Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
08/1999
08/19/1999WO1999026930A3 Benzylidene pyrazolones and use as herbicide
08/19/1999WO1999015894A3 Method of identification of leads or active compounds
08/19/1999DE19806438A1 New pyrimidinyloxy-propionic acid derivatives useful as endothelin receptor antagonists in treatment of e.g. cardiac insufficiency, restenosis, hypertension, kidney failure, asthma and prostate cancer
08/19/1999DE19806348A1 3,4-Dihydrochinolin-Derivate und ihre Verwendung in Arzneimitteln 3,4-dihydroquinoline derivatives and their use in medicaments
08/19/1999CA2321218A1 Condensed heterocyclic system derivatives, preparation, pharmaceutical compositions containing them
08/19/1999CA2320378A1 Cyclic dipeptides and azetidinone compounds and their use in treating cns injury and neurodegenerative disorders
08/18/1999EP0936221A1 Novel 2,4-dioxopyrrolidine and 2,4-dioxotetrahydrofuran derivatives and medicines containing the same as the active ingredient
08/18/1999EP0936216A1 Novel acetamide derivatives and protease inhibitors
08/18/1999EP0935597A2 Dihydropyrones with improved antiviral activity
08/18/1999CN1226246A Noval tricyclic N-cyanoimines useful as inhibitors of farnesyl-protein transferase
08/18/1999CN1226243A Benzodihydropyran derivative
08/18/1999CN1226238A Sulphonyl-mercapto-triazolyl derivative and their use as microbiocides
08/18/1999CN1226237A Thiocyano-triazolyl derivatives and their use as microbicides
08/18/1999CN1226235A Mercapto-imidazolyl derivatives and their use as microbicides
08/18/1999CN1044707C Substituted aminoalkylaminopyridine, preparation method, its use and medicinal composition containing same compound
08/17/1999US5939560 Inhibitors of DP-mediated processes, compositions and therapeutic methods thereof
08/17/1999US5939559 Herbicides from pyrazole ketones
08/17/1999US5939552 Resolution of enantiomorphs with batch system chromatography or moving bed chromatography
08/17/1999US5939462 NPY5 receptor antagonists and methods for using same
08/17/1999US5939447 Substituted benzopyrans
08/17/1999US5939440 Fungicides and bactericides
08/17/1999US5939439 Enzyme inhibitors in carriers for ras proteins
08/12/1999WO1999040086A1 Pyran derivatives and use thereof
08/12/1999WO1999040085A1 Benzofuran-4-carboxamides and their therapeutic use
08/12/1999WO1999040084A1 Salts of paroxetine
08/12/1999WO1999040081A1 Novel antifungal compounds and process for producing the same
08/12/1999WO1999040080A1 Hydroxamic and carboxylic acid derivatives
08/12/1999WO1999040075A1 Sulfonamide derivatives, process for producing the same and utilization thereof
08/12/1999WO1999040072A1 Five-membered, benzo-condensed heterocycles used as antithrombotic agents
08/12/1999WO1999040071A1 Urocanic acid derivatives
08/12/1999WO1999040068A2 2-aminoquinoline derivatives having d4-agonistic activity
08/12/1999DE19805431A1 Heteroaromatische Oligoamide als Affinitätsliganden Heteroaromatic oligoamides as affinity ligands
08/12/1999CA2319652A1 Salts of paroxetine
08/12/1999CA2319494A1 5-membered heterocyclic condensed benzoderivatives, the preparation thereof and their use as pharmaceuticals
08/12/1999CA2319060A1 Urocanic acid derivatives
08/12/1999CA2317478A1 Benzofuran-4-carboxamides and their therapeutic use
08/12/1999CA2317476A1 Hydroxamic and carboxylic acid derivatives
08/12/1999CA2317017A1 Sulfonamide derivatives, their production and use
08/11/1999EP0934931A2 3-Benzylidene-2-indolinones and their analogues as tyrosine kinase activity modulators
08/11/1999EP0934930A1 Process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds from N-(perfluoroalkylmethyl)arylimidoyl chloride compounds
08/11/1999EP0934929A1 Process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds from N-(arylmethylene)-1-chloro-1-(perfluoroalkyl) methylamine compounds
08/11/1999EP0934527A1 Non radioactive receptor assay suitable for quantitative and qualitative analysis of trace amounts of receptor binding analyte
08/11/1999EP0934314A1 N-substituted azaheterocyclic compounds
08/11/1999EP0934313A1 N-substituted azaheterocyclic compounds
08/11/1999EP0934312A1 1,4-disubstituted piperazines
08/11/1999EP0934311A2 New heterocyclylmethyl-substituted pyrazol derivates
08/11/1999EP0934309A1 New pyridyl alkane acid amides as cytostatics and immunosuppressives
08/11/1999EP0934308A1 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling chemical synaptic transmission
08/11/1999EP0934307A1 Substituted azabicylic compounds and their use as inhibitors of the production of tnf and cyclic amp phosphodiesterase
08/11/1999EP0934303A2 Compounds useful for inhibition of farnesyl protein transferase
08/11/1999EP0934298A1 NOVEL (+)-ENANTIOMERS OF $i(CIS)-3,4-CHROMAN DERIVATIVES USEFUL IN THE PREVENTION OR TREATMENT OF ESTROGEN RELATED DISEASES OR SYNDROMES
