Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
03/1999
03/18/1999CA2302284A1 Ureido and thioureido derivatives of 4-amino-2(5h)-furanones and 4-amino-2(5h)-thiophenones as antitumor agents
03/18/1999CA2247551A1 Novel imidazolidine derivatives, their preparation, their use and pharmaceutical preparations comprising them
03/17/1999EP0902028A1 Tetrazoline herbicides
03/17/1999EP0902027A1 Indole and indazole derivatives, process for their preparation and the pharmaceutical compositions containing them
03/17/1999EP0902022A1 Novel benzofuranone derivatives and process for producing the same
03/17/1999EP0902018A2 2-(Arylphenyl)amino-imidazoline derivatives
03/17/1999EP0901489A1 Antagonists of gonadotropin releasing hormone
03/17/1999EP0901488A1 2,4-diaminopyrimidine derivatives
03/17/1999EP0901487A1 Novel 2,3 disubstituted-4(3h)-quinazolinones
03/17/1999EP0901483A2 Benzofurans and benzopyrans as chronobiological agents
03/17/1999EP0901482A1 Benzofuran carboxamides and their therapeutic use
03/17/1999EP0901480A1 Process for preparing oxiranemethanamine derivatives
03/17/1999EP0901478A1 Thiocyano-triazolyl derivatives and their use as microbicides
03/17/1999EP0901477A1 Sulphonyl-mercapto-triazolyl derivatives and their use as microbicides
03/17/1999EP0901474A1 Aryl pyrimidine derivatives
03/17/1999EP0901472A1 Mercapto-imidazolyl derivatives and their use as microbicides
03/17/1999EP0901470A1 Indole derivatives useful as endothelin receptor antagonists
03/17/1999EP0901469A1 Arylalkylpiperazine compounds as antioxidants
03/17/1999EP0626962B1 Substituted phenylheterocyclic herbicides
03/17/1999EP0626954B1 Benzocycloheptenes, benzoxepines and benzothiepines
03/17/1999EP0603404B1 Process for producing glycide derivative
03/17/1999CN1211252A Coralyne analogs as topoisomerase inhibitors
03/17/1999CN1211248A Novel substituted N-methyl-N-(4-(4-(1H-benzimidazol-2-yl) [1,4] diazepan-1-yl)-1-(aryl) butyl) benzamides useful for treatment of allergic diseases
03/17/1999CN1211247A Novel substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl) butyl) benzamides useful for treatment of allergic diseases
03/17/1999CN1211246A Novel substituted N-methyl-N-(4-(1H-benzimidazol-2-yl-amino) piperidin-1-yl)-2-(aryl) butyl) benzamides useful for treatment of allergic diseases
03/17/1999CN1211240A Quinazoline derivatives as antitumor agents
03/17/1999CN1211238A Benzimidazole derivatives
03/17/1999CN1211183A Methods for preparation of biphenyl isoxazole sulfonamides
03/16/1999US5883253 Process for the preparation of aromatic O-sulfocarboxylic acids and sulfonylureas
03/16/1999US5883252 Aspartyl protease inhibitors
03/16/1999US5883251 Enzyme inhibitors
03/16/1999US5883116 3-(2'-alkoxybenzylidenyl)-2-indolinone and analogues thereof for the treatment of disease
03/16/1999US5883113 Tyrosine kinase inhibitors; antiproliferative and anticarcinogenic agents; diabetes, arthritis, restenosis, atherosclerosis
03/16/1999US5883102 Pharmaceutically active compounds
03/16/1999US5883099 Treatment of athersclerosis, pancreatitis obesity or hyperglycemia
03/16/1999US5883098 Used as tachykinin antagonists in the treatment of respiratory diseases, ophthalmic diseases and inflammatory diseases
03/16/1999US5883096 Di-n-substituted piperazine derivatives; alzheimer*s disease, cognition activators; synergistic mixtures with acetylcholinesterase inhibitors
03/16/1999US5883090 Endothelin receptor antagonists
03/16/1999CA2131545C Substituted pyrimidines and their use as pesticides
03/11/1999WO1999011658A1 Meta-benzamidine derivatives as serin protease inhibitors
03/11/1999WO1999011657A1 1-amino-7-isoquinoline derivatives as serine protease inhibitors
03/11/1999WO1999011640A1 Epoxysuccinamide derivatives
03/11/1999WO1999011633A1 Triazines with an adenosine antagonistic effect
03/11/1999WO1999011632A1 6,7-asymmetrically disubstituted quinoxalinecarboxylic acid deri vatives, addition salts thereof, and processes for the preparation of both
03/11/1999WO1999011627A1 2-substituted phenyl-benzimidazole antibacterial agents
03/11/1999WO1999011619A1 Phenylindole derivatives as 5-ht2a receptor ligands
03/11/1999WO1999011267A1 Pyrazinone thrombin inhibitors
03/11/1999WO1999011258A1 Lymphocyte function antigen-1 antagonists
03/11/1999WO1998056771A3 Piperazine derivatives and their use as anti-inflammatory agents
03/11/1999WO1998051672A3 A method for the preparation of tertiary amines, a compound useful therefor and alpha-2-receptor active tetrahydroisoquinoline derivatives
03/11/1999CA2302161A1 6,7-asymmetrically disubstituted quinoxalinecarboxylic acid derivatives, addition salts thereof, and processes for the preparation of both
