| Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687) |
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| 09/12/2008 | WO2008091580A3 Fungicidal amides |
| 09/12/2008 | WO2008089933A3 Benzoquinazole derivatives |
| 09/12/2008 | WO2008070016A3 Inhibitors of akt activity |
| 09/12/2008 | WO2008012227A8 Pyrazoles as glucokinase activators |
| 09/12/2008 | WO2004078116A9 P38 inhibitors and methods of use thereof |
| 09/12/2008 | CA2680177A1 Metalloprotease inhibitors containing a heterocyclic moiety |
| 09/12/2008 | CA2680173A1 Metalloprotease inhibitors containing a heterocyclic moiety |
| 09/12/2008 | CA2679305A1 Pyrrole compounds |
| 09/12/2008 | CA2679249A1 Compounds and compositions as modulators of gpr119 activity |
| 09/12/2008 | CA2679101A1 Heterocyclic compounds, compositions comprising them and methods of their use |
| 09/11/2008 | US20080221206 less anesthetic activity, but with more anti-inflammatory and spasmolytic activity; asthma, rhinitis, allergic urticaria, chronic lung inflammation associated with eosinophilia, following the example of atopic asthma and chronic intestinal inflammation, as colitis for instance |
| 09/11/2008 | US20080221196 Pharmaceutically active isoindoline derivatives |
| 09/11/2008 | US20080221178 Benzimidazole Derivatives,Compositions Containing Them, Preparation Thereof and Uses Thereof |
| 09/11/2008 | US20080221122 cancer and non-cancer diseases associated with vascular proliferation; mitoxantrone resistant, taxol resistant cancers |
| 09/11/2008 | US20080221116 for the treatment of benign prostatic hypertrophy and/or lower urinary tract symptoms; with finasteride |
| 09/11/2008 | US20080221103 4-(3-Methyl-2,5-dioxo-2,5-dihydro-1H-pyrrol-1-ylamino)-6-(methylthio)-2-phenylpyrimidine-5-carbonitrile; having significant in vitro TNF- alpha inhibitory activity useful for the treatment of various inflammatory diseases such as arthritis, inflammatory bowel disease, psoriasis, asthma, COPD, cancer etc. |
| 09/11/2008 | US20080221100 Soluble epoxide hydrolase inhibitors |
| 09/11/2008 | US20080221095 increased potency and selectivity in relation to currently known MMP-13, MMP-8 and MMP-3 inhibitors; treating rheumatoid arthritis, osteoarthritis or inflammation; squaramide or benzoxazinone moiety |
| 09/11/2008 | US20080221094 Metalloprotease inhibitors containing a squaramide moiety |
| 09/11/2008 | US20080221093 Metalloprotease inhibitors containing a heterocyclic moiety |
| 09/11/2008 | US20080221086 Novel Inhibitors of Glutaminyl Cyclase |
| 09/11/2008 | US20080221082 of the alpha V beta 3 integrin receptor; , thromboembolic events, cardiovascular disorders, lung diseases, disorders of the CNS, the kidney, the gastrointestinal tract or inflammation |
| 09/11/2008 | US20080216606 Grinding to uniform particle size; heating; pressurization;; extraction from ores, concentrates |
| 09/10/2008 | EP1967519A1 3,4-dihydrobenzoxazine compound and inhibitor of vanilloid receptor type 1 (vr1) activity |
| 09/10/2008 | EP1967517A1 Probe for diagnosis of conformational disease |
| 09/10/2008 | EP1966195A2 5-aryl isoxazolines for controlling invertebrate pests |
| 09/10/2008 | EP1966187A1 Piperazine compounds useful as antagonists of c-c chemokines (ccr2b and ccr5) for the treatment of inflammatory diseases |
| 09/10/2008 | EP1966176A1 Heterocyclic gaba-b modulators |
| 09/10/2008 | EP1966171A1 Improved process for the preparation of 4-(benzimidazolylmethylamino)-benzamides and the salts thereof |
| 09/10/2008 | EP1966170A2 Estrogen modulators |
| 09/10/2008 | EP1966167A1 Diaryltriazolmethylamine derivatives, preparation and therapeutic use thereof |
| 09/10/2008 | EP1966151A1 Polycyclic indazole derivatives that are erk inhibitors |
| 09/10/2008 | EP1966144A1 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors |
| 09/10/2008 | EP1966134A1 Novel fused pyrrole derivatives |
| 09/10/2008 | EP1966132A2 Compounds which modulate the cb2 receptor |
