptor
01/23/2008EP1667635A4 Sulfonylaminovalerolactams and derivatives thereof as factor xa inhibitors
01/23/2008EP1636215B1 Furazanobenzimidazoles
01/23/2008EP1569934B1 Cyclopropyl compounds as ccr5 antagonists
01/23/2008EP1432313B1 N-thio-nicotinamide derivatives and related compounds for use as pesticides
01/23/2008EP1322619B1 Isoquinolinone potassium channel inhibitors
01/23/2008EP1272178B1 Bilirubin or biliverdin degradation fragments
01/23/2008EP1257547B1 1,3-disubstituted pyrrolidines as alpha-2-adrenoceptor antagonists
01/23/2008EP1020465B1 Stereoisomeric indole compounds, process for the preparation of the same, and use thereof
01/23/2008EP0812321B1 Prokinetic oxadiazoles
01/23/2008CN101111488A Novel compounds
01/23/2008CN101111486A 抗糖尿病二环化合物 Antidiabetic bicyclic compound
01/23/2008CN101111247A Preventive or therapeutic agent for herpesvirus-related disease
01/23/2008CN101108849A Benzo**azine compound having crystal structure and method of producing the same
01/23/2008CN101108830A Cyclic compound, process for producing the same, and pest control agent
01/23/2008CN100363361C Hetaryl-substd. heterocycles
01/23/2008CN100363348C PgD2 receptor antagonists for the treatment of inflammatory diseases
01/23/2008CN100363346C Small molecular inhibiting agent for coronavirus main proteinase, its preparation method and uses
01/22/2008US7321063 Sulfonamide inhibitors of aspartyl protease
01/22/2008US7320995 Lung melanoma metastasis, rheumatoid arthritis, 1-isopropylsulfonyl-2-amino-6-(2-(2,6-difluorophenyl)-5-(phenyl)-imidazol-4-yl)-benzimidazole
01/22/2008US7320994 {2-[1-(3,5-bis-trifluoromethyl-benzyl)-5-pyridin-4-yl-1H-[1,2,3]triazol-4-yl]-pyridin-3-yl}-(2-chloro-phenyl)-methanone; anxiety, depression, psychosis, and schizophrenia and other psychotic disorders; neurodegenerative disorders, multiple sclerosis and amyotrophic lateral sclerosis
01/22/2008US7320993 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic useful as cytostatic and immuosuppressive agents
01/22/2008US7320989 E.g., {4-Chloro-3-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethoxy]phenyl}-(2-methylquinolin-4-yl)amine; congestive heart failure, stroke, antiischemic, -arrhythmia, -arthritis, -diabetic, -inflammatory, -ulcer and hypotensive agents; urogenital, bone, respiratory, cardiovascular and nervous systems disorders
01/22/2008US7320978 Inflammations of the respiratory system, locomotor system traumas, and edemas; 1-{[5-(4-Chlorophenyl)-4-(2,4-dichlorophenyl)-1,3-oxazol-2-yl]carbonyl}-4-(3-methylphenyl)piperazine
01/22/2008US7320973 5,11-Dihydrodiaryl[b,e][1,4,]oxazepine derivatives for gastrointestinal disorder treatment; irritable bowel syndrome
01/22/2008CA2305807C Substituted fused heterocyclic compounds
01/22/2008CA2281721C Phthalazines with angiogenesis inhibiting activity
01/17/2008WO2008008518A1 Substituted diazepan orexin receptor antagonists
01/17/2008WO2008008327A2 Xinafoate salt of a substituted 5-oxazol-2-yl-quinoline compound
01/17/2008WO2008008022A1 Isoindoline derivatives for the treatment of arrhythmias
01/17/2008WO2008007390A2 An improved process for purification of zolmitriptan
01/17/2008WO2008006795A2 Indole compounds
01/17/2008WO2008006794A1 Indole compounds having affinity to the ep1 receptor
01/17/2008WO2008006793A1 Indole compounds
01/17/2008WO2008006790A1 Indole compounds
01/17/2008WO2008006583A1 Pyrimidine derivatives as alk-5 inhibitors
01/17/2008WO2008006561A1 Substituted isoxalines, pharmaceutical compositions containing same, methods of preparing same, and uses of same
01/17/2008WO2008006560A1 Substituted sulphoximines as tie2 inhibitors and salts thereof, pharmaceutical compositions comprising same, methods of preparing same and uses of same
01/17/2008WO2008006479A1 2-(heteroaryl) alkyl indazole 6-phenyl and thienyl methyl amide as thrombin inhibitors
01/17/2008WO2008006372A1 (3-aryl-piperazin-1-yl), (2-aryl-morpholin-4-yl) and (2-aryl- thiomorpholin-4-yl) derivatives of 6,7-dialkoxyquinazoline, 6,7- dialkoxyphtalazine and 6,7-dialkoxyisoquinoline
01/17/2008WO2007084413B1 Methods for treating hepatitis c
01/17/2008WO2007074078A3 Aryl-isoxazol-4-yl-imidazole derivatives
01/17/2008WO2007019080A3 Tricyclic beta-secretase inhibitors for the treatment of alzheimer's disease
01/17/2008WO2006056930A3 Novel 4 -aminopiperidine derivatives as plasmepsin ii inhibitors
01/17/2008US20080015242 Use of N-[3-[2-[2-(3-methylindazol-6-yloxy)ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide or salt for treating diabetes, obesity, hyperlipidemia and urinary incontinence; drug interaction side effect reduction
01/17/2008US20080015238 Cycloalkylmethoxy-substituted acetic acid derivatives, processes for their preparation and their use as pharmaceuticals
01/17/2008US20080015237 New compounds i/418
01/17/2008US20080015234 Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
01/17/2008US20080015233 2,4,6-Substituted Pyridyl Derivative Compounds Useful as Beta-Secretase Inhibitors for the Treatment of Alzheimer's Disease
01/17/2008US20080015232 Schweinfurthin analogues
01/17/2008US20080015225 Dimeric Piperidine Derivatives
01/17/2008US20080015204 Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
01/17/2008US20080015203 Such as 3-[(1S)-2-hydroxy-1-methylethoxy]-5-[4-(methylsulfonyl)phenoxy]-N-1,3-thiazol-2-ylbenzamide; glucokinases (Glk)
01/17/2008US20080015192 Inhibitors of polo-like kinases
01/17/2008US20080015191 Pyrazines and Pyridines and Derivatives Thereof as Therapeutic Compounds
01/17/2008US20080015190 Inhibitors of Histone Deacetylase