08/11/1999EP0934296A1 Chroman derivatives
08/11/1999EP0934295A1 Novel bi-aromatic dibenzofuran derivatives and their use in human and veterinary medicine and in cosmetics
08/11/1999EP0934291A1 Protease inhibitors
08/11/1999EP0934283A2 Arthropodicidal and fungicidal cyclic amides
08/11/1999EP0934281A1 1-phenyl-benzimidazole compounds and their use as baga- a? receptor modulators
08/11/1999EP0934280A1 Pde iv inhibiting 2-cyanoiminoimidazole derivatives
08/11/1999EP0934276A1 Anthranilic acid derivatives as multi drug resistance modulators
08/11/1999EP0934274A1 Substituted pyridines and biphenyls as anti-hypercholesterinemic, anti-hyperlipoproteinemic and anti-hyperglycemic agents
08/11/1999EP0934264A1 Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists
08/11/1999EP0789706A4 Sugar modified nucleosides and their use for synthesis of oligonucleotides
08/11/1999EP0741724B1 Neuroprotective chroman compounds
08/11/1999EP0584223B1 Novel immunosuppressive compounds
08/11/1999CN1225635A Substituted pyrazolyl-pyrazole derivatives, process for their prepn. and their use as agents with herbicidal effect
08/11/1999CN1225633A Taxane derivatives and drugs contg. same
08/11/1999CN1225629A Novel pyrrole derivatives
08/11/1999CN1225360A Substituted imidazolidine derivatives, their prepn., their use and pharmaceutical prepn. comprising them
08/11/1999CN1044605C Benzopyran and oxazine derivative
08/10/1999US5936128 5,6-dihydropyrone derivatives as protease inhibitors and antiviral agents
08/10/1999US5935992 Substituted 1,2,3,4-tetrahydro-2-dibenzofuranamines and 2-aminocyclohepta 6,!benzofurans
08/10/1999US5935987 Transdermal delivery of 3,4-diarylchromans
08/10/1999US5935982 Methods of treating retroviral infection and compounds useful therefor
08/10/1999US5935977 Substituted vinyl pyridine derivative and drugs containing the same
08/10/1999US5935973 Affinity for 5-ht1a, alpha1, alpha2 and/or d2 receptors; antidepressants, anxiolytic agents, psychoses, dyskinesias, parkinson's disease, hypotensive agents, tourette's syndrome, obsessive-compulsive behaviour, panic attacks, social phobias
08/10/1999US5935972 Benzofuran derivatives as tachykinin antagonists
08/10/1999US5935966 Compounds that block the activation of transcription factors through inhibition of a family of specific kinases, decreasing proinflammatory proteins to treat autoimmune diseases and as general antiinflammatory agents
08/10/1999US5935963 Piperazinones, their production and use
08/10/1999US5935961 Compounds such as n-methyl 2-(2-(6'-(3?,4?-dichlorophenyl)-pyridazin-3'-on-2'yl)-methylphenyl)-2 -methoxyiminoacetamide useful against powdery mildew, blight in cucumbers, tomatoes, and wheat for example
08/10/1999US5935957 Compounds, compositions and methods for treating influenza
08/10/1999US5935954 Compounds with improved multi-drug resistance activity
08/10/1999US5935907 Phenylacetylene derivatives
08/10/1999CA2260698A1 Pyrrolidine and piperidine derivatives
08/10/1999CA2011144C Nicotinic acid derivatives and pharmaceutical compositions comprising same
08/10/1999CA1340695C Antibacterial agents
08/09/1999CA2260735A1 Process for the preparation of 2-aryl-5-(perfluoroalkyl) pyrrole compounds from n-(arylmethylene)-1-chloro-1-(perfluoroalkyl) methylamine compounds
08/09/1999CA2260699A1 Process for the preparation of 2-aryl-5-(perfluoroalkyl) pyrrole compounds from n-(perfluoroalkylmethyl) arylimidoyl chloride compounds
08/05/1999WO1999038846A1 Immunosuppressive agents
08/05/1999WO1999038845A1 Ppar-gamma modulators
08/05/1999WO1999038844A1 Method for preparing an n-[(aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
08/05/1999WO1999038514A1 Cyclic amine modulators of chemokine receptor activity
08/05/1999WO1999024398A3 Urea derivatives and their use as integrin inhibitors
08/05/1999WO1995031429A8 Photocleavable agents and conjugates for the detection and isolation of biomolecules
08/05/1999DE19903870A1 New 3,3,5,5-tetraalkyl-2-oxo-1,4-piperazine derivatives, used as light, heat and oxygen stabilizers e.g. in photographic and reprographic materials and in paper
08/05/1999DE19804085A1 New benzo-condensed heterocyclic compounds useful in treatment of thrombosis and prevention of vascular occlusion
08/05/1999CA2319781A1 Cyclic amine modulators of chemokine receptor activity
08/05/1999CA2318601A1 Method for preparing an n-[(aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
08/04/1999EP0933372A1 Sulphonamide derivatives as prodrugs of aspartyl protease inhibitors
08/04/1999EP0932403A1 Use of condensated (hetaryl-substituted) 1-benzal-3-pyrazol derivates for treating special diseases of the cardiovascular and the central nervous systems
08/04/1999EP0755387B1 Oxidative purification of biomass extracts containing taxol and cephalomannine using ozone and girard reagents
08/04/1999EP0701555B1 Indazole derivatives