| 09/10/2008 | EP1965807A2 S1p receptor modulating compounds and use thereof |
| 09/10/2008 | EP1965645A2 Isoxazolines for controlling invertebrate pests |
| 09/10/2008 | EP1597240B1 Bicyclic heterocycles, medicaments containing said compounds, use thereof, and method for the production thereof |
| 09/10/2008 | EP1438053B1 Pyrimidine derivatives, pharmaceutical agent containing said compounds, use and method for making same |
| 09/10/2008 | EP1437349B9 Substituted isoxazoles and the use thereof as antibiotics |
| 09/10/2008 | EP1323710B1 Nitrogenous five-membered ring compounds |
| 09/10/2008 | CN101263139A Isoxazolo derivatives as GABA A alpha5 inverse agonists |
| 09/10/2008 | CN101263138A Salicylate and gentisate salts of a piperazine compound |
| 09/10/2008 | CN101263137A Compound having oxadiazole ring structure bonded with aromatic heterocyclic ring and organic electroluminescent device |
| 09/10/2008 | CN101263133A New pyridine analogues |
| 09/10/2008 | CN101263125A Quinazoline derivatives useful in cancer treatment |
| 09/10/2008 | CN101263124A Quinazoline derivatives useful in cancer treatment |
| 09/10/2008 | CN101263116A Novel heterobicyclic derivatives useful as inhibitors of liver carnitine palmitoyl transferase |
| 09/10/2008 | CN101260106A Raf kinase inhibitor, preparing method and use thereof |
| 09/10/2008 | CN101260075A Aralkylpiperidine derivative and application thereof in preparing analgesic and sedative medicament |
| 09/09/2008 | US7423159 Agent for preventing or treating neuropathy |
| 09/09/2008 | US7423156 Optionally fused oxazolyl- or thiazolyl-aminophenylbenzoyl(cyclo)alkanoic acid derivatives, e.g., trans-(1R,2R)-2-({3'-fluoro-4'-,[(6-fluoro-1,3-benzothiazol-2-yl)amino]-1,1'-biphenyl-4-yl}carbonyl)cyclopentanecarboxylic acid; diacylglycerol O-acyltransferase type 1 inhibitors |
| 09/09/2008 | US7423150 Substituted benzazoles and methods of their use as inhibitors of Raf kinase |
| 09/09/2008 | US7423148 Small molecule PI 3-kinase inhibitors and methods of their use |
| 09/09/2008 | US7423147 Therapy of Histamine H3 receptor mediated diseases |
| 09/09/2008 | US7423058 Inhibitors of hepatitis C virus NS3 protease |
| 09/09/2008 | US7423052 Piperidine compounds for use as orexin receptor antagoinst |
| 09/09/2008 | US7423049 e.g., 2-(5-fluoro-2-tolyl)-4-(4-aminocarbonylpiperazinylmethyl)-6-[a-aminocarbonyl-2,6-dichlorobenzyl]pyridine; mitogen-activated protein kinase inhibitor; antiinflammatory agent, autoimmune diseases |
| 09/09/2008 | US7423048 eating disorders of disturbed fundus such as dyspepsia, early satiety, bloating, anorexia; fundic relaxation; 1-(1-((2,3-dihydro(1,4)dioxino(2,3-b)pyridin-3-yl)methyl) -4- piperidinyl)-2-imidazolidinone; improved pharmacokinetics, less vasoconstriction, side effect reduction, sustain release |
| 09/09/2008 | US7423040 Stable crystalline form of bifeprunox mesylate, dosage forms thereof and methods for using same |
| 09/09/2008 | US7423038 Compounds and compositions as protein kinase inhibitors |
| 09/09/2008 | US7423037 Morpholine derivatives as norepinephrine reuptake inhibitors |
| 09/09/2008 | US7423036 Long-acting betamimetics for the treatment of respiratory complaints |
| 09/09/2008 | US7423030 1-amino-phthalazine derivatives, the preparation and the therapeutic use thereof |
| 09/09/2008 | CA2252163C D-proline derivatives |
| 09/09/2008 | CA2225756C Substituted cyanophenyl uracils |
| 09/04/2008 | WO2008106047A2 Carbamate compounds |
| 09/04/2008 | WO2008105607A1 Heteroaryl-imidazole derivatives as cannabinoid cb1 receptor antagonists |
| 09/04/2008 | WO2008105515A1 Novel hydroxamic acid derivative |
| 09/04/2008 | WO2008105442A1 Sulfonamide derivative |
| 09/04/2008 | WO2008105408A1 Novel pyrrole derivative having ureide group and aminocarbonyl group as substituents |
| 09/04/2008 | WO2008104875A1 Oxazolidinones as cholesterol absorption inhibitors |
| 09/04/2008 | WO2008104869A1 Nicotinamide derivatives as inhibitors of h-pgds and their use for treating prostaglandin d2 mediated diseases |