03/11/1999CA2301520A1 Pyrazinone thrombin inhibitors
03/10/1999EP0900568A2 AMPA antagonists for the treatment of dyskinesias associated with dopamine agonist therapy
03/10/1999EP0900215A1 N-3 substituted pyrimidin-4-ones with aii antagonistic activity
03/10/1999EP0900211A1 Thiadiazolyl(thio)ureas useful as matrix metalloprotease inhibitors
03/10/1999EP0900208A1 Acyl mercapto-triazolyl derivatives and the use thereof as microbicides
03/10/1999EP0900207A1 Pyrazinone thrombin inhibitors
03/10/1999EP0900083A1 Novel substituted imidazole compounds
03/10/1999CN1210535A Taxane derivatives having pyridil substituted C13 side chain, their preparation and their use as anti-tumor agents
03/10/1999CN1210534A Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
03/10/1999CN1210532A Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
03/10/1999CN1210530A Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
03/10/1999CN1210528A Dihydrobenzofuran compounds useful as anti-inflammatory agents
03/10/1999CN1210527A Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
03/10/1999CN1210522A 2,4-diamino-1,3,5-iriazines, processes for their preparation and their use as herbicides and plant-growth regulators
03/09/1999US5880296 Racemic mixture is resolved by selective crystallization with the appropriate optically pure enantiomer of 2-phenylglycinol; antidepressant, migraine drug synthesis
03/09/1999US5880295 Process for the preparation of diamine intermediates useful in the synthesis of HIV protease inhibitors
03/09/1999US5880147 Amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prohylactic use
03/09/1999US5880141 Controlling, modulating and inhibiting tyrosine kinase signal transduction
03/09/1999US5879929 Enzymatic processes for the resolution of enantiomeric mixtures of lactams useful as intermediates in the preparation of taxanes
03/09/1999CA1340430C Preparation of antihypercholesterolemic tetrazole compounds and intermediates thereof
03/04/1999WO1999010524A1 A method of treating cancer
03/04/1999WO1999010339A1 2-aminopyridines containing fused ring substituents as nos inhibitors
03/04/1999WO1999010338A2 Benzylidene- and cinnamylidene-anabaseines as neuronal nicotinic alpha-7 receptor agonists
03/04/1999WO1999010331A1 Arylpyridazinones as prostaglandin endoperoxide h synthase biosynthesis inhibitors
03/04/1999WO1999010328A1 Heterocyclic substituted 4-benzoyl-pyrazole as herbicides
03/04/1999WO1999010325A1 Benzylidene-1,3-dihydro-indol-2-one derivatives as receptor tyrosine kinase inhibitors, particularly of raf kinases
03/04/1999WO1999009987A1 Method for treating premenstrual or late luteal phase syndrome
03/04/1999WO1999009984A1 Pyrrolidine and piperidine modulators of chemokine receptor activity
03/04/1999WO1999009983A1 4-aryl-3-aminoquinoline-2-one derivatives as potassium channel modulators
03/04/1999WO1998055454A3 Benzofurans and benzothophenes as suppressors of neurodegeneration
03/04/1999WO1998053790A3 Compounds that inhibit the binding of vascular endothelial growth factor to its receptors
03/04/1999DE19738084A1 New 3-aryl-methyl-uracil derivatives
03/04/1999CA2301857A1 A method of treating cancer
03/04/1999CA2301549A1 4-aryl-3-aminoquinoline-2-one derivatives as potassium channel modulators
03/04/1999CA2298979A1 Method for treating premenstrual or late luteal phase syndrome
03/04/1999CA2298813A1 Pyrrolidine and piperidine modulators of chemokine receptor activity
03/04/1999CA2245755A1 2-(arylphenyl)amino-imidazoline derivatives
03/03/1999EP0899263A2 Fused pyrimidine derivatives and medicaments thereof for a blood oxygen partial pressure amelioration
03/03/1999EP0898569A1 Piperidines and pyrrolidines
03/03/1999EP0898565A1 Substituted pyridines/pyrimidines, process for their production and their use as pest control agents
03/03/1999EP0805993A4 Photochromic substituted naphthopyran compounds
03/03/1999EP0777666B1 Substituted piperidines useful for the treatment of allergic diseases
03/03/1999EP0724570B1 Amidino derivatives useful as nitric oxide synthase inhibitors
03/03/1999EP0674641B1 Pyrrolopyrimidines as crf antagonists
03/03/1999EP0626957B1 Styril derivatives and processes for their preparation
03/03/1999CN1209805A Noval fused pyrrolecarboxamides and new class of GABA brain receptor ligands
03/03/1999CN1209803A Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method therefor
03/03/1999CN1209744A Vitronectin receptor antagonists
03/03/1999CN1042335C 1-acylpiperidine compounds, preparation method, medicinal composition and use thereof