| 09/04/2008 | WO2008104754A1 Novel pyrimidine derivatives 698 |
| 09/04/2008 | WO2008104512A2 Novel polymorphs of aprepitant and processes for preparation |
| 09/04/2008 | WO2008104472A1 2, 4 -diaminopyrimidine derivatives and their use as p2x antagonists or as prodrugs thereof |
| 09/04/2008 | WO2008104135A1 A method for the preparation of zolmitriptan |
| 09/04/2008 | WO2008104134A2 A method for the preparation of zolmitriptan |
| 09/04/2008 | WO2008104077A1 Small molecule inhibitors of protein arginine methyltransferases (prmts) |
| 09/04/2008 | WO2008047229A3 Biaryl ether urea compounds |
| 09/04/2008 | US20080214645 Administering 2-(1H-1-Indol-3-ylsulfanyl)benzyl]dimethyl amine; general anxiety disorder, social anxiety disorder, post traumatic stress disorder, obsessive compulsive disorder, panic disorder, panic attacks, specific phobias, social phobia and agoraphobia |
| 09/04/2008 | US20080214644 [2-(4-Fluoro-]. H-indol-3-ylsulfanyl)benzyl]dimethyl amine; depression, anxiety disorders including general anxiety disorder, social anxiety disorder, post traumatic stress disorder, obsessive compulsive disorder, panic disorder, panic attacks |
| 09/04/2008 | US20080214623 N-(2,2-Dimethylpropyl)-6-{3-fluoro-5-[(3-isoxazolylamino)carbonyl]-2-methylphenyl}-3-pyridinecarboxamide; inhibitors of p38 kinase |
| 09/04/2008 | US20080214620 Novel inhibitors of glutaminyl cyclase |
| 09/04/2008 | US20080214617 antitumor agents; anticancer agents; structurally related to the leptomycin family; Leptolstatin |
| 09/04/2008 | US20080214608 4-Amino-3,3-dimethylpiperidine; reduced toxicity, and improved pharmacology and pharmacokinetics |
| 09/04/2008 | US20080214565 Oxazolidinone Derivatives as Antimicrobials |
| 09/04/2008 | US20080214546 N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase |
| 09/04/2008 | US20080214545 4-{3-tert-butyl-5-[({[4-(pyridin-4-yloxy)phenyl]amino}carbonyl)amino]-1H-pyrazol-1-yl}-N-(2-pyrrolidin-1-ylethyl)benzamide; antiproliferatives; angiogenesis inhibitors |
| 09/04/2008 | US20080214544 N-(4-(6-(1-methyl-6-oxo-2-(phenylamino)-1,6-dihydropyrimidin-5-yl)pyridin-3-yloxy)pyridin-2-yl)pyrrolidine-1-carboxamide; anticarcinogenics, antiproliferatives, angiogenesis inhibitors; hepatocyte growth factor mediated diseases |
| 09/04/2008 | US20080214543 Antiandrogen; prostate cancer; excellent oral pharmacokinetics |
| 09/04/2008 | US20080214542 1-(5-methoxyisoindolin-2-yl)-6-[4-(3-trifluoromethylphenyl)piperazin-1-yl]hexan-1-one; amidation of an isoindole with a 4-phenylpyrimidinylalkanoic acid or amination of a N-haloalkylcarbonyl isoindole with a 4-phenylpyrimidine; antidepressant, neuroleptic agent; drug abuse, impotency, Parkinson's Disease |
| 09/04/2008 | US20080214539 Benzisoxazole Piperidine Compounds and Methods of Use Thereof |
| 09/04/2008 | US20080214537 Bridged phenanthridines |
| 09/04/2008 | US20080214536 4-((4aR,10bR)-8,9-Dimethoxy-1,2,3,4,4a,10b-hexahydro-phenanthridin-6-yl)-N-(2-methoxyethyl)-N-methyl-benzamide; phosphodiesterase 4 inhibitors; respiratory system disorders |
| 09/04/2008 | US20080214533 Anticoagulants, thrombolytic agents; amidating a p-(hydroxy-protected alkylamino)aniline with a (hetero)arylaminocarbonyl-(hetero)aryl carboxylic acid; deblocking, reacting with cyanogen bromide and cyclizing |
| 09/04/2008 | US20080214526 Macrocyclic Compounds and Compositions Useful as Bace Inhibitors |
| 09/04/2008 | US20080214524 e.g. N-[2-(3-fluorophenyl)ethyl]-N'-isoquinolin-5-ylurea; opioid receptor inhibitor; analgesic, antiinflammatory agent; inflammatory thermal hyperalgesia, urinary incontinence and bladder overactivity |
| 09/04/2008 | US20080214448 Compounds, Methods and Formulations for the Oral Delivery of a Glucagon-Like Peptide (Glp)-1 Compound or a Melanocortin-4 Receptor (Mc4) Agonist Peptide |
| 09/04/2008 | US20080213822 Methods for diagnosing celiac sprue and reagents useful